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69

抑制剂 & 化合物

5

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T25480	H 256 H-256,H256,Pro-thr-glu-phe-CH2NH-phe-arg-glu
	H 256 is a pepsin heptapeptide inhibitor.
T34189	PTZ-256 phenothiazine derivative,PTZ256
	PTZ-256 is a phenothiazine derivative with chemical name: 3-(10H-phenothiazin-10-yl)propane-1-amine. PTZ-256 has molecule weight 256, therefore, we call it as PTZ-256.
T35249	YG 19-256
	YG 19-256 is a biochemical.
TF0032	NDSB-256
	NDSB-256 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 TF0032，CAS号为 81239-45-4。
T32739	Libexin Lomapect,Toparten,HK 256,HK-256,Prenoxdiazine hydrochloride,HK256
	Libexin is a cough suppressant.
T30233	AWD-G256
	AWD-G256 是一种抗心律失常物质，AWD-G256 对卒中量、肺压和全身血压没有显著影响。
T6798	Tretazicar 5-Aziridino-2,4-dinitrobenzamide,CB1954,NSC 115829	DNA Alkylator/Crosslinker; DNA Alkylation	DNA Damage/DNA Repair
	Tretazicar (NSC-115829) 是一种抗肿瘤前药，由 NAD(P)H 醌氧化还原酶 2 激活。它在酶促活化后生成细胞毒性双功能烷基剂，可以形成 DNA-DNA 链间交联。
T30233L	G256 HCl（134867-97-3 Free base)

TP1238L	ACTH 1-14 acetate(25696-21-3 free base) Adrenocorticotropic Hormone Fragment 1-14 acetate	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	ACTH 1-14 acetate(25696-21-3 free base) (Adrenocorticotropic Hormone Fragment 1-14 acetate) 是促肾上腺皮质激素的片段，可调节皮质醇和雄激素的产生。促肾上腺皮质激素 (ACTH)，也称为促肾上腺皮质激素，由垂体前叶产生和分泌。作为对生物应激的反应，ACTH 是下丘脑-垂体-肾上腺轴的重要组成部分。
T8943	AKOS025692697	Others	Others
	AKOS025692697 是一种生化产品。
T6054	GSK256066	PDE	Metabolism
	GSK256066 是高亲和力的、选择性的PDE4抑制剂，IC50=3.2 pM，被开发用于慢性阻塞性肺病的研究。
T36569	KR-32568	Sodium Channel	Membrane transporter/Ion channel
	KR-32568是一种钠/氢交换器1（NHE-1）抑制剂（IC50：230 nM）。KR-32568具有强大的心脏保护作用。当使用浓度为10μM 时，它能在离体的缺血大鼠心脏模型中恢复心脏收缩功能。KR-32568（0.3mg/kg）在缺血和再灌注损伤的大鼠模型中减少了心肌梗死的大小。
T15430	GSK2256294A GSK 2256294	Others; Epoxide Hydrolase	Metabolism; Others
	GSK2256294A (GSK 2256294) 是重组人、大鼠和小鼠 sEH 的有效特异性抑制剂，IC50 分别为 27 pM、61 pM 和 189 pM。
T15806	LY2562175	FXR; Autophagy	Autophagy; Metabolism
	LY2562175 是一种有效的选择性 FXR 激动剂，其EC50值为 193 nM。
T2281	GSK2256098 GSK 2256098,GSK-2256098,GTPL7939	Apoptosis; FAK	Angiogenesis; Apoptosis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	GSK2256098 (GTPL7939) 是一种选择性FAK 激酶抑制剂，抑制胰腺癌细胞的生长和存活。
T8562	A 425619 1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA	TRP/TRPV Channel	Membrane transporter/Ion channel
	A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) 是一种有效的 TRPV1 拮抗剂。
T13169	TM-25659	Others	Others
	TM-25659是一种具有 PDZ 结合图案的转录协同激活剂（TAZ）的调节剂，具有抗骨质疏松和抗肥胖的活性。
T15432	GSK256073	GPR; Others	Endocrinology/Hormones; GPCR/G Protein; Others
	GSK256073 是一种口服有活性的GPR109A 选择性激动剂，也是一种持久的人HCA2激动剂(pEC50:7.5) 。它能够减少脂降解，而显著改善葡萄糖稳态，对 2 型糖尿病和血脂异常具有潜在的研究价值。
T5428	BIX 02565	LRRK2; S6 Kinase	Autophagy; MAPK; PI3K/Akt/mTOR signaling
	BIX 02565 是核糖体 S6 激酶 2 (RSK2) 抑制剂，IC50为 1.1 nM。
T72073	AKOS037652256
	AKOS037652256可作为 TRPML 调节剂，可用于治疗如溶酶体积存病、肌肉萎缩症、与年龄相关的常见神经退行性疾病、氧化应激或活性氧(ROS)相关疾病以及衰老等与 TRPML 活性相关的疾病。
T71181	GSK256073 Tris
	GSK256073 is an agonist of G-protein coupled receptor 109A (GPR109A). It acts by reducing serum glucose in subjects with type 2 diabetes mellitus.
TP1465	IRL-1620 TFA (142569-99-1 free base) IRL-1620 TFA
	IRL-1620 (TFA) is a potent selective endothelin receptor B (ETB) agonist with a Ki value of 16pm.
T69811	AGI25696
	AGI-25696 is a MATA2 inhibitor that are useful as therapeutic agents for treating malignancies. AGI-25696 showed in vivo activity in MTAP null tumors. Note: The correct structure of AGI-25696 is CAS#2201065-84-9. Many vendors mistakenly listed CAS#2201066-35-3 as its AGI25696. J. Med. Chem. 2021, 64, 8, 4430–4449 published AGI25696 structure (it is CAS#2201065-84-9).
T68927	AY 25674
	AY 25674 is a drug with antiallergic properties which has been shown to inhibit passive anaphylaxis in rat.
T30551	BN 52256 BN52256,BN-52256
	BN 52256 helps reduce arrhythmias.
T27464	GSK2565363C
	GSK2565363C is a betulin derivative wth antitumor activity.
T25249	CID-2562757 CID 2562757
	CID-2562757 is an antagonist of α6β2 specific nAChR.
T15361	FW1256	Others	Others
	FW1256 is a phenyl analog. It also a slow-releasing hydrogen sulfide (H2S) donor. FW1256 inhibits NF-κB activity and causes cell apoptosis. FW1256 shows potent anti-inflammatory effects. It also has the potential for cancer and cardiovascular disease trea
T68263	MDL-72567
	MDL-72567 is a dihydropyridine calcium antagonist that causes vasodilation and direct sinus bradycardia.
T70005	LY3325656
	LY3325656 is a GPR142 agonist suitable for clinical testing in human. LY3325656 demonstrated anti-diabetic benefits in pre-clinical studies and ADME/PK properties suitable for human dosing. LY3325656 is the first GPR142 agonist molecule advancing to phase 1 clinic trials for the treatment of Type 2 diabetes.
T36533	SCH 725674
	SCH 725674 is an antifungal macrolide originally isolated from Aspergillus. It inhibits the growth of S. cerevisiae and C. albicans in vitro (MICs = 8 and 32 μg/ml, respectively).
T23690	AI 3-25614 AI-3-25614,AI3-25614
	AI 3-25614 is a pesticide.
T73372	GNE-2256
	GNE-2256 (molecule 19) 是一种具有口服活性的IRAK4(白介素 1 受体关联激酶 4) 抑制剂 (IRAK4Ki=1.4 nM ; IL-6IC50=190 nM)。
T23873	CEP-2563 CEP 2563
	CEP-2563 is a prodrug of CEP-751. It also used as an antitumor agent, inhibiting protein kinases.
T71547	MDL-25637
	MDL-25637 is a glucosidase inhibitor.
T27906	LY 25648 LY-25648,LY25648
	LY 25648 is an antagonist of leukotriene B4.
T16095	MK-4256	Others	Others
	MK-4256 is an effective and selective SSTR3 antagonist (IC50s: 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively).
T12423	PF-06256142	Others	Others
	PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).
T10259	AGI-25696	Others; Methionine Adenosyltransferase (MAT)	Chromatin/Epigenetic; Others
	AGI-25696 是甲硫氨酸腺苷转移酶 2A (MATA2) 的抑制剂。 AGI-25696 在体内阻断 MTAP 缺失肿瘤的生长，可用于癌症治疗的研究。
T31642	ENT 25642 ENT 25,642,ENT25642,AC 35,217,BRN 2168785,CL-35217,ENT-25642,CL-35217;AC 35,217
	ENT 25642 is a bio-active chemical. Detailed information has not been published.
T29143	VU6004256 VU 6004256,VU-6004256
	VU6004256 is a selective positive allosteric modulator (PAM) of muscarinic receptor M1.
T28102	MRS2567 MRS-2567,MRS 2567
	MRS2567 is a potent P2Y6 nucleotide receptors antagonists.
T70995	GSK-256066
	GSK-256066 is a PDE4 inhibitor.
T31641	ENT 25641 AC 28,865 AI3-25641,Benzenesulfonamide, p-hydroxy-, dimethyl phosphate,American cyanamid CL-28865,ENT25641,ENT-25641
	ENT 25641 is a bio-active chemical. Detailed information has not been published.
T39522	HTL22562
	HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.
T24037	EPZ-025654 HCl EPZ 025654,EPZ-025654,GSK35336023,EPZ025654,GSK-35336023,GSK 35336023
	EPZ-025654 is an effective and selective inhibitor of arginine methyltransferase CARM1.
T29760	AI 3-25610
	AI 3-25610 is a bioactive chemical.
T16511	PF2562	Dopamine Receptor	GPCR/G Protein; Neuroscience
	PF2562 is a dopamine D1 ligand. It is used as a dopamine D1 agonist or partial agonist. PF2562 binds to human D1 receptor (Ki: 113 nM). PF2562 shows activity against human D1 cAMP (EC50: 568 nM in HTRF assay).
T70724	GSK-2256098 HCl
	GSK-2256098 HCl is a focal adhesion kinase-1 (FAK) inhibitor with potential antiangiogenic and antineoplastic activities.
T71653	GS-9256	HCV Protease	Microbiology/Virology; Proteases/Proteasome
	GS-9256为选择性HCV NS3蛋白酶抑制剂，展现出优良的药代动力学特性及抗病毒活性。

化合物

Cat.No: T25480

Synonym: H-256,H256,Pro-thr-glu-phe-CH2NH-phe-arg-glu

Cat.No: T34189

Synonym: phenothiazine derivative,PTZ256

Cat.No: T35249

Cat.No: TF0032

Cat.No: T32739

Synonym: Lomapect,Toparten,HK 256,HK-256,Prenoxdiazine hydrochloride,HK256

Cat.No: T30233

Cat.No: T6798

Synonym: 5-Aziridino-2,4-dinitrobenzamide,CB1954,NSC 115829

Target: DNA Alkylator/Crosslinker, DNA Alkylation

G256 HCl（134867-97-3 Free base)

Cat.No: T30233L

ACTH 1-14 acetate(25696-21-3 free base)

Cat.No: TP1238L

Synonym: Adrenocorticotropic Hormone Fragment 1-14 acetate

Target: Adrenergic Receptor

Cat.No: T8943

Target: Others

Cat.No: T6054

Target: PDE

Cat.No: T36569

Target: Sodium Channel

Cat.No: T15430

Synonym: GSK 2256294

Target: Others, Epoxide Hydrolase

Cat.No: T15806

Target: FXR, Autophagy

Cat.No: T2281

Synonym: GSK 2256098,GSK-2256098,GTPL7939

Target: Apoptosis, FAK

Cat.No: T8562

Synonym: 1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA

Target: TRP/TRPV Channel

Cat.No: T13169

Target: Others

Cat.No: T15432

Target: GPR, Others

Cat.No: T5428

Target: LRRK2, S6 Kinase

Cat.No: T72073

Cat.No: T71181

IRL-1620 TFA (142569-99-1 free base)

Cat.No: TP1465

Synonym: IRL-1620 TFA

Cat.No: T69811

Cat.No: T68927

Cat.No: T30551

Synonym: BN52256,BN-52256

Cat.No: T27464

Cat.No: T25249

Synonym: CID 2562757

Cat.No: T15361

Target: Others

Cat.No: T68263

Cat.No: T70005

Cat.No: T36533

Cat.No: T23690

Synonym: AI-3-25614,AI3-25614

Cat.No: T73372

Cat.No: T23873

Synonym: CEP 2563

Cat.No: T71547

Cat.No: T27906

Synonym: LY-25648,LY25648

Cat.No: T16095

Target: Others

Cat.No: T12423

Target: Others

Cat.No: T10259

Target: Others, Methionine Adenosyltransferase (MAT)

Cat.No: T31642

Synonym: ENT 25,642,ENT25642,AC 35,217,BRN 2168785,CL-35217,ENT-25642,CL-35217;AC 35,217

Cat.No: T29143

Synonym: VU 6004256,VU-6004256

Cat.No: T28102

Synonym: MRS-2567,MRS 2567

Cat.No: T70995

Cat.No: T31641

Synonym: AC 28,865 AI3-25641,Benzenesulfonamide, p-hydroxy-, dimethyl phosphate,American cyanamid CL-28865,ENT25641,ENT-25641

Cat.No: T39522

Cat.No: T24037

Synonym: EPZ 025654,EPZ-025654,GSK35336023,EPZ025654,GSK-35336023,GSK 35336023

Cat.No: T29760

Cat.No: T16511

Target: Dopamine Receptor

GSK-2256098 HCl

Cat.No: T70724

Cat.No: T71653

Target: HCV Protease

Cat. No.	Product Name	Target	Signaling Pathways
T6926	Palmitoylethanolamide Mackpeart DR 14V,帕米醇,N-palmitoylethanolamine,Loramine P 256,Impulsin,AM 3112,Palmidrol	Influenza Virus; Endogenous Metabolite; PPAR	DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
	Palmitoylethanolamide (Impulsin) 是一种内源性脂肪酸酰胺。它有消炎药、降压药、神经保护剂和抗惊厥药的作用。在给药后，Palmitoylethanolamide 可抑制促炎介质从活化肥大细胞的释放。
T5802	Stearyl glycyrrhetinate	Antiviral; Antibacterial	Immunology/Inflammation; Microbiology/Virology
	Stearyl glycyrrhetinate 是甘草提取物中的主要成分之一，具有抗菌作用，对金黄色葡萄球菌菌株的 MIC 大于 256 mg/L。
T3S1955	7-Ethylcamptothecin	Others	Others
	7-Ethylcamptothecin 是一种喜树碱类似物。其中喜树碱是一种细胞毒性生物碱，从喜树中分离出得到，对 L1210 白血病和 Walker 256 癌肉瘤模型具有很强的抗肿瘤活性。
TN3450	Artanin	Antifection	Microbiology/Virology
	Artanin displays promising inhibition against both MSSA and MRSA with minimal inhibitory concentrations (MICs) of 8-64 ug/ml, but very weak against Gram-negative pathogen and yeast with MICs of 256 to ≥1024 ug/ml.
TN1165	(Rac)-Myrislignan 1-(3,4-dimethoxyphenyl)-2-(4-allly-2,6-dimethoxyphenoxy)propan-1-ol,rac-myrislignan,ALPHA-[1-[2,6-二甲氧基-4-(2-丙烯-1-基)苯氧基]乙基]-4-羟	Others	Others
	1-(3,4-Dimethoxyphenyl)-2-(4-allly-2,6-dimethoxyphenoxy)propan-1-ol shows anti-staphylococcal activity against a total of five multidrug-resistant (MDR) and methicillin-resistant Staphylococcus aureus strains and the minimum inhibitory concentrations (MIC

天然产物

Palmitoylethanolamide

Cat.No: T6926

Synonym: Mackpeart DR 14V,帕米醇,N-palmitoylethanolamine,Loramine P 256,Impulsin,AM 3112,Palmidrol

Target: Influenza Virus, Endogenous Metabolite, PPAR

Stearyl glycyrrhetinate

Cat.No: T5802

Target: Antiviral, Antibacterial

7-Ethylcamptothecin

Cat.No: T3S1955

Target: Others

Cat.No: TN3450

Target: Antifection

(Rac)-Myrislignan

Cat.No: TN1165

Synonym: 1-(3,4-dimethoxyphenyl)-2-(4-allly-2,6-dimethoxyphenoxy)propan-1-ol,rac-myrislignan,ALPHA-[1-[2,6-二甲氧基-4-(2-丙烯-1-基)苯氧基]乙基]-4-羟

Target: Others

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