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222

抑制剂 & 化合物

19

天然产物

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Cat. No. Product Name Target Signaling Pathways
T10341 Antitumor agent-19

Others Others
Antitumor agent-19 是一种肿瘤相关巨噬细胞的调节剂,在 RAW 264.7 细胞和 BMDM 细胞中的 EC50 分别为 17.18 μM 和 18.87 μM。
T10342 Antitumor agent-2

Others Others
Antitumor agent-2 具有抗炎和抗肿瘤活性,可用于研究癌症。
T39889 Antitumor agent-23

Antitumor agent-23 exhibits potent antitumoral activity, as demonstrated by its GI50 values of 38, 48, 5, 27, 80, and 28 nM against the lymphoma cell lines GRANTA-519, KARPAS-422, KARPAS-299, RAMOS, DAUDI, and RAJI respectively.
T39523 Antitumor agent-28

Antitumor agent-28 is a compound that specifically targets and inhibits the activity of the ataxia telangiectasia mutated (ATM) kinase. By doing so, it effectively impedes the progression of ATM-mediated diseases and demonstrates significant anti-cancer activity.
T12443 Antitumor agent-4

Others Others
Antitumor agent-4 is a butenylphenyl phosphate derivative, is an agent of mammary cancer and anovulatory sterility.
T14296 Antitumor agent-3

Others Others
Antitumor agent-3 is a potent compound. It comprises a new imidazopyridine having excellent antitumor activity as an active ingredient.
T3389 Antitumor agent-21

TRX818

Others Others
Antitumor agent-21 (TRX818) 是一种具有潜在的抗癌、抗炎、抗增殖、抗激素作用和抑制血管生成拟态作用的芳基-喹啉衍生物。
T72572 Antitumor agent-85

Antitumor agent-85 是一种 G-quadruplex(G4) 配体,具有稳定不同 G4-DNA 结构的能力。Antitumor agent-85 具有高效的抗肿瘤特性。
T74494 Antitumor agent-63

Antitumor agent-63(Compound 40),一种20 (S)-O-linked camptothecin (CPT) 糖复合物,作为抗肿瘤剂,对正常细胞展现出无毒性。该化合物表现出高稳定性和低topoisomeraseI (Topo I)直接抑制活性。
T79249 Antitumor agent-101

Histone Methyltransferase Chromatin/Epigenetic
Antitumor agent-101是一种针对赖氨酸甲基转移酶G9a/GLP的选择性共价抑制剂,其对G9a的IC50为8.5 nM,对GLP为5.5 nM。在PANC-1异种移植模型中,Antitumor agent-101展现了其抗肿瘤活性。
T83011 Antitumor agent-105

Antitumor agent-105(Compound 37)是一种对A549、H1299、H460、HCT116、MDA-MB-231细胞线显示出抗肿瘤活性的化合物,其IC50值分别为6.7、8.3、4.3、4.4、6.7μM。
T64128 Antitumor agent-56

Antitumor agent-56 是一种口服具有活力的 triptolide 衍生物,能够明显抑制黑色素瘤的生长,表现出抗肿瘤、抗炎和 NO 释放作用。
T64034 Antitumor agent-45

Antitumor agent-45 对 c-Met 表达具有抑制作用,能够将 A549 细胞的细胞阻滞在 G0/G1 和 G2/M 期,并诱导其凋亡。
T79434 Antitumor agent-103

Apoptosis Apoptosis
Antitumor agent-103(compound 24l)是一种诱导凋亡(apoptosis)的化合物,具备抗增殖及抗克隆形成的特性。该化合物能够导致细胞周期在G0/G1期发生阻滞,并且刺激NO的产生,表现出显著的抗肿瘤活性。
T62480 Antitumor agent-51

Antitumor agent-51 能够有效的、选择性的抑制骨肉瘤细胞的生长和迁移,作用于 MNNG/HOS 细胞 (IC50: 21.9 nM)。Antitumor agent-51 毒性较低,生物利用度极高。
T72525 Antitumor agent-48

Antitumor agent-48 是一种具有抗肿瘤活性的 2,3-dehydrosilybin 衍生物。Antitumor agent-48 对 MCF-7、NCI-H1299、HepG2 和 HT29 细胞具有细胞毒活性,IC50值分别为 8.06 µM、13.1 µM、16.51 µM 和 12.44 µM。
T63001 Antitumor agent-72

Antitumor agent-72 是一种有效的抗癌剂。Antitumor agent-72 具有抗癌活性,并通过激活 caspase-3 和裂解PARP 诱导细胞凋亡 (apoptosis)。Antitumor agent-72 可用于癌症研究。
T72575 Antitumor agent-90

Antitumor agent-90 对 PC 14 细胞和 MKN 45 细胞具有细胞毒性。Antitumor agent-90 可用于癌症研究。
T61616 Antitumor agent-38

Antitumor agent-38 is a highly effective antitumor compound that exhibits antiproliferative activity towards cancer cells. It induces cell cycle arrest specifically at the late S and G2/M phase, while not impeding microtubule formation or altering cell morphology [1].
T64071 Antitumor agent-42

Antitumor agent-42 能够抑制微管多聚和 NO 释放,表现出抗血管生成、抑制集落形成和诱导凋亡作用。
T61313 Antitumor agent-70

Antitumor agent-70 (compound 8b) is a highly potent multi-targeted kinase inhibitor, particularly targeting c-Kit. It demonstrates remarkable anti-tumor activity and the ability to induce cell apoptosis. This compound also exhibits strong inhibition of multiple myeloma, with an IC 50 value of 0.12 μM. Therefore, Antitumor agent-70 holds great potential as an effective therapy for combating cancer, especially in cases involving c-Kit. [1]
T74605 Antitumor agent-64

Antitumor agent-64 (Compound 8d),一种薯蓣皂苷元衍生物,对A549细胞系展示出显著的细胞毒性。通过线粒体相关途径促进A549细胞的凋亡(apoptosis)。
T83002 Antitumor agent-49

Antitumor agent-49 (Compound 10) 是一款 Harmine 和呋喃杂化的衍生物,带有 NO 供体且表现出抗肿瘤特性。该化合物对 HepG2 细胞线展现出显著的细胞毒性,其 IC50 值为 1.79 µM,并且能在体外产生大量的 NO。
T72523 Antitumor agent-46

Antitumor agent-46 是一种抗肿瘤剂。Antitumor agent-46 对 MCF-7 细胞具有明显更高的抗增殖活性,IC50值为 2.08 µM。
T63494 Antitumor agent-60

Antitumor agent-60 是有效的抗肿瘤药物,靶向RAS-RAF 信号通路,可与CRAF 结合 (Kd: 721.3 nM)。Antitumor agent-60 能增加癌细胞中p53和ROS 水平,使细胞核呈椭圆形和不规则形态。Antitumor agent-60 够将细胞的细胞周期阻滞在 G2/M 期,并诱导细胞凋亡 (apoptosis)。在 A549 肿瘤移植模型中,Antitumor agent-60 具有一定的抑制肿瘤生长能力。
T61806 Antitumor agent-44

Antitumor agent-44 (Compound 5n) elicits potent antitumor effects by inducing disruption of mitochondrial homeostasis, cell cycle arrest, and apoptosis in human adenocarcinoma cells. Moreover, Antitumor agent-44 demonstrates significant anti-tumor activity in a lung cancer cell xenograft mice model [1].
T63513 Antitumor agent-71

Antitumor Agent-71 是一种抗肿瘤化合物,对微管蛋白 (tubulin) 的聚集表现出抑制作用。Antitumor Agent-71 拥有抗增殖作用,对肿瘤细胞系的 IC50值范围为3.98-15.70 μM。
T72524 Antitumor agent-47

Antitumor agent-47 是一种具有抗肿瘤活性的水飞蓟宾衍生物。Antitumor agent-47 对 NCI-H1299 和 HT29 细胞具有细胞毒活性,IC50值分别为 8.07 µM 和 6.27 µM。
T72571 Antitumor agent-84

Antitumor agent-84 是一种G-quadruplex(G4) 配体,具有稳定不同 G4-DNA 结构的能力。Antitumor agent-84 具有高效的抗肿瘤特性。
T62814 Antitumor agent-77

Antitumor agent-77 对癌细胞的生长和迁移具有抑制作用,具有抗癌作用。Antitumor agent-77 能够抑制 GPx-4 和提高 COX2 引发铁下垂。Antitumor agent-77 可以激活肿瘤细胞固有凋亡通路 (Bax-Bcl-2-caspase-3),阻碍肿瘤细胞上皮间质转化 (EMT) 过程。
T78911 Antitumor agent-112

Apoptosis Apoptosis
Antitumor agent-112(compound 3a)为一有效抗肿瘤剂,能诱导细胞凋亡(apoptosis)。该化合物对A549细胞展现细胞毒活性,具有91.35 μM的IC50值。
T64222 Antitumor agent-55

Antitumor agent-55 (compound 5q) 是一种有效的抗肿瘤剂,能够有效的抑制PC3 (IC50: 0.91 μM)。Antitumor agent-55 能够将 PC3 的细胞周期阻滞 G1/S 期,诱导其凋亡,抑制细胞迁移,阻碍 PC3 的形成。
T63271 Antitumor agent-62

Antitumor agent-62 是释放 NO 的抗肿瘤剂,对癌细胞表现出抗增殖作用,能够激活线粒体凋亡 (apoptosis) 通路,能够将细胞周期阻滞到 G2/M 期。
T64014 Antitumor agent-58

Antitumor agent-58 是一种抗肿瘤剂,对 MGC-803 细胞的集落形成和细胞迁移具有有效的抑制作用,并能够诱导 MGC-803 细胞的线粒体功能障碍。Antitumor agent-58 可以激活 p38 和 JNK 信号通路,并诱导 MGC-803 细胞凋亡 (apoptosis)。Antitumor agent-58 对携带 MGC-803 细胞的异种移植模型的肿瘤生长表现出有效的抑制活性。
T61868 Antitumor agent-66

Antitumor agent-66 (Compound 4) is a derivative of (-)-cleistenolide, showcasing potential as a research tool for cancer diseases [1].
T82999 Antitumor agent-93

Antitumor agent-93 (化合物 7D) 为抗癌剂,对MDA-MB-231与HCT-116等多种肿瘤细胞系生长抑制效果显著。
T72570 Antitumor agent-83

Antitumor agent-83 是一种促凋亡蛋白 BAX 的激活剂,对肿瘤细胞有显著的抗增殖作用。Antitumor agent-83 通过诱导 BAX 的构象激活介导细胞凋亡 (Apoptosis),对 A549 细胞周期有抑制作用。Antitumor agent-83 具有良好的体外代谢稳定性和 CYP 谱。
T83010 Antitumor agent-106

Antitumor agent-106 (化合物 42),对肺癌和结肠癌细胞系展现出显著的抑制效果,IC50值介于4.2-6.6 µM。
T83007 Antitumor agent-120

Antitumor agent-120 (compound 1) 为一类黄酮化合物,来源于葛根提取。本化合物对LNCaP和PC3癌细胞的抑制作用不明显,表现出IC50s均大于50 μM。
T75078 Antitumor agent-86

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Antitumor agent-86 (compound 5a) 对MCF-7乳腺癌细胞线具有IC50值2.62 µM的抑制活性。该化合物通过促进细胞凋亡和引发细胞周期阻滞来表现其抗癌效能,并对RAS/PI3K/Akt/JNK信号传导途径具有靶向作用。
T62510 Antitumor agent-75

Antitumor agent-75 是一种新型的、有效的抗肿瘤剂。Antitumor agent-75 对癌症和正常人类细胞系具有细胞毒性作用。Antitumor agent-75 结合使用 Antitumor agent-74 时对人肺腺癌(细胞系 A549 )表现出高度选择性的细胞毒作用 (IC50: 2.8 μM)。Antitumor agent-75 能够用于研究癌症。
T62033 Antitumor agent-65

Antitumor agent-65 (Compound 5) 是 (-)-cleistenolide 的类似物/衍生物。Antitumor agent-65在癌症疾病的研究具有潜力。
T60505 Antitumor agent-43

Antitumor agent-43 (Compound 4B) 是一种有效的抗肿瘤剂,可诱导细胞周期阻滞在G2/M 期。Antitumor agent-43对 T-24 细胞的IC50值为0.5 μM。
T64022 Antitumor agent-37

Antitumor agent-37 表现出有效的抗增殖和抗转移效果。Antitumor agent-37 能够诱导严重的 DNA 损伤,进而导致 γ-H2AX 和 p53 的高表达。Antitumor agent-37 可利用线粒体凋亡通路 Bcl-2/Bax/caspase3,诱导肿瘤细胞凋亡 (apoptosis)。Antitumor agent-37 可以抑制 PD-L1 的表达,提高肿瘤组织中 CD3+ 和 CD8+ T 浸润细胞,明显改善免疫反应。
T62835 Antitumor agent-54

Antitumor agent-54 (Compound C11) 是一种 14-3-3η 蛋白抑制剂 (KD: 35 μM)。Antitumor agent-54 能够抑制几种典型的人肝癌细胞系。Antitumor agent-54 可以将细胞周期阻滞在 G1-S 期,并诱导细胞凋亡,表现出良好的代谢稳定性。
T72561 Antitumor agent-82

Antitumor agent-82是一种有效的抗肿瘤剂。Antitumor agent-82 显示出抗增殖活性。Antitumor agent-82 通过 ATG5/ATG7信号通路诱导细胞自噬 (Autophagy)。
T83001 Antitumor agent-67

Antitumor agent-67 (compound 3) 是一种高选择性抗肿瘤化合物,针对癌细胞具备显著选择性毒性,且对正常细胞损害低。该化合物经 NQO1 激活后,有效地释放鬼臼毒素(Podophyllotoxin),以消灭肿瘤细胞。在 HepG2 异种移植肿瘤模型中,Antitumor agent-67 展现出强效的肿瘤抑制能力而无显著毒副作用。
T79463 Antitumor agent-110

Apoptosis Apoptosis
Antitumor agent-110 (compound 13) 是一种抗癌咪唑四嗪,具备良好的渗透性,能够阻滞细胞周期于G2/M期并诱导apoptosis。
T79466 Antitumor agent-111

c-Met/HGFR Tyrosine Kinase/Adaptors
Antitumor agent-111(compound 46)是一款c-Met激酶抑制剂,IC50为46 nM,显示出抗肿瘤和抗增殖特性。该化合物能够导致细胞周期在G0/G1期停滞,并诱发细胞凋亡(apoptosis)。
T78909 Antitumor agent-97

Apoptosis Apoptosis
Antitumor agent-97(化合物 42)是一种有效抑制MGC 803细胞增殖与自噬(autophagy)并诱导细胞凋亡(apoptosis)的抗癌剂。该化合物还可增强MGC 803细胞中ROS的积累,适用于癌症研究。

化合物

Antitumor agent-19
Cat.No: T10341
Synonym:
Target: Others
Antitumor agent-2
Cat.No: T10342
Synonym:
Target: Others
Antitumor agent-23
Cat.No: T39889
Synonym:
Target:
Antitumor agent-28
Cat.No: T39523
Synonym:
Target:
Antitumor agent-4
Cat.No: T12443
Synonym:
Target: Others
Antitumor agent-3
Cat.No: T14296
Synonym:
Target: Others
Antitumor agent-21
Cat.No: T3389
Synonym: TRX818
Target: Others
Antitumor agent-85
Cat.No: T72572
Synonym:
Target:
Antitumor agent-63
Cat.No: T74494
Synonym:
Target:
Antitumor agent-101
Cat.No: T79249
Synonym:
Target: Histone Methyltransferase
Antitumor agent-105
Cat.No: T83011
Synonym:
Target:
Antitumor agent-56
Cat.No: T64128
Synonym:
Target:
Antitumor agent-45
Cat.No: T64034
Synonym:
Target:
Antitumor agent-103
Cat.No: T79434
Synonym:
Target: Apoptosis
Antitumor agent-51
Cat.No: T62480
Synonym:
Target:
Antitumor agent-48
Cat.No: T72525
Synonym:
Target:
Antitumor agent-72
Cat.No: T63001
Synonym:
Target:
Antitumor agent-90
Cat.No: T72575
Synonym:
Target:
Antitumor agent-38
Cat.No: T61616
Synonym:
Target:
Antitumor agent-42
Cat.No: T64071
Synonym:
Target:
Antitumor agent-70
Cat.No: T61313
Synonym:
Target:
Antitumor agent-64
Cat.No: T74605
Synonym:
Target:
Antitumor agent-49
Cat.No: T83002
Synonym:
Target:
Antitumor agent-46
Cat.No: T72523
Synonym:
Target:
Antitumor agent-60
Cat.No: T63494
Synonym:
Target:
Antitumor agent-44
Cat.No: T61806
Synonym:
Target:
Antitumor agent-71
Cat.No: T63513
Synonym:
Target:
Antitumor agent-47
Cat.No: T72524
Synonym:
Target:
Antitumor agent-84
Cat.No: T72571
Synonym:
Target:
Antitumor agent-77
Cat.No: T62814
Synonym:
Target:
Antitumor agent-112
Cat.No: T78911
Synonym:
Target: Apoptosis
Antitumor agent-55
Cat.No: T64222
Synonym:
Target:
Antitumor agent-62
Cat.No: T63271
Synonym:
Target:
Antitumor agent-58
Cat.No: T64014
Synonym:
Target:
Antitumor agent-66
Cat.No: T61868
Synonym:
Target:
Antitumor agent-93
Cat.No: T82999
Synonym:
Target:
Antitumor agent-83
Cat.No: T72570
Synonym:
Target:
Antitumor agent-106
Cat.No: T83010
Synonym:
Target:
Antitumor agent-120
Cat.No: T83007
Synonym:
Target:
Antitumor agent-86
Cat.No: T75078
Synonym:
Target: Akt
Antitumor agent-75
Cat.No: T62510
Synonym:
Target:
Antitumor agent-65
Cat.No: T62033
Synonym:
Target:
Antitumor agent-43
Cat.No: T60505
Synonym:
Target:
Antitumor agent-37
Cat.No: T64022
Synonym:
Target:
Antitumor agent-54
Cat.No: T62835
Synonym:
Target:
Antitumor agent-82
Cat.No: T72561
Synonym:
Target:
Antitumor agent-67
Cat.No: T83001
Synonym:
Target:
Antitumor agent-110
Cat.No: T79463
Synonym:
Target: Apoptosis
Antitumor agent-111
Cat.No: T79466
Synonym:
Target: c-Met/HGFR
Antitumor agent-97
Cat.No: T78909
Synonym:
Target: Apoptosis
Cat. No. Product Name Target Signaling Pathways
T83000 Antitumor agent-89

Antitumor agent-89(Compd OTS-5)为源自天然的化合物,其活性表现为轻度抑制fMLP诱导的超氧化物生成。
T3366 Cephalotaxine

ZINC19795976,三尖杉碱,(-)-Cephalotaxine,Cephalotaxlen

Antiviral; Influenza Virus Immunology/Inflammation; Microbiology/Virology
Cephalotaxine (ZINC19795976) 是从头孢紫杉中分离得到的一种生物碱,具有抗白血病和抗病毒活性,如抗 Zika 病毒。
T2763 Panaxadiol

人参二醇,20(R)-Panaxadiol

Others; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism; Others
Panaxadiol (20(R)-Panaxadiol) 是从人参根中获得,具有神经保护和抗肿瘤作用,能够抑制程序性细胞死亡配体-1(PD-L1)的表达和肿瘤增殖。
T1257 Bestatin

Ubenimex,乌苯美司

Others; Aminopeptidase; Antibacterial; Antibiotic; LTR Immunology/Inflammation; Metabolism; Microbiology/Virology; Others
Bestatin (Ubenimex) 是 CD13 (Aminopeptidase N)/APN 和 leukotriene A4 hydrolase 抑制剂,可用于癌症研究。
T2731 Usnic Acid

Usniacin,松萝酸,地衣酸

Antibacterial; Autophagy Autophagy; Microbiology/Virology
Usnic Acid (Usniacin) 是地衣次生代谢产物,具有独特的二苯并呋喃骨架。它是一种抗菌剂、抗肿瘤剂和酶抑制剂。
T3774 Gracillin

山药,纤细薯蓣皂苷

cell cycle arrest Cell Cycle/Checkpoint
Gracillin 是一种甾体皂苷,从植物的根里提取得到,有抗肿瘤作用。
T5853 Rubitecan

RFS 2000,鲁比特康,9-Nitrocamptothecin

Topoisomerase DNA Damage/DNA Repair
Rubitecan (9-Nitrocamptothecin) 是一种与喜树碱相关的半合成药物,具有有效的抗肿瘤和抗病毒特性。它是一种 DNA 拓扑异构酶 I 抑制剂,以浓度依赖性方式抑制 DNA 拓扑异构酶 I 并在无细胞试验中增加超螺旋 DNA 的比例。
TN3284 8-Hydroxyodoroside A

Others Others
An antitumor agent containing at least one compound selected from the group consisting of nerigoside, oleandrigenin, sarmentoside, oleaside A, oleandrin, 8β-hydroxy odoroside A, narciclasine, trans-dihydronarciclasine and bisdeoxynarciclasine is provided, this antitumor agent has an advantage of having an excellent therapeutic effect of tumor and less side effects.
T40519 Indicine N-oxide

(+)-Indicine N-oxide,Indicine N-oxide,NSC132319

Indicine N-oxide (NSC 132319), a pyrrolizidine alkaloid, serves as an antitumor agent in pediatric cancer and solid tumors research.
TN4251 Indicine

Others Others
Indicine N-oxide is a more active antitumor agent than its free base Indicine.
T78497 λ-Carrageenan

λ-Carrageenan是广泛应用于基础研究的海藻多糖,常用作促炎剂,并具有有效的抗肿瘤活性。
T75563 Vanicoside E

Vanicoside E 是一种抗氧化和抗癌剂。Vanicoside E 抑制L-Tyrosine 和L-DOPA,IC50为 45.23 μM 和 189.96 μM。
T75520 Aplyronine A

Aplyronine A是具有特异性肌动蛋白解聚活性、抗肿瘤及促凋亡功能的化合物,适用于癌症、肌肉收缩、细胞运动和细胞分裂等研究领域。
TMA1743 Ergosterol peroxide

ERK; VEGFR; p38 MAPK; Wnt/beta-catenin; Akt; JAK; CDK; JNK; STAT; Antifection Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling; Stem Cells; Tyrosine Kinase/Adaptors
Ergosterol peroxide is an inhibitor of osteoclast differentiation, which has antiviral, trypanocidal, antitumor, and antiangiogenic actions, it can stimulate Foxo3a activity by inhibiting pAKT and c-Myc and activating pro-apoptotic protein Puma and Bax to
T80996 Theasaponin E1

Theasaponin E1,一种可从茶籽分离的茶皂苷,对人肿瘤细胞系K562和HL60展示了抗肿瘤潜能。此外,Theasaponin E1具备醌还原酶(QR)诱导活性,有助于作为抗癌预防药物的研究。
T14121 Actinonin

(-)-Actinonin

Aminopeptidase Metabolism
Actinonin ((-)-Actinonin) is a naturally occurring antibacterial agent produced by Actinomyces and a potent reversible peptide deformylase (PDF) inhibitor with a Ki of 0.28 nM, it also is an apoptosis inducer. Actinonin inhibits aminopeptidase M, aminopeptidase N and leucine aminopeptidase, it also inhibits MMP-1, MMP-3, MMP-8, MMP-9, and hmeprin α with Ki values of 300 nM, 1,700 nM, 190 nM, 330 nM, and 20 nM, respectively. Actinonin has antiproliferative and antitumor activities[1][2][3][4][5].
TN4652 Niazimicin

NF-κB; PI3K; AChR; Antifection Microbiology/Virology; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling
Niazimicin are NF-B and PI3K inhibitors, which shows antimicrobial, hypotensive and spasmolytic activities. Niazimicin has potent antitumor promoting activity in the two-stage carcinogenesis in mouse skin using 7,12-dimethylbenz(a)anthracene (DMBA) as ini
T81168 Shishijimicin C

Shishijimicin C 是由子囊菌 Didemnum proliferum 分离得到的一种新型抗肿瘤剂,具有显著的细胞毒性和抗肿瘤活性。作为点击化学试剂,Shishijimicin C 含有Alkyne基团,能够通过铜催化的叠氮-炔环加成反应(CuAAc)与含Azide基团的分子反应。
T81170 Shishijimicin A

Shishijimicin A是一款从子囊菌Didemnum proliferum中分离出的新型抗肿瘤剂,具备突出的细胞毒性及抗肿瘤活性。作为点击化学试剂,Shishijimicin A内含Alkyne基团,能够与含Azide基团的分子通过铜催化的叠氮-炔环加成反应(CuAAc)进行作用。

天然产物

Antitumor agent-89
Cat.No: T83000
Synonym:
Target:
Cephalotaxine
Cat.No: T3366
Synonym: ZINC19795976,三尖杉碱,(-)-Cephalotaxine,Cephalotaxlen
Target: Antiviral, Influenza Virus
Panaxadiol
Cat.No: T2763
Synonym: 人参二醇,20(R)-Panaxadiol
Target: Others, HIF/HIF Prolyl-Hydroxylase
Bestatin
Cat.No: T1257
Synonym: Ubenimex,乌苯美司
Target: Others, Aminopeptidase, Antibacterial, Antibiotic, LTR
Usnic Acid
Cat.No: T2731
Synonym: Usniacin,松萝酸,地衣酸
Target: Antibacterial, Autophagy
Gracillin
Cat.No: T3774
Synonym: 山药,纤细薯蓣皂苷
Target: cell cycle arrest
Rubitecan
Cat.No: T5853
Synonym: RFS 2000,鲁比特康,9-Nitrocamptothecin
Target: Topoisomerase
8-Hydroxyodoroside A
Cat.No: TN3284
Synonym:
Target: Others
Indicine N-oxide
Cat.No: T40519
Synonym: (+)-Indicine N-oxide,Indicine N-oxide,NSC132319
Target:
Indicine
Cat.No: TN4251
Synonym:
Target: Others
λ-Carrageenan
Cat.No: T78497
Synonym:
Target:
Vanicoside E
Cat.No: T75563
Synonym:
Target:
Aplyronine A
Cat.No: T75520
Synonym:
Target:
Ergosterol peroxide
Cat.No: TMA1743
Synonym:
Target: ERK, VEGFR, p38 MAPK, Wnt/beta-catenin, Akt, JAK, CDK, JNK, STAT, Antifection
Theasaponin E1
Cat.No: T80996
Synonym:
Target:
Actinonin
Cat.No: T14121
Synonym: (-)-Actinonin
Target: Aminopeptidase
Niazimicin
Cat.No: TN4652
Synonym:
Target: NF-κB, PI3K, AChR, Antifection
Shishijimicin C
Cat.No: T81168
Synonym:
Target:
Shishijimicin A
Cat.No: T81170
Synonym:
Target:
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