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78

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T14495 Baloxavir

Baloxavir acid,S-033447

Influenza Virus Microbiology/Virology
Baloxavir (S-033447) 是衍生自前药 Baloxavir marboxil,是流感病毒聚合酶 PA 亚基的一流帽依赖性核酸内切酶抑制剂。它抑制病毒 RNA 的转录和复制,具有强大的抗病毒活性。
T4686 Simeprevir

TMC435,西咪匹韦,TMC-435350,Olysio

HCV Protease; SARS-CoV Microbiology/Virology; Proteases/Proteasome
Simeprevir (TMC435) 是一种有效的 HCV NS3/4A 蛋白酶抑制剂,抑制 HCV 复制,EC50 为 7.8 nM。它也是 SARS-CoV-2 3CLpro 抑制剂。
T8972 FIT-039

Others; DNA/RNA Synthesis; CDK; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
FIT-039 是一种选择性和 ATP 竞争性的口服活性 CDK9 抑制剂,对CKD9/cyclin T1的IC50为 5.8 μM。它抑制HSV-1(IC50为 0.69 μM),HSV-2,人腺病毒和人CMV 的复制。它可抑制耐药性HSV 和其他 DNA 病毒,是有前途的抗病毒药物。
T5539 GS-443902

瑞德西韦代谢物

Nucleoside Antimetabolite/Analog; HCV Protease; SARS-CoV; DNA/RNA Synthesis; RSV; Drug Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; Proteases/Proteasome
Remdesivir triphosphate 是一种有效的病毒 RNA 依赖的 RNA 聚合酶抑制剂,对RSVRdRp 和 HCVRdRp 的IC50分别为 1.1 µM 和 5 µM。它是 Remdesivir 的活性三磷酸代谢物。
T10493 Beclabuvir

BMS-791325

Others Others
Beclabuvir is an allosteric inhibitor that binds to thumb site 1 of the HCV NS5B RNA-dependent RNA polymerase. It inhibits recombinant NS5B proteins from HCV genotypes 1, 3, 4, and 5 (IC50 < 28 nM).
T15282 Filibuvir

PF-00868554

HCV Protease; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
Filibuvir (PF-00868554) 是 HCV NS5B RNA 依赖性 RNA 聚合酶的选择性非共价抑制剂。 Filibuvir 抑制基因型 1a 和 1b 复制子,EC50 为 59 nM。
T9617 RdRP-IN-2

SARS-CoV Microbiology/Virology
RdRP-IN-2 是一种依赖于 RNARNA 聚合酶 (RdRp) 抑制剂。它显著抑制 SARS-CoV-2 RdRp,IC50 为 41.2 µM。它还抑制猫冠状病毒 (FIPV) 复制。
T6833 Favipiravir

T-705,6-Fluoro-3-oxo-3,4-dihydropyrazine-2-carboxamide,法匹拉韦,法维拉韦

Others; SARS-CoV; Influenza Virus; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Favipiravir (T-705) 是一种有效且选择性的 RNA 依赖性 RNA 聚合酶抑制剂,用于治疗流感病毒感染。
T1501 Rifabutin

LM-427,Ansamycin,利福布汀,利福布丁

HSP; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Rifabutin (LM-427) 是半合成的安莎霉素抗生素,抑制 DNA 依赖性 RNA 聚合酶,有抗分枝杆菌作用。
T27696 JTK-109

JTK109

HCV Protease Microbiology/Virology; Proteases/Proteasome
JTK-109 是一种丙型肝炎病毒 NS5B RNA 依赖性 RNA 聚合酶抑制剂,可抑制 G1b 和 G3a 亚基因组复制子和重组酶。
T9618 HeE1-2Tyr

SARS-CoV Microbiology/Virology
HeE1-2Tyr 是 一种pyridobenzothiazole,抑制黄病毒 RNA 依赖性 RNA 聚合酶。HeE1-2Tyr 在体外对Dengue, West Nile 和 SARS-CoV-2 RdRps 有显著的抑制活性(IC50为 27.6 µM) 。
TQ0090 Nesbuvir

HCV-796

HCV Protease Microbiology/Virology; Proteases/Proteasome
Nesbuvir 是一种选择性丙型肝炎病毒(HCV)非结构蛋白5B(NS5B)RNA 依赖性聚合酶抑制剂。Nesbuvir 对含1b HCV 复制子的肝癌细胞的 IC50为9nM。
T10491 Galidesivir

BCX4430,Immucillin-A

Others Others
Galidesivir (BCX4430) 是一种广谱抗病毒化合物,是一种腺苷类似物,能抑制病毒 RNA 依赖的 RNA 聚合酶 (RdRp) 活性。Galidesivir 在体外对多种 RNA 病毒病原体有抑制作用,可减少受感染动物的肺部感染。
T82568 DHX9-IN-2

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
DHX9-IN-2 是一种针对ATP依赖型RNA解螺旋酶A(DHX9)的抑制剂,具有抗癌和抗肿瘤活性,可用于研究癌症。
T3489 Dasabuvir

ABT-333,达塞布韦

HCV Protease Microbiology/Virology; Proteases/Proteasome
Dasabuvir (ABT-333) 是丙型肝炎病毒非结构蛋白 5B 的非核苷抑制剂,是一种 RNA 依赖性 RNA 聚合酶,具有抗 HCV 的潜在活性。
T63253 AVG-233

DNA/RNA Synthesis; RSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
AVG-233 是一种可口服的RNA 依赖性 RNA 聚合酶 (RdRp) 抑制剂,具有抗病毒活性,可阻断呼吸道合胞病毒和 SARS-CoV-2 复制。AVG-233 可用于研究呼吸道合胞病毒感染。
T7766 Remdesivir

瑞德西韦,GS-5734

SARS-CoV; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Remdesivir (GS-5734) 是一种核苷类似物,一种广谱的抗病毒化合物,通过抑制病毒的 RNA 依赖性 RNA 聚合酶发挥活性。Remdesivir 对埃博拉病毒、SARS 病毒、MERS病毒等均有活性,对 COVID-19 有潜在治疗价值。
T1154 Rifaximin

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Rifaximin 是一种胃肠道选择性抗生素,与细菌 DNA 依赖性 RNA 聚合酶的 β 亚基结合,抑制细菌 RNA 合成。与革兰氏阴性菌(MIC:8-50 毫克/毫升)相比,它对革兰氏阳性菌株(MIC:0.03-5 毫克/毫升)的敏感性更高。
T11760 KIN101

3-(4-Bromophenyl)-7-[(methylsulfonyl)oxy]-4-oxo-4H-chromene,3-(4-溴苯基)-4-氧代-7-[(甲磺酰基)氧基]-4H-色烯

HCV Protease; Influenza Virus; RSV; Antifection Microbiology/Virology; Proteases/Proteasome
KIN101 (3-(4-Bromophenyl)-7-[(methylsulfonyl)oxy]-4-oxo-4H-chromene) 是 IRF-3 依赖性信号传导的异黄酮激动剂,可诱导 IRF-3 核易位。 它对 RNA 病毒、HCV 和 RSV 具有抗病毒活性。
T61334 DMA-135 hydrochloride

DMA-135 HCl

Virus Protease Microbiology/Virology
DMA-135 hydrochloride (DMA-135 HCl) 靶向 RNA 的抗病毒活性化合物,抑制肠道病毒 71 型 (EV71)IRES依赖的翻译和复制。DMA-135 hydrochloride 可用于研究肠道病毒感染。
T19836 2-Aminopurine

DNA/RNA Synthesis; PKA Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Tyrosine Kinase/Adaptors
2-Aminopurine 是一种鸟苷和腺苷的荧光类似物,是基于荧光衰变的 DNA 结构探针。当它插入寡核苷酸后,其荧光会通过与天然碱基堆积而被高度淬灭。它可用于核酸的结构和动力学的探测。
T77520 AOH1996

Apoptosis; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
AOH1996 是一种具有口服活性的复制体组分 PCNA (增殖细胞核抗原) 配体,靶向转录-复制冲突 (TRC)。AOH1996 可干扰 PCNA 与其结合蛋白的相互作用,导致 DNA 复制应激,诱导细胞凋亡 (apoptosis)。AOH1996 通过稳定 PCNA 和 RNA 聚合酶 II 的相互作用从而导致蛋白酶体依赖的 rpb1 降解和致命的 DNA 损伤。AOH1996 与 DNA 损伤剂具有协同作用,可抑制肿瘤细胞生长。
T79404 A09-003

Apoptosis; BCL; CDK Apoptosis; Cell Cycle/Checkpoint
A09-003 是一种新型细胞周期蛋白依赖性激酶-9 CDK-9 抑制剂。A09-003 能够抑制多种白血病细胞系的增殖,抑制hi髓系细胞白血病序列-1蛋白增加。A09-003还能诱导细胞凋亡,降低 RNA 聚合酶 II 活性,降低 Mcl-1 表达。
T27260 Emivirine

MKC442,MKC-442,MKC 442,DRG-0302,DRG 0302,DRG0302

HIV Protease Microbiology/Virology; Proteases/Proteasome
Emivirine (MKC-442) 是一种有效和选择性的人类免疫缺陷病毒1型(HIV-1)的非核苷逆转录酶抑制剂。
T40267 RdRP-IN-3

RdRP-IN-3, a potential anti-influenza drug candidate, functions by inhibiting the activity of RNA-dependent RNA polymerase (RdRp).
T71748 RK-0404678

RK-0404678 is a novel inhibitor of dengue virus NS5 RNA-dependent RNA polymerase (RdRp), inhibiting the DENV type 2 (DENV2) RdRp activities.
T28538 Rifamycin SV

Rifamycin SV, a natural antibiotic, blocks RNA-polymerase transcription initiation, modulating ß2m aggregation; inhibits prokaryotic DNA-dependent RNA synthesis and protein synthesis.
T10491L Galidesivir hydrochloride

BCX 4430 hydrochloride,Immucillin-A hydrochloride

Others Others
Galidesivir hydrochloride is an inhibitor of viral RNA-dependent RNA polymerase (RdRp). It inhibits SARS-CoV-2 by tightly binding to its RdRp.
T21225 Rifamycin

Rifocin,Rifamycin SV

Rifamycin, a natural antibiotic, inhibits prokaryotic DNA-dependent RNA synthesis and protein synthesis, leading to the block of RNA-polymerase transcription initiation.
T71825 BEPP monohydrochloride

BEPP monohydrochloride is a double-strand RNA-dependent protein kinase (PKR) activator.
T27485 GSK-625433

GSK-625433, a homochiral inhibitor of the hepatitis C virus (HCV) RNA-dependent RNA polymerase, has the ability to inhibit the polymerase of both HCV genotypes 1a and 1b.
T62160 AS-136A

AS-136A 是一种麻疹病毒 RNA 依赖性 RNA 聚合酶(RdRp)的、口服具有活力的非核苷抑制剂,能够作用于麻疹病毒 (IC50: 2 μM)。
T63598 DENV-IN-4

DENV-IN-4 是 DENV 的有效抑制剂 (DENV EC50=4.79 μM, Vero CC50>100 μM, SI>20.9)。DENV-IN-4 能够减少 DENV2 的表达水平,具有浓度依赖性,并可抑制依赖性 RNA 聚合酶 (RNA-dependent RNA polymerase, RdRp) 的活性,表现出抗病毒效果。
T11062 dmDNA31

Others Others
dmDNA31 is a rifamycin antibiotic that can inhibit the DNA-dependent RNA polymerase of bacteria and has strong bactericidal activity against Staphylococcus aureus.
T70855 Favipiravir sodium

Favipiravir sodium is a selective inhibitor of viral RNA-dependent RNA polymerase with activity against many RNA viruses, influenza viruses, West Nile virus, yellow fever virus, foot-and-mouth disease virus as well as other flaviviruses, arenaviruses, bunyaviruses and alphaviruses.
T79233 RdRP-IN-6

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
RdRP-IN-6(化合物27),其针对RNA依赖型RNA聚合酶(RdRP)的抑制IC90值为14.1 μM,适用于抗病毒和抗癌研究领域。
T25106 Aranotin

L53185,Lilly 53185,L 53185,L-53185,Antibiotic A 21101-IL

Aranotin 是一种从金黄色蜘蛛中分离的真菌毒素,具有对抗脊髓灰质炎病毒、柯萨奇病毒、犀牛和副流感病毒等 RNA 病毒的活性。Aranotin 通过阻碍 RNA 依赖性RNA 聚合酶的活性来抑制病毒RNA 的合成。
T11352 Galidesivir triphosphate

BCX4430-triphosphate,Immucillin-A triphosphate,BCX6870

Others Others
Galidesivir triphosphate is a substrate for viral RNA-dependent RNA polymerase (RDRP), resulting in termination of viral RNA replication and thus serves as an antiviral. Galidesivir triphosphate inhibits HCV NS5B RNA polymerase activity and protects mice against Ebola. Galidesivir triphosphate (Immucillin-A triphosphate) is converted by the prodrug Galidesivir.
T67814 TMC-649128 PM

TMC-649128 PM 是HCV NS5B RNA 依赖性RNA 聚合酶的有效核苷抑制剂,EC(50)值为1.2 muM,大鼠体内生物利用度中等(F=14%)。
T40616 8-Azido-ATP

8-Azidoadenosine 5'-triphosphate,8-N3-ATP,8-Azido-ATP

8-Azido-ATP is a nucleotide analog that demonstrates photo-reactivity properties. It offers utility in the precise labeling and identification of proteins, particularly those involved in DNA-dependent RNA polymerase activity.
T38616 Teprasiran

QPI-1002

Teprasiran (QPI-1002) is an RNA-based compound that transiently suppresses p53-dependent apoptosis, a process involved in the development of acute kidney injury (AKI).
T35533 6-Hydroxypyridin-3-ylboronic Acid

6-Hydroxypyridin-3-ylboronic acid is a heterocyclic building block.1,2It has been used in the synthesis of non-nucleoside inhibitors of hepatitis C virus (HCV) RNA-dependent RNA polymerase nonstructural protein 5B (NS5B).16-Hydroxypyridin-3-ylboronic acid has also been used in the synthesis of mammalian target of rapamycin (mTOR) inhibitors.2 1.Hendricks, R.T., Spencer, S.R., Blake, J.F., et al.3-Hydroxyisoquinolines as inhibitors of HCV NS5b RNA-dependent RNA polymeraseBioorg. Med. Chem. Lett.1...
T41177 Galidesivir dihydrochloride

BCX 4430

Galidesivir is a viral RNA-dependent RNA polymerase (RdRP) inhibitor and broad spectrum antiviral nucleotide.In vitro, galidesivir displays antiviral activity against a range of RNA viruses, including bunyaviruses, arenaviruses, paramyxoviruses, coronaviruses, and flaviviruses (EC50values range from 3 μM to >100 μM). Galidesivir protects against Ebola and Marburg viral infection in animal models.
T73323 RdRP-IN-5

Influenza Virus Microbiology/Virology
RdRP-IN-5 (compound 20) 为一种抑制流感病毒RNA依赖性RNA聚合酶(RdRP)的有效药物,适用于该病毒研究。
T72792 trans-RdRP-IN-5

trans-RdRP-IN-5 是一种有效的流感病毒 RNA 依赖性 RNA 聚合酶 (RdRP) 抑制剂。trans-RdRP-IN-5 可用于流感病毒的研究。
T72896 cis-RdRP-IN-5

cis-RdRP-IN-5 是一种有效的流感病毒 RNA 依赖性 RNA 聚合酶 (RdRP) 抑制剂。cis-RdRP-IN-5 可用于流感病毒的研究。
T83251 7-51A

Influenza Virus Microbiology/Virology
7-51A为一有效PB2抑制剂,其通过ITC测定的KD值仅为1.64 nM;PB2为流感RNA依赖性RNA聚合酶(RdRP)的关键亚基。
T63073 Cap-dependent endonuclease-IN-19

Cap-dependent endonuclease-IN-19 是一种螺环吡啶酮衍生物,是一种 cap-dependent 核酸内切酶 (CEN) 的有效抑制剂。Cap-dependent endonuclease-IN-19 能够强效的抑制甲型流感病毒的 RNA 聚合酶活性。
T35658 3'-Deoxyuridine-5'-triphosphate trisodium

3'-Deoxyuridine-5'-triphosphate trisodium (3'-dUTP trisodium) is a nucleotide analogue that inhibits DNA-dependent RNA polymerases I and II. 3'-Deoxyuridine-5'-triphosphate trisodium strongly and competitively inhibits the incorporations of UTP into RNA with a Ki value of 2.0 μM[1]. 3'-Deoxyuridine-5'-triphosphate (3'-dUTP) is synthesized starting from cordycepin in good yield. 3'-Deoxyuridine-5'-triphosphate strongly and competitively inhibits the incorporations of UTP into RNA by the RNA polym...
T82569 DHX9-IN-1

DHX9-IN-1,作为ATP依赖性RNA解螺旋酶A (DHX9) 的抑制剂,表现出9.45 nM的IC50值,并具有抗肿瘤活性。

化合物

Baloxavir
Cat.No: T14495
Synonym: Baloxavir acid,S-033447
Target: Influenza Virus
Simeprevir
Cat.No: T4686
Synonym: TMC435,西咪匹韦,TMC-435350,Olysio
Target: HCV Protease, SARS-CoV
FIT-039
Cat.No: T8972
Synonym:
Target: Others, DNA/RNA Synthesis, CDK, HSV
GS-443902
Cat.No: T5539
Synonym: 瑞德西韦代谢物
Target: Nucleoside Antimetabolite/Analog, HCV Protease, SARS-CoV, DNA/RNA Synthesis, RSV, Drug Metabolite
Beclabuvir
Cat.No: T10493
Synonym: BMS-791325
Target: Others
Filibuvir
Cat.No: T15282
Synonym: PF-00868554
Target: HCV Protease, DNA/RNA Synthesis
RdRP-IN-2
Cat.No: T9617
Synonym:
Target: SARS-CoV
Favipiravir
Cat.No: T6833
Synonym: T-705,6-Fluoro-3-oxo-3,4-dihydropyrazine-2-carboxamide,法匹拉韦,法维拉韦
Target: Others, SARS-CoV, Influenza Virus, DNA/RNA Synthesis
Rifabutin
Cat.No: T1501
Synonym: LM-427,Ansamycin,利福布汀,利福布丁
Target: HSP, DNA/RNA Synthesis, Antibacterial, Antibiotic
JTK-109
Cat.No: T27696
Synonym: JTK109
Target: HCV Protease
HeE1-2Tyr
Cat.No: T9618
Synonym:
Target: SARS-CoV
Nesbuvir
Cat.No: TQ0090
Synonym: HCV-796
Target: HCV Protease
Galidesivir
Cat.No: T10491
Synonym: BCX4430,Immucillin-A
Target: Others
DHX9-IN-2
Cat.No: T82568
Synonym:
Target: DNA/RNA Synthesis
Dasabuvir
Cat.No: T3489
Synonym: ABT-333,达塞布韦
Target: HCV Protease
AVG-233
Cat.No: T63253
Synonym:
Target: DNA/RNA Synthesis, RSV
Remdesivir
Cat.No: T7766
Synonym: 瑞德西韦,GS-5734
Target: SARS-CoV, DNA/RNA Synthesis
Rifaximin
Cat.No: T1154
Synonym:
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
KIN101
Cat.No: T11760
Synonym: 3-(4-Bromophenyl)-7-[(methylsulfonyl)oxy]-4-oxo-4H-chromene,3-(4-溴苯基)-4-氧代-7-[(甲磺酰基)氧基]-4H-色烯
Target: HCV Protease, Influenza Virus, RSV, Antifection
DMA-135 hydrochloride
Cat.No: T61334
Synonym: DMA-135 HCl
Target: Virus Protease
2-Aminopurine
Cat.No: T19836
Synonym:
Target: DNA/RNA Synthesis, PKA
AOH1996
Cat.No: T77520
Synonym:
Target: Apoptosis, DNA/RNA Synthesis
A09-003
Cat.No: T79404
Synonym:
Target: Apoptosis, BCL, CDK
Emivirine
Cat.No: T27260
Synonym: MKC442,MKC-442,MKC 442,DRG-0302,DRG 0302,DRG0302
Target: HIV Protease
RdRP-IN-3
Cat.No: T40267
Synonym:
Target:
RK-0404678
Cat.No: T71748
Synonym:
Target:
Rifamycin SV
Cat.No: T28538
Synonym:
Target:
Galidesivir hydrochloride
Cat.No: T10491L
Synonym: BCX 4430 hydrochloride,Immucillin-A hydrochloride
Target: Others
Rifamycin
Cat.No: T21225
Synonym: Rifocin,Rifamycin SV
Target:
BEPP monohydrochloride
Cat.No: T71825
Synonym:
Target:
GSK-625433
Cat.No: T27485
Synonym:
Target:
AS-136A
Cat.No: T62160
Synonym:
Target:
DENV-IN-4
Cat.No: T63598
Synonym:
Target:
dmDNA31
Cat.No: T11062
Synonym:
Target: Others
Favipiravir sodium
Cat.No: T70855
Synonym:
Target:
RdRP-IN-6
Cat.No: T79233
Synonym:
Target: DNA/RNA Synthesis
Aranotin
Cat.No: T25106
Synonym: L53185,Lilly 53185,L 53185,L-53185,Antibiotic A 21101-IL
Target:
Galidesivir triphosphate
Cat.No: T11352
Synonym: BCX4430-triphosphate,Immucillin-A triphosphate,BCX6870
Target: Others
TMC-649128 PM
Cat.No: T67814
Synonym:
Target:
8-Azido-ATP
Cat.No: T40616
Synonym: 8-Azidoadenosine 5'-triphosphate,8-N3-ATP,8-Azido-ATP
Target:
Teprasiran
Cat.No: T38616
Synonym: QPI-1002
Target:
6-Hydroxypyridin-3-ylboronic Acid
Cat.No: T35533
Synonym:
Target:
Galidesivir dihydrochloride
Cat.No: T41177
Synonym: BCX 4430
Target:
RdRP-IN-5
Cat.No: T73323
Synonym:
Target: Influenza Virus
trans-RdRP-IN-5
Cat.No: T72792
Synonym:
Target:
cis-RdRP-IN-5
Cat.No: T72896
Synonym:
Target:
7-51A
Cat.No: T83251
Synonym:
Target: Influenza Virus
Cap-dependent endonuclease-IN-19
Cat.No: T63073
Synonym:
Target:
3'-Deoxyuridine-5'-triphosphate trisodium
Cat.No: T35658
Synonym:
Target:
DHX9-IN-1
Cat.No: T82569
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T17143 Toyocamycin

丰加霉素,Vengicide

Apoptosis; Others; IRE1; Antibiotic; Antifungal Apoptosis; Cell Cycle/Checkpoint; Microbiology/Virology; Others
Toyocamycin (Vengicide) 是放线菌类产生的腺苷类似物,为 X 盒结合蛋白 1 (XBP1) 抑制剂,抑制 IRE1α 诱导的 ATP 依赖性 XBP1 mRNA 的断裂,IC50值为 80 nM。它还诱导凋亡。
T5003 Rifamycin sodium

Rifamycin sodium salt,利福霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Rifamycin sodium (Rifamycin sodium salt) salt 是从地中海曲霉或其突变体的发酵中分离出来的一种安沙霉素抗生素家族。它对革兰氏阳性菌和某些革兰氏阴性菌有抗生素活性。
T8347 Rifamycin S

Reactive Oxygen Species; ROS; Antibacterial; Antibiotic Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Rifamycin S 是一种 DNA 依赖性 RNA 聚合酶抑制剂,是一种醌和一种针对革兰氏阳性细菌的抗生素试剂。它是涉及两个电子的可逆氧化还原系统的氧化形式。它能产生活性氧并抑制微粒体脂质过氧化,可研究肺结核和麻风病。
TN1258 3-Acetyl-beta-boswellic acid

3-O-Acetyl-beta-boswellic acid,3-乙酰基-BETA-乳香酸

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
3-Acetyl-beta-boswellic acid 是一种乳香酸,分离自乳香锯缘胶树脂。
T5075 Phytic acid potassium

植酸二钾盐,Inositol hexakisphosphate dipotassium salt,Phytic acid dipotassium salt,Fytic Acid dipotassium salt,Inositol polyphosphate dipotassium salt

Others; Endogenous Metabolite Metabolism; Others
Phytic acid potassium (Inositol polyphosphate dipotassium salt) 是内源性代谢产物的一种。
TN2222 Sotetsuflavone

Others Others
Sotetsuflavone is a potent inhibitor of DENV-NS5 RdRp (Dengue virus NS5 RNA-dependent RNA polymerase) with an IC50 of 0.16 μM, is the most active compound of this series.
T11233 Erythromycin thiocyanate

Antibacterial Microbiology/Virology
Erythromycin thiocyanate acts by binding to bacterial 50S ribosomal subunits and inhibits RNA-dependent protein synthesis by blockage of transpeptidation and/or translocation reactions, without affecting synthesis of nucleic acid .Erythromycin thiocyanate

天然产物

Toyocamycin
Cat.No: T17143
Synonym: 丰加霉素,Vengicide
Target: Apoptosis, Others, IRE1, Antibiotic, Antifungal
Rifamycin sodium
Cat.No: T5003
Synonym: Rifamycin sodium salt,利福霉素钠
Target: Antibacterial, Antibiotic
Rifamycin S
Cat.No: T8347
Synonym:
Target: Reactive Oxygen Species, ROS, Antibacterial, Antibiotic
3-Acetyl-beta-boswellic acid
Cat.No: TN1258
Synonym: 3-O-Acetyl-beta-boswellic acid,3-乙酰基-BETA-乳香酸
Target: DNA/RNA Synthesis
Phytic acid potassium
Cat.No: T5075
Synonym: 植酸二钾盐,Inositol hexakisphosphate dipotassium salt,Phytic acid dipotassium salt,Fytic Acid dipotassium salt,Inositol polyphosphate dipotassium salt
Target: Others, Endogenous Metabolite
Sotetsuflavone
Cat.No: TN2222
Synonym:
Target: Others
Erythromycin thiocyanate
Cat.No: T11233
Synonym:
Target: Antibacterial
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