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159

抑制剂 & 化合物

14

天然产物

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Cat. No. Product Name Target Signaling Pathways
T37591 IMP-1710

DUB Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination
IMP-1710 是一种选择性 UCH-L1 抑制剂,在荧光偏振测定中的 IC50 值为 38 nM。
T9350 IMP-1088

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
IMP-1088 是一种人N-肉豆蔻酰基转移酶NMT1和NMT2双重抑制剂,对 HsNMT1 和 HsNMT2 的IC50小于1 nM,对 HsNMT1 的Kd 小于210 pM。它有保护宿主细胞免受病毒感染的细胞毒作用,通过阻断鼻病毒的 N-肉豆蔻酰化蛋白来阻断鼻病毒的复制。
T73362 C-di-IMP

Cyclic-di-IMP

C-di-IMP (Cyclic-di-IMP) 是一种STING 激动剂。C-di-IMP 可用于肿瘤的研究。
T68322 IMP-321

IMP-321 is a soluble dimeric recombinant form of LAG-3 and first-in-class antigen presenting cell activator.
T82760 C-di-IMP disodium

Cyclic-di-IMP disodium

STING Immunology/Inflammation
C-di-IMP二钠是一种效果显著的STING激动剂,主要在肿瘤领域的研究中应用。
T37729 IMP-1700

IMP-1700 is an inhibitor of bacterial DNA repair.1It potentiates the activity of the quinolone antibiotic ciprofloxacin against methicillin-resistantS. aureus(MRSA) with a combination index value of 0.7. IMP-1700 inhibits the ciprofloxacin-induced bacterial SOS response, a process that repairs DNA damage, in a reporter assay in a concentration-dependent manner. It is also active againstE. coli, as well as methicillin-resistant and -sensitive S. aureus, when used alone (EC50s = 0.5, 0.21, and 3.8...
T36984 Cyclic di-IMP (sodium salt)

Cyclic di-IMP (sodium salt) (c-di-IMP) is a synthetic second messenger structurally related to the bacterial second messengers cyclic di-GMP and cyclic di-AMP . C-di-IMP has adjuvant properties when co-administered with antigens in vitro and by mucosal routes in vivo. C-di-IMP enriches the population of MHC class I and II, CD80, CD86, CD40, and CD54 positive dendritic cells derived from murine bone marrow. It also stimulates macrophages at 500 ng/ml. Mice immunized with β-galactosidase (β-gal) p...
T9593 Senaparib

IMP4297

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Senaparib (IMP4297) 是一种选择性和口服有效的PARP1/2抑制剂,具有强效的抗肿瘤活性。
T78247 Ieramilimab

IMP701,LAG525

Ieramilimab(LAG525;IMP701)是一款针对LAG-3的人源化IgG4单克隆抗体,它通过结合到LAG-3来阻断其与MHC-II 分子的相互作用。
T78332 Eftilagimod alfa

IMP321,LAG-3Ig

Eftilagimod alfa为重组LAG-3Ig融合蛋白,具有MHC II 类分子结合能力。该药物通过介导抗原提呈细胞(APC)的激活进而激活CD8 T细胞,可用于研究转移性黑色素瘤及转移性乳腺癌。
T16028 IMB-XH1

Mcl1-IN-2,7-[(2-吡啶基氨基)-2-噻吩基甲基]-8-喹啉醇

BCL; Antibacterial Apoptosis; Microbiology/Virology
IMB-XH1 (Mcl1-IN-2) 是一种骨髓细胞因子 1 抑制剂。它也是非竞争性的 Delhi metallo-β-lactamase(NDM-1) 抑制剂。它对金属 β-内酰胺酶 NDM-1,IMP-4,ImiS 和 L1 的 IC50值分别为 0.4637 μM,3.980 μM,0.2287 μM 和 1.158 μM。
T70760 NVP018

NVP018, also known as BC 556, is a potent inhibitor of hepatitis B virus, hepatitis C virus (HCV), and HIV-1 replication, shows minimal inhibition of major drug transporters, and has a high barrier to generation of both HCV and HIV-1 resistance..
T62685 IMP2-IN-2

IMP2-IN-2 是一种有效的、选择性的 IMP2 抑制剂,抑制 IMP2 与 RNA_A 和 RNA_B 相互作用的 IC50 值分别为 120.9 μM 和 236.7 μM。IMP2-IN-2 能够用于研究癌症。
T61946 IMP2-IN-1

IMP2-IN-1 (compound 4) 是有效的IMP2抑制剂,对 IMP2 RNA 的IC50为 81.3-127.5 μM。IMP2-IN-1 降低 SW480 细胞中 IMP2 水平。IMP2-IN-1 显著抑制分化和未分化 Huh7 细胞的活力。
T11007L Levofloxacin Hydrochloride Impurity A

Levofloxacin Hydrochloride Impurity A(117707-40-1 Free base),左氧氟沙星杂质A(盐酸盐)

Antibacterial Microbiology/Virology
Levofloxacin Hydrochloride Impurity A 是一种喹诺酮类药物,具有广谱抗菌作用。
T1698 Carvedilol EP IMpurity E

Carvedilol USP E,Carvedilol Impurity E,卡维地洛杂质

Others Others
Carvedilol EP IMpurity E (Carvedilol USP E) 用作药物中间体。
T8752 BAR 501 impurity

GPCR19 GPCR/G Protein
BAR 501 impurity 在 BAR501 制剂中发现的一种杂质,可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。
T0550 Domperidone EP Impurity A

5-氯-1,3-二氢-1-(4-哌啶基)-2H-苯并咪唑-2-酮

Others Others
Domperidone EP Impurity A 用作医药中间体。
T40867 Simpinicline

OC-02

AChE Neuroscience
Simpinicline (OC-02)(OC-02)是一种高选择性烟碱乙酰胆碱受体(nAChR)激动剂,可激活三叉神经副交感神经通路,可用于治疗干眼症。
T9084 Cetirizine Impurity B dihydrochloride

De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride,西替利嗪杂质B二盐酸盐,西替利嗪杂质04

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Cetirizine Impurity B dihydrochloride (De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride) 是 Cetirizine dihydrochloride 的杂质。Cetirizine 是一种抗组胺剂,是口服有活力的、特异性 H1受体拮抗剂。它能够抑制过敏反应期间嗜酸性粒细胞趋化,可以标记抗过敏特性。
T9042 Teriflunomide impurity 3

4-Amino-N-(4-trifluoromethylphenyl)benzamide

COX Immunology/Inflammation; Neuroscience
Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) 是一种选择性COX-1抑制剂,IC50为 30 µM。
T67847 Imatinib impurities3

Bcr-Abl; PDGFR; c-Kit Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Imatinib impurities3是一种蛋白激酶抑制剂,对 ABL1 wt、KIT wt 和 PDGFRR wt 的 IC50值分别为6.95μM 、0.245μM 和0.139μM 。
T1690 BroMhexine IMpurity B

Others Others
BroMhexine IMpurity B 试剂用于制备 Ambroxol 和 Bromhexine (B678600) 代谢物 Ambroxol EP Impurity E。
T4196 Betahistine EP Impurity C

NSC19005

Others; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience; Others
Betahistine EP Impurity C (NSC19005) 是 Betahistine 的杂质。 Betahistine 是可口服的组胺 H1 受体激动剂和 H3 受体的拮抗剂,可用作血管扩张剂,用于类风湿性关节炎的研究。
T68921 Impromidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Impromidine hydrochloride 是一种非常有效和特异性的组胺H2受体激动剂,可用于进行心血管研究。
T1689 Enalapril IMpurity B

(+)-N-[1-(S)-Ethoxycarbonxyl-3-phenylpropyl]-L-alanine,依那普利杂质B

Others Others
Enalapril IMpurity B ((+)-N-[1-(S)-Ethoxycarbonxyl-3-phenylpropyl]-L-alanine) 是 Moexipril 中间体,是 Imidapril 的主要代谢物。
T61326 AIMP2-DX2-IN-1

Others Others
AIMP2-DX2-IN-1 是一种有效的 AIMP2-DX2 抑制剂,具有潜在的抗肿瘤活性,可用于研究淋巴癌。
T0667 Flecainide Impurity D

Others Others
Flecainide Impurity D 在工业中用作中间体。
T1357 TriMetazidine EP IMpurity-D

Others Others
TriMetazidine EP IMpurity-D 是合成 TriMetazidine 的起始原料,是合成多种化合物的中间体。
T12961 Sofosbuvir impurity F

索非布韦杂质 F,Sofosbuvir 3',5'-Bis-(S)-phosphate

HCV Protease Microbiology/Virology; Proteases/Proteasome
Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) 既是 Sofosbuvir 的非对映异构体,也是 Sofosbuvir 的杂质,Sofosbuvir 是 HCV RNA 复制的抑制剂。
T12962 Sofosbuvir impurity G

HCV Protease Microbiology/Virology; Proteases/Proteasome
Sofosbuvir impurity G 是 Sofosbuvir 的非对映异构体,是 Sofosbuvir 的杂质。其中 Sofosbuvir 能够抑制 HCVRNA 的复制,具有抗丙型肝炎病毒作用。
T31204 Darapladib-impurity

Others Others
Darapladib-impurity 是 Darapladib 的杂质。Darapladib 对脂蛋白相关磷脂酶 A2 (Lp-PLA2)有抑制作用。
T1733 Ciprofloxacin EP IMpurity A

Q-Acid,Fluoroquinolonic Acid,环丙羧酸,Ciprofloxacin Impurity A

Antibiotic Microbiology/Virology
Ciprofloxacin EP IMpurity A (Fluoroquinolonic Acid) 是一种抗生素和抗菌剂。
T67853 Rivaroxaban Impurity

Rivaroxaban-10

Factor Xa Metabolism
Rivaroxaban Impurity (Rivaroxaban-10) 是一种强效凝血因子Xa 抑制剂,IC50=66 nM。
T3097 Mycophenolic Acid Impurity

马替麦考酚酸杂质,5,7-dihydroxy-4-methylphthalide

Others Others
Mycophenolic Acid Impurity (5,7-dihydroxy-4-methylphthalide) 是一种免疫抑制药物和有效的抗增殖剂,可用于代替旧的抗增殖剂 azathioprine。它通常用作三联疗法的一部分,包括钙调神经磷酸酶抑制剂(ciclosporin 或 tacrolimus)和prednisolone。它还可用于研究选择表达编码 XGPRT(黄嘌呤鸟嘌呤磷酸核糖基转移酶)的大肠杆菌基因的动物细胞。
T4058 R-IMPP

Others; Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism; Others
R-IMPP 是抗 PCSK9分泌的药物 (IC50=4.8 μM),靶向作用于 80S 核糖体,抑制 PCSK9 蛋白的翻译。
T3445 Importazole

Apoptosis; Others Apoptosis; Others
Importazole 是一种核转运受体 importin-β 小分子抑制剂。
T38740 Rivastigmine carbamate impurity

利凡斯的明氨基甲酸酯杂质;利瓦斯的明氨基甲酸酯杂质;卡巴拉汀氨基甲酸酯杂质;利斯的明氨基甲酸酯杂质,3-Nitrophenyl ethyl(methyl)carbamate

Rivastigmine carbamate impurity (3-Nitrophenyl ethyl(methyl)carbamate) is a byproduct found in Rivastigmine, which is recognized as a powerful and orally active inhibitor of cholinesterase (ChE). Specifically, Rivastigmine effectively inhibits both butyrylcholinesterase (BChE) and acetylcholinesterase (AChE), with IC50 values of 0.037 μM and 4.15 μM, respectively.
T35430 Afatinib impurity 11

Afatinib impurity 11 is an impurity of Afatinib. Afatinib is an irreversible EGFR family inhibitor with IC50s of 0.5 nM, 0.4 nM, 10 nM and 14 nM for EGFRwt, EGFRL858R, EGFRL858R/T790M and HER2, respectively[1]. [1]. Li D, et al. BIBW2992, an irreversible EGFR/HER2 inhibitor highly effective in preclinical lung cancer models. Oncogene. 2008 Aug 7;27(34):4702-11.
T38577 Remdesivir O-desphosphate acetonide impurity

Remdesivir O-desphosphate acetonide impurity is a contaminant found in Remdesivir. Remdesivir (GS-5734) is a nucleoside analogue known for its potent antiviral properties, particularly in inhibiting SARS-CoV-2 (COVID-19) infection in vitro.
T12958 Sofosbuvir impurity C

Others Others
Sofosbuvir impurity C is the less active impurity of Sofosbuvir. Sofosbuvir is an active HCV RNA replication inhibitor in the HCV replicon assay,with potent anti-hepatitis C virus (HCV) activity.
T73969 Febuxostat impurity 6

Febuxostat impurity 6 是 Febuxostat 一种杂质。Febuxostat 是选择性黄嘌呤氧化酶 (XO) 抑制剂,Ki 为 0.6 nM。
T37628 Ibuprofen impurity 1

Ibuprofen impurity 1 is an Ibuprofen impurity. Ibuprofen is an anti-inflammatory inhibitor targeting COX-1 and COX-2 with IC50s of 13 μM and 370 μM, respectively[1]. [1]. Noreen Y, et al. Development of a radiochemical cyclooxygenase-1 and -2 in vitro assay for identification of natural products as inhibitors of prostaglandin biosynthesis. J Nat Prod. 1998 Jan;61(1):2-7.
T73962 Cetirizine Impurity C dihydrochloride

Cetirizine Impurity C dihydrochloride 为Cetirizine杂质之一,属于羟嗪的羧化代谢物,是第二代抗组胺剂中的一个。其为具有特异性且口服有效的H1受体(histamine H1-receptor)长效拮抗剂。
T73964 Hydroxychloroquine Impurity F

Hydroxychloroquine Impurity F为Hydroxychloroquine的一种杂质,后者为合成抗疟疾剂,能抑制Toll样受体7/9(TLR7/9)信号传导,并有效抑制SARS-CoV-2感染。
T126193 Diosmin Impurity 5

Diosmin Impurity 5 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126193。
T37817 Terazosin dimer impurity dihydrochloride

Terazosin dimer impurity dihydrochloride, a dimeric form of Terazosin, is a chemical impurity found in Terazosin. Terazosin itself is a derivative of quinazoline and acts as a competitive and orally active α1-adrenoceptor antagonist[1].
T40752 Ibuprofen Impurity F

Ibuprofen Impurity F is a known impurity of Ibuprofen, which acts as an anti-inflammatory inhibitor that selectively targets both COX-1 and COX-2 enzymes. It exhibits inhibitory activity with IC50 values of 13 μM and 370 μM for COX-1 and COX-2, respectively.
T12963 Sofosbuvir impurity H

HCV Protease Microbiology/Virology; Proteases/Proteasome
Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir. Sofosbuvir (PSI-7977) is a diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.
T40941 Olmesartan lactone impurity

Olmesartan lactone impurity is a cyclic ester impurity derived from Olmesartan, which is an angiotensin II receptor (AT1R) antagonist with potential applications in the study of high blood pressure.

化合物

IMP-1710
Cat.No: T37591
Synonym:
Target: DUB
IMP-1088
Cat.No: T9350
Synonym:
Target: Others, DNA/RNA Synthesis
C-di-IMP
Cat.No: T73362
Synonym: Cyclic-di-IMP
Target:
IMP-321
Cat.No: T68322
Synonym:
Target:
C-di-IMP disodium
Cat.No: T82760
Synonym: Cyclic-di-IMP disodium
Target: STING
IMP-1700
Cat.No: T37729
Synonym:
Target:
Cyclic di-IMP (sodium salt)
Cat.No: T36984
Synonym:
Target:
Senaparib
Cat.No: T9593
Synonym: IMP4297
Target: PARP
Ieramilimab
Cat.No: T78247
Synonym: IMP701,LAG525
Target:
Eftilagimod alfa
Cat.No: T78332
Synonym: IMP321,LAG-3Ig
Target:
IMB-XH1
Cat.No: T16028
Synonym: Mcl1-IN-2,7-[(2-吡啶基氨基)-2-噻吩基甲基]-8-喹啉醇
Target: BCL, Antibacterial
NVP018
Cat.No: T70760
Synonym:
Target:
IMP2-IN-2
Cat.No: T62685
Synonym:
Target:
IMP2-IN-1
Cat.No: T61946
Synonym:
Target:
Levofloxacin Hydrochloride Impurity A
Cat.No: T11007L
Synonym: Levofloxacin Hydrochloride Impurity A(117707-40-1 Free base),左氧氟沙星杂质A(盐酸盐)
Target: Antibacterial
Carvedilol EP IMpurity E
Cat.No: T1698
Synonym: Carvedilol USP E,Carvedilol Impurity E,卡维地洛杂质
Target: Others
BAR 501 impurity
Cat.No: T8752
Synonym:
Target: GPCR19
Domperidone EP Impurity A
Cat.No: T0550
Synonym: 5-氯-1,3-二氢-1-(4-哌啶基)-2H-苯并咪唑-2-酮
Target: Others
Simpinicline
Cat.No: T40867
Synonym: OC-02
Target: AChE
Cetirizine Impurity B dihydrochloride
Cat.No: T9084
Synonym: De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride,西替利嗪杂质B二盐酸盐,西替利嗪杂质04
Target: Histamine Receptor
Teriflunomide impurity 3
Cat.No: T9042
Synonym: 4-Amino-N-(4-trifluoromethylphenyl)benzamide
Target: COX
Imatinib impurities3
Cat.No: T67847
Synonym:
Target: Bcr-Abl, PDGFR, c-Kit
BroMhexine IMpurity B
Cat.No: T1690
Synonym:
Target: Others
Betahistine EP Impurity C
Cat.No: T4196
Synonym: NSC19005
Target: Others, Histamine Receptor
Impromidine hydrochloride
Cat.No: T68921
Synonym:
Target: Histamine Receptor
Enalapril IMpurity B
Cat.No: T1689
Synonym: (+)-N-[1-(S)-Ethoxycarbonxyl-3-phenylpropyl]-L-alanine,依那普利杂质B
Target: Others
AIMP2-DX2-IN-1
Cat.No: T61326
Synonym:
Target: Others
Flecainide Impurity D
Cat.No: T0667
Synonym:
Target: Others
TriMetazidine EP IMpurity-D
Cat.No: T1357
Synonym:
Target: Others
Sofosbuvir impurity F
Cat.No: T12961
Synonym: 索非布韦杂质 F,Sofosbuvir 3',5'-Bis-(S)-phosphate
Target: HCV Protease
Sofosbuvir impurity G
Cat.No: T12962
Synonym:
Target: HCV Protease
Darapladib-impurity
Cat.No: T31204
Synonym:
Target: Others
Ciprofloxacin EP IMpurity A
Cat.No: T1733
Synonym: Q-Acid,Fluoroquinolonic Acid,环丙羧酸,Ciprofloxacin Impurity A
Target: Antibiotic
Rivaroxaban Impurity
Cat.No: T67853
Synonym: Rivaroxaban-10
Target: Factor Xa
Mycophenolic Acid Impurity
Cat.No: T3097
Synonym: 马替麦考酚酸杂质,5,7-dihydroxy-4-methylphthalide
Target: Others
R-IMPP
Cat.No: T4058
Synonym:
Target: Others, Serine/threonin kinase
Importazole
Cat.No: T3445
Synonym:
Target: Apoptosis, Others
Rivastigmine carbamate impurity
Cat.No: T38740
Synonym: 利凡斯的明氨基甲酸酯杂质;利瓦斯的明氨基甲酸酯杂质;卡巴拉汀氨基甲酸酯杂质;利斯的明氨基甲酸酯杂质,3-Nitrophenyl ethyl(methyl)carbamate
Target:
Afatinib impurity 11
Cat.No: T35430
Synonym:
Target:
Remdesivir O-desphosphate acetonide impurity
Cat.No: T38577
Synonym:
Target:
Sofosbuvir impurity C
Cat.No: T12958
Synonym:
Target: Others
Febuxostat impurity 6
Cat.No: T73969
Synonym:
Target:
Ibuprofen impurity 1
Cat.No: T37628
Synonym:
Target:
Cetirizine Impurity C dihydrochloride
Cat.No: T73962
Synonym:
Target:
Hydroxychloroquine Impurity F
Cat.No: T73964
Synonym:
Target:
Diosmin Impurity 5
Cat.No: T126193
Synonym:
Target:
Terazosin dimer impurity dihydrochloride
Cat.No: T37817
Synonym:
Target:
Ibuprofen Impurity F
Cat.No: T40752
Synonym:
Target:
Sofosbuvir impurity H
Cat.No: T12963
Synonym:
Target: HCV Protease
Olmesartan lactone impurity
Cat.No: T40941
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4685 INOSINIC ACID

Inosine 5′-monophosphate,IMP,5'-肌苷酸,I-5'-P

Endogenous Metabolite Metabolism
Inosinic acid (IMP) 是内源性代谢产物。
TMS1830 Disodium 5'-inosinate

Disodium Inosinate,肌苷酸二钠盐,Sodium Inosinate,5'-IMP disodium salt

Others Others
Disodium 5'-inosinate (5'-IMP disodium salt) 是一种食品添加剂,可从通过糖的细菌发酵获得。
T5073 Inosine 5'-monophosphate disodium salt hydrate

Inosine 5'-monophosphate disodium salt,5'-IMP-Na2,肌苷5-单磷酸二钠盐水合物,Disodium 5'-inosinate monohydrate

Others; Endogenous Metabolite Metabolism; Others
Inosine 5'-monophosphate disodium salt hydrate (Inosine 5'-monophosphate disodium salt) 或肌苷酸是次黄嘌呤的核糖核苷酸,是嘌呤合成过程中形成的第一个核苷酸。
T4593 ISOPIMPINELLIN

5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen

Antiviral; DNA/RNA Synthesis; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology
Isopimpinellin (4,9-Dimethoxypsoralen) 是从 Pimpinella saxifrage 根部分离得到的一种天然产物,具有抗病毒和抗利什曼病活性。
T5776 pimpinellin

Apoptosis; Anti-infection Apoptosis; Microbiology/Virology
Pimpinellin 是贯众的一种成分,可通过诱导肿瘤细胞凋亡抑制肿瘤细胞的生长,可作为具有 GABA 受体活性的蛋白质的拮抗剂。
TN2213 Imperialine 3-β-D-glucoside

Sipeimine-3-beta-D-glucoside,西贝母碱苷

Others Others
Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) 是 Imperialine 的糖苷。它对多重耐药肿瘤细胞表现出抗肿瘤特性。
T2845 Imperatorin

Ammidin,8-Isoamylenoxypsoralen,欧前胡素,8-Isopentenyloxypsoralene,Marmelosin,Pentosalen

TRP/TRPV Channel; AChR; AChE; NOD Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; NF-κB
Imperatorin (8-Isopentenyloxypsoralene) 是NO synthesis 和BChE 的抑制剂,IC50分别为 9.2 μmol 和 31.4 μmol。它也是TRPV1的微弱激动剂,EC50为 12.6±3.2 μM。
TN1369 Alloimperatorin

Prangenidin,别欧前胡素

Others Others
Alloimperatorin (Prangenidin) 是一种从Angelica dahurica 的提取得到的香豆素类化合物,具有抗肿瘤作用。
TN2024 Oxyimperatorin

Others Others
Oxyimperatorin 是一种香豆素,分离自当归。
T2846 Isoimperatorin

Antibacterial; AChE Microbiology/Virology; Neuroscience
Isoimperatorin 是 Angelica dahurica 根的甲醇提取物,是一种抗炎剂,有效抑制乙酰胆碱酯酶,IC50为 74.6 μM。
T83522 (S)-(+)-Imperanene

(S)-(+)-Imperanene 是从 Imperata cylindrica 中分离得到的化合物,后者具有明显的利尿和抗炎作用。
TN3380 Alloisoimperatorin

AChR Neuroscience
Alloisoimperatorin is a candidate of AChE inhibitors, it displays potent antioxidant effects against the DPPH radical and against renal epithelial cell injury by using AAPH to generate peroxyl radicals in vitro. Alloisoimperatorin has estrogenic activity
TN6498 Stevia impurity (13-[(2-O-6-deoxy-β-D-glucopyranosyl-3-O-β-D-glucopyranosyl-β-D-glucopyranosyl)oxy]ent-kaur-16-en-19-oic acid β-D-glucopyranosyl ester)

Stevia impurity (13-[(2-O-6-deoxy-β-D-glucopyranosyl-3-O-β-D-glucopyranosyl-β-D-glucopyranosyl)oxy]ent-kaur-16-en-19-oic acid β-D-glucopyranosyl ester) 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6498,CAS号为 1309929-72-3。
T5084 Xanthosine dihydrate

黄苷二水合物

Others; Endogenous Metabolite Metabolism; Others
Xanthosine dihydrate 是衍生自黄嘌呤和核糖的核苷,能够提高牛和山羊的乳腺干细胞数量和产奶量。

天然产物

INOSINIC ACID
Cat.No: T4685
Synonym: Inosine 5′-monophosphate,IMP,5'-肌苷酸,I-5'-P
Target: Endogenous Metabolite
Disodium 5'-inosinate
Cat.No: TMS1830
Synonym: Disodium Inosinate,肌苷酸二钠盐,Sodium Inosinate,5'-IMP disodium salt
Target: Others
Inosine 5'-monophosphate disodium salt hydrate
Cat.No: T5073
Synonym: Inosine 5'-monophosphate disodium salt,5'-IMP-Na2,肌苷5-单磷酸二钠盐水合物,Disodium 5'-inosinate monohydrate
Target: Others, Endogenous Metabolite
ISOPIMPINELLIN
Cat.No: T4593
Synonym: 5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen
Target: Antiviral, DNA/RNA Synthesis, Parasite
pimpinellin
Cat.No: T5776
Synonym:
Target: Apoptosis, Anti-infection
Imperialine 3-β-D-glucoside
Cat.No: TN2213
Synonym: Sipeimine-3-beta-D-glucoside,西贝母碱苷
Target: Others
Imperatorin
Cat.No: T2845
Synonym: Ammidin,8-Isoamylenoxypsoralen,欧前胡素,8-Isopentenyloxypsoralene,Marmelosin,Pentosalen
Target: TRP/TRPV Channel, AChR, AChE, NOD
Alloimperatorin
Cat.No: TN1369
Synonym: Prangenidin,别欧前胡素
Target: Others
Oxyimperatorin
Cat.No: TN2024
Synonym:
Target: Others
Isoimperatorin
Cat.No: T2846
Synonym:
Target: Antibacterial, AChE
(S)-(+)-Imperanene
Cat.No: T83522
Synonym:
Target:
Alloisoimperatorin
Cat.No: TN3380
Synonym:
Target: AChR
Stevia impurity (13-[(2-O-6-deoxy-β-D-glucopyranosyl-3-O-β-D-glucopyranosyl-β-D-glucopyranosyl)oxy]ent-kaur-16-en-19-oic acid β-D-glucopyranosyl ester)
Cat.No: TN6498
Synonym:
Target:
Xanthosine dihydrate
Cat.No: T5084
Synonym: 黄苷二水合物
Target: Others, Endogenous Metabolite
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