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Targets Recommended: ROS

10

抑制剂 & 化合物

31

天然产物

1

化合物库

8

重组蛋白

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Cat. No. Product Name
L4600 植物来源化合物库

3048 compounds
3048 个植物来源天然产物的独特集合,来自277类植物的精心之选;

化合物库

植物来源化合物库
Cat.No: L4600
Compounds: 3048
Cat. No. Product Name Target Signaling Pathways
T13538 AlbA-DCA

ROS Immunology/Inflammation
AlbA-DCA is a conjugate formed by the attachment of Albiziabioside A to a dichloroacetate acid subunit. It can induce a marked increase in intracellular ROS and alleviate the accumulation of lactic acid in the tumor microenvironment, and also selectively
T20600 Kaolin

Clay 347,Hydrated aluminum silicate,Bolus alba,HSDB 630,Altowhite,China clay,高岭土

Others Others
Kaolin (Bolus alba) 是一种以高岭石族矿物为主的粘土。 Kaolin 提高了这种监测血友病治疗方法的敏感性。
T21358 Dalbavancin

BI 397,BI-397,VER 001,A-A 1,BI397,VER-001,Dalbavancin HCl,达巴万星

Antibacterial; Antibiotic Microbiology/Virology
Dalbavancin (BI-397) HCl 是一种半合成的脂糖肽抗生素,对革兰氏阳性细菌有杀菌活性。Dalbavancin 抑制金黄色葡萄球菌和炭疽芽孢杆菌的 MIC90分别为 0.06 μg/mL 和 0.25 μg/mL。
T7725 Albaconazole

W 0027,UR-9825,UR9825,W-0027

P450; Antifungal Metabolism; Microbiology/Virology
Albaconazole (W-0027)是一种小分子真菌细胞色素P450家族成员51 (fungal CYP51A1)抑制剂。它可用于治疗真菌感染、皮肤和肌肉骨骼疾病,可用于研究外阴阴道念珠菌病、Chagas病和泌尿生殖系统疾病。
T75253 Dalbavancin hydrochloride

Dalbavancin hydrochloride (MDL-63397 hydrochloride)为半合成脂糖肽类抗生素,有效对抗革兰氏阳性菌。其对金黄色葡萄球菌与炭疽芽孢杆菌的MIC90分别为0.06 μg/mL与0.25 μg/mL。
T125711 Eclalbasaponin IV

Eclalbasaponin IV 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125711,CAS号为 158511-61-6。
T29830 Albacarcin V

NSC354844,NSC-354844,NSC 354844

Albacarcin V is a biochemical.
T125712 Eclalbasaponin III

Eclalbasaponin III 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125712,CAS号为 158511-60-5。
T124310 Albanin A

Albanin A 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124310。
T81970 Kuwanon T

Kuwanon T为一种源自桑树根皮的异戊二烯黄酮类化合物,能抵御t-BHP诱导的氧化应激,其EC50值为30.32 μM。

化合物

AlbA-DCA
Cat.No: T13538
Synonym:
Target: ROS
Kaolin
Cat.No: T20600
Synonym: Clay 347,Hydrated aluminum silicate,Bolus alba,HSDB 630,Altowhite,China clay,高岭土
Target: Others
Dalbavancin
Cat.No: T21358
Synonym: BI 397,BI-397,VER 001,A-A 1,BI397,VER-001,Dalbavancin HCl,达巴万星
Target: Antibacterial, Antibiotic
Albaconazole
Cat.No: T7725
Synonym: W 0027,UR-9825,UR9825,W-0027
Target: P450, Antifungal
Dalbavancin hydrochloride
Cat.No: T75253
Synonym:
Target:
Eclalbasaponin IV
Cat.No: T125711
Synonym:
Target:
Albacarcin V
Cat.No: T29830
Synonym: NSC354844,NSC-354844,NSC 354844
Target:
Eclalbasaponin III
Cat.No: T125712
Synonym:
Target:
Albanin A
Cat.No: T124310
Synonym:
Target:
Kuwanon T
Cat.No: T81970
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3384 Wedelolactone

蟛蜞菊内酯,IKK Inhibitor II

Apoptosis; NF-κB; Lipoxygenase; Caspase Apoptosis; Metabolism; NF-κB; Proteases/Proteasome
Wedelolactone (IKK Inhibitor II) 是来自旱莲草的一种天然产物,通过阻断 IκBα 的磷酸化和降解来抑制细胞中 NF-κB 介导的基因转录,具有抗癌,抗炎和抗氧化活性。
TN7121 d-Epigalbacin

(-)-Zuonin A,表加巴辛

JNK MAPK
d-Epigalbacin ((-)-Zuonin A) 是一种天然木质素。d-Epigalbacin 是一种强效、选择性的JNKs 抑制剂,JNK1、JNK2和JNK3的IC50s 分别为1.7μM、2.9μM 和1.74μM。
TN1600 Eclalbasaponin I

Others Others
Eclalbasaponin I 分离自鳢肠中,具有抗肿瘤作用,能够抑制肝癌细胞 smmc-7721 的增殖(IC50:111.1703 μg/ml)。
TN3371 Albatrelin G

Others Others
Albatrelin G shows weak cytotoxic activity to cell lines HL-60, SMMC-7721, A-549, and MCF-7, in vitro.
T75602 Albanol B

Albanol B 是一种芳基苯并呋喃衍生物,可从桑葚中分离得到。Albanol B 具有抗阿尔茨海默病、抗菌和抗氧化活性。Albanol B 抑制癌细胞增殖,下调 CDK1表达。Albanol B 还会诱导细胞周期停滞在 G2/M 期,诱导细胞凋亡 (apoptosis)。Albanol B 诱导线粒体 ROS 产生并增加 AKT 和 ERK1/2的磷酸化水平。
T2S1115 Albaspidin AA

Antifection Microbiology/Virology
Albaspidin AA displays strong antibacterial activity against the vegetative form of P. larvae (MIC ranging from 0.168-220 uM). It may have in vitro nematocidal activity against L4 stage larvae.
T29831 Albaspidin

Albaspidin is a biochemical.
TN3370 Albatrelin C

Others Others
Albatrelin C is a natural product from Albatrellus ovinus.
TN3369 Albatrelin A

Others Others
Albatrelin A is a natural product from Albatrellus ovinus.
TN1365 Albaspidin AP

Fatty Acid Synthase Metabolism
Albaspidin-AP, -PP, -PB inhibit Fatty acid synthase (FAS) with IC50 values ranging from 23.1+/-1.4 to 71.7+/-3.9 microM, they could be considered to be a promising class of FAS inhibitors, and FAS is emerging as a potential therapeutic target to treat can
T13706 Glucosinalbate

Others Others
Glucosinalbate 是一种天然产物,分离自拟南芥。
TN2212 Glucosinalbate potassium

白芥子钾盐,Sinalbin potassium salt

Others Others
Sinalbin potassium salt is a natural product
TQ0301 Kuwanon A

NO Synthase Immunology/Inflammation
Kuwanon A 抑制一氧化氮的产生 (IC50: 10.5 μM)。Kuwanon A 是从桑树 (Morus alba L.) 中分离出来的黄酮衍生物。
TN1261 3-O-Caffeoylquinic acid methyl ester

Others Others
3-O-Caffeoylquinic acid methyl ester 是 Pyrrosia calvata 的成分之一。
TN7027 Benzoylalbiflorin

Paeonivayin,苯甲酰芍药内酯苷

Others Others
Benzoylalbiflorin (Paeonivayin) 是一种分离自 Radix Paeoniae Alba 的单萜。其中 Radix Paeoniae Alba 是传统中药,已用于研究类风湿关节炎,能够缓解炎症,闭经,鼻出血,腹痛和其他症状。
TN1949 Moracin C

桑辛素 C,5-(6-羟基-2-苯并呋喃基)-2-(3-甲基-2-丁烯基)-1,3-苯二醇

ROS; NO Synthase Immunology/Inflammation
Moracin C 是一种发现于Morus mesozygia、Morus alba var. multicaulis 中的天然化合物,是一种抗炎剂。Moracin C 可抑制细胞中的一氧化氮(NO)释放和LPS 激活的活性氧(ROS)。
T5742 Isodemethylwedelolactone

异去甲蟛蜞菊内酯,Isodemethylwedelolacton

Others Others
Isodemethylwedelolactone (Isodemethylwedelolacton) 是一种促凝剂,也是溶血性成分,分离自 Eclipta alba
T5S0689 Demethylwedelolactone

去甲蟛蜞菊内酯,去甲基蟛蜞内酯

Serine Protease Proteases/Proteasome
Demethylwedelolactone 是一种分离自 Eclipta alba 中的 coumestan 天然产物。它能抑制乳腺癌细胞的移动和侵袭,是一种有效的trypsin 抑制剂(IC50:3.0 μM)。
T3773 Oxypaeoniflorin

氧化芍药苷,Oxypaeoniflora

Others Others
Oxypaeoniflorin (Oxypaeoniflora) 从 Paeoniae 中分离得到的单萜糖苷化合物,是一种抗氧化剂,是具有神经保护和抗炎作用。
TN1252 3'-Geranyl-3-prenyl-2',4',5,7-tetrahydroxyflavone

Apoptosis Apoptosis
3'-Geranyl-3-prenyl-2',4',5,7-tetrahydroxyflavone 是一种来自桑叶的黄酮类化合物,具有细胞毒性,可诱导细胞凋亡。
T2830 Betulinic acid

白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid

Apoptosis; Mitophagy; NF-κB; HIV Protease; Topoisomerase; Endogenous Metabolite; Aminopeptidase; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Betulinic acid (ALS-357) 是从白桦树皮中分离出来的一种五环三萜类天然产物,是真核细胞拓扑异构酶 I 的抑制剂,IC50值为 5 μM,具有抗逆转录病毒、抗疟疾、抗癌和抗炎特性。
TN1956 Mulberrofuran G

Phosphatase; HBV; Glucosidase Metabolism; Microbiology/Virology
Mulberrofuran G分离自自 Morus alba L.,具有抗乙型肝炎病毒活性,可保护缺血损伤诱导的细胞死亡。Mulberrofuran G 是一种 PTP1B 和 α-葡萄糖苷酶的双重抑制剂,可用于研究阿尔茨海默症。
TN1950 Moracin M

PDE Metabolism
Moracin M 是桑白皮中的一种酚类成分,有效的磷酸二酯酶 4 (PDE4) 抑制剂,对于 PDE4D2,PDE4B2,PDE5A1 和 PDE9A2 的 IC50 分别为 2.9 μM,4.5 μM,> 40 μM 和 > 100 μM。Moracin M 具有抗炎活性。
T82054 Ipalbine

Ipalbine为源自Ipomoea alba L的六氢吲哚生物碱类化合物。
T81742 Mulberrofuran B

Mulberrofuran B,一种从Morus alba乙醇提取物中分离得到的化合物,展现了抗氧化活性。
T38524 Paeoniflorin sulfite

During the sulfur-fumigation process of Paeoniae Radix Alba, Paeoniflorin, which serves as a principal constituent, can be converted into Paeoniflorin sulfite.
TN2814 23-Hydroxybetulin

Others Others
23-Hydroxybetulin is a natural product from Betula alba L.
TN4401 Kuwanol C

Others Others
Kuwanol C 是一种天然产物,存在于Morus alba L。
TN2453 Kuwanol A

Others Others
Kuwanol A is a natural product from Morus alba L.
T83479 1,2,6,7,8,9-Hexahydro-1,6,6-trimethyl-3,11-dioxanaphth[2,1-e]azulene-10,12-dione

1,2,6,7,8,9-Hexahydro-1,6,6-trimethyl-3,11-dioxanaphth[2,1-e]azulene-10,12-dione 是一种从丹参酮 (Salvia miltiorrhiza f. alba) 中提取的化学物质,具有二氢异丹参酮结构,显示出细胞毒性和抗肿瘤的活性。
TN1953 Morusinol

桑根皮醇,桑树醇

ERK; MEK; Autophagy; Ras Autophagy; GPCR/G Protein; MAPK
Morusinol 是从桑树根皮中提取出的类黄酮。 Morusinol 具有抗血小板和抗癌活性,在体内抑制动脉血栓形成,通过诱导自噬、G2/M 细胞周期阻滞、抑制细胞侵袭和迁移以及靶向 Ras/MEK/ERK 通路发挥抗肿瘤活性。

天然产物

Wedelolactone
Cat.No: T3384
Synonym: 蟛蜞菊内酯,IKK Inhibitor II
Target: Apoptosis, NF-κB, Lipoxygenase, Caspase
d-Epigalbacin
Cat.No: TN7121
Synonym: (-)-Zuonin A,表加巴辛
Target: JNK
Eclalbasaponin I
Cat.No: TN1600
Synonym:
Target: Others
Albatrelin G
Cat.No: TN3371
Synonym:
Target: Others
Albanol B
Cat.No: T75602
Synonym:
Target:
Albaspidin AA
Cat.No: T2S1115
Synonym:
Target: Antifection
Albaspidin
Cat.No: T29831
Synonym:
Target:
Albatrelin C
Cat.No: TN3370
Synonym:
Target: Others
Albatrelin A
Cat.No: TN3369
Synonym:
Target: Others
Albaspidin AP
Cat.No: TN1365
Synonym:
Target: Fatty Acid Synthase
Glucosinalbate
Cat.No: T13706
Synonym:
Target: Others
Glucosinalbate potassium
Cat.No: TN2212
Synonym: 白芥子钾盐,Sinalbin potassium salt
Target: Others
Kuwanon A
Cat.No: TQ0301
Synonym:
Target: NO Synthase
3-O-Caffeoylquinic acid methyl ester
Cat.No: TN1261
Synonym:
Target: Others
Benzoylalbiflorin
Cat.No: TN7027
Synonym: Paeonivayin,苯甲酰芍药内酯苷
Target: Others
Moracin C
Cat.No: TN1949
Synonym: 桑辛素 C,5-(6-羟基-2-苯并呋喃基)-2-(3-甲基-2-丁烯基)-1,3-苯二醇
Target: ROS, NO Synthase
Isodemethylwedelolactone
Cat.No: T5742
Synonym: 异去甲蟛蜞菊内酯,Isodemethylwedelolacton
Target: Others
Demethylwedelolactone
Cat.No: T5S0689
Synonym: 去甲蟛蜞菊内酯,去甲基蟛蜞内酯
Target: Serine Protease
Oxypaeoniflorin
Cat.No: T3773
Synonym: 氧化芍药苷,Oxypaeoniflora
Target: Others
3'-Geranyl-3-prenyl-2',4',5,7-tetrahydroxyflavone
Cat.No: TN1252
Synonym:
Target: Apoptosis
Betulinic acid
Cat.No: T2830
Synonym: 白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid
Target: Apoptosis, Mitophagy, NF-κB, HIV Protease, Topoisomerase, Endogenous Metabolite, Aminopeptidase, Autophagy
Mulberrofuran G
Cat.No: TN1956
Synonym:
Target: Phosphatase, HBV, Glucosidase
Moracin M
Cat.No: TN1950
Synonym:
Target: PDE
Ipalbine
Cat.No: T82054
Synonym:
Target:
Mulberrofuran B
Cat.No: T81742
Synonym:
Target:
Paeoniflorin sulfite
Cat.No: T38524
Synonym:
Target:
23-Hydroxybetulin
Cat.No: TN2814
Synonym:
Target: Others
Kuwanol C
Cat.No: TN4401
Synonym:
Target: Others
Kuwanol A
Cat.No: TN2453
Synonym:
Target: Others
1,2,6,7,8,9-Hexahydro-1,6,6-trimethyl-3,11-dioxanaphth[2,1-e]azulene-10,12-dione
Cat.No: T83479
Synonym:
Target:
Morusinol
Cat.No: TN1953
Synonym: 桑根皮醇,桑树醇
Target: ERK, MEK, Autophagy, Ras
Cat. No. Product Name Species Expression System
TMPH-03193 Alba Protein, Pyrococcus furiosus, Recombinant (His & SUMO)

DNA/RNA-binding protein Alba

Pyrococcus furiosus E. coli
Binds double-stranded DNA tightly but without sequence specificity. It is distributed uniformly and abundantly on the chromosome, suggesting a role in chromatin architecture. However, it does not significantly compact DNA. Binds rRNA and mRNA in vivo. May play a role in maintaining the structural and functional stability of RNA, and, perhaps, ribosomes. Alba Protein, Pyrococcus furiosus, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molec...
TMPY-03962 AFM Protein, Human, Recombinant (His)

afamin,ALBA,ALB2,ALF

Human HEK293 Cells
Afamin is an 87 kDa glycoprotein with five predicted N-glycosylation sites. Afamin's glycan abundance contributes to conformational and chemical inhomogeneity presenting great challenges for molecular structure determination. Afamin, a human plasma glycoprotein and putative transporter of hydrophobic molecules, has been shown to act as extracellular chaperone for poorly soluble, acylated Wnt proteins, forming a stable, soluble complex with functioning Wnt proteins. The 2.1-Å crystal structure of...
TMPH-03197 Que a 1 Protein, Quercus alba, Recombinant (B2M & His)

Quercus alba E. coli
N/A. Que a 1 Protein, Quercus alba, Recombinant (B2M & His) is expressed in E. coli expression system with N-6xHis-B2M tag. The predicted molecular weight is 19.4 kDa and the accession number is P85126.
TMPY-04523 Influenza A H1N1 (A/Albany/12/1951) Hemagglutinin/HA1 Protein (His)

Harvey rat sarcoma viral oncogene homolog

H1N1 HEK293 Cells
Influenza A H1N1 (A/Albany/12/1951) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.2 kDa and the accession number is A4U7A6.1.
TMPY-04886 Influenza A H1N1 (A/Albany/12/1951) Hemagglutinin/HA Protein (His)

Harvey rat sarcoma viral oncogene homolog

H1N1 Baculovirus Insect Cells
Influenza A H1N1 (A/Albany/12/1951) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59.3 kDa and the accession number is A4U7A6.
TMPY-05006 Alpha Lactalbumin/LALBA Protein, Human, Recombinant (His)

α Lactalbumin/LALBA,LYZL7,lactalbumin alpha,lactalb...

Human HEK293 Cells
Alpha Lactalbumin/LALBA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 15.5 kDa and the accession number is A0A080YV01.
TMPY-00187 Alpha Lactalbumin/LALBA Protein, Human, Recombinant (mFc)

LYZL7,lactalbumin α,lactalbumin alpha,α Lactalbumin/LALB...

Human HEK293 Cells
Alpha Lactalbumin/LALBA Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 40.5 kDa and the accession number is A0A080YV01.
TMPY-05938 Influenza A H3N2 (A/Albany/18/1968) Neuraminidase/NA Protein (His)

NA Protein

H3N2 HEK293 Cells
Influenza A H3N2 (A/Albany/18/1968) Neuraminidase/NA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 50.8 kDa and the accession number is A4JZ31.

重组蛋白

Alba Protein, Pyrococcus furiosus, Recombinant (His & SUMO)
Cat.No: TMPH-03193
Species: Pyrococcus furiosus
Expression System: E. coli
AFM Protein, Human, Recombinant (His)
Cat.No: TMPY-03962
Species: Human
Expression System: HEK293 Cells
Que a 1 Protein, Quercus alba, Recombinant (B2M & His)
Cat.No: TMPH-03197
Species: Quercus alba
Expression System: E. coli
Influenza A H1N1 (A/Albany/12/1951) Hemagglutinin/HA1 Protein (His)
Cat.No: TMPY-04523
Species: H1N1
Expression System: HEK293 Cells
Influenza A H1N1 (A/Albany/12/1951) Hemagglutinin/HA Protein (His)
Cat.No: TMPY-04886
Species: H1N1
Expression System: Baculovirus Insect Cells
Alpha Lactalbumin/LALBA Protein, Human, Recombinant (His)
Cat.No: TMPY-05006
Species: Human
Expression System: HEK293 Cells
Alpha Lactalbumin/LALBA Protein, Human, Recombinant (mFc)
Cat.No: TMPY-00187
Species: Human
Expression System: HEK293 Cells
Influenza A H3N2 (A/Albany/18/1968) Neuraminidase/NA Protein (His)
Cat.No: TMPY-05938
Species: H3N2
Expression System: HEK293 Cells
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