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Search Results for " anti-asthmatic "

16

抑制剂 & 化合物

5

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T21404	Fluticasone furoate Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate	Glucocorticoid Receptor	Endocrinology/Hormones
	Fluticasone furoate (Avamys) 是一种合成的三氟化皮质类固醇，衍生自氟替卡松，Kd 为 0.3 nM。Fluticasone furoate 具有有效的抗炎、抗哮喘活性和低全身暴露。Fluticasone furoate 可用作过敏性鼻炎治疗研究的鼻喷雾剂。
T12215	Nexopamil racemate (Rac)-Nexopamil	Calcium Channel; 5-HT Receptor	GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
	Nexopamil racemate（(Rac)-Nexopamil）是 Nexopamil 的外消旋体。Nexopamil racemate 具有潜在的抗哮喘和抗溃疡活性。
T28529	RG 7152 RG7152,RG-7152	Leukotriene Receptor	GPCR/G Protein
	RG 7152 是白三烯 D4 拮抗剂,具有抗哮喘作用，可作用于研究哮喘。
T16026	MCI826	P-gp; LTR	Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
	MCI826 是一种具有有效性和选择性的 P-glycoprotein (P-gp)和肽白三烯（p-LTs）拮抗剂，在豚鼠晚期哮喘模型中显示出抗哮喘活性。
T26519	Ablukast Ro 23-3544,阿鲁司特	Leukotriene Receptor	GPCR/G Protein
	Ablukast (Ro 23-3544) 是白三烯受体的选择性拮抗剂，也是LTD4受体拮抗剂。可改善 LTC4 和抗原诱导的支气管狭窄。
T11581	HSR6071	Others	Others
	HSR6071 是一种新型具有口服活性和有效性的抗过敏制剂，能抑制被动皮肤过敏反应 (PCA)。HSR6071 在大鼠实验性哮喘模型中显示出抗哮喘活性。
T0212	Seratrodast 塞曲司特,AA 2414,ABT-001	COX; Prostaglandin Receptor; PPAR	DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
	Seratrodast (ABT-001) 是一种血栓素 A2 受体 (TP) 拮抗剂，用于治疗哮喘。
T0117	Suplatast (Tosilate) IPD 1151T,甲磺司特,Suplatast tosilate,Suplatast Tosylate	IL Receptor; Interleukin	Immunology/Inflammation
	Suplatast Tosilate (IPD 1151T) 是一种口服有活性的 Th2 细胞因子抑制剂，能够阻碍 Th2 细胞产生 IL-4 和 IL-5 ，并对 IgE 的合成具有抑制作用。它是一种抗过敏剂，它具有抗纤维化、抗哮喘及抗炎特性。
T15344	Minocromil 米诺罗米,FPL59360	Others	Others
	Minocromil is a new agent of Anti-asthmatic.
T26589	Albifylline
	Albifylline is a xanthine derivates with anti-asthmatic activity. Albifylline may cause a significant reduction of shock-induced leukocyte adhesions to the sinusoidal endothelium in the liver after hemorrhagic shock. Albifylline also improves microvascula
T10508	Asthma relating compound 1	Others	Others
	Asthma relating compound 1 is an anti-asthmatic compound.
T26595	Allosamidin A-82516,A 82516,A82516
	Allosamidin, a chitinase inhibitor and typical secondary metabolite of Streptomyces, may be used as a pesticide and anti-asthmatic agent.
T28296	Parogrelil hydrochloride INDI-702,NM-702,NT-702,NM702,INDI702
	Parogrelil is a phosphodiesterase (PDE3/PDE5A) inhibitor potentially for the treatment of intermittent. Parogrelil suppress the asthmatic response in guinea pigs, with both bronchodilating and anti-inflammatory effects. Parogrelil improves reduced walking
T61794	LASSBio-1632
	LASSBio-1632 is a novel anti-asthmatic lead candidate that selectively inhibits PDE4A and PDE4D isoenzymes, leading to the suppression of airway hyper-reactivity (AHR) and TNF-α production in lung tissue. With high experimental BBB permeability, LASSBio-1632 (7j) efficiently crosses the blood-brain barrier through passive diffusion [1].
T62598	Pitavastatin sodium
	Pitavastatin (NK-104) sodium 是一种有效的羟甲基戊二酰-CoA(HMG-CoA) 还原酶抑制剂，也是一种高效的肝细胞低密度脂蛋白胆固醇 (LDL-C) 受体诱导剂。Pitavastatin sodium 在 HepG2 细胞中，能够抑制乙酸合成胆固醇 (IC50: 5.8 nM) 。Pitavastatin sodium 表现出抗动脉粥样硬化、抗哮喘、抗骨关节炎、神经保护、抗肿瘤、肝保护和肾保护作用。
T7072	Pitavastatin
	Pitavastatin (NK-104) 是有效的羟甲基戊二酰-CoA(HMG-CoA)还原酶抑制剂。Pitavastatin 抑制乙酸合成胆固醇，在 HepG2 细胞中的IC50为 5.8 nM。Pitavastatin 是一种高效的肝细胞低密度脂蛋白胆固醇 (LDL-C) 受体诱导剂。Pitavastatin 具有抗动脉粥样硬化、抗哮喘、抗骨关节炎、抗肿瘤、神经保护、肝保护和肾保护等作用。

化合物

Fluticasone furoate

Cat.No: T21404

Synonym: Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate

Target: Glucocorticoid Receptor

Nexopamil racemate

Cat.No: T12215

Synonym: (Rac)-Nexopamil

Target: Calcium Channel, 5-HT Receptor

Cat.No: T28529

Synonym: RG7152,RG-7152

Target: Leukotriene Receptor

Cat.No: T16026

Target: P-gp, LTR

Cat.No: T26519

Synonym: Ro 23-3544,阿鲁司特

Target: Leukotriene Receptor

Cat.No: T11581

Target: Others

Cat.No: T0212

Synonym: 塞曲司特,AA 2414,ABT-001

Target: COX, Prostaglandin Receptor, PPAR

Suplatast (Tosilate)

Cat.No: T0117

Synonym: IPD 1151T,甲磺司特,Suplatast tosilate,Suplatast Tosylate

Target: IL Receptor, Interleukin

Cat.No: T15344

Synonym: 米诺罗米,FPL59360

Target: Others

Cat.No: T26589

Asthma relating compound 1

Cat.No: T10508

Target: Others

Cat.No: T26595

Synonym: A-82516,A 82516,A82516

Parogrelil hydrochloride

Cat.No: T28296

Synonym: INDI-702,NM-702,NT-702,NM702,INDI702

Cat.No: T61794

Pitavastatin sodium

Cat.No: T62598

Cat.No: T7072

Cat. No.	Product Name	Target	Signaling Pathways
T8208	androsin	Others	Others
	Androsin 分离于印度胡黄连中，具有抗哮喘作用。
T2950	Schisandrin Wuweizi alcohol-A,Wuweizichun-A,Schizandrol-A,Schizandrol,五味子醇甲	Autophagy	Autophagy
	Schisandrin (Wuweizi alcohol-A) 是一种从五味子中分离出来的联苯环辛烯类木脂素，可逆转大鼠的记忆障碍，具有保肝、抗氧化、抗哮喘、抗癌和抗炎作用。
T2S2173	(E)-Naringenin chalcone Isosalipurpol,柚皮苷查尔酮,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone,柚皮素查耳酮	Others	Others
	Naringenin chalcone (Isosalipurpol) 是一种黄酮醇生物合成的中间体，在查耳酮异构酶的作用下，自发代谢成柚皮素。它具有抗炎和抗过敏活性。
TN3367	Akuammidine	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 microM at mu-, delta- and kappa-opioid binding sites, respectively.
TN2511	Britannilactone diacetate 1,6-O,O-Diacetylbritannilactone	IL Receptor; PARP; ROS; MAPK; Caspase; JAK; JNK; STAT	Angiogenesis; Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; JAK/STAT signaling; MAPK; Proteases/Proteasome; Stem Cells
	1,6-O,O-Diacetylbritannilactone(OODBL) has anti-inflammatory activity, it has a potential therapeutic efficacy on inflammatory diseases especially allergic airway disease as a lead compound. OODBL has anti-asthmatic activity, it reduces leukotriene C4 pro

天然产物

Cat.No: T8208

Target: Others

Cat.No: T2950

Synonym: Wuweizi alcohol-A,Wuweizichun-A,Schizandrol-A,Schizandrol,五味子醇甲

Target: Autophagy

(E)-Naringenin chalcone

Cat.No: T2S2173

Synonym: Isosalipurpol,柚皮苷查尔酮,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone,柚皮素查耳酮

Target: Others

Cat.No: TN3367

Target: Opioid Receptor

Britannilactone diacetate

Cat.No: TN2511

Synonym: 1,6-O,O-Diacetylbritannilactone

Target: IL Receptor, PARP, ROS, MAPK, Caspase, JAK, JNK, STAT

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