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Targets Recommended: Apelin receptor DNA/RNA Synthesis

185

抑制剂 & 化合物

21

天然产物

12

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T61487 APE1-IN-1

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
APE1-IN-1 是一种可透过血脑屏障且有效的无嘌呤/嘧啶内切酶 1 (APE1) 抑制剂,具有潜在的抗肿瘤活性,可增强烷基化剂甲基甲烷磺酸盐对癌细胞的细胞毒性。
T73299 APE1-IN-2

Apoptosis Apoptosis
APE1-IN-2(compound AP1)是一种具有抗癌活性的Pt(IV)前体,靶向BER关键蛋白APE1。该化合物能诱导细胞内铂的积累,并激活DNA损伤反应及凋亡信号。
T6507 Gabapentin hydrochloride

加巴喷丁盐酸盐,Neurontin HCl,Gabapentin HCl

Calcium Channel; GABA Receptor Membrane transporter/Ion channel; Metabolism; Neuroscience
Gabapentin hydrochloride (Neurontin HCl) 是GABA 类似物,可用于缓解神经性疼痛。
TP1101 Nonapeptide-1 acetate salt (158563-45-2 free base)

Melanostatine-5 acetate salt,Nonapeptide-1 acetate salt

Melanocortin Receptor GPCR/G Protein; Neuroscience
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) 是一种肽激素,是一种有效的 α-黑色素细胞刺激素 (α-MSH) 拮抗剂,IC50 为 11 nM。
T7769 Nonapeptide-1

Met-Pro-D-Phe-Arg-D-Trp-Phe-Lys-Pro-Val-,九胜肽-1,Melanostatine™ 5

Others Others
Nonapeptide-1 (Melanostatine™ 5) 可以抑制黑色素的合成,这使得它对治疗某些皮肤病很感兴趣。
T20494L Acetyl tetrapeptide-15 Acetate

Skinasensyl Acetate,Acetyl tetrapeptide-15 Acetate (928007-64-1 Free base)

Acetyl tetrapeptide-15 Acetate (Skinasensyl Acetate) 是一种用于敏感皮肤的化妆品中的合成肽,是 endomorphin-2 衍生物, 通过内啡肽样通路扩大 μ-阿片受体中的神经元兴奋性阈值范围,可用于研究由皮肤高反应性产生的炎症性和神经性疼痛。
T40622 Mapenterol hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Mapenterol hydrochloride 是 β2 肾上腺素受体激动剂。
T1629 Rifapentine

MDL473,Rifapentina,Rifapentinum,DL 473,利福喷丁,Priftin,Cyclopentylrifampicin

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Rifapentine (Rifapentinum) 是可用于肺结核的抗生素。
T6411 Biapenem

CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627

Antibacterial; Antibiotic Microbiology/Virology
Biapenem (CLI 86815) 是不经肠道的广谱碳青霉烯抗生素。
T0464 Carbetapentane citrate

托可拉斯,Pentoxyverine citrate,咳必清

AChR Neuroscience
Carbetapentane citrate (Pentoxyverine citrate) 能够选择性抑制咳嗽中枢,具有轻度的阿托品样作用和局麻作用。
TP1260 [Pyr1]-Apelin-13

[pGlu1]-Apelin-13,人牛吡啶APELIN-13

Apelin receptor GPCR/G Protein
[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) 是一种高效的、内源性 apelin 受体选择性激动剂。
TP2313 Acetyl Tetrapeptide-5 acetate

Acetyl Tetrapeptide-5 acetate(820959-17-9 free base)

Others Others
Acetyl Tetrapeptide-5 acetate(820959-17-9 free base) 有助于减少眼部浮肿,改善皮肤弹性以及整体光滑度。
T64318 Capecitabine-2',3'-cyclic Carbonate

Others Others
Capecitabine-2',3'-cyclic Carbonate 是一种抗增殖化合物。
T14083 Abaperidone

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Abaperidone 是一种有效的 5-HT2A 受体和多巴胺 D2 受体拮抗剂,对 5-HT2A 受体的 IC50 为 6.2 nM,对多巴胺 D2 受体的IC50 为 17 nM。Abaperidone是一种潜在的非典型抗精神化合物,可降低大鼠纹状体和前额叶皮层中的基础hsp70 mRNA表达。
TP2092L Apelin-17 (human, bovine) acetate

Apelin-17 (human, bovine) acetate(217082-57-0 free base)

HIV Protease Microbiology/Virology; Proteases/Proteasome
Apelin-17 (human, bovine) acetate(217082-57-0 free base) 是一种内源性 apelin 受体激动剂。有效抑制毛喉素刺激的 cAMP 积累 (pIC50 = 9.94)。
T21249L Myristoyl Pentapeptide-17 Acetate

Myristoyl Pentapeptide-17 Acetate(959610-30-1 Free base)

Others Others
Myristoyl Pentapeptide-17 Acetate 是一种小肽。促进关键成分的输送,从而有效促进睫毛生长,使睫毛变长变浓密,强韧秀发,显着强化眼部表情。
TP2204L CCK Octapeptide, non-sulfated acetate

CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)

cholecystokinin GPCR/G Protein
CCK Octapeptide, non-sulfated acetate 是一种合成的胆囊收缩素脱硫酸肽。
T38318L Acetyl Pentapeptide-1 acetate

Histone Demethylase Chromatin/Epigenetic
Acetyl Pentapeptide-1 acetate 是一种组蛋白脱乙酰酶抑制剂。
T68023L Tolnapersine TFA

Tolnapersine TFA(70312-00-4 Free base)

Dopamine Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Tolnapersine TFA 是混合多巴胺激动剂和α肾上腺素受体拮抗剂。
TP2365L Acetyl tetrapeptide-9 Acetate

Acetyl tetrapeptide-9 Acetate(928006-50-2 Free base)

Others Others
Acetyl tetrapeptide-9 Acetate 在刺激基底膜多糖(lumican)和胶原蛋白 I 的合成中发挥作用。
TP2419 V-9-M Cholecystokinin nonapeptide

V 9 M,Prepro CCK Fragment V-9-M,Val-pro-val-glu-ala-val-asp-pro-met,Cholecystokinin Precursor (24-32),V9M,V-9-M

Beta Amyloid Neuroscience
V-9-M Cholecystokinin nonapeptide (Prepro CCK Fragment V-9-M) 是胆囊收缩素(CCK)的前体化合物。胆囊收缩素(CCK)是一种刺激胆囊收缩和胰腺外分泌的脑肠肽,可从狗和猫的小肠中提取的,可以引起胆囊收缩。
T4990 Cefcapene pivoxil hydrochloride hydrate

Cefcapene Pivoxil Hydrochloride,盐酸头孢卡品酯

Antibacterial; Antibiotic Microbiology/Virology
Cefcapene pivoxil hydrochloride hydrate 是一种头孢菌素的前药,具有口服活性和广谱抗菌活性。它可研究掌跖脓疱病等感染性疾病。
T68087 Inaperisone

Others Others
Inaperisone 是一种新型的中枢作用的肌肉松弛剂,对排尿反射有抑制作用。Inaperisone 可能通过间接作用于脑干的GABAB 受体来抑制排尿反射。
T68165 Trapencaine

Trapencaine 是一种新合成的氨基甲酸型局部麻醉剂,诱导的肥大细胞膜上钠通道的构象变化。
T39823L Apelin-12 acetate

Apelin-12 acetate (229961-08-4 Free base)

Apelin receptor; p38 MAPK; JNK GPCR/G Protein; MAPK
Apelin-12 acetate 对 APJ 受体具有高亲和力。 Apelin-12 acetate 抑制凋亡相关 MAPKs 家族的 JNK 和 p38 MAPK 信号通路,从而为神经元提供保护。
T7656 Apelin-13

Apelin-13 是存在于中枢和外周神经系统由13个氨基酸组成的多肽序列,是 G 蛋白偶联受体angiotensin II protein J (APJ) 的内源性配体,对 APJ 的 EC50 值为 0.37 nM。Apelin-13 具有扩张血管和降压活性,可用于研究 2 型糖尿病综合征。
T4991 Ertapenem sodium

厄他培南钠,MK-826,L-749345,尔他培南钠

Antibacterial; Antibiotic Microbiology/Virology
Ertapenem sodium (MK-826) 是碳青霉烯,是一种 β-内酰胺抗生素,具有广谱抗菌活性。
T0702 Gabapentin

Neurontin,Gabapentine,加巴喷丁,Aclonium

Calcium Channel; GABA Receptor Membrane transporter/Ion channel; Metabolism; Neuroscience
Gabapentin (Neurontin) 是GABA 类似物,是一种抗癫痫药,可用于缓解神经性疼痛。
T68035 Capeserod

SL-650155,SL-65.0155

5-HT Receptor GPCR/G Protein; Neuroscience
Capeserod 是一种潜在的 5-HT4 receptor(5-羟色胺受体4)激动剂,可用于研究消化系统疾病和神经系统疾病。
T3497 Ocaperidone

奥卡哌酮,Ocaperidona,R79598

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Ocaperidone (Ocaperidona) 是5-HT2和多巴胺D2的拮抗剂,也是5-HT1A 的激动剂,有安定作用。
TP2364L Acetyl tetrapeptide-3 Acetate

Acetyl tetrapeptide-3 Acetate(827306-88-7 Free base)

Others Others
Acetyl tetrapeptide-3 Acetate 是一种仿生肽。
T7847 Apelin-13 triTFA(217082-58-1(free base))

Others Others
Apelin-13 triTFA(217082-58-1(free base)) 是 APJ 受体的内源性配体,可激活该 G 蛋白偶联受体,EC50 值为 0.37 nM。
T8833 2-chloro-5-(16,18-dioxo-17-azapentacyclo[6.6.5.0~2,7~.0~9,14~.0~15,19~]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoic acid

Others Others
2-chloro-5-(16,18-dioxo-17-azapentacyclo[6.6.5.0~2,7~.0~9,14~.0~15,19~]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoic acid 可用于合成多种有机化合物。
TP2496 Octapeptide-2 Acetate

Octapeptide-2 Acetate(1374396-34-5 Free base)

Others Others
Octapeptide-2 Acetate 作为一种促进毛发生长的活性物质,是一种双层封装的仿生肽,有助于促进细胞生长和迁移。它通过激活毛囊的干细胞来促进头发生长。 它比天然蛋白质更稳定且作用时间更长。
TP2497 Myristoyl Tetrapeptide-12 Acetate

醋酸肉蔻酰四胜肽-12,Myristoyl Tetrapeptide-12 Acetate(959610-24-3 Free base)

Others Others
Myristoyl Tetrapeptide-12 Acetate (Myristoyl Tetrapeptide-12 Acetate (959610-24-3 Free base)) 是肉豆蔻酸和 Tetrapeptide-12 的反应产物,是一种刺激头发和睫毛生长并增强睫毛和/或眉毛外观的肽。 Myristoyl tetrapeptide-12 可以增加角质形成细胞的增殖,改善外观、紧致弹性和皮肤厚度。
TP2316 Myristoyl Hexapeptide-23 Acetate

Others Others
Myristoyl Hexapeptide-23 Acetate 有抗粉刺作用。
TP1042 Palmitoyl Tetrapeptide-3

Rigin,棕榈酰四肽-7/棕榈酰四肽-3

Others Others
Palmitoyl Tetrapeptide-3 (Rigin) 是一种具有刺激吞噬活性的合成多肽,对应人免疫球蛋白重链的第 341-344 氨基酸序列。
TP1341L Polymyxin B nonapeptide acetate

Polymyxin B nonapeptide acetate(86408-36-8 free base)

Antibacterial; Antibiotic Microbiology/Virology
Polymyxin B nonapeptide acetate(86408-36-8 free base) 是一种阳离子环肽。 Polyxin B 九肽是 polyxin B 经酶解产生的衍生物。与 polyxin B 相比,polyxin B 九肽毒性低,缺乏杀菌活性,仍具有破坏革兰氏阴性菌外膜的能力。
TP2499 Human IgE Pentapeptide HEPP acetate

Human IgE Pentapeptide HEPP acetate (62087-72-3 Free base)

Human IgE Pentapeptide HEPP acetate 是一种五肽,在几种不同体系中均不能产生 IgE 抑制作用,可用于治疗结膜炎。
T11894 Lusaperidone

R107474

Adrenergic Receptor GPCR/G Protein; Neuroscience
Lusaperidone (R107474) 是一种有效的α2肾上腺素受体 (adrenergic receptor) 拮抗剂,是 α (2)-肾上腺素受体的潜在放射性配体,对 α2A和α2C 具有抑制作用, Ki 值分别为0.13和0.15 nM。
T6398 Azaperone

R-1929,Fluoperidol,阿扎哌隆,Stresnil,NSC 170976,Suicalm

Others; Dopamine Receptor GPCR/G Protein; Neuroscience; Others
Azaperone (Fluoperidol) 是多巴胺拮抗剂,具有一些抗组胺和抗胆碱特性,具有止吐活性。
TP2489 Tetrapeptide-21 Acetate

Tetrapeptide-21 Acetate(960608-17-7 Free base)

Others Others
Tetrapeptide-21 Acetate 是一种新型生物活性纯四肽,具有基于皮肤自身结构的抗衰老特性,可用于护肤配方。
TP2384L Hexapeptide-10 Acetate

Hexapeptide-10 Acetate(146439-94-3 Free base)

Integrin Cytoskeletal Signaling
Hexapeptide-10 Acetate (Hexapeptide-10 Acetate) 是一种合成肽。它增加层粘连蛋白 V 和 α6-整合素的合成以促进细胞结合,具有非凡的可见皮肤重组和紧致能力。
T8953L Acetyl hexapeptide 38 Acetate

Acetyl hexapeptide 38 Acetate(1400634-44-7 free base)

Others Others
Acetyl hexapeptide 38 Acetate(1400634-44-7 free base) 丰胸肽,是一种乙酰化六肽,能显着刺激脂肪合成部位的使用,增加胸部或脸颊的体积,塑造完美身材。
T26235 Sulfaperin

磺胺培林,Methylsulfadiazin,Archisulfa,Chemiopen,Demosulfan,Anastaf,Isosulfamerazine

Antibacterial Microbiology/Virology
Sulfaperin (Chemiopen) 是一种磺胺类抗菌剂。
TP1318 Antennapedia Peptide TFA(188842-14-0 free base)

Antennapedia Peptide(TFA)

Others Others
Antennapedia Peptide TFA (188842-14-0 free base) 是一种 16 个氨基酸的肽,是细胞穿透肽家族的成员,最初来源于果蝇转录因子 Antennapedia 的 60 个氨基酸长的同源域。
TP2492 Hexapeptide-9 Acetate

Hexapeptide-9 Acetate(1228371-11-6 Free base)

Others Others
Hexapeptide-9 Acetate 是一种胶原蛋白肽,通过与皮肤细胞自然相互作用来帮助强化结构组织,从而促进再生过程。
TP2490 Palmitoyl Hexapeptide-12 Acetate

Palmitoyl Hexapeptide-12 Acetate(171263-26-6 Free base)

Others Others
Palmitoyl Hexapeptide-12 Acetate (Palmitoyl Hexapeptide-12 Acetate (171263-26-6 Free base)) 可以促进胶原蛋白、弹性蛋白和透明质酸的增殖。可用于改善皮肤含水量,增加真皮层厚度,减少细纹。
T1408 Capecitabine

Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978

Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Capecitabine (Capecitibine) 是一种可口服的前药,可由胸苷磷酸化酶催化转变为其活性代谢物 Fluorouracil。
TP1616L Hsp70-derived octapeptide acetate

Hsp70-derived octapeptide acetate(736171-62-3 free base)

Others Others
Hsp70-derived octapeptide acetate (Hsp70-derived octapeptide acetate)(736171-62-3 free base) 是一组含有四肽重复 (TPR) 的蛋白质,已显示与 70 kDa 热休克同源蛋白 (hsc70) 的 C 末端结构域相互作用。在本研究中,含 TPR 的蛋白质,包括 hsc70 相互作用蛋白 (CHIP)、TPR1 和人富含谷氨酰胺的 TPR 含蛋白 (hSGT) 的 C 端,对 DnaJ 和 hsc70 对荧光素酶重折叠的影响进行了调查。

化合物

APE1-IN-1
Cat.No: T61487
Synonym:
Target: DNA/RNA Synthesis
APE1-IN-2
Cat.No: T73299
Synonym:
Target: Apoptosis
Gabapentin hydrochloride
Cat.No: T6507
Synonym: 加巴喷丁盐酸盐,Neurontin HCl,Gabapentin HCl
Target: Calcium Channel, GABA Receptor
Nonapeptide-1 acetate salt (158563-45-2 free base)
Cat.No: TP1101
Synonym: Melanostatine-5 acetate salt,Nonapeptide-1 acetate salt
Target: Melanocortin Receptor
Nonapeptide-1
Cat.No: T7769
Synonym: Met-Pro-D-Phe-Arg-D-Trp-Phe-Lys-Pro-Val-,九胜肽-1,Melanostatine™ 5
Target: Others
Acetyl tetrapeptide-15 Acetate
Cat.No: T20494L
Synonym: Skinasensyl Acetate,Acetyl tetrapeptide-15 Acetate (928007-64-1 Free base)
Target:
Mapenterol hydrochloride
Cat.No: T40622
Synonym:
Target: Adrenergic Receptor
Rifapentine
Cat.No: T1629
Synonym: MDL473,Rifapentina,Rifapentinum,DL 473,利福喷丁,Priftin,Cyclopentylrifampicin
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Biapenem
Cat.No: T6411
Synonym: CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627
Target: Antibacterial, Antibiotic
Carbetapentane citrate
Cat.No: T0464
Synonym: 托可拉斯,Pentoxyverine citrate,咳必清
Target: AChR
[Pyr1]-Apelin-13
Cat.No: TP1260
Synonym: [pGlu1]-Apelin-13,人牛吡啶APELIN-13
Target: Apelin receptor
Acetyl Tetrapeptide-5 acetate
Cat.No: TP2313
Synonym: Acetyl Tetrapeptide-5 acetate(820959-17-9 free base)
Target: Others
Capecitabine-2',3'-cyclic Carbonate
Cat.No: T64318
Synonym:
Target: Others
Abaperidone
Cat.No: T14083
Synonym:
Target: Dopamine Receptor, 5-HT Receptor
Apelin-17 (human, bovine) acetate
Cat.No: TP2092L
Synonym: Apelin-17 (human, bovine) acetate(217082-57-0 free base)
Target: HIV Protease
Myristoyl Pentapeptide-17 Acetate
Cat.No: T21249L
Synonym: Myristoyl Pentapeptide-17 Acetate(959610-30-1 Free base)
Target: Others
CCK Octapeptide, non-sulfated acetate
Cat.No: TP2204L
Synonym: CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)
Target: cholecystokinin
Acetyl Pentapeptide-1 acetate
Cat.No: T38318L
Synonym:
Target: Histone Demethylase
Tolnapersine TFA
Cat.No: T68023L
Synonym: Tolnapersine TFA(70312-00-4 Free base)
Target: Dopamine Receptor, Adrenergic Receptor
Acetyl tetrapeptide-9 Acetate
Cat.No: TP2365L
Synonym: Acetyl tetrapeptide-9 Acetate(928006-50-2 Free base)
Target: Others
V-9-M Cholecystokinin nonapeptide
Cat.No: TP2419
Synonym: V 9 M,Prepro CCK Fragment V-9-M,Val-pro-val-glu-ala-val-asp-pro-met,Cholecystokinin Precursor (24-32),V9M,V-9-M
Target: Beta Amyloid
Cefcapene pivoxil hydrochloride hydrate
Cat.No: T4990
Synonym: Cefcapene Pivoxil Hydrochloride,盐酸头孢卡品酯
Target: Antibacterial, Antibiotic
Inaperisone
Cat.No: T68087
Synonym:
Target: Others
Trapencaine
Cat.No: T68165
Synonym:
Target:
Apelin-12 acetate
Cat.No: T39823L
Synonym: Apelin-12 acetate (229961-08-4 Free base)
Target: Apelin receptor, p38 MAPK, JNK
Apelin-13
Cat.No: T7656
Synonym:
Target:
Ertapenem sodium
Cat.No: T4991
Synonym: 厄他培南钠,MK-826,L-749345,尔他培南钠
Target: Antibacterial, Antibiotic
Gabapentin
Cat.No: T0702
Synonym: Neurontin,Gabapentine,加巴喷丁,Aclonium
Target: Calcium Channel, GABA Receptor
Capeserod
Cat.No: T68035
Synonym: SL-650155,SL-65.0155
Target: 5-HT Receptor
Ocaperidone
Cat.No: T3497
Synonym: 奥卡哌酮,Ocaperidona,R79598
Target: Dopamine Receptor, 5-HT Receptor
Acetyl tetrapeptide-3 Acetate
Cat.No: TP2364L
Synonym: Acetyl tetrapeptide-3 Acetate(827306-88-7 Free base)
Target: Others
Apelin-13 triTFA(217082-58-1(free base))
Cat.No: T7847
Synonym:
Target: Others
2-chloro-5-(16,18-dioxo-17-azapentacyclo[6.6.5.0~2,7~.0~9,14~.0~15,19~]nonadeca-2,4,6,9,11,13-hexaen-17-yl)benzoic acid
Cat.No: T8833
Synonym:
Target: Others
Octapeptide-2 Acetate
Cat.No: TP2496
Synonym: Octapeptide-2 Acetate(1374396-34-5 Free base)
Target: Others
Myristoyl Tetrapeptide-12 Acetate
Cat.No: TP2497
Synonym: 醋酸肉蔻酰四胜肽-12,Myristoyl Tetrapeptide-12 Acetate(959610-24-3 Free base)
Target: Others
Myristoyl Hexapeptide-23 Acetate
Cat.No: TP2316
Synonym:
Target: Others
Palmitoyl Tetrapeptide-3
Cat.No: TP1042
Synonym: Rigin,棕榈酰四肽-7/棕榈酰四肽-3
Target: Others
Polymyxin B nonapeptide acetate
Cat.No: TP1341L
Synonym: Polymyxin B nonapeptide acetate(86408-36-8 free base)
Target: Antibacterial, Antibiotic
Human IgE Pentapeptide HEPP acetate
Cat.No: TP2499
Synonym: Human IgE Pentapeptide HEPP acetate (62087-72-3 Free base)
Target:
Lusaperidone
Cat.No: T11894
Synonym: R107474
Target: Adrenergic Receptor
Azaperone
Cat.No: T6398
Synonym: R-1929,Fluoperidol,阿扎哌隆,Stresnil,NSC 170976,Suicalm
Target: Others, Dopamine Receptor
Tetrapeptide-21 Acetate
Cat.No: TP2489
Synonym: Tetrapeptide-21 Acetate(960608-17-7 Free base)
Target: Others
Hexapeptide-10 Acetate
Cat.No: TP2384L
Synonym: Hexapeptide-10 Acetate(146439-94-3 Free base)
Target: Integrin
Acetyl hexapeptide 38 Acetate
Cat.No: T8953L
Synonym: Acetyl hexapeptide 38 Acetate(1400634-44-7 free base)
Target: Others
Sulfaperin
Cat.No: T26235
Synonym: 磺胺培林,Methylsulfadiazin,Archisulfa,Chemiopen,Demosulfan,Anastaf,Isosulfamerazine
Target: Antibacterial
Antennapedia Peptide TFA(188842-14-0 free base)
Cat.No: TP1318
Synonym: Antennapedia Peptide(TFA)
Target: Others
Hexapeptide-9 Acetate
Cat.No: TP2492
Synonym: Hexapeptide-9 Acetate(1228371-11-6 Free base)
Target: Others
Palmitoyl Hexapeptide-12 Acetate
Cat.No: TP2490
Synonym: Palmitoyl Hexapeptide-12 Acetate(171263-26-6 Free base)
Target: Others
Capecitabine
Cat.No: T1408
Synonym: Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
Hsp70-derived octapeptide acetate
Cat.No: TP1616L
Synonym: Hsp70-derived octapeptide acetate(736171-62-3 free base)
Target: Others
Cat. No. Product Name Target Signaling Pathways
T6520 Grape Seed Extract

Grape Seed P.E.,葡萄籽提取物

Apoptosis; Others Apoptosis; Others
Grape Seed Extract (Grape Seed P.E.) 是葡萄植物 Vitis vinifera 的种子分泌物,能诱导人类结肠直肠癌细胞凋亡,具有抗炎和抗增殖作用。它对脂肪代谢酶、胰脂肪酶和脂蛋白脂肪酶有抑制作用。
T4S1869 12-Epinapelline

12-表欧乌头碱,12-表-欧乌头碱

Others Others
12-Epinapelline 是一种二萜生物碱,分离自Aconitum baikalense 中。它具有抗炎作用,能刺激成纤维细胞前体克隆的生长。
T7068 Eicosapentaenoic acid ethyl ester

Icosapent ethyl,顺-二十碳五烯酸乙酯,EPA ethyl ester,Ethyl eicosapentaenoate

Others; Endogenous Metabolite Metabolism; Others
Eicosapentaenoic acid ethyl ester (Ethyl eicosapentaenoate) 是 一种ω-3 脂肪酸剂和人内源性代谢物。
T19295 Docosapentaenoic acid 22n-3

Endogenous Metabolite Metabolism
Docosapentaenoic acid 22n-3 是在所有动物细胞膜中发现的磷脂组成成分。
T5368 Eicosapentaenoic Acid

Histone Demethylase; Others; Endogenous Metabolite Chromatin/Epigenetic; Metabolism; Others
Eicosapentaenoic Acid 是一种 ω-3 脂肪酸。
T75650 Rivulariapeptolides 1121

Rivulariapeptolides 1121,作为一种高效的选择性丝氨酸蛋白酶抑制剂,对胰凝蛋白酶、弹性蛋白酶和蛋白酶K展示出了显著的抑制活性,其IC50值分别为35.52 nM、13.24 nM和48.05 nM。
T75649 Rivulariapeptolides 1185

Rivulariapeptolides 1185 是一种高效的选择性丝氨酸蛋白酶抑制剂,其对胰凝蛋白酶、弹性蛋白酶和蛋白酶 K 的 IC50分别为 13.17 nM、23.59 nM 和 55.26 nM。
TN4338 Isovouacapenol C

Others Others
Isovouacapenol C是一种天然产物,属于豆科云实属,其产品编号为 TN4338,CAS号为 455255-15-9。Isovouacapenol C可用作对照参考。
TN3531 Borapetoside D

Others Others
Borapetoside D是一种天然产物,属于防己科青牛胆属,其产品编号为 TN3531,CAS号为 151200-48-5。Borapetoside D可用作对照参考。
T40347 Eicosapentaenoic acid methyl ester

Eicosapentaenoic acid methyl ester is a degradation product derived from monogalactosyl diacylglycerol, which is an apoptosis-inducing anticancer compound.
TN3533 Borapetoside F

Others Others
Borapetoside F是一种天然产物,属于防己科青牛胆属,其产品编号为 TN3533,CAS号为 151200-50-9。Borapetoside F可用作对照参考。
T83660 3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic Acid

C18:5 n-3,C18:5(3Z,6Z,9Z,12Z,15Z),all-cis-3,6,9,12,15-Octadecapentaenoic Acid

3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic acid 是一种在 G. kowalevskii 中发现的微藻 PUFA,常作为微藻和甲藻的化学分类生物标志物使用。
T75648 Rivulariapeptolides 1155

Rivulariapeptolides 1155 是一种有效的丝氨酸蛋白酶 (serine protease) 抑制剂,对糜蛋白酶、弹性蛋白酶、蛋白蛋白酶 K 的 IC50分别为 41.84、4.94、56.54 nM。
TN3795 Dehydroborapetoside B

Others Others
Dehydroborapetoside B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3795,CAS号为 1221178-16-0。
TN6827 Hapepunine

Hapepunine is a natural product.
TN3530 Borapetoside B

Others Others
Borapetoside B是一种天然产物,属于防己科青牛胆属,其产品编号为 TN3530,CAS号为 104901-05-5。Borapetoside B可用作对照参考。
T72152 Eicosapentaenoic Acid sodium

二十碳五烯酸钠盐,Timnodonic acid sodium,EPA sodium

Eicosapentaenoic Acid (EPA) sodium 为口服活性 ω-3 长链多不饱和脂肪酸 (ω-3 LC-PUFAs)。其通过DNA去甲基化,促进肿瘤抑制基因CCAAT/增强子结合蛋白δ (C/EBPδ)的重新表达,并通过H-RAS内含子1 CpG岛的去甲基化,激活U937白血病细胞中RAS/ERK/C/EBPβ途径。此外,该化合物能够促进血管平滑肌细胞松弛和血管舒张。
TN5302 Withaperuvin C

Withaperuvin C may have anti-inflammatory activity with lipopolysaccharide (LPS)-activated murine macrophage RAW 264.7 cells.
TN3532 Borapetoside E

Others Others
Borapetoside E has anti-hyperglycemic activity, it can significantly reduce serum glucose levels at dose-dependent manners in alloxan-induced hyperglycemic mice and db/db type 2 diabetic mice.
T75651 Rivulariapeptolides 988

Rivulariapeptolides 988作为一种高效选择性丝氨酸蛋白酶抑制剂,对胰凝蛋白酶、弹性蛋白酶和蛋白酶K的IC50分别为95.46 nM、15.29 nM和85.50 nM。
TN4264 Isoapetalic acid

胡桐,海棠木

HIV Protease; Antifection Microbiology/Virology; Proteases/Proteasome
Isoapetalic acid and apetalic acid exhibit cytotoxic activities towards both cancer cell lines(human breast cancer (MCF-7) and human lung carcinoma (A-549) cell lines) and both Gram-positive bacteria(two Gram-positive bacteria, S. aureus and B. subtilis a

天然产物

Grape Seed Extract
Cat.No: T6520
Synonym: Grape Seed P.E.,葡萄籽提取物
Target: Apoptosis, Others
12-Epinapelline
Cat.No: T4S1869
Synonym: 12-表欧乌头碱,12-表-欧乌头碱
Target: Others
Eicosapentaenoic acid ethyl ester
Cat.No: T7068
Synonym: Icosapent ethyl,顺-二十碳五烯酸乙酯,EPA ethyl ester,Ethyl eicosapentaenoate
Target: Others, Endogenous Metabolite
Docosapentaenoic acid 22n-3
Cat.No: T19295
Synonym:
Target: Endogenous Metabolite
Eicosapentaenoic Acid
Cat.No: T5368
Synonym:
Target: Histone Demethylase, Others, Endogenous Metabolite
Rivulariapeptolides 1121
Cat.No: T75650
Synonym:
Target:
Rivulariapeptolides 1185
Cat.No: T75649
Synonym:
Target:
Isovouacapenol C
Cat.No: TN4338
Synonym:
Target: Others
Borapetoside D
Cat.No: TN3531
Synonym:
Target: Others
Eicosapentaenoic acid methyl ester
Cat.No: T40347
Synonym:
Target:
Borapetoside F
Cat.No: TN3533
Synonym:
Target: Others
3(Z),6(Z),9(Z),12(Z),15(Z)-Octadecapentaenoic Acid
Cat.No: T83660
Synonym: C18:5 n-3,C18:5(3Z,6Z,9Z,12Z,15Z),all-cis-3,6,9,12,15-Octadecapentaenoic Acid
Target:
Rivulariapeptolides 1155
Cat.No: T75648
Synonym:
Target:
Dehydroborapetoside B
Cat.No: TN3795
Synonym:
Target: Others
Hapepunine
Cat.No: TN6827
Synonym:
Target:
Borapetoside B
Cat.No: TN3530
Synonym:
Target: Others
Eicosapentaenoic Acid sodium
Cat.No: T72152
Synonym: 二十碳五烯酸钠盐,Timnodonic acid sodium,EPA sodium
Target:
Withaperuvin C
Cat.No: TN5302
Synonym:
Target:
Borapetoside E
Cat.No: TN3532
Synonym:
Target: Others
Rivulariapeptolides 988
Cat.No: T75651
Synonym:
Target:
Isoapetalic acid
Cat.No: TN4264
Synonym: 胡桐,海棠木
Target: HIV Protease, Antifection
Cat. No. Product Name Species Expression System
TMPJ-00464 APE Protein, Human, Recombinant

APEX,Apurinic-Apyrimidinic Endonuclease 1,APE

Human E. coli
Apurinic-Apyrimidinic Endonuclease 1 (APE1) is required for efficient DNA base excision repair. When the DNA glycosylase remove the damaged bases, APE1 cleaves the AP site to allow resynthesis and ligation to complete repair. APE1 stimulates the DNA binding activity of many transcription factors, which participate in cancer promotion and progression. APE1 regulates the redox state of multiple transcription factors, such as c-Jun, c-Fos, NF-kB, p53. APEN is also involved in calcium-dependent down...
TMPY-02433 APE1/APEX1 Protein, Human, Recombinant (His)

APEX,HAP1,APX,APE,APEX nuclease (...

Human E. coli
The enzyme is known to be a redox factor (Ref-1) stimulating DNA binding activity of AP-1 binding proteins such as Fos and Jun as well as a multifunctional DNA repair enzyme having 5' AP endonuclease, DNA 3' repair diesterase, 3'-5' exonuclease and DNA 3'-phosphatase activities.Although Apex mRNA was expressed ubiquitously, the levels varied significantly, suggesting organ- or tissue-specific expression of the Apex gene. The highest level was observed in the testis, relatively high levels in the...
TMPY-04471 APEG1 Protein, Human, Recombinant (His)

SPEG complex locus,BPEG,SPEGalpha,SPEGβ,APEG-1,SPEG...

Human E. coli
Striated muscle preferentially expressed protein kinase, also known as aortic preferentially expressed protein 1, APEG-1, SPEG and KIAA1297, is a protein that belongs to the protein kinase superfamily and CAMK Ser/Thr protein kinase family. SPEG / APEG-1 contains two fibronectin type-III domains, nine Ig-like (immunoglobulin-like) domains, two protein kinase domains. Isoform 1 of SPEG is preferentially expressed in striated muscle. Non-kinase form such as isoform 3 of SPEG is predominantly expre...
TMPH-00334 Candidapepsin-6 Protein, Candida albicans, Recombinant (His)

SAP6,Candidapepsin-6,Secreted aspartic protease 6,A...

Candida albicans E. coli
Candidapepsin-6 Protein, Candida albicans, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 39.8 kDa and the accession number is P43095.
TMPH-00332 Candidapepsin-2 Protein, Candida albicans (strain WO-1), Recombinant (His)

Aspartate protease 2,ACP 2,Secreted aspartic protease 2,Cand...

Candida albicans E. coli
Candidapepsin-2 Protein, Candida albicans (strain WO-1), Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 42.3 kDa and the accession number is C4YMJ3.
TMPY-05947 Influenza A H1N2 (A/swine/Papenburg/IDT12653/2010) Neuraminidase/NA Protein (His)

H1N2 HEK293 Cells
Influenza A H1N2 (A/swine/Papenburg/IDT12653/2010) Neuraminidase/NA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.6 kDa and the accession number is V5J546.
TMPH-03502 Chaperonin GroEL Protein, Shigella dysenteriae serotype 1, Recombinant (His & Myc & SUMO)

groEL,Chaperonin GroEL,hypB,60 kDa chapero...

Shigella dysenteriae E. coli
Together with its co-chaperonin GroES, plays an essential role in assisting protein folding. The GroEL-GroES system forms a nano-cage that allows encapsulation of the non-native substrate proteins and provides a physical environment optimized to promote and accelerate protein folding. Chaperonin GroEL Protein, Shigella dysenteriae serotype 1, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 66.9 kDa and t...
TMPH-00333 Candidapepsin-2 Protein, Candida albicans, Recombinant (His)

Candidapepsin-2,Aspartate protease 2,SAP2,PRA2,Secr...

Candida albicans E. coli
Candidapepsin-2 Protein, Candida albicans, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 42.4 kDa and the accession number is P0CS83.
TMPH-00888 APEH Protein, Human, Recombinant (His)

Acylamino-acid-releasing enzyme,Acylaminoacyl-peptidase,Oxid...

Human E. coli
This enzyme catalyzes the hydrolysis of the N-terminal peptide bond of an N-acetylated peptide to generate an N-acetylated amino acid and a peptide with a free N-terminus. It preferentially cleaves off Ac-Ala, Ac-Met and Ac-Ser. APEH Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 85.2 kDa and the accession number is P13798.
TMPY-06739 Pol d 5 Protein, Mediterranean paper wasp, Recombinant

Mediterranean paper wasp P. pastoris (Yeast)
Pol d 5 Protein, Mediterranean paper wasp, Recombinant is expressed in P. pastoris yeast expression system. The predicted molecular weight is 20 kDa.
TMPH-00388 Chaperonin GroEL Protein, Chlamydia trachomatis, Recombinant (His & SUMO)

Cpn60,mopA,60 kDa chaperonin,Chaperonin-60...

Chlamydia trachomatis E. coli
Together with its co-chaperonin GroES, plays an essential role in assisting protein folding. The GroEL-GroES system forms a nano-cage that allows encapsulation of the non-native substrate proteins and provides a physical environment optimized to promote and accelerate protein folding. Chaperonin GroEL Protein, Chlamydia trachomatis, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 74.0 kDa and the accession number is P0C0...
TMPY-06675 Met e 1 Protein, Metapenaeus ensis, Recombinant

Metapenaeus ensis E. coli
Met e 1 Protein, Metapenaeus ensis, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 32.7 kDa.

重组蛋白

APE Protein, Human, Recombinant
Cat.No: TMPJ-00464
Species: Human
Expression System: E. coli
APE1/APEX1 Protein, Human, Recombinant (His)
Cat.No: TMPY-02433
Species: Human
Expression System: E. coli
APEG1 Protein, Human, Recombinant (His)
Cat.No: TMPY-04471
Species: Human
Expression System: E. coli
Candidapepsin-6 Protein, Candida albicans, Recombinant (His)
Cat.No: TMPH-00334
Species: Candida albicans
Expression System: E. coli
Candidapepsin-2 Protein, Candida albicans (strain WO-1), Recombinant (His)
Cat.No: TMPH-00332
Species: Candida albicans
Expression System: E. coli
Influenza A H1N2 (A/swine/Papenburg/IDT12653/2010) Neuraminidase/NA Protein (His)
Cat.No: TMPY-05947
Species: H1N2
Expression System: HEK293 Cells
Chaperonin GroEL Protein, Shigella dysenteriae serotype 1, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-03502
Species: Shigella dysenteriae
Expression System: E. coli
Candidapepsin-2 Protein, Candida albicans, Recombinant (His)
Cat.No: TMPH-00333
Species: Candida albicans
Expression System: E. coli
APEH Protein, Human, Recombinant (His)
Cat.No: TMPH-00888
Species: Human
Expression System: E. coli
Pol d 5 Protein, Mediterranean paper wasp, Recombinant
Cat.No: TMPY-06739
Species: Mediterranean paper wasp
Expression System: P. pastoris (Yeast)
Chaperonin GroEL Protein, Chlamydia trachomatis, Recombinant (His & SUMO)
Cat.No: TMPH-00388
Species: Chlamydia trachomatis
Expression System: E. coli
Met e 1 Protein, Metapenaeus ensis, Recombinant
Cat.No: TMPY-06675
Species: Metapenaeus ensis
Expression System: E. coli
TargetMol Loading
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