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29

抑制剂 & 化合物

8

天然产物

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Cat. No. Product Name Target Signaling Pathways
T9497 Niraparib tosylate monohyrate

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Niraparib tosylate monohyrate 也称为 MK-4827,是一种聚 (ADP-核糖) 聚合酶 (PARP) 抑制剂,具有潜在的抗肿瘤活性。 MK4827 抑制 PARP 活性,增强 DNA 链断裂的积累,促进基因组不稳定性和细胞凋亡。 PARP 蛋白家族通过碱基切除修复 (BER) 途径检测和修复单链 DNA 断裂。
T6207 SC144

Apoptosis; Interleukin Apoptosis; Immunology/Inflammation
SC144 是一种口服活性 gp130 抑制剂。它结合 gp130,诱导 gp130 磷酸化(S782) 和去糖基化,消除 Stat3 磷酸化和核易位,进一步抑制下游靶基因的表达。它对 gp130 配体触发的信号转导有明显的抑制作用,可诱导人卵巢癌细胞凋亡。
T3231 Niraparib

尼拉帕尼,MK-4827

Apoptosis; Others; PARP Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
Niraparib (MK-4827) 是一种 PARP 抑制剂,可以抑制 PARP1 和 PARP2 (IC50=3.8/2.1 nM),具有选择性。Niraparib 具有抗肿瘤活性,可以抑制 DNA 损伤修复、诱导细胞凋亡。
T4102 Goserelin acetate

醋酸戈舍瑞林,Fertilan,ICI-118630 acetate,Zoladex

Apoptosis; GNRH Receptor Apoptosis; GPCR/G Protein
Goserelin acetate (Fertilan) 是一种促性腺激素释放激素 (GnRH/LHRH) 十肽类似物,能作为GnRH 激动剂。它可研究乳腺癌、上皮性卵巢癌和前列腺癌。
T3353 Niraparib hydrochloride

尼拉帕利盐酸盐,MK-4827 hydrochloride,MK-4827 (hydrochloride)

Apoptosis; Others; PARP Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
Niraparib hydrochloride (MK-4827 hydrochloride) 是一种具有口服活性的PARP1和PARP2抑制剂,IC50值分别为 3.8 nM 和 2.1 nM。它抑制 DNA 损伤修复,诱导凋亡并具有抗肿瘤活性。
T6892 Niraparib tosylate

尼拉帕利,MK-4827 (tosylate),MK 4827 tosylate,Niraparib (MK-4827) tosylate,尼拉帕尼对苯甲磺酸盐

Apoptosis; PARP Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Niraparib tosylate (MK-4827(tosylate)) 是一种高效的,具有生物口服利用度的PARP1和PARP2抑制剂,IC50分别为 3.8 和 2.1 nM。它抑制 DNA 损伤修复,诱导凋亡并具有抗肿瘤活性。
T24997 ABT-510 acetate

ABT 510 acetate

Apoptosis Apoptosis
ABT-510 acetate 是一种内源性抗血管生成的 TSP 肽抑制剂,是一种凝血酶原类似物,具有抗炎抗癌和抗血管生成活性,能诱导肿瘤细胞凋亡并抑制上皮性卵巢癌正位、同种异体模型中的卵巢肿瘤生长。ABT-510 acetate 可减少小鼠炎症性肠病模型的血管生成和炎症反应,可用于癌症 (尤其是上皮性卵巢癌) 以及炎症性肠病 (IBD) 的研究。
T78646 Estrogen receptor antagonist 8

Estrogen/progestogen Receptor Endocrinology/Hormones
Estrogen receptor antagonist 8 作为一种雌激素受体(ER)拮抗剂,具有抗子宫活性和潜在的抗肿瘤活性,可用于研究卵巢功能障碍。
T76749 Zilovertamab

Cirmtuzumab,UC-961

Others Others
Zilovertamab (UC-961) 是一种人源化抗 ROR1 单克隆抗体,可切断 Wnt5a 诱导的 ROR1 信号通路,在卵巢癌和子宫内膜癌细胞中显示出抗增殖活性。可用于研究淋巴癌。
T37376 PHY34

Autophagy Autophagy
PHY34是一种晚期自噬抑制剂,具有纳摩尔水平的抑制作用。在体内,PHY34具有抗高级别浆液性卵巢癌(HGSOC)活性。
T77408 Abagovomab

ACA 125

Others Others
Abagovomab (Anti-Human CA-125 Recombinant Antibody) 是一种独特型靶向肿瘤相关抗原 CA-125 的鼠源单克隆抗体。Abagovomab 由小鼠杂交瘤细胞产生。Abagovomab 可用于研究卵巢癌。
T76766 Mirvetuximab

M9346A

Antifolate Cell Cycle/Checkpoint
Mirvetuximab (M9346A) 是一种新型叶酸受体α (FRα) 靶向 anti-FOLR1 (folate receptor 1) 的单克隆抗体。Mirvetuximab soravtansine 常与铂类化合物或与其他化合物偶联成为抗体-药物偶联物用来治疗卵巢癌和其他 FRα 阳性的癌症。
T64167 Ifebemtinib

IN-10018,BI-853520

FAK Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Ifebemtinib (BI-853520) 是一种具有口服活性和强效性的粘附斑激酶 (FAK) 抑制剂 (IC50=1 nM),具有抗肿瘤活性,可抑制恶性胸膜间皮瘤中的球状体形成和原位肿瘤生长,可用于研究乳腺癌和卵巢癌。
T0005 Aspirin

阿司匹林,Acetylsalicylate,Acetylsalicylic Acid,邻乙酰水杨酸,ASA

Mitophagy; Virus Protease; COX; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Aspirin (Acetylsalicylic Acid) 是一种选择性 COX 抑制剂,具有多种药理活性。它是组蛋白去乙酰化酶抑制剂,可上调细胞周期阻滞蛋白 p21,抑制携带 COX-1 的卵巢 Y 细胞。 它还抑制 HUVEC 和新生大鼠心室心肌细胞中 COX-2 的表达,分别减少 PG 的产生和 ERK 和 NF-KB 的下调。
T36674 DMU-212

Apoptosis; ERK Apoptosis; MAPK
DMU-212 是具有口服活性的白藜芦醇的甲基化衍生物,表现出抗分裂、抗增殖、抗氧化和促进细胞凋亡的活性。它通过诱导凋亡和激活ERK1/2蛋白阻止有丝分裂。
T36083 DS-7423

PI3K; mTOR PI3K/Akt/mTOR signaling
DS-7423 是PI3K 和mTOR 的有效抑制剂,抑制PI3Kα 和 mTOR 的IC50分别为15.6 nM 和 34.9 nM。DS-7423表现出抗癌活性。
T41070 LP-184

LP-184 (Compound 6), referred to as an acylfulvene analog, demonstrates the ability to inhibit tumor growth with noteworthy anti-cancer efficacy observed across multiple cell lines, including ovarian, colon, prostate, and pancreatic.
T82664 CTX-2026

CTX-2026是一种与CD277结合的纯人源抗体,在卵巢肿瘤模型中表现出抗肿瘤活性,适用于癌症研究。
T39586 Cantrixil

TRX-E-002-1

Cantrixil (TRX-E-002-1) is a second-generation super-benzopyran (SBP) compound, derived from TRX-E-002. It elicits an increase in phosphorylated c-Jun levels, leading to caspase-mediated apoptosis in ovarian cancer cells. Cantrixil exhibits potent pan anti-cancer activity against various cancer phenotypes.
T61909 Estrogen receptor antagonist 7

Estrogen receptor antagonist7 (compound 13) 是高效ER拮抗剂,能够抑制乳腺癌细胞与卵巢癌细胞生长,展现出抗癌及抗子宫营养活性。
T78296 IMAB027

ASP1650

IMAB027 (ASP1650)是针对CLDN6 (Claudin 6)的特异性单克隆抗体,CLDN6作为一种紧密连接蛋白,其在多种人类癌症中异常高表达,尤其显著于卵巢癌。IMAB027展现出抗肿瘤特性,并能诱导表达CLDN6的卵巢癌和睾丸癌细胞走向凋亡。
T76871 Navicixizumab

Navicixizumab (OMP-305B83) 是一种双特异性抗 VEGF 和抗 DLL4抑制抗体。Navicixizumab 可以与紫杉醇结合用于癌症研究。Navicixizumab 可用于卵巢癌、原发性腹膜癌或输卵管癌的研究。
T76879 Vesencumab

Vesencumab (MNRP-1685A)是一种针对neuropilin-1 (NRP-1)的IG1抗体。通过与NRP-1结合,Vesencumab 阻断了NRP-1与VEGFR-2的偶联,展现出抗血管生成和抗肿瘤的活性。此化合物适用于转移性实体瘤,如卵巢癌的研究。
T63168 VEGFR-2-IN-26

VEGFR-2-IN-26 (compound 5h) 是一种 VEGFR-2 的高效抑制剂 (IC50: 15.5 nM)。VEGFR-2-IN-26 对白血病、中枢神经系统、非小肺、卵巢、肾、前列腺和乳腺癌细胞表现出良好的抗增殖作用。
T71287 CDKI-83

CDKI-83 is a potent CDK9 inhibitor. The compound shows effective anti-proliferative activity in human tumour cell lines with GI50 <1 μM, and is capable of inducing apoptosis in A2780 human ovarian cancer cells as determined by the activated caspase-3, Annexin V/PI double staining and accumulated cells at the sub-G1 phase of cellcycle. The research results suggest that combined inhibition of CDK9 and CDK1 may result in the effective induction of apoptosis and CDKI-83 has the potential to be devel...
T71218 AEZS-112

AEZS-112, also known as ZEN012, is an orally active small mol. anti-cancer drug which inhibits the polymn. of tubulin at low micromolar concns. AEZS 112 dose-dependently increased non-vital hypodiploid cells and the cytotoxic effect was least pronounced in G2 phase of the cell cycle, indicating cell death during mitosis, as detd. by FACS anal. AEZS 112 showed anti-tumor activity in human ovarian and endometrial cancer cell lines at low micromolar concns., which could not be abrogated by caspase ...
T77816 Deruxtecan analog 2

Deruxtecananalog 2(示例9 P3)是一种含活性分子-linker的Deruxtecan类似物,由Camptothecin(一种对多种癌症如结直肠癌、乳腺癌、肺癌和卵巢癌具有抗肿瘤活性的Topo I抑制剂)和linker组成,主要用于开发针对EGFR2的抗体药物偶联物(ADC)活性分子。
T62572 Enclomiphene hydrochloride

Enclomiphene ((E)-Clomiphene) hydrochloride 是一种口服具有活力的、有效的非甾体雌激素受体 (estrogen receptor) 拮抗剂,具有抗雌激素作用。Enclomiphene hydrochloride 能够用于研究卵巢功能障碍、睾酮缺乏、男性性腺功能减退症和 type 2 型糖尿病。
T35993 Epitalon (acetate)

Epitalon is a synthetic tetrapeptide with anti-aging properties.1,2,3,4 Dietary administration of epitalon (0.00001% w/w) reduces levels of lipid peroxidation products in aged D. melanogaster tissue homogenates.1 Epitalon (1 μg/animal) delays age-related estrous shutdown and decreases the frequency of bone marrow cell chromosomal aberrations in female mice.2 It decreases spontaneous mammary gland and ovarian tumor development and metastasis in aged female mice.3 Epitalon also stimulates melatoni...

化合物

Niraparib tosylate monohyrate
Cat.No: T9497
Synonym:
Target: PARP
SC144
Cat.No: T6207
Synonym:
Target: Apoptosis, Interleukin
Niraparib
Cat.No: T3231
Synonym: 尼拉帕尼,MK-4827
Target: Apoptosis, Others, PARP
Goserelin acetate
Cat.No: T4102
Synonym: 醋酸戈舍瑞林,Fertilan,ICI-118630 acetate,Zoladex
Target: Apoptosis, GNRH Receptor
Niraparib hydrochloride
Cat.No: T3353
Synonym: 尼拉帕利盐酸盐,MK-4827 hydrochloride,MK-4827 (hydrochloride)
Target: Apoptosis, Others, PARP
Niraparib tosylate
Cat.No: T6892
Synonym: 尼拉帕利,MK-4827 (tosylate),MK 4827 tosylate,Niraparib (MK-4827) tosylate,尼拉帕尼对苯甲磺酸盐
Target: Apoptosis, PARP
ABT-510 acetate
Cat.No: T24997
Synonym: ABT 510 acetate
Target: Apoptosis
Estrogen receptor antagonist 8
Cat.No: T78646
Synonym:
Target: Estrogen/progestogen Receptor
Zilovertamab
Cat.No: T76749
Synonym: Cirmtuzumab,UC-961
Target: Others
PHY34
Cat.No: T37376
Synonym:
Target: Autophagy
Abagovomab
Cat.No: T77408
Synonym: ACA 125
Target: Others
Mirvetuximab
Cat.No: T76766
Synonym: M9346A
Target: Antifolate
Ifebemtinib
Cat.No: T64167
Synonym: IN-10018,BI-853520
Target: FAK
Aspirin
Cat.No: T0005
Synonym: 阿司匹林,Acetylsalicylate,Acetylsalicylic Acid,邻乙酰水杨酸,ASA
Target: Mitophagy, Virus Protease, COX, Autophagy
DMU-212
Cat.No: T36674
Synonym:
Target: Apoptosis, ERK
DS-7423
Cat.No: T36083
Synonym:
Target: PI3K, mTOR
LP-184
Cat.No: T41070
Synonym:
Target:
CTX-2026
Cat.No: T82664
Synonym:
Target:
Cantrixil
Cat.No: T39586
Synonym: TRX-E-002-1
Target:
Estrogen receptor antagonist 7
Cat.No: T61909
Synonym:
Target:
IMAB027
Cat.No: T78296
Synonym: ASP1650
Target:
Navicixizumab
Cat.No: T76871
Synonym:
Target:
Vesencumab
Cat.No: T76879
Synonym:
Target:
VEGFR-2-IN-26
Cat.No: T63168
Synonym:
Target:
CDKI-83
Cat.No: T71287
Synonym:
Target:
AEZS-112
Cat.No: T71218
Synonym:
Target:
Deruxtecan analog 2
Cat.No: T77816
Synonym:
Target:
Enclomiphene hydrochloride
Cat.No: T62572
Synonym:
Target:
Epitalon (acetate)
Cat.No: T35993
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5755 Aloesin

Tyrosinase Proteases/Proteasome
Aloesin 是芦荟的活性成分之一,能够通过 MAPK 信号通路发挥抗癌作用,并具有抗炎、紫外线保护和抗菌作用。
T8206 Cycleanine

Others Others
Cycleanine 是一种高效血管选择性Ca- 拮抗剂,具有缓解疼痛、肌肉松弛和抗炎作用。它还具有有效的抗菌、抗真菌、抗疟原虫和细胞毒活性。
TN2064 Physcion 8-O-β-D-glucopyranoside

大黄素甲醚-8-O-Β-D-葡萄糖苷,Physcion 8-O-beta-D-monoglucoside

TNF Apoptosis
Physcion 8-O-β-D-glucopyranoside (Physcion 8-O-beta-D-monoglucoside) 具有抗炎和抗癌活性。Physcion 8-O-β-D-glucopyranoside 可用于常见恶性肿瘤的研究。
T4S0998 Trifolirhizin

红车轴草根甙/三叶豆紫檀苷,三叶豆紫檀苷

TNF; Tyrosinase Apoptosis; Proteases/Proteasome
Trifolirhizin 是一种从苦参根中分离出的 pterocarpan 黄酮类化合物。它具有酪氨酸酶高抑制活性,IC50=506 μM。它具有抗炎和抗癌的潜能。
TN3447 Arjunglucoside I

Arjunglucoside I has anti-inflammatory activity, it exhibits significant activity against carrageenan-induced paw edema in rat. It also shows antiproliferative activity against the A2780 human ovarian cancer cell line with an IC(50) value of 1.2 microM.
TN4168 Grifolin

Others Others
Grifolin has anti-cancer effects, it induces apoptosis and promotes cell cycle arrest in the A2780 human ovarian cancer cell line via inactivation of the ERK1/2 and Akt pathways; it enhances the differentiation and proliferation of oligodendrocyte precurs
TN5474 Bonducellin

Bonducellin has anti-inflammatory activities, it can significantly and dose-dependently inhibit the inflammatory mediators; nitric oxide (NO), and cytokines [tumor necrosis factor (TNF)-alpha and interleukin (IL)-12. Bonducellin shows weak antimalarial ac
TN3364 Agrimonolide

Apoptosis; Dehydrogenase; p38 MAPK; ROS; JAK Angiogenesis; Apoptosis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; MAPK; Metabolism; Stem Cells
Agrimonolide 是一种来自异香豆素的化合物,主要存在于草药Agrimonia pilosa Ledeb 中,具有显著的生物活性。Agrimonolide 通过抑制脂多糖(LPS)诱导的JAK-STATs 和p38 MAPKs 信号通路的激活而发挥抗炎作用。Agrimonolide 及其衍生物去甲阿戈莫内德已显示出能够有效提高肝细胞中胰岛素介导的糖原水平,可能在调节胰岛素抵抗的HepG2细胞中发挥关键作用。Agrimonolide 通过靶向卵巢癌细胞中的SCD1,对癌症的进展和诱导细胞死亡和凋亡表现出抑制作用。特别是,Agrimonolide 对A2780和SKOV-3细胞的增殖、迁移和侵袭表现出剂量依赖性的抑制,同时促进细胞凋亡。该化合物还被发现能诱导铁介导的细胞死亡,同时增加活性氧(ROS)和总铁的水平。Agrimonolide 很容易穿过血脑屏障,表明其在神经系统疾病的治疗应用方面具有潜力。

天然产物

Aloesin
Cat.No: T5755
Synonym:
Target: Tyrosinase
Cycleanine
Cat.No: T8206
Synonym:
Target: Others
Physcion 8-O-β-D-glucopyranoside
Cat.No: TN2064
Synonym: 大黄素甲醚-8-O-Β-D-葡萄糖苷,Physcion 8-O-beta-D-monoglucoside
Target: TNF
Trifolirhizin
Cat.No: T4S0998
Synonym: 红车轴草根甙/三叶豆紫檀苷,三叶豆紫檀苷
Target: TNF, Tyrosinase
Arjunglucoside I
Cat.No: TN3447
Synonym:
Target:
Grifolin
Cat.No: TN4168
Synonym:
Target: Others
Bonducellin
Cat.No: TN5474
Synonym:
Target:
Agrimonolide
Cat.No: TN3364
Synonym:
Target: Apoptosis, Dehydrogenase, p38 MAPK, ROS, JAK
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