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45

抑制剂 & 化合物

15

天然产物

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Cat. No. Product Name Target Signaling Pathways
T9705 TL-895

BTK Angiogenesis; Tyrosine Kinase/Adaptors
TL-895 是口服有效的,ATP 竞争性的,以及高度选择性和不可逆的BTK 抑制剂,IC50和Ki 分别为 1.5 nM 和 11.9 nM。TL-895在 JAKi 复发/难治性骨髓纤维化、急性髓系白血病、COVID-19 和癌症方面有研究的价值。
T4121 Bicyclol

SY801,双环醇

HBV; Autophagy Autophagy; Microbiology/Virology
Bicyclol (SY801) 是一种抗肝炎 HBV 和 HCV 药物。
T2162 Maribavir

BW1263W94,GW257406X,Benzimidavir,马立巴韦,1263W94

Others; HCV Protease Microbiology/Virology; Others; Proteases/Proteasome
Maribavir (GW257406X) 是一种可口服的苯并咪唑核苷化合物,具有抗巨细胞病毒的活性。
T61793 HIV-IN-6

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-IN-6 是一种 HIV 病毒抑制剂,可抑制HIV 病毒的复制。HIV-IN-6 具有抗HIV 病毒的活性,通过靶向与病毒 Nef 蛋白相互作用的 Src 家族激酶 (SFK) (如 Hck) 而起作用。
T1370 2-Amino-5-Fluorophenol

Others Others
2-Amino-5-Fluorophenol(2-AF)用于合成各种药物和化合物,包括抗癌药、抗炎药和其他药物,以及抗微生物、抗真菌和抗病毒的化合物。
T5396 Letermovir

AIC246,MK-8828,莱莫维韦

Others; HCV Protease Microbiology/Virology; Others; Proteases/Proteasome
Letermovir (AIC246) 是一种新型抗 CMV 抑制剂,靶向病毒末端酶,抑制其活性。
T38343 Quercetin pentaacetate

Pentaacetylquercetin

RSV Microbiology/Virology
Quercetin pentaacetate (Pentaacetylquercetin) 具有多种生物活性,包括抗氧化、抗炎和抗癌特性。 Quercetin pentaacetate 与 RSV 相互作用并抑制病毒在细胞表面的粘附。
T15777 Loxoribine

RWJ 21757,7-Allyl-8-oxoguanosine,洛索立宾

Influenza Virus; TLR Immunology/Inflammation; Microbiology/Virology
Loxoribine (RWJ 21757) 是一种鸟苷类似物,是一种口服生物可利用的选择性 Toll 样受体 (TLR) 7 激动剂。 具有抗病毒和抗肿瘤活性。它是一种新型的强效免疫刺激剂,具有较广谱的免疫生物学活性。
T8736 Cidofovir dihydrate

HPMPC,(S)-HPMPC,GS 0504,西多福韦二水合物

Others Others
Cidofovir dihydrate (HPMPC) 是注射型巨细胞病毒 DNA 聚合酶抑制剂,通过选择性抑制病毒 DNA 聚合酶来抑制 CMV 复制,从而阻止病毒复制和转录。
T67833 HIV-1 inhibitor-54

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 inhibitor-54 是一种有效的 HIV-1 抑制剂,在 MT-4 细胞中对 WT HIV-1 (菌株 IIIB) x 显示出抗 HIV 活性(EC50 : 32 nM)。HIV-1 inhibitor-54 可用于研究病毒感染。
T73375 CK2-IN-4

Casein Kinase Metabolism; Stem Cells
CK2-IN-4 是一种蛋白激酶 (CK2) 抑制剂 ,IC50 值为 8.6 µM。 CK2-IN-4 具有潜在的抗癌啊和抗炎活性,可用于研究病毒感染和肾小球肾炎的疾病。
TNU0007 3'-Deoxy-3'-fluoroadenosine

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
3'-Deoxy-3'-fluoroadenosine 是一种嘌呤核苷类似物,具有广泛的抗肿瘤活性和抗病毒活性,对蜱传脑炎病毒(TBEV),寨卡病毒和西尼罗河病毒(WNV)具有抑制作用,EC50分别为1.1μM、 0.1 μM和4.7 1.5 μM。3'-Deoxy-3'-fluoroadenosine可用于研究肿瘤疾病。
T60540 Netivudine

Netivudine 是一种有效的核苷类逆转录酶抑制剂(NRTIs),是一种核苷类似物,具有抗水痘带状疱疹病毒活性,可用于治疗人类免疫缺陷病毒(HIV)感染。Netivudine 通过抑制逆转录酶起作用,通过抑制作用减少体内的病毒载量,减缓疾病的进展。
T67801 GS-6620 PM

GS-6620 PM 是GS-6620的衍生物。GS-6620是一种口服的抗丙型肝炎病毒聚合酶抑制剂,是一种新型强效的C-核苷腺嘌呤类似物单磷酸酯原药。GS-6620对其他病毒的活性有限,对密切相关的牛病毒性腹泻病毒仅保持部分活性(EC50,1.5μM)。
T28701 SC-58272

SC58272

SC-58272 is an inhibitor of N-myristoyltransferase (Nmt), a target for anti-fungal and anti-viral therapy.
T40971 Dehydroandrographolide succinate potassium sodium salt

Dehydroandrographolide succinate (potassium sodium salt), derived from the herbal medicine Andrographis paniculata (Burm f) Nees, is a versatile compound highly utilized for the treatment of viral pneumonia and viral upper respiratory tract infections due to its potent immunostimulatory, anti-infective, and anti-inflammatory properties.
TQ0030 Tomeglovir

托美洛韦,BAY 38-4766

HCV Protease Microbiology/Virology; Proteases/Proteasome
Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).
T61824 NIOCH 14

NIOCH 14 is an antiviral agent and pro-drug with demonstrated potency against orthopoxviruses. It exhibits significant efficacy in reducing infection rates and lung viral load in mice. NIOCH 14 is particularly useful for anti-smallpox research [1] [2], as it displays marked anti-orthopoxvirus activity.
T63412 DB772 hydrate

DB772 hydrate 是一种牛病毒性腹泻病毒 (BVDV) 抑制剂,同时表现出抗朊病毒作用。
T40949 5'-O-TBDMS-N2-ibu-dG

5'-O-TBDMS-N2-ibu-dG

5'-O-TBDMS-N2-ibu-dG is a nucleoside derivative that possesses potent anti-bovine viral diarrhea virus activity. It serves as a valuable compound for the synthesis of lead compounds with such activity.
T61856 Antiviral agent 10

Antiviral agent 10 是一种可抑制呼吸道合胞病毒 (RSV) 的抗病毒剂。
T36651 Anti-MERS-2E6 mAb

Anti-MERS-2E6 mAb

Anti-MERS-2E6 mAb (MERS-2E6), a human IgG1 neutralizing antibody, is expressed in CHO cells. It effectively competes with the virus Spike protein for binding to the CD26 receptor, consequently inhibiting viral invasion into host cells.
T60709 Acyclovir monophosphate

Acyclovir monophosphate 是抗单纯疱疹病毒 (HSV)剂,并且具有抗肿瘤活性。Acyclovir monophosphate 通过抑制病毒 DNA 聚合酶从而阻断 DNA 合成,同时能终止病毒 DNA 的链延伸。
T61606 Indomethacin sodium

Indomethacin sodium, a powerful and orally active inhibitor of COX1/2, exhibits IC50 values of 18 nM and 26 nM for COX-1 and COX-2, respectively. Apart from its potent anti-inflammatory effects, this compound possesses notable anticancer and anti-infective activities. Since it has such versatile attributes, it finds useful applicability in cancer, inflammation, and viral infection research [1] [2] [3].
T61613 SARS-CoV-2-IN-17

SARS-CoV-2-IN-17 (Compound 16) is a highly effective inhibitor of SARS-CoV-2 nucleocapsid protein (NPro). It demonstrates potent anti-viral activity, with an EC50 value of 2.18 μM. Furthermore, SARS-CoV-2-IN-17 binds to NPro with a low Kd value of 7.82 μM, highlighting its potency as a NPro ligand [1].
T83046 Anti-Influenza agent 5

Influenza Virus Microbiology/Virology
Anti-Influenza agent 5 (Compound IIB-2)为查耳酮类衍生物,具有抑制流感病毒核输出的活性。该化合物能有效抑制对Oseltamivir具有耐药性的病毒株,主要通过阻断流感病毒核蛋白输出作用来抑制病毒复制。
T61080 L-I-OddU

L-I-OddU, a potent and selective anti-Epstein-Barr virus (EBV) agent, is a L-5'-halo-dioxolane nucleoside analogue. It demonstrates antiviral activity by effectively suppressing replicative EBV DNA and viral protein synthesis [1] [2]. With an EC 50 value of 0.03 μM, L-I-OddU exhibits high potency against EBV while maintaining low cytotoxicity, as indicated by its CC 50 value of 1000 nM.
T38946 C8 Dihydroceramide

C8 Dihydroceramide

C8 Dihydroceramide acts as a negative control for C8 Ceramide, a cell-permeable analog of natural ceramides. C8 Ceramide, also known as N-Octanoyl-D-erythro-sphingosine, exhibits potent chemotherapeutic properties and anti-proliferation effects. Additionally, it stimulates dendritic cells to enhance T cell responses during viral infections. In vitro studies have also shown that C8 Ceramide induces a slight activation of protein kinase (PKC) [4].
T70859 ent-Abacavir

ent-Abacavir is an enatiomer of Abacavir. Abacavir is a carbocyclic 2'-deoxyguanosine nucleoside reverse transcriptase inhibitor and an anti-HIV drug used to treat HIV infection. Intracellular enzymes convert Abacavir to its active form, carbovir-triphosphate (CBV-TP), which then selectively inhibits HIV reverse transcriptase by incorporating into viral DNA. Abacavir is metabolized in the liver by uridine diphosphate glucuronyltransferase and alcohol dehydrogenase resulting in inactive glucuroni...
T78756 Yhhu6669

HBV Microbiology/Virology
Yhhu6669为抗HBV药物,能够抑制HBVDNA。该化合物通过诱导无DNA衣壳的形成,从而抑制HBV复制,且能有效降低AAV/HBV感染小鼠中的HBVDNA及HBcAg水平,展现出优良的药代动力学特性。
T82215 HEP-1

Human ezrin peptide (324-337)

HEP-1 (Human ezrin peptide (324-337)) 是一种具抗HIV活性的口服多肽,能增强乙型肝炎疫苗接种后的抗体滴度,表现出潜在的抗病毒感染研究价值。
T77158 Diridavumab

Diridavumab为一种针对HA茎的单克隆抗体。它能稳定HA的融合前结构,阻断细胞膜与病毒膜在核内体内因pH变化引起的融合。此抗体主要用于H2流感病毒研究。
T69731 Remdesivir maleate

Remdesivir, also known as GS-5734, is a prodrug form of the antiviral nucleoside analog GS-44152. Remdesivir is a broad spectrum anti-viral drug that has shown to inhibit SARS-CoV-2, in vitro and in vivo. Efficacy of remdesivir against Ebola virus has been demonstrated. Remdesivir inhibits SARS-CoV-2 replication, reduces viral load, and exerts protective effects in SARS-CoV-2 infected animals. Remdesivir also reduces the pathological process, alleviates mild symptoms, and improves pulmonary les...
T62888 Influenza A virus-IN-7

Influenza A virus-IN-7 (compound 16r) 是一种有效的、口服具有活力的甲型流感病毒抑制剂 (IC50: 3.43 μM, CC50>100 μM)。Influenza A virus-IN-7 具有抗 IAV 作用,细胞毒性低,对病毒 RNA 的转录和复制表现出抑制作用。
T80657 SARS-CoV-2 3CLpro-IN-15

Virus Protease Microbiology/Virology
SARS-CoV-2 3CLpro-IN-15(compound a)为β-硝基苯乙烯型抑制剂,专门针对SARS-CoV-2的3CL蛋白酶(3CLpro)而设计。该化合物能有效抑制病毒的复制转录过程,是研发抗COVID-19候选先导化合物的关键因素。
T68957 Eprociclovir dihydrate

Eprociclovir dihydrate is a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applied onto the affected cornea, ameliorated clinica...
T70027 Eprociclovir potassium

Eprociclovir potassium is a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applied onto the affected cornea, ameliorated clinica...
T38340 10-Norparvulenone

10-Norparvulenone is a fungal metabolite originally isolated fromMicrosphaeropsis.1It decreases viral sialidase activity in, and increases survival of, MDCK cells infected with the mouse-adapted influenza virus A/PR/8/34 when used at a concentration of 1 μg/ml. 1.Fukami, A., Nakamura, T., Kim, Y.P., et al.A new anti-influenza virus antibiotic, 10-norparvulenone from Microsphaeropsis sp. FO-5050J. Antibiot. (Tokyo)53(10)1215-1218(2000)
T71291 EICAR

EICAR is a drug which acts as an inhibitor of the enzyme IMP dehydrogenase. It is a nucleoside derivative which has both anti-cancer and antiviral effects, and was originally developed for the treatment of leukemia, but was unsuccessful in human clinical trials. It has broad spectrum antiviral effects with activity against vaccinia virus, Semliki forest virus, Junin virus, reovirus, influenza, measles virus and respiratory syncytial virus among others, although it is not active against SARS. T...
T69817 Eprociclovir Na

Eprociclovir Na is the salt form of Eprociclovir, also known as A-5021, a new acyclovir analogue and a potent inhibitor of EHV1 replication and may have potential for the treatment and/or prophylaxis of infections with this virus. Eprociclovir possess potent anti-herpetic activity against most human herpesviruses. A-5021 proved to be about 15-fold more potent than acyclovir in inhibiting viral replication. Eprociclovir inhibits murine herpetic keratitis. A-5021 eyedrops, which are easily applie...
T82937 ATV041

ATV041是一种结合了布洛芬和核苷酸类似物的口服活性化合物。该化合物优化了口服药物动力学(PK)特性和组织分布,显示出对抗小鼠肝炎病毒(MHV)的能力。ATV041能够剂量依赖性地降低病毒载量,减少组织损伤并减轻病毒引发的炎症。
T69081 KRH-1636

KRH-1636 is an orally active, selective and extremely potent CXC chemokine receptor 4 antagonist. KRH-1636 exhibits a potent and selective anti-HIV-1 activity. KRH-1636 efficiently blocked replication of various T cell line-tropic (X4) HIV type 1 (HIV-1) in MT-4 cells and peripheral blood mononuclear cells through the inhibition of viral entry and membrane fusion via the CXC chemokine receptor (CXCR)4 coreceptor but not via CC chemokine receptor 5. KRH-1636 also inhibits binding of the CXC chem...
T83143 Alloferon 1

Alloferon 1 是一种具有抗病毒和抗肿瘤功能的肽。它能激活人外周血淋巴细胞的天然细胞毒性,诱导IFN合成,并在小鼠体内增强其抗病毒和抗肿瘤的防御机制。此外,Alloferon 1 在 λ-角叉菜胶诱导的足水肿模型中展现出抗炎作用。它可从双翅目昆虫丽蝇Calliphora vicina的血液中提取。
T79567 Antiviral agent 35

Influenza Virus Microbiology/Virology
Antiviralagent 35 (compound 4d) 作为一种口服抗流感病毒药物,针对流感病毒复制的早期阶段有效。该化合物能够阻断流感病毒引发的ROS积聚、自噬及细胞凋亡,同时在肺部感染的小鼠模型中,抑制RIG-1通路所介导的炎症响应。Antiviralagent 35展现出低细胞毒性(CC50>800 μM,MDCK细胞)且对H1N1(A/Weiss/43)展现出显著的抗病毒活性,EC50为2.28 μM。
T37295 Ganglioside GM1 Asialo Mixture

Ganglioside GM1 asialo is a component of cellular lipid rafts and can be formed by the cleavage of the sialic acid residue from ganglioside GM1 by neuraminidase. Ganglioside GM1 asialo is a glycolipid receptor for P. aeruginosa flagellin and stimulates defensive responses in host cells, including extracellular ATP release, calcium mobilization, and ERK1/2 phosphorylation when stimulated by flagellin and an anti-ganglioside GM1 asialo antibody. The percentage of ganglioside GM1 asialo-positive na...

化合物

TL-895
Cat.No: T9705
Synonym:
Target: BTK
Bicyclol
Cat.No: T4121
Synonym: SY801,双环醇
Target: HBV, Autophagy
Maribavir
Cat.No: T2162
Synonym: BW1263W94,GW257406X,Benzimidavir,马立巴韦,1263W94
Target: Others, HCV Protease
HIV-IN-6
Cat.No: T61793
Synonym:
Target: HIV Protease
2-Amino-5-Fluorophenol
Cat.No: T1370
Synonym:
Target: Others
Letermovir
Cat.No: T5396
Synonym: AIC246,MK-8828,莱莫维韦
Target: Others, HCV Protease
Quercetin pentaacetate
Cat.No: T38343
Synonym: Pentaacetylquercetin
Target: RSV
Loxoribine
Cat.No: T15777
Synonym: RWJ 21757,7-Allyl-8-oxoguanosine,洛索立宾
Target: Influenza Virus, TLR
Cidofovir dihydrate
Cat.No: T8736
Synonym: HPMPC,(S)-HPMPC,GS 0504,西多福韦二水合物
Target: Others
HIV-1 inhibitor-54
Cat.No: T67833
Synonym:
Target: HIV Protease
CK2-IN-4
Cat.No: T73375
Synonym:
Target: Casein Kinase
3'-Deoxy-3'-fluoroadenosine
Cat.No: TNU0007
Synonym:
Target: Nucleoside Antimetabolite/Analog
Netivudine
Cat.No: T60540
Synonym:
Target:
GS-6620 PM
Cat.No: T67801
Synonym:
Target:
SC-58272
Cat.No: T28701
Synonym: SC58272
Target:
Dehydroandrographolide succinate potassium sodium salt
Cat.No: T40971
Synonym:
Target:
Tomeglovir
Cat.No: TQ0030
Synonym: 托美洛韦,BAY 38-4766
Target: HCV Protease
NIOCH 14
Cat.No: T61824
Synonym:
Target:
DB772 hydrate
Cat.No: T63412
Synonym:
Target:
5'-O-TBDMS-N2-ibu-dG
Cat.No: T40949
Synonym: 5'-O-TBDMS-N2-ibu-dG
Target:
Antiviral agent 10
Cat.No: T61856
Synonym:
Target:
Anti-MERS-2E6 mAb
Cat.No: T36651
Synonym: Anti-MERS-2E6 mAb
Target:
Acyclovir monophosphate
Cat.No: T60709
Synonym:
Target:
Indomethacin sodium
Cat.No: T61606
Synonym:
Target:
SARS-CoV-2-IN-17
Cat.No: T61613
Synonym:
Target:
Anti-Influenza agent 5
Cat.No: T83046
Synonym:
Target: Influenza Virus
L-I-OddU
Cat.No: T61080
Synonym:
Target:
C8 Dihydroceramide
Cat.No: T38946
Synonym: C8 Dihydroceramide
Target:
ent-Abacavir
Cat.No: T70859
Synonym:
Target:
Yhhu6669
Cat.No: T78756
Synonym:
Target: HBV
HEP-1
Cat.No: T82215
Synonym: Human ezrin peptide (324-337)
Target:
Diridavumab
Cat.No: T77158
Synonym:
Target:
Remdesivir maleate
Cat.No: T69731
Synonym:
Target:
Influenza A virus-IN-7
Cat.No: T62888
Synonym:
Target:
SARS-CoV-2 3CLpro-IN-15
Cat.No: T80657
Synonym:
Target: Virus Protease
Eprociclovir dihydrate
Cat.No: T68957
Synonym:
Target:
Eprociclovir potassium
Cat.No: T70027
Synonym:
Target:
10-Norparvulenone
Cat.No: T38340
Synonym:
Target:
EICAR
Cat.No: T71291
Synonym:
Target:
Eprociclovir Na
Cat.No: T69817
Synonym:
Target:
ATV041
Cat.No: T82937
Synonym:
Target:
KRH-1636
Cat.No: T69081
Synonym:
Target:
Alloferon 1
Cat.No: T83143
Synonym:
Target:
Antiviral agent 35
Cat.No: T79567
Synonym:
Target: Influenza Virus
Ganglioside GM1 Asialo Mixture
Cat.No: T37295
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T6S1369 Vitexin

牡荆素,Apigenin-8-C-glucoside

Antioxidant oxidation-reduction
Vitexin 是一种存在于多种药用植物(如榕树、螺旋藻)中的 c-糖基化的黄酮。 它具有广泛的药理作用,包括抗氧化,抗癌,抗炎,抗痛觉过敏和神经保护作用。
T2982 Xanthone

Genicide,呫吨酮,氧杂蒽酮,Xanthenone,Benzophenone oxide

Apoptosis; Others; Influenza Virus; Antibacterial; Antifungal Apoptosis; Microbiology/Virology; Others
Xanthone (Xanthenone) 是一种从山竹果中分离得到的天然产物,具有抗炎,抗氧化,抗肿瘤,抗过敏,抗细菌,抗真菌和抗病毒活性。在癌变的不同阶段可控制细胞分裂和生长,凋亡,炎症和转移。
T5S0018 Betulonic acid

路路通酸,(+)-Betulonic acid,Betunolic acid,Liquidambaric acid

Parasite; HSV Microbiology/Virology
Betulonic acid (Liquidambaric acid) 是一种在许多植物中存在的三萜类天然产物,具有抗肿瘤,抗炎,抗寄生虫和抗病毒的活性。
TN1788 Isookanin

Amylase Metabolism
Isookanin 在多种疾病领域有研究价值,包括肿瘤,皮疹,蛇和昆虫叮咬,糖尿病,腹泻。它可作为抗病毒剂对抗 HSV 和水痘带状疱疹病毒。它也具有抗氧化特性。
T13229 Tunicamycin

Influenza Virus; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Tunicamycin 是一种抗生素的混合物,通过阻断 GlcNAc 磷酸转移酶 (GPT),抑制 N-连接糖基化。Tunicamycin 具有抗肿瘤活性,还具有抗细菌、抗真菌和抗病毒活性。
T2S1975 Ponicidin

冬凌草乙素,Rubescensine B

Apoptosis; JAK; STAT Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
Ponicidin (Rubescensine B) 是来源于冬凌草的一种二萜,具有免疫调节、抗炎、抗病毒和抗癌作用。它可诱导胃癌细胞凋亡,降低 JAK2 和 STAT3 的磷酸化水平。
T40660 Kansuinine B

IL Receptor; SARS-CoV Immunology/Inflammation; Microbiology/Virology
Kansuinine B 抑制由 IL-6 诱导的 Stat3 活化。 Kansuinine B 具有抗病毒活性,可用于 COVID-19 研究。
T75675 Nepasaikosaponin K

Antiviral Immunology/Inflammation
Nepasaikosaponin K 是一种从柴胡根中分离出来小分子化合物,具有抗流感和抗病毒活性,可用于研究病毒感染。
T0875 Acetylcysteine

乙酰半胱氨酸,N-Acetyl-L-cysteine,LNAC,NAC,易咳净

Apoptosis; TNF; Ferroptosis; Influenza Virus; Reactive Oxygen Species; ROS; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Acetylcysteine (NAC) 是半胱氨酸的 N-乙酰衍生物,是一种 ROS 抑制剂和粘液溶解剂。Acetylcysteine 可诱导细胞凋亡,可用于减少粘液的厚度,还具有抗流感病毒活性。
TN1622 Ermanin

堪非醇3,4'-二-O-甲醚

NOS; Influenza Virus; COX; HIV Protease; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ermanin 是一种从 Tanacetum microphyllum 中分离出来的类黄酮。Ermanin抑制血小板聚集,具有抗结核和抗病毒/细菌特性。Ermanin 可抑制 iNOS 和 COX-2 的表达,从而具有抗炎活性。Ermanin 可能具有抗 HIV-1 活性。Ermanin 在较低浓度下可有效地抑制 Dione juno 幼虫。
T6519 Gramine

NSC 16892,芦竹碱,Donaxine

Adiponectin receptor; Reverse Transcriptase; Adrenergic Receptor GPCR/G Protein; Microbiology/Virology; Neuroscience
Gramine (Donaxine) 是从芦竹中得到的一种生物碱,是脂联素受体激动剂,对 AdipoR2 和 AdipoR1 的 IC50值分别为 3.2 和 4.2 µM。它也是小鼠和人β2-肾上腺素受体激动剂,具有抗肿瘤、抗炎和抗病毒作用。
T4S0999 (2S)-Isoxanthohumol

Isoxanthohumol,(2S)-异黄腐酚,异黄腐醇

Virus Protease; HSV Microbiology/Virology
(2S)-Isoxanthohumol 是一种由啤酒花原异戊烯基二氢黄酮 Isoxanthohumol 的微生物转化代谢物。
TN5005 Shegansu B

Influenza Virus Microbiology/Virology
Shegansu B exhibits significant in vitro anti-influenza viral activity in MDCK cells.
T8521 Gnetin D

Gnetin D exhibits significant in vitro anti-influenza viral activity in MDCK cells, with IC(50) values from 0.67 to 11.99 ug/mL.
TN2176 Sanggenol A

Influenza Virus; Antifection Microbiology/Virology
Sanggenol A 抑制甲型流感病毒和肺炎球菌神经氨酸酶,因此可作为双重作用的抗感染试剂。

天然产物

Vitexin
Cat.No: T6S1369
Synonym: 牡荆素,Apigenin-8-C-glucoside
Target: Antioxidant
Xanthone
Cat.No: T2982
Synonym: Genicide,呫吨酮,氧杂蒽酮,Xanthenone,Benzophenone oxide
Target: Apoptosis, Others, Influenza Virus, Antibacterial, Antifungal
Betulonic acid
Cat.No: T5S0018
Synonym: 路路通酸,(+)-Betulonic acid,Betunolic acid,Liquidambaric acid
Target: Parasite, HSV
Isookanin
Cat.No: TN1788
Synonym:
Target: Amylase
Tunicamycin
Cat.No: T13229
Synonym:
Target: Influenza Virus, Antibacterial, Antibiotic, Antifungal
Ponicidin
Cat.No: T2S1975
Synonym: 冬凌草乙素,Rubescensine B
Target: Apoptosis, JAK, STAT
Kansuinine B
Cat.No: T40660
Synonym:
Target: IL Receptor, SARS-CoV
Nepasaikosaponin K
Cat.No: T75675
Synonym:
Target: Antiviral
Acetylcysteine
Cat.No: T0875
Synonym: 乙酰半胱氨酸,N-Acetyl-L-cysteine,LNAC,NAC,易咳净
Target: Apoptosis, TNF, Ferroptosis, Influenza Virus, Reactive Oxygen Species, ROS, Endogenous Metabolite
Ermanin
Cat.No: TN1622
Synonym: 堪非醇3,4'-二-O-甲醚
Target: NOS, Influenza Virus, COX, HIV Protease, Antibacterial, Antibiotic
Gramine
Cat.No: T6519
Synonym: NSC 16892,芦竹碱,Donaxine
Target: Adiponectin receptor, Reverse Transcriptase, Adrenergic Receptor
(2S)-Isoxanthohumol
Cat.No: T4S0999
Synonym: Isoxanthohumol,(2S)-异黄腐酚,异黄腐醇
Target: Virus Protease, HSV
Shegansu B
Cat.No: TN5005
Synonym:
Target: Influenza Virus
Gnetin D
Cat.No: T8521
Synonym:
Target:
Sanggenol A
Cat.No: TN2176
Synonym:
Target: Influenza Virus, Antifection
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