76
27
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T25365 |
EGA
|
Others | Others |
EGA 抑制致命毒素的中毒,并阻止多种其他酸依赖性细菌毒素和病毒进入哺乳动物细胞。EGA 是研究膜运输的有力工具,可用于治疗传染病。 | |||
T62899 |
Tau-aggregation and neuroinflammation-IN-1
|
Microtubule Associated; NO Synthase | Cytoskeletal Signaling; Immunology/Inflammation |
Tau-aggregation and neuroinflammation-IN-1 是一种有效的 Tau 蛋白聚集体抑制剂, 对 AcPHF6 和全长 tau 蛋白聚集体显示出显著的抑制活性。Tau-aggregation and neuroinflammation-IN-1具有抗炎活性且可减少 NO 释放。Tau-aggregation and neuroinflammation-IN-1 对 LSP 刺激的 BV2 细胞具有低细胞毒性。Tau-aggregation and neuroinflammation-IN-1 可逆转冈田酸诱导的大鼠记忆障碍。 | |||
T2671 |
Regadenoson
CVT-3146,瑞加德松,Lexiscan |
Adenosine Receptor | GPCR/G Protein; Neuroscience |
Regadenoson (CVT-3146) 是一种腺苷衍生物和选择性 A2A 腺苷受体激动剂,具有冠状动脉舒张活性,对大鼠和猪腺苷 A2A 受体的Ki 分别为 290 和 1120 nM。它是血管扩张剂,可增加啮齿动物血脑屏障的通透性。 | |||
T75129 |
Luxdegalutamide
ARV-766 |
Androgen Receptor; PROTACs | Endocrinology/Hormones; PROTAC |
Luxdegalutamide (ARV-766) 是一种可口服且有效的蛋白水解靶向嵌合体 (PROTAC) 的蛋白质降解剂。Luxdegalutamide降解野生型雄激素受体 AR,也降解包括最普遍的致病性 AR L702H、H875Y 和 T878A 突变相关的 AR LBD 突变体。 | |||
T1551 |
Tegaserod maleate
HTF-919,马来酸替加色罗,SDZ-HTF-919 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tegaserod maleate (SDZ-HTF-919) 是选择性5-HT4受体的部分激动剂和5-HT2B 受体的拮抗剂,用于治疗肠易激综合征和便秘。 | |||
T19335 |
Danegaptide Hydrochloride
GAP-134 (Hydrochloride),ZP 1609 Hydrochloride,(4R)-甘氨酰基-4-(苯甲酰基氨基)-L-脯氨酸盐酸盐 |
Gap Junction Protein | Cytoskeletal Signaling |
Danegaptide Hydrochloride (GAP-134 (Hydrochloride)) 是一种具有口服活性的间隙连接蛋白选择性修饰剂,具有抗心律不齐的作用。 | |||
T68141 |
Seganserin
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Seganserin 是一种非选择性5-羟色胺2-HT 受体拮抗剂,可逆转了氟西汀和喹帕嗪对黄体酮诱导的食欲亢进,抑郁和痛觉的抑制作用,逆转氟西汀和喹帕嗪诱导的抗抑郁和镇痛作用。 | |||
T20992 |
MEGA-9
Nonanoyl-N-Methylglucamide |
Serine Protease | Proteases/Proteasome |
MEGA-9 (Nonanoyl-N-Methylglucamide) 可溶解膜蛋白,可用作非离子去污剂。 | |||
T5432 |
Eganelisib
IPI-549 |
PI3K | PI3K/Akt/mTOR signaling |
Eganelisib (IPI-549) 是 PI3Kγ的选择性抑制剂,其 IC50=16 nM,选择性是其他脂类和蛋白质激酶的 100 倍以上。 | |||
T1378 |
Tegafur
Fluorafur,替加氟,FT-207,NSC 148958,FT 207 |
Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Tegafur (FT 207) 是一种前药,在肝脏中被细胞色素 P-450 酶逐渐转化为氟尿嘧啶。它是抗代谢物氟尿嘧啶的同源物,具有抗肿瘤活性。 | |||
T13111 |
Tegadifur
40497S,FD 1 |
Others | Others |
Tegadifur (40497S) 是一种可口服的抗肿瘤化合物,具有抗新陈代谢作用,常与尿嘧啶林和治疗直肠腺癌。 | |||
T24610 |
Pegamotecan
Prothecan,PEG-camptothecin,PEG-beta-CPT |
Topoisomerase | DNA Damage/DNA Repair |
Pegamotecan (PEG-camptothecin)是一种拓扑异构酶I(TOP1)抑制剂,具有抗癌活性,它可用于治疗食管癌、非小细胞肺癌和胰腺癌。 | |||
T30191L |
Atecegatran TFA
Atecegatran TFA(917904-13-3 Free base),AR-H067637 TFA |
Others | Others |
Atecegatran TFA 常被当作一种抗凝血剂,可用来治疗心血管疾病。 | |||
T22263 |
Bavdegalutamide
ARV-110 |
Androgen Receptor | Endocrinology/Hormones |
Bavdegalutamide (ARV-110) 是一种雄激素受体 (AR) 的 PROTAC 降解剂。 Bavdegalutamide 可用于前列腺癌的研究。 Bavdegalutamide 具有口服活性和选择性,并促进 AR 的泛素化和降解。 | |||
T60680 |
Tegaserod
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tegaserod 是一种可口服的 5-HT4R 激动剂和 5-HT2B 受体拮抗剂,对多种5-羟色胺受体具有抑制作用。 Tegaserod 具有抗肿瘤活性,用于治疗肠易激综合征 (IBS)。 | |||
T25364L |
Efegatran sulfate
LY294468 sulfate,GYKI-14766 sulfate,LY 294468 sulfate,LY-294468 sulfate |
Thrombin | Proteases/Proteasome |
Efegatran sulfate (LY294468 sulfate) 是一种有效的凝血酶抑制剂,可用于治疗血栓类疾病。 | |||
T10988L |
Degarelix acetate(214766-78-6 free base)
|
GNRH Receptor | GPCR/G Protein |
Degarelix acetate(214766-78-6 free base) 是促性腺激素释放激素受体 (GnRHR) 的竞争性可逆拮抗剂。 | |||
T38260 |
SP 600125, negative control
JNK Inhibitor II, negative control |
Others | Others |
SP 600125, negative control 是 SP 600125 的甲基化类似物,可用作SP 600125的阴性对照,对 DTP3和GADD45β/MKK7(生长停滞和 DNA 损伤诱导型 β/介原活化蛋白激酶激酶 7)具有抑制作用,能够恢复活化。SP 600125, negative control 对 JNK2 和 JNK3 的 IC50s 分别为 18 和 24 μM。 | |||
T5642 |
Tegatrabetan
BC2059 |
Wnt/beta-catenin | Cytoskeletal Signaling; Stem Cells |
Tegatrabetan (BC2059) 是β-Catenin 拮抗剂,能够破坏 β-catenin 与转导素 β 样蛋白 1 (TBL1) 结合。 | |||
TP1489 |
Risuteganib
|
||
Risuteganib is a synthetic RGD (arginyl-glycyl-aspartic acid)-class peptide that regulates the functions of multiple integrin isoforms. | |||
T10988 |
Degarelix
|
GNRH Receptor | GPCR/G Protein |
Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist. | |||
T76235 |
Peceleganan
|
||
Peceleganan (PL-5) 是一种合成的肽类似物,由天蚕素 A (1-10) × 蜂毒素 B (3-18) 杂化而成,具有 (10+16) 的结构。该化合物具有抑制伤口感染的作用。 | |||
T76272 |
Pegapamodutide
|
||
Pegapamodutide (LY-2944876) 是一种glucagon-GLP-1 receptor 激动剂,可用于 2 型糖尿病和肥胖症的研究。 | |||
T19336 |
Danegaptide
ZP 1609,GAP-134 |
Others | Others |
Danegaptide (GAP-134), has been identified as a potent and selective second generation gap junction modifier with oral bioavailability.a small modified dipeptide. | |||
T78666 |
Egaptivon pegol
ARC 1779 |
Integrin | Cytoskeletal Signaling |
Egaptivon pegol (ARC1779)为一种核酸适配体,能够阻断von Willebrand Factor (VWF)与血小板GPIb受体的结合,从而展现其抗血栓功能。 | |||
T30192 |
Atecegatran metoxil
Atecegatran fexenetil,AZD-0837,AZD 0837,AZD0837 |
Others | Others |
Atecegatran Metoxil (Atecegatran Fexenetil ,AZD0837) is an oral direct thrombin inhibitor,which currently in clinical development for the prevention of stroke and systemic embolic events in patients with atrial fibrillation. AZD0837 is a selective and re | |||
TF0069 |
HEGA-10
|
Others | Others |
HEGA-10 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0069,CAS号为 139361-84-5。 | |||
T28011 |
Megazol
CL 64855,CL-64855,CL64855 |
Others | Others |
Megazol is a nitroimidazole based drug that cures some protozoan infections. A study of nitroimidazoles found the drug extremely effective against T. cruzi and T. brucei which cause Chagas disease and African sleeping sickness, respectively. | |||
T39781 |
Aβ/tau aggregation-IN-1
|
Others | Others |
Aβ/tau aggregation-IN-1 is a potent inhibitor of Aβ 1-42 β-sheet formation and tau aggregation. It exhibits K D values of 160 μM and 337 μM with Aβ 1-42 and tau, respectively. Additionally, Aβ/tau aggregation-IN-1 can penetrate the blood-brain barrier efficiently. | |||
T39706 |
Pegaptanib sodium
|
Others | Others |
Pegaptanib sodium, an RNA aptamer specifically targeting vascular endothelial growth factor (VEGF)-165, holds great promise for investigating neovascular age-related macular degeneration (AMD). | |||
TF0101 |
C-HEGA-9
|
Others | Others |
C-HEGA-9 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0101,CAS号为 864434-14-0。 | |||
TF0025 |
HEGA-8
|
Others | Others |
HEGA-8 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0025,CAS号为 869652-63-1。 | |||
T76235L |
Peceleganan acetate
|
||
Peceleganan (PL-5) acetate,一种人工合成的肽类似物,由天蚕素 A (1-10) 和蜂毒素 B (3-18) 杂化而成,具有 (10+16) 的结构。该化合物有效抑制伤口感染。 | |||
T81530 |
Pegacaristim
|
||
Pegacaristim是一种单克隆抗体,具有促进血小板生成的活性。 | |||
T78291 |
Tregalizumab
BT-061 |
||
Tregalizumab为人源化抗CD4单克隆抗体(IgG1型),体外能选择性激活调节性T细胞(Tregs)功能。适用于研究自身免疫性疾病(因Treg功能不足)及过敏反应。 | |||
TF0074 |
Mega-10
|
Others | Others |
Mega-10 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0074,CAS号为 85261-20-7。 | |||
T30191 |
Atecegatran
metabolite of AZD0837,atecegatran metoxil |
Others | Others |
Atecegatran 常被当作一种抗凝血剂属于,可用来治疗心血管疾病。 | |||
T69914 |
Variegatic acid
|
Others | Others |
Variegatic acid is a natural inhibitor of β-hexosaminidase release and tumor necrosis factor (TNF)-α secretion from rat basophilic leukemia (RBL 2H3) cells, with IC50 values of 10.4 μM and 16.8 μM, respectively, also inhibiting PKC β1 activity with an IC50 value of 36.2 μM. | |||
T78094 |
Eglumegad hydrochloride
LY354740 hydrochloride,Eglumetad hydrochloride |
Others | Others |
Eglumegad (LY354740) hydrochloride是一种高效且选择性的group II (mGlu2/3) receptor激动剂,其对人mGlu2和mGlu3受体的IC50值分别是5和24 nM。该化合物能够保护神经元不受NMDA毒性影响,并表现出抗焦虑及抗精神病样作用。 | |||
T41227 |
ARCC 4 negative control
|
Others | Others |
ARCC 4 negative control is a negative control for ARCC 4. Binds androgen receptors (AR) without inducing degradation. | |||
T70233 |
Efegatran HCl
|
Others | Others |
Efegatran, also known as GYKI-14166, RGH-2958 and LY294468, a thrombin inhibitor which is being developed by IVAX for the potential treatment of thromboembolic disorders. | |||
T124876 |
Steganacin
|
Others | Others |
Steganacin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124876,CAS号为 41451-68-7。 | |||
T13160 |
Timegadine
替美加定,SR1368 |
COX | Immunology/Inflammation; Neuroscience |
Timegadine is a competitive inhibitor of COX and lipo-oxygenase, with IC50s ranging from 5 nM (washed rabbit platelets) to 20 μM (rat brain) for COX and 100 μM for lipo-oxygenase both in the cytosol fraction of horse platelet homogenates and in washed rabbit platelets. | |||
T77146 | Regavirumab | ||
Regavirumab (MCA C23)为针对巨细胞病毒(CMV)、人血清白蛋白(HSA)及氨基乙酸的人源单克隆抗体。 | |||
T76283 |
Iseganan
|
||
Iseganan 是一种抗菌肽,表现出广谱的抗细菌和抗真菌活性,可用于口腔粘膜炎的研究。 | |||
T14525 |
Begacestat
GSI-953 |
Beta Amyloid | Neuroscience |
Begacestat is a selective thiophene sulfonamide amyloid precursor protein gamma-secretase inhibitor (Aβ40,IC50=15 nM),and for the treatment of Alzheimer's disease. | |||
TF0102 |
C-HEGA-11
|
Others | Others |
C-HEGA-11 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0102,CAS号为 864434-16-2。 | |||
T74811 |
tau/Aβ40 aggregation-IN-1
|
Others | Others |
tau/Aβ40 aggregation-IN-1 (Compound 20) 是一种tau 和Aβ40聚集抑制剂,其IC50分别为 1.8 μM 和 1.3 μM 。 | |||
T79038 |
Tau protein aggregation-IN-1
|
Others | Others |
Tau protein aggregation-IN-1(化合物 0c)是一种针对Tau protein聚集的抑制剂。该化合物主要应用于研究蛋白质折叠障碍类疾病,包括阿尔茨海默病、痴呆、帕金森病、亨廷顿舞蹈病及基于朊病毒引起的海绵状脑病。 | |||
T70255 |
Elapegademase
|
Others | Others |
Elapegademase is an Adenosine Deaminase Inhibitor |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN7038 |
Regaloside H
|
Others | Others |
Regaloside H 是一种糖异生抑制剂,是一种苯丙酸甘油糖苷。它能够抑制大鼠肝癌细胞中葡萄糖的产生。 | |||
TN6489 |
Regaloside A
|
Others | Others |
Regaloside A 是一种从百合中提取出的苯丙烷,在 160 ppm 时显示出 DPPH 自由基清除活性。Regaloside A 具有抗炎活性和抗抑郁活性。 | |||
TN7232 |
Pegamine
|
||
pegamine 是一种在Peganum harmala 和Peganum nigellastrum 中发现的天然产品,是一种新型的生物碱。 | |||
TN2139 |
Regaloside B
鸦胆子苦醇,王百合苷 B |
NOS; COX; NO Synthase | Immunology/Inflammation; Neuroscience |
Regaloside B 是从麝香百合中分离出来的一种苯丙烷,可抑制iNOS 和COX-2的表达,具有抗炎活性。 | |||
TC0022 |
Desoxypeganine
Deoxypeganine |
AChE | Neuroscience |
Desoxypeganine (Deoxypeganine) 是胆碱酯酶的抑制剂。它优先作用于丁酰胆碱酯酶,作为单胺氧化酶 A 而不是单胺氧化酶 B 的选择性抑制剂。它在酒精滥用的药理学治疗中的潜在用途,以减少酒精滥用者的渴望和抑郁,并且也可能有用作为戒烟辅助。 | |||
TN6490 |
Regaloside C
|
Others | Others |
Regaloside C 是一种从百合属的中分离出来的甘油葡糖苷,具有抗炎作用。 | |||
TN7117 |
regaloside I
|
Others | Others |
Regaloside I 是百合中的单体成分,可能是保护人类皮肤成纤维细胞免受 UVA 诱导的形态变化的主要成分。 | |||
TN5778 | cis-Shegansu B | ||
cis-Shegansu B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5778,CAS号为 865474-99-3。 | |||
TN3990 |
Erysenegalensein E
|
Antifection | Microbiology/Virology |
Erysenegalensein E是一种天然产物,属于豆科刺桐属,其产品编号为 TN3990,CAS号为 154992-17-3。Erysenegalensein E可用作对照参考。 | |||
TN6201 |
(1R,6R,9R)-6,9,11-Trihydroxy-4,7-megastigmadien-3-one 11-O-glucoside
|
||
(1R,6R,9R)-6,9,11-Trihydroxy-4,7-megastigmadien-3-one 11-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6201,CAS号为 289914-68-7。 | |||
TN6838 |
Degalactotigonin
|
||
Degalactotigonin is a natural product. | |||
TN5337 |
Megastigm-7-ene-3,5,6,9-tetraol
|
||
Megastigm-7-ene-3,5,6,9-tetraol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5337,CAS号为 276870-26-9。 | |||
T38592 |
Regaloside F
|
Others | Others |
Regaloside F is a phenolic glycerol glucoside that can be found in Lily bulbs. | |||
TN4511 |
Megastigm-7-ene-3,4,6,9-tetrol
|
Others | Others |
Megastigm-7-ene-3,4,6,9-tetrol is a natural product from Apollonias barbujana. | |||
TN5005 |
Shegansu B
|
Influenza Virus | Microbiology/Virology |
Shegansu B exhibits significant in vitro anti-influenza viral activity in MDCK cells. | |||
TN5456 |
Isoerysenegalensein E
|
||
Isoerysenegalensein E shows anti-estrogenic activity comparable to that of 4-hydroxytamoxifen, a typical estrogen receptor antagonist. It shows significant cytotoxicity against HL-60 cells, it induces apoptosis in HL-60 cells through activation of the cas | |||
TN4709 | omega-Benzoyl oxyphloracetophenone | Others | Others |
omega-Benzoyl oxyphloracetophenone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4709,CAS号为 65982-77-6。 | |||
TN5338 |
6,9,10-Trihydroxy-7-megastigmen-3-one
|
||
6,9,10-Trihydroxy-7-megastigmen-3-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5338,CAS号为 476682-97-0。 | |||
T81303 |
Regaloside E
|
||
Regaloside E为自Lilium longiflorum Thunb. 提取的天然化合物。 | |||
TN1920 |
Megastigm-7-ene-3,5,6,9-tetraol
|
Others | Others |
Megastigm-7-ene-3,5,6,9-tetraol is a natural product | |||
TN4990 |
Seneganolide
|
Antifection | Microbiology/Virology |
Seneganolide has insect antifeeding activity. Seneganolide A has antifungal activity. | |||
T81302 |
Regaloside K
|
||
Regaloside K (Compd 1) 是从Easter Lily (Lilium longiflorum Thunb.) 提取的天然化合物。 | |||
TN6045 |
Spegatrine
|
||
Spegatrine is a natural product from Rauvolfia verticillata. | |||
T39610 |
Guattegaumerine
|
Others | Others |
Guattegaumerine, a bisbenzylisoquinoline alkaloid, exhibits antimitotic, cytotoxic, and neuroprotective activities. | |||
TN2140 |
Regaloside D
王百合苷,王百合苷D |
Others | Others |
Regaloside D 是一种分离于 Lilium Longiflorum 的苯丙素。 | |||
TN5332 |
Cucumegastigmane I
|
||
Cucumegastigmane I是一种天然产物,属于葫芦科栝楼属,其产品编号为 TN5332,CAS号为 929881-46-9。Cucumegastigmane I可用作对照参考。 | |||
T81529 |
Peganumine A
|
Others | Others |
Peganumine A,一种天然产物,源自Peganum harmala,具备对HL-60、MCF-7、PC-3、HepG2细胞线显示出细胞毒性作用,其IC50值依次为5.8、38.5、40.2、55.4 µM[1]< /sup>。 |