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34
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T28865 |
STAT3-IN-B9
STAT3 IN B9,B9 |
STAT | JAK/STAT signaling; Stem Cells |
STAT3-IN-B9 (B9) 是异常 STAT3 激活的抑制剂,可抑制 MDA-MB-468、MDA-MB-231 和 DU145 等肿瘤细胞的增殖。 | |||
T21527 |
HBX 41108
HBX-41108,7-氯-9-氧代-9H-茚并[1,2-B]吡嗪-2,3-二甲腈 |
DUB; p53 | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination |
HBX 41108 (HBX-41108) 是一种泛素特异性蛋白酶 7 的非竞争性抑制剂,IC50为 424 nM。它诱导 p53 依赖的凋亡,抑制 USP7 介导的 p53 去泛素化以稳定 p53 并抑制癌细胞生长。 | |||
T60671 |
MAO-B-IN-9
|
Beta Amyloid; Serotonin Transporter; Monoamine Oxidase | Neuroscience |
MAO-B-IN-9是一种可穿过血脑屏障的单胺氧化酶B MAO-B 抑制剂(IC50:0.18μM),具有有效性、选择性和时间依赖性。MAO-B-IN-9具有神经保护作用,可以防止Aβ1-42诱导的神经元细胞死亡,这可能与Aβ1-42的抗聚集作用有关。 | |||
T21660L |
b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate (72122-59-9 Free base) |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
b-Casomorphin (1-3) Acetate 是一种具有阿片样物质作用的三肽。 | |||
TNU0266 |
9-(β-D-Xylofuranosyl)adenine
Xylosyladenine,Adenine xyloside |
Nucleoside Antimetabolite/Analog | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
9-(β-D-Xylofuranosyl)adenine (Adenine xyloside) 是一种腺嘌呤核苷类似物,是一种潜在的平滑肌血管扩张剂。9-(β-D-Xylofuranosyl)adenine 具有抗癌活性。 | |||
T38193L |
β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate(76622-84-9 Free base) |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
β-Endorphin (1-27) (human) acetate 存在于大脑垂体和下丘脑中,具有镇痛活性。 β-Endorphin (1-27) (human) acetate 是一种阿片受体激动剂,对 μ-阿片受体和 δ-阿片受体具有较好的亲和力。 | |||
T60053 |
Hamaline
9-(4-chlorobenzyl)-6-methoxy-1-methyl-4,9-dihydro-3H-pyrido[3,4-b]indole |
COX | Immunology/Inflammation; Neuroscience |
Hamaline (9-(4-chlorobenzyl)-6-methoxy-1-methyl-4,9-dihydro-3H-pyrido[3,4-b]indole) 是一种底物选择性环氧合酶 2 (COX-2) 抑制剂。 | |||
TP2359 |
FMOC-DL-7-AZATRYPTOPHAN
2-({[(9H-fluoren-9-yl)methoxy]carbonyl}amino)-3-{1H-pyrrolo[2,3-b]pyridin-3-yl}propanoic acid |
Others | Others |
FMOC-DL-7-AZATRYPTOPHAN (2-({[(9H-fluoren-9-yl)methoxy]carbonyl}amino)-3-{1H-pyrrolo[2,3-b]pyridin-3-yl}propanoic acid) 是肽。 | |||
T7302 |
CU-CPT9b
CU-CPT-9b,TLR8-specific antagonist 1 |
TLR | Immunology/Inflammation |
CU-CPT9b (TLR8-specific antagonist 1) 是 toll 样受体 8 (TLR8) 的拮抗剂,Kd 为 21 nM。它抑制由 TLR8 激动剂 R-848 在过表达 TLR8 的 HEK-Blue 细胞中诱导的 NF-ĸB 活化,IC50 值为 0.7 nM。 | |||
T12579 |
RAMB4
PTP1B-IN-9 |
Proteasome | Proteases/Proteasome; Ubiquitination |
RAMB4 (PTP1B-IN-9) 是一种泛素-蛋白酶体系统(UPS)应激源,是通过抑制 20S 蛋白酶体催化活性物质上游泛素介导的蛋白质降解而产生。它能够在不影响 20S 蛋白酶体催化活性的情况下触发泛素蛋白酶体系统 (UPS) 应激反应。 | |||
T67703 |
mTOR inhibitor 9b
|
mTOR | PI3K/Akt/mTOR signaling |
mTOR inhibitor 9b 是一种酶抑制剂,对蛋白激酶mTOR 和磷脂酰肌醇 3-激酶 PIK3CA 具有抑制作用,IC50分别为 0.76nm 和1.262 µM。mTOR inhibitor 9b 具有抗癌活性,可用来研究白血病、皮肤癌、乳腺癌、肺癌和结肠癌。 | |||
T13112L1 |
Tat-NR2B9c acetate
Tat-NR2B9c acetate (500992-11-0 Free base),NA-1 acetate |
Others | Others |
Tat-NR2B9c acetate (NA-1 acetate) 是一种突触后密度 95 (PSD-95) 抑制剂,对 PSD-95d2 (PSD-95 PDZ domain 2) 和 PSD-95d1 的 EC50 值分别为 6.7 nM 和 670 nM。它破坏 PSD-95/NMDAR 相互作用,抑制 NR2A 和 NR2B 与 PSD-95 的结合,IC50 值分别为 0.5 μM 和 8 μM。它还抑制神经元一氧化氮合酶 (nNOS)/PSD-95 相互作用,并具有神经保护功效。 | |||
TP1126 |
InsB 9-23
Insulin B chain (9-23) |
||
InsB (9-23) is an insulin B-chain peptide that binds to a class II histocompatibility complex (MHC) allele called I-Ag7. | |||
T21608L |
β-Interleukin I (163-171), human Acetate
β-Interleukin I (163-171), human Acetate(106021-96-9 Free base) |
Others | Others |
β-Interleukin I (163-171), human Acetate 是一种参与调节免疫反应、炎症反应和造血的肽。 | |||
T20889 |
AalphaC
2-Amino-alpha-carboline,Aalpha C,2-氨基-9H-吡啶[2,3-b]吲哚,Aalpha-C |
Others | Others |
AalphaC (2-Amino-alpha-carboline) 是一种潜在的致癌物质。 | |||
TP1645 |
β-Amyloid (1-9)
β-Amyloid 1-9 |
||
This is an N-terminal fragment of beta amyloid. It consists of amino acid residues 1 to 9. Truncated beta amyloid peptide (10-40) still forms amyloid fibrils and shows fibril polymorphism. | |||
T21609L |
Beta-Sheet Breaker Peptide iAβ5 Acetate
Beta-Sheet Breaker Peptide iAβ5 Acetate(182912-74-9 Free base) |
Others | Others |
Beta-Sheet Breaker Peptide iAβ5 Acetate 抑制大鼠脑模型中的淀粉样蛋白生成。 | |||
T13524 | 9-cis-β-Carotene | Others | Others |
9-cis-β-Carotene, a precursor of retinal, is cleaved by beta-carotene oxygenase 1 (BCMO1) to produce 9-cis-retinal. It inhibits photoreceptor degeneration and restores retinal function in vivo. | |||
T61935 |
B-Raf IN 9
|
||
B-Raf IN 9 (compound 8b) 是有效的B-Raf 抑制剂(IC50= 24.79 nM)。B-Raf IN 9 将细胞周期阻滞于 G2/M 期,诱导凋亡。B-Raf IN 9 对人前列腺癌 PC-3 细胞表现出较强的抗肿瘤活性(IC50= 7.83 μM)。 | |||
T7167 |
Purvalanol B
NG 95,(2R)-2-[[6-[(3-氯-4-羧基苯基)氨基]-9-(1-甲基乙基)-9H-嘌呤-2-基]氨基]-3-甲基-1-丁醇 |
CDK; Parasite | Cell Cycle/Checkpoint; Microbiology/Virology |
Purvalanol B (NG 95) 是选择性可逆的 ATP 竞争性 CDK 抑制剂。它在一系列其他蛋白激酶 (IC50>1000 nM) 中显示出对 CDK 的选择性。它抑制耐氯喹菌株 P. falciparum 的生长。 | |||
T79896 |
Cbl-b-IN-9
|
E1/E2/E3 Enzyme | Ubiquitination |
Cbl-b-IN-9(Compound 300)为针对casitas B系淋巴瘤(Cbl-b)及c-Cbl的抑制剂,其IC50值分别为5.6 nM与4.7 nM。 | |||
T80463 |
Dynorphin B (1-9)
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Dynorphin B (1-9)为Dynorphin B的N-端裂解产物,属于神经肽类。其形成受到半胱氨酸肽酶非选择性抑制剂N-ethylmaleimide的阻断。 | |||
T35655 |
2,6-Dichloropurine-9-β-D-riboside
|
||
2,6-Dichloropurine-9-β-D-riboside is a building block.1,2It has been used in the synthesis of photoaffinity probes for nucleotide binding sites in proteins. 1.Wower, J., Hixson, S.S., Sylvers, L.A., et al.Synthesis of 2,6-diazido-9-(β-D-ribofuranosyl)purine 3',5'-bisphosphate: Incorporation into transfer RNA and photochemical labeling of Escherichia coli ribosomesBioconjug. Chem.5(2)158-161(1994) 2.Seiter, M.S., Bauer, M.P., Bogel, P.D., et al.Synthesis of novel spin-labeled photoaffinity deriva... | |||
T31672 |
Erythrofuranosyladenine
9-β-D-Erythrofuranosyladenine,ETA |
||
Erythrofuranosyladenine(9-beta-D-Erythrofuranosyladenine, ETA) is a nontoxic MTAP substrate. Erythrofuranosyladenine is an effective salvage agent for methylthioadenosine phosphorylase–selective therapy of T-cell acute lymphoblastic leukemia with L-alanos | |||
TNU0267 |
9-(b-D-Xylofuranosyl)guanine
|
||
9-(b-D-Xylofuranosyl)guanine is a Nucleoside Derivative - Xylo-nucleoside. | |||
TNU0382 |
8-Bromo-9-(b-D-xylofuranosyl)guanine
|
||
8-Bromo-9-(b-D-xylofuranosyl)guanine is a Nucleoside Derivative - Xylo-nucleoside; 8-Modified purine nucleoside. | |||
TNU0384 |
8-Benzyloxy-9-(b-D-xylofuranosyl)guanine
|
||
8-Benzyloxy-9-(b-D-xylofuranosyl)guanine is a Nucleoside Derivative - Xylo-nucleoside; 8-Modified purine nucleoside. | |||
T82579 |
Dermaseptin-B9
|
||
Dermaseptin-B9为Phyllomedusinae亚科青蛙分离得到的一种抗菌肽。 | |||
TNU1411 | 2,6-Bis(4-morpholinyl)-9-b-D-ribofuranosyl-9H-purine | ||
Nucleoside Derivatives –6-Subtituted nucleosides;2-Substituted nucleosides | |||
T74841 | NF-κB-IN-9 | ||
NF-κB-IN-9 是一种靶向核因子 NF-κB 的声敏剂 (λex/λem=489/628 nm)。NF-κB-IN-9 由于分子中有两个白藜芦醇单元,而对 NF-κB 信号表现出强烈的抑制作用。NF-κB-IN-9 具有抗肿瘤活性,并对癌细胞表现出显着的声细胞毒性。NF-κB-IN-9 在小鼠移植模型中具有生物安全性。 | |||
TNU0291 | 1,N6-Etheno-9-(b-D-xylofuranosyl)adenosine | ||
Nucleoside Derivatives - Tricyclic nucleosides; Xylo-nucleosides | |||
TNU0154 |
6-Methoxy-9-(3-deoxy-3-fluoro-b-D-ribofuranosyl)-9H-purine
|
||
Nucleoside Derivatives –Fluoro-modified nucleosides, 6-Modified purine nucleosides, 3’-Modified nucleosides | |||
TNU0385 |
1-Amino-8-benzyloxy-9-(b-D-xylofuranosyl)guanine
|
||
1-Amino-8-benzyloxy-9-(b-D-xylofuranosyl)guanine is a Nucleoside Derivative - Xylo-nucleoside; 8-Modified purine nucleoside; Amino nucleoside. | |||
T13112 |
Tat-NR2B9c
Tat-NR2Bct,NA-1 |
NO Synthase; iGluR | Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience |
Tat-NR2B9c (NA-1) 是一种突触后密度-95(PSD-95)抑制剂,具有神经保护和抗癫痫作用。Tat-NR2B9c 可抑制PSD-95d2、 PSD-95d1 和 PSD-95,可阻止NMDA诱导的神经元NADPH氧化酶的激活,从而阻断超氧化物的产生,可减少中风后急性期的缺血性损伤。 | |||
TNU1077 |
6-Chloro-2-hydroxy-9-(2,3,5-tri-O-acetyl)-b-D-ribofuranosyl-9H-purine
|
||
Nucleoside Derivatives - Halo-nucleoside | |||
TNU1591 | 5-Aza-9-(b-D-xylofuranosyl) cytosine; 5-Aza-xylo-cytidine | ||
5-Aza-9-(b-D-xylofuranosyl) cytosine; 5-Aza-xylo-cytidine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TNU1591。 | |||
TNU0383 | 7-Allyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl) guanine | ||
Nucleoside Derivatives - Xylo nucleosides, 8-Modified purine nucleosides; N-Methylated alkylated nucleosides | |||
TNU0386 |
1-Amino-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl) guanine
|
||
1-Amino-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl) guanine is a Nucleoside Derivative - Xylo-nucleoside; 8-Modified purine nucleoside; Amino nucleoside. | |||
TNU0394 | 7-Cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-ribofuranosyl)guanine | ||
7-Cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-ribofuranosyl)guanine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TNU0394。 | |||
T81037 |
Tat-HA-NR2B9c
|
||
Tat-HA-NR2B9 是一种包括HIV-1 Tat细胞膜转导结构域片段、流感病毒血凝素(HA)表位标签以及NR2B(NR2B9c) C端9个氨基酸的化学复合物。该化合物能够降低大鼠缺血性脑损伤的梗塞面积,同时促进神经功能的恢复。 | |||
TNU0388 |
7-Cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl) guanine
|
||
Nucleoside Derivatives - Xylo-nucleosides; 8-Modified purine nucleosides; N-Methylated alkylated nucleosides | |||
TNU0387 | 1-Amino-7-cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl)guanine | ||
Nucleoside Derivatives - Xylo-nucleosides; 8-Modified purine nucleosides; Amino nucleosides; N-Methylated alkylated nucleosides | |||
TNU1301 |
6-Chloro-7-deaza-9-(2’,3’,5’-tri-O-acetyl-b-D-ribofuranosyl)purine
|
||
Nucleoside Derivatives - 7-Deazapurine nucleosides; Halo-nucleosides; Scaffolds and Templates | |||
TNU0992 | 9-(5(R)-C-Methyl-2,3,5-tri-O-benzoyl-b-D-ribofuranosyl)-6-chloropurine | ||
9-(5(R)-C-Methyl-2,3,5-tri-O-benzoyl-b-D-ribofuranosyl)-6-chloropurine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TNU0992。 | |||
TNU1002 |
6-chloro-purine-9-b-D-(2-O-acetyl-3,5-di-O-benzoyl)xylo-furanoside
|
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Nucleoside Derivatives - Xylo-nucleoside; Halo-nucleoside; Scaffolds and Templates | |||
T78266 |
Anti-Mouse LAG-3 Antibody (C9B7W)
|
||
Anti-MouseLAG-3Antibody为针对小鼠LAG-3的Rat源IgG1抗体抑制剂。 | |||
TNU1086 | 6-Chloro-2-fluoropurine-9-b-D-(3,5-bis-O-(p-toluoyl)-2-deoxy)riboside | ||
Nucleoside Derivatives - Fluoro-modified nucleoside; Halo-nucleoside | |||
T66996 | (4aR,4bS,6aS,7S,9aS,9bS,11aR)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid | ||
(4aR,4bS,6aS,7S,9aS,9bS,11aR)-4a,6a-Dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66996,CAS号为 104239-97-6。 | |||
T65298 |
(4aR,4bS,6aS,7S,9aS,9bS,11aR)-Methyl 4a,6a-dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylate
|
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(4aR,4bS,6aS,7S,9aS,9bS,11aR)-Methyl 4a,6a-dimethyl-2-oxo-2,4a,4b,5,6,6a,7,8,9,9a,9b,10,11,11a-tetradecahydro-1H-indeno[5,4-f]quinoline-7-carboxylate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T65298。 | |||
T66280 |
2-Chloro-4-(4-fluorophenyl)-5,6,7,8,9,10-hexahydrocycloocta[b]pyridine
|
||
2-Chloro-4-(4-fluorophenyl)-5,6,7,8,9,10-hexahydrocycloocta[b]pyridine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66280,CAS号为 132813-14-0。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4589 |
9'''-Methyl salvianolate B
9’’’-丹酚酸B单甲酯,9'''-丹酚酸B单甲酯,9'''-MethyllithosperMate B |
Others | Others |
9'''-MethyllithosperMate B 是一种从 Cynoglossum columnaeTen 中获得的一种天然提取物。 | |||
T4961 |
9''-Methyl salvianolate B
9'-Methyl lithospermate B,9’-丹酚酸B单甲酯,9''-丹酚酸B单甲酯 |
Others | Others |
9'-Methyl lithospermate B 是一种酚类化合物,提取自 RadixSalvia miltiorrhizae。 | |||
TN3317 |
9-Epiblumenol B
|
Others | Others |
9-Epiblumenol B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3317,CAS号为 22841-42-5。 | |||
TN6251 |
Blumenol B 9-O-glucoside
Dihydrovomifoliol 9-O-glucoside |
||
Blumenol B 9-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6251,CAS号为 114226-08-3。 | |||
TNU0052 |
Nebularine
9-(beta-D-Ribofuranosyl)-9H-purine |
Apoptosis | Apoptosis |
Nebularine (9-(beta-D-Ribofuranosyl)-9H-purine),是一种嘌呤核苷类似物,具有广谱的抗肿瘤活性,针对惰性淋巴恶性肿瘤并诱导凋亡。Nebularine的抗癌机制依赖于抑制DNA合成。 | |||
TN3327 |
9-O-Methyl-4-hydroxyboeravinone B
|
Others | Others |
9-O-Methyl-4-hydroxyboeravinone B is a promising candidate for cancer therapy. | |||
TMO2681 |
Xanthosine
9-Beta-D-Ribofuranosylxanthine,黄嘌呤核苷,Xanthine riboside |
Others; Endogenous Metabolite | Metabolism; Others |
Xanthosine (9-Beta-D-Ribofuranosylxanthine) 是黄嘌呤核苷,它能够提高山羊和牛的乳腺干细胞数量和产奶量。 | |||
T0062 |
Folic acid
Folate,Vitamin B9,Pteroylglutamic acid,Vitamin M,叶酸,Folacin |
DNA/RNA Synthesis; Endogenous Metabolite | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism |
Folic acid (Vitamin B9) 是维生素B9,是合成DNA/RNA,新细胞产生和维持的必要成分。 | |||
T1506 |
Vidarabine
Adenine Arabinoside,阿糖腺苷,9-β-D-Arabinofuranosyladenine,Vira-A,Arabinosyladenine,Ara-A |
Nucleoside Antimetabolite/Analog; Tyrosine Kinases; DNA/RNA Synthesis; Antibiotic; HSV | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Vidarabine (Adenine Arabinoside) 是从链霉菌分离的核苷类抗生素,能抗单纯性疱疹和水痘-带状疱疹病毒。它对 HSV-1 和 HSV-2 的 IC50值分别为 9.3 μg/ml 和 11.3 μg/ml。 | |||
TN1471 |
Cassiaside C
决明子苷C,Toralactone 9-O-β-D-gentiobioside |
Others; Endogenous Metabolite | Metabolism; Others |
Cassiaside C (Toralactone 9-O-β-D-gentiobioside) 是一种萘酚类化合物,从决明子种子中分离得到,对晚期糖基化终产物 (AGE) 的形成具有抑制作用。 | |||
TN6909 |
Polyporusterone B
猪苓酮B,(1R,2R,4S,5R,7R,11R,14S,15R)-14-[(2R,3R)-2,3-dihydroxy-6-methyl-5-methylideneheptan-2-yl]-4,5,11-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,?.011,1?]heptadec-9-en-8-one |
Others | Others |
Polyporusterone B ((1R,2R,4S,5R,7R,11R,14S,15R)-14-[(2R,3R)-2,3-dihydroxy-6-methyl-5-methylideneheptan-2-yl]-4,5,11-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,?.011,1?]heptadec-9-en-8-one) 是一种三萜羧酸,从Polyporus umbellatusFries 中分离得到。它对自由基诱导的红细胞裂解 (溶血) 具有抑制作用。 | |||
TN4537 | Methyl 8-hydroxy-3-(2-methoxy-2-oxoethyl)-6-methyl-9-oxo-9H-furo[3,4-b]chromene-1-carboxylate | Others | Others |
Methyl 8-hydroxy-3-(2-methoxy-2-oxoethyl)-6-methyl-9-oxo-9H-furo[3,4-b]chromene-1-carboxylate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4537,CAS号为 96287-41-1。 | |||
T83551 | (9S)-Macrocidin B | ||
(9S)-Macrocidin B 的除草活性不如macrocidin A。 | |||
TN2410 |
Uncinatone
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Others | Others |
Uncinatone is a natural product from the stems and roots of Clerodendrum philippinum var. simplex | |||
TN1631 |
Eupalinolide K
[3AR-[3AR*,4R*(E),6E,9S*,10E,11AR*]]-4-羟基-2-甲基-2-丁烯酸 2,3,3A,4,5,8,9,11A-八氢-9-羟基-6,10-二甲基-3-亚甲基-2-氧代环癸五烯并[B]呋喃-4-基酯,野马追内酯 K,野马追内酯K |
STAT | JAK/STAT signaling; Stem Cells |
Eupalinolide K 是来自野马追的一种倍半萜内酯,是 STAT3抑制剂,可作为迈克尔反应受体。 | |||
TN2413 |
Diacetylpiptocarphol
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Others | Others |
Diacetylpiptocarphol has antiplasmodial activity | |||
TN1880 |
Lucidenic acid B
Lucidenicacid B |
Apoptosis; Caspase | Apoptosis; Proteases/Proteasome |
Lucidenic acid B (Lucidenicacid B) 是从灵芝中提取得到的天然化合物,可诱导caspase-9 和 caspase-3 的活化和 PARP 的裂解,可通过线粒体介导诱导人白血病细胞凋亡 。 Lucidenic acid B通过灭活MAPK / ERK信号转导途径和降低NF-kappaB和AP-1的结合活性来抑制PMA诱导的人肝癌细胞侵袭。。Lucidenic acid B 对细胞周期和坏死细胞没有影响。 | |||
T36473 |
trans-Nerolidol
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trans-Nerolidol is a sesquiterpene that has been found in various plants, includingC. sativa, and has diverse biological activities, including antimicrobial, antioxidant, anticancer, and insecticidal properties.1,2,3,4In a disc assay,trans-nerolidol inhibits the growth ofS. aureus,B. subtilis,E. coli, andS. cerevisiaewith zones of inhibition measuring 10, 9, 10, and 4 mm, respectively.2It reduces viability of CaCo-2 adenocarcinoma cells with an IC50value of 28.7 mg/L and reduces production of re... | |||
T4S0181 |
Hinokiflavone
日本扁柏黄酮,扁柏双黄酮 |
MMP; BCL; E1/E2/E3 Enzyme | Apoptosis; Proteases/Proteasome; Ubiquitination |
Hinokiflavone 是pre-mRNA 剪接活性的新型调节剂,通过抑制剪接体装配来阻止pre-mRNA 底物的剪接,特别是阻止 B complex 的形成。它是SUMO protease 蛋白酶抑制剂,能够抑制前哨蛋白特异性蛋白酶 1 的活性。 | |||
T83545 |
(E)-(-)-Aspongopusamide B
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(E)-(-)-Aspongopusamide B (Compound 9) 是从昆虫Aspongopus chinensis 分离得到的一种天然产物。 | |||
TN6026 |
Deoxyisocalyciphylline B
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Deoxyisocalyciphylline B是一种天然产物,属于交让木科虎皮楠属,其产品编号为 TN6026,CAS号为 619326-75-9。Deoxyisocalyciphylline B可用作对照参考。 | |||
TN5705 | Muricarpone B | ||
Muricarpone B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5705,CAS号为 886226-15-9。 | |||
TN4786 |
Picrasin B acetate
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Others | Others |
Picrasin B acetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4786,CAS号为 30315-04-9。 | |||
TN6668 |
Rheumone B
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Rheumone B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6668,CAS号为 2095596-67-9。 | |||
TN3969 | Epiguajadial B | Others | Others |
Epiguajadial B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3969,CAS号为 1411629-26-9。 | |||
TN5553 | Valeriotriate B | ||
Valeriotriate B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5553,CAS号为 862255-64-9。 | |||
TN5931 |
Alstonic acid B
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Alstonic acid B是一种天然产物,属于夹竹桃科鸡骨常山属,其产品编号为 TN5931,CAS号为 1159579-45-9。Alstonic acid B可用作对照参考。 | |||
TN2577 | 11,12-Di-O-acetyltenacigenin B | Others | Others |
11,12-Di-O-acetyltenacigenin B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2577,CAS号为 857897-01-9。 | |||
T75441 | (8′α,9′β-Dihydroxy)-3-farnesylindole | ||
(8'α,9'β-Dihydroxy)-3-farnesylindole 对枯草芽孢杆菌具有较强的抑制活性(EC509.8μM)。 | |||
TN5632 | Sarcandrone B | ||
Sarcandrone B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5632,CAS号为 1190225-48-9。 | |||
TN5196 |
Turmeronol A
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Others | Others |
Turmeronol A and turmeronol B are inhibitors of soybean lipoxygenase, they inhibited soybean lipoxygenase at the IC50 values of 16 uM and 9 uM, respectively. | |||
T79976 |
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside
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HBV | Microbiology/Virology |
Dihydrodehydrodiconiferyl alcohol 9-O-β-D-xylopyranoside 作为一种抗HBV剂,在Hep G2.2.15细胞系上能够抑制HBsAg和HBeAg的分泌,其IC50值分别约为1.67 mM和>2.15 mM。 | |||
T31471 |
Dihydroisoalantolactone
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Dihydroisoalantolactone is found in herbs and spices. Dihydroisoalantolactone is isolated from roots of Inula helenium (elecampane). This compound Aliphatic heteropolycyclic, belongs to the class of organic compounds known as eudesmanolides, secoeudesmano | |||
T37452 |
Stephacidin B
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Stephacidin B is a fungal metabolite that has been found inA. ochraceus.1Dimeric stephacidin B is rapidly converted to a monomer, avrainvillamide ,in vitro.2Stephacidin B is cytotoxic to a variety of cancer cells, including testosterone-independent PC3 and -sensitive LNCaP prostate cancer cells (IC50s = 0.37 and 0.06 μM, respectively) and estradiol-independent SK-BR-3 and -sensitive MCF-7 breast cancer cells (IC50s = 0.32 and 0.27 μM, respectively).1It induces apoptosis in HepG2 and Huh7 hepatoc... |