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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T6231 Tebipenem Pivoxil

ME1211,Orapenem,替​比​培​南​匹​酯

Antibacterial; Antibiotic Microbiology/Virology
Tebipenem Pivoxil (Orapenem) 是一种碳青霉烯类新型口服抗生素。
T1491 Atovaquone

Atavaquone,阿托伐醌

Others; P450; Dehydrogenase; Antibiotic; Parasite Metabolism; Microbiology/Virology; Others
Atovaquone (Atavaquone) 是具有口服活性的选择性寄生虫线粒体细胞色素bc1复合物的抑制剂。它抑制人类和P. falciparum 细胞色素bc1活性,IC50值分别为 460 nM 和 2.0 nM。它有抗疟作用,有潜力用于疟疾、弓形体病、肺孢子虫肺炎和巴贝斯虫病的相关研究。
T23133 Pentamidine

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine 是抗微生物剂,会干扰 DNA 的生物合成。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它可用于冈比亚锥虫病,抗锑利什曼病和卡氏肺孢子虫肺炎的研究,有抗肿瘤活性,抗菌活性。
T4267 Tulathromycin A

CP 472295,Draxxin,Tulathromycin,托拉菌素 A

Antibacterial; Antibiotic Microbiology/Virology
Tulathromycin A (CP 472295) 是一种大环内酯类抗生素,靶向细菌核糖体抑制蛋白质合成 (IC50=0.26 µM),具有免疫调节作用。它可研究牛和猪的呼吸道疾病。
T4201 Avibactam sodium

阿维巴坦,AVE-1330A,阿维巴坦钠,NXL-104

Antibacterial; Antibiotic Microbiology/Virology
Avibactam sodium (NXL-104) 是一种可逆的 β-内酰胺酶抑制剂,抑制 TEM-1,P99和KPC-2 β-内酰胺酶,IC50分别为8、80和38 nM。
T2691 Oritavancin diphosphate

奥利万星二磷酸盐,LY333328 diphosphate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Oritavancin diphosphate (LY333328 diphosphate) 是一种新型半合成的糖肽抗生素, 可研究革兰氏阳性菌感染。
T5189 Omadacycline

PTK 0796,Amadacycline

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Omadacycline (Amadacycline) 是一种具有口服活性的氨基甲基环素抗菌剂,是四环素类抗生素。它与 30S 核糖体亚基结合,抑制细菌蛋白质合成。它可用于研究急性细菌性皮肤和皮肤结构感染,感染性肺炎和尿路感染。
T1654 Pentamidine isethionate

Pentamidine isethionate salt,Pentamidine diisethionate,喷他脒羟乙磺酸盐

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine isethionate (Pentamidine diisethionate) 是抗微生物剂,会干扰 DNA 的生物合成。它抑制寄生虫Leishmania infantum,IC50为 2.5 μM。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它有抗肿瘤和抗菌活性。
T7804 Garenoxacin mesylate hydrate

Garenoxacin mesylate [USAN],加雷沙星甲磺酸盐,BMS284756 (Mesylate hydrate)

Antibacterial Microbiology/Virology
Garenoxacin mesylate hydrate (Garenoxacin mesylate [USAN]) 是一种新型口服 des-fluoro(6) 喹诺酮,具有强抗菌活性,抗呼吸道病原体。
T23132 Pentamidine dihydrochloride

喷他脒二盐酸盐,MP-601205 dihydrochloride

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine dihydrochloride (MP-601205 dihydrochloride) 是一种抗微生物剂,会干扰 DNA 的生物合成。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它可用于冈比亚锥虫病,抗锑利什曼病和卡氏肺孢子虫肺炎的研究,有抗肿瘤活性,抗菌活性。
T0331 Moxifloxacin hydrochloride

盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Moxifloxacin hydrochloride (BAY12-8039 HCl) 是一种口服有效的 8-甲氧基喹诺酮类抗菌药物,可研究感染性肺炎,急性细菌性鼻窦炎和慢性支气管炎的急性细菌性加重。
T7179 Garenoxacin

BMS284756,加雷沙星

Antibacterial Microbiology/Virology
Garenoxacin (BMS284756) 是一种新型的口服 des-fluoro(6) 喹诺酮,有抗菌活性,可抑制呼吸道病原体。
T79088 Chlamydia pneumoniae-IN-1

Chlamydia pneumoniae-IN-1 (compound 55),一种抗衣原体的苯并咪唑类化合物,对肺炎衣原体具有高度抑制作用,在10 μM 浓度下能够抑制99%的肺炎衣原体生长,并对宿主细胞的活力产生95%的抑制效果。此外,Chlamydia pneumoniae-IN-1 对CV-6菌株亦显示出明显的抗菌活性,其最小抑菌浓度(MIC)为12.6 μM。
T12242 Norvancomycin hydrochloride

Desmethyl-vancomycin hydrochloride,盐酸去甲万古霉素

Antibacterial Microbiology/Virology
Norvancomycin hydrochloride (Desmethyl-vancomycin hydrochloride) 可用于葡萄球菌所致的心内膜炎、骨髓炎、肺炎、败血症或软组织感染。
T11785 KT203

MAGL Metabolism
KT203 是一种具有选择性和高效性的 α/β 水解酶结构域 6 (ABHD6) 抑制剂,具有潜在的抗病毒和抗炎活性,可用于研究肺炎。
T17210 Vaborbactam

RPX7009

Antibacterial Microbiology/Virology
Vaborbactam (RPX7009)是一种 β-内酰胺酶抑制剂,常与美罗培南共同作用来研究肺炎和 CRE 感染。
T22387 NSC 55655

5-[(2-nitrophenyl)methylidene]thiazolidine-2,4-dione

Others Others
NSC 55655 (5-[(2-Nitrophenyl)methylene]-2,4-thiazolidinedione) 具有抗菌和抗氧化活性,抑制 B. subtilis, S. aureus, K. pneumonia, E. coli, S. typhi ,A. niger 和 C. albicans 的增殖,可用于糖尿病。
T11815 Lanopepden

GSK 1322322,GSK-1322322B,GSK-1322322J

Antibiotic Microbiology/Virology
Lanopepden (GSK 1322322) 是一种有效的肽去甲酰酶抑制剂,抑制金黄色葡萄球菌,抑制 ATCC 29213 和 ATCC 25923 菌株,可用于研究肺炎、皮肤病和传染病。
T77125 Otilimab

GSK 3196165,MOR103

CSF-1R Tyrosine Kinase/Adaptors
Otilimab (GSK 3196165) 是一种人源化抗粒细胞-巨噬细胞集落刺激因子 (GM-CSF) 单克隆抗体。Otilimab 具有抗炎活性,通过阻断 GM-CSF 与其细胞表面受体的相互作用来调节 GM-CSF 的生物学功能,可用于研究治疗重症 COVID-19 肺炎。
T10987 Decarboxy Moxifloxacin

Others Others
Decarboxy Moxifloxacin 是一种莫西沙星的脱羧化合物。Moxifloxacin 是一种能够口服的 8-甲氧基喹诺酮类抗菌药物,可用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎。
T4553 Procaine penicillin G

普鲁卡因青霉素,Duphapen,Hydracillin,Hostacillin

Antibiotic Microbiology/Virology
Procaine penicillin G (Duphapen) 是一种抗生素,可用于治疗多种细菌感染。具体来说,它用于梅毒、炭疽、口腔感染、肺炎、白喉、蜂窝组织炎和动物咬伤。
T1492 Gemifloxacin mesylate

LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。
T39933 Bexotegrast

PLN-74809

Integrin Cytoskeletal Signaling
Bexotegrast (PLN-74809)是一种具有口服活性和强效性的 αvβ6和αvβ1 整合素抑制剂,具有抗纤维化作用,抑制 αvβ6 和 αvβ1 诱导的 TGF-β 激活,可用于研究特发性肺纤维化(IPF)和非特异性间质性肺炎(NSIP)。
T11836 Lefamulin acetate

BC-3781 acetate,醋酸来法莫林

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Lefamulin acetate (BC-3781 acetate) 是具有口服活性的抗生素。它是用于人体细菌感染的全身研究的半合成截短侧耳素。它与 50S 细菌核糖体的肽基转移酶peptidyl transferase 中心结合抑制蛋白质合成,并阻止了转移RNA 与肽转移的结合。
T1283 Clinafloxacin

克林沙星,PD 127391,CI-960,AM-1091

Antibacterial; Antibiotic Microbiology/Virology
Clinafloxacin (CI-960) 是一种高效广谱氟喹诺酮类抗生素,抑制革兰氏阳性、革兰氏阴性和厌氧病原体。它对金黄色葡萄球菌的 DNA 促旋酶和拓扑异构酶 IV 有抑制作用,IC50值分别为 0.92 µg/ml 和 1.62 µg/ml。
T16428 Pafuramidine

DB289

Others Others
Pafuramidine is an orally bioavailable prodrug of furamidine. It has activity against Pneumocystis pneumonia (IC50 value: 4.5 nM)
T1293L Gatifloxacin sesquihydrate

Gatifloxacin

Gatifloxacin sesquihydrate, a bacterial DNA gyrase inhibitor, is used to treat tuberculosis and pneumonia.
T32891 l-Primaquine

BRN0019337,BRN-0019337,BRN 0019337

l-Primaquine is used to treat and prevent malaria and to treat Pneumocystis pneumonia.
T19198 Atovaquone-d4

阿托伐醌D4

Others Others
Atovaquone D4 is the deuterium-labeled Atovaquone. Atovaquone is a medication used to treat or prevent pneumocystis babesia, malaria, toxoplasmosis, and pneumonia.
T38586 Grepafloxacin

dl-Grepafloxacin,OPC-17116

Grepafloxacin (OPC-17116) is a fluoroquinolone antibiotic that is administered orally. It possesses strong efficacy against community-acquired respiratory pathogens, notably Streptococcus pneumonia. Grepafloxacin exhibits excellent tissue penetration and demonstrates a promising pharmacodynamic profile.
TP2139 AMY-101

Cp40

Others Others
AMY-101 TFA (Cp40 TFA) is a peptidic inhibitor of the central complement component C3 (KD: 0.5 nM). It shows a favorable anti-inflammatory activity in models with COVID-19 severe pneumonia with systemic hyper inflammation.
T28997 TP-271

TP271

TP-271, a tetracyclines antibiotic, is used potentially for the treatment of community-acquired bacterial pneumonia (CABP).
T36993 Moxifloxacin N-Sulfate (sodium salt)

Moxifloxacin N-sulfate is a metabolite of moxifloxacin . Moxifloxacin is a fluoroquinolone antibiotic. Formulations containing moxifloxacin have been used in the treatment of bacterial infections, including sinusitis, chronic bronchitis, and pneumonia.
T23622 Acorafloxacin HCl

JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl

Acorafloxacin is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and skin structure infections and community-acquired pneumonia.
T10420 Avarofloxacin

JNJ-Q2

Others Others
Avarofloxacin (JNJ-Q2) is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and community-acquired pneumonia and skin structure infections.
T19678 Cefaloridine

Cephaloridine,Sch 11527

Cefaloridine is a first-generation semisynthetic derivative of cephalosporin C. It is unique among cephalosporins in that it exists as a zwitterion. Cephaloridine was very effective to cure pneumococcal pneumonia. It has a high clinical and bacteriologica
TP2139L AMY-101 TFA

Cp40 TFA

Others Others
AMY-101 TFA (Cp40 TFA) is a peptidic inhibitor of the central complement component C3 (KD: 0.5 nM). It shows a favorable anti-inflammatory activity in models with COVID-19 severe pneumonia with systemic hyper inflammation.
T39862 Trimethoprim lactate

Trimethoprim lactic is a bacteriostatic antibiotic and an orally active dihydrofolate reductase inhibitor. Trimethoprim lactic is active against a wide range of Gram-positive and Gram-negative aerobic bacteria . Trimethoprim lactic has the potential for urinary tract infections, Shigellosis and Pneumocystis pneumonia treatment.
T9931 meplazumab

Others Others
meplazumab 是一种人源化抗 CD147 抗体,作为 COVID-19 肺炎患者的附加疗法。
T61123 Antibacterial agent 111

Antibacterial agent 111 (Compound 3) exhibits potent antibacterial activity against B. cereus and K. pneumonia, with MIC values of 3.90 μg/mL and 0.49 μg/mL, respectively. It achieves this antibacterial effect by strongly binding to specific residues of tyrosyl-tRNA synthetase [1].
T60569 Sulfametrole

Sulfametrole 是具有口服活性的抗菌剂,可用于传染病相关的研究,如艾滋病毒、严重肺炎和尿路感染。
T40971 Dehydroandrographolide succinate potassium sodium salt

Dehydroandrographolide succinate (potassium sodium salt), derived from the herbal medicine Andrographis paniculata (Burm f) Nees, is a versatile compound highly utilized for the treatment of viral pneumonia and viral upper respiratory tract infections due to its potent immunostimulatory, anti-infective, and anti-inflammatory properties.
T77174 Efmarodocokin alfa

Efmarodocokin alfa为人IL-22与IgG4可结晶片段的融合蛋白,具有激活IL-22信号的功能。该化学物质主要用于重症COVID-19肺炎的研究。
T60238 Acloproxalap

Acloproxalap 是一种基于喹啉的醛清除剂,可用于研究有毒醛积累的疾病,如眼部、皮肤等炎症性疾病,肺炎等呼吸系统疾病,器官疾病以及病毒感染相关性综合症等。
T70642 Lanopepden camsylate

Lanopepden, also known as GSK-1322322 or GSK-322, is a potent and selective peptide deformylase inhibitor with good in vitro activity against bacteria associated with community-acquired pneumonia and skin infections. GSK1322322 had bactericidal activity against S. pneumoniae, H. influenzae, S. pyogenes, and S. aureus, demonstrating a ≥ 3-log(10) decrease in the number of CFU/ml at 4× MIC within 24 h in 29 of the 33 strains tested. GSK1322322 represents a valuable alternative therapy for the trea...
T71266 Omadacycline HCl

Omadacycline, also known as PTK 0796 and Amadacyclin, is a novel first-in-class aminomethylcycline with potent activity against important skin and pneumonia pathogens, including community-acquired methicillin-resistant Staphylococcus aureus (MRSA), β-hemolytic streptococci, penicillin-resistant Streptococcus pneumoniae, Haemophilus influenzae, and Legionella. Omadacycline is active against strains expressing the two main forms of tetracycline resistance (efflux and ribosomal protection). The pri...
T76320 FIZZ-1 (32-51) (mouse)

FIZZ-1 (32-51) (mouse) 是一种富含半胱氨酸的分泌性蛋白,主要在过敏性气道炎症中被巨噬细胞、支气管上皮细胞及II型肺泡上皮细胞高度表达,具有对肺成纤维细胞的抗凋亡功能,广泛应用于过敏性肺炎的研究领域。
T74821 Nemonoxacin

Nemonoxacin (TG-873870) 是一种口服有效的广谱抗生素,对多种葡萄球菌、链球菌、肠球菌、淋病奈瑟菌和流感嗜血杆菌显示出强效的抑制活性。适用于研究细菌感染和社区获得性肺炎。
T37283 1-Palmitoyl Lysophosphatidic Acid (sodium salt)

1-Palmitoyl lysophosphatidic acid (1-Palmitoyl LPA) is a LPA analog containing palmitic acid at the sn-1 position. LPA binds to one of five different G protein-coupled receptors (GPCRs) to mediate a variety of biological responses including cell proliferation, smooth muscle contraction, platelet aggregation, neurite retraction, and cell motility. In addition to playing a role in the aforementioned biological responses, 1-palmitoyl LPA enhances the action of β-lactam antibiotics (ampicillin, pipe...
T76990 Suvratoxumab

Suvratoxumab (MEDI4893) 是一种长效且具有亲和力高的人源化抗 α-毒素单克隆抗体(IgG1κ 型)。Suvratoxumab 能有效中和 α-毒素 (一种关键的金黄色葡萄球菌毒力因子)。Suvratoxumab 可提高免疫功能低下的小鼠肺炎模型的存活率并减少肺损伤。Suvratoxumab 还可增强Vancomycin 或Linezolid 的抗菌活性。

化合物

Tebipenem Pivoxil
Cat.No: T6231
Synonym: ME1211,Orapenem,替​比​培​南​匹​酯
Target: Antibacterial, Antibiotic
Atovaquone
Cat.No: T1491
Synonym: Atavaquone,阿托伐醌
Target: Others, P450, Dehydrogenase, Antibiotic, Parasite
Pentamidine
Cat.No: T23133
Synonym:
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Tulathromycin A
Cat.No: T4267
Synonym: CP 472295,Draxxin,Tulathromycin,托拉菌素 A
Target: Antibacterial, Antibiotic
Avibactam sodium
Cat.No: T4201
Synonym: 阿维巴坦,AVE-1330A,阿维巴坦钠,NXL-104
Target: Antibacterial, Antibiotic
Oritavancin diphosphate
Cat.No: T2691
Synonym: 奥利万星二磷酸盐,LY333328 diphosphate
Target: Others, Antibacterial, Antibiotic
Omadacycline
Cat.No: T5189
Synonym: PTK 0796,Amadacycline
Target: ribosome, Antibacterial, Antibiotic
Pentamidine isethionate
Cat.No: T1654
Synonym: Pentamidine isethionate salt,Pentamidine diisethionate,喷他脒羟乙磺酸盐
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Garenoxacin mesylate hydrate
Cat.No: T7804
Synonym: Garenoxacin mesylate [USAN],加雷沙星甲磺酸盐,BMS284756 (Mesylate hydrate)
Target: Antibacterial
Pentamidine dihydrochloride
Cat.No: T23132
Synonym: 喷他脒二盐酸盐,MP-601205 dihydrochloride
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Moxifloxacin hydrochloride
Cat.No: T0331
Synonym: 盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl
Target: Topoisomerase, Antibacterial, Antibiotic
Garenoxacin
Cat.No: T7179
Synonym: BMS284756,加雷沙星
Target: Antibacterial
Chlamydia pneumoniae-IN-1
Cat.No: T79088
Synonym:
Target:
Norvancomycin hydrochloride
Cat.No: T12242
Synonym: Desmethyl-vancomycin hydrochloride,盐酸去甲万古霉素
Target: Antibacterial
KT203
Cat.No: T11785
Synonym:
Target: MAGL
Vaborbactam
Cat.No: T17210
Synonym: RPX7009
Target: Antibacterial
NSC 55655
Cat.No: T22387
Synonym: 5-[(2-nitrophenyl)methylidene]thiazolidine-2,4-dione
Target: Others
Lanopepden
Cat.No: T11815
Synonym: GSK 1322322,GSK-1322322B,GSK-1322322J
Target: Antibiotic
Otilimab
Cat.No: T77125
Synonym: GSK 3196165,MOR103
Target: CSF-1R
Decarboxy Moxifloxacin
Cat.No: T10987
Synonym:
Target: Others
Procaine penicillin G
Cat.No: T4553
Synonym: 普鲁卡因青霉素,Duphapen,Hydracillin,Hostacillin
Target: Antibiotic
Gemifloxacin mesylate
Cat.No: T1492
Synonym: LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate
Target: DNA gyrase, Topoisomerase, Antibacterial
Bexotegrast
Cat.No: T39933
Synonym: PLN-74809
Target: Integrin
Lefamulin acetate
Cat.No: T11836
Synonym: BC-3781 acetate,醋酸来法莫林
Target: ribosome, Antibacterial, Antibiotic
Clinafloxacin
Cat.No: T1283
Synonym: 克林沙星,PD 127391,CI-960,AM-1091
Target: Antibacterial, Antibiotic
Pafuramidine
Cat.No: T16428
Synonym: DB289
Target: Others
Gatifloxacin sesquihydrate
Cat.No: T1293L
Synonym: Gatifloxacin
Target:
l-Primaquine
Cat.No: T32891
Synonym: BRN0019337,BRN-0019337,BRN 0019337
Target:
Atovaquone-d4
Cat.No: T19198
Synonym: 阿托伐醌D4
Target: Others
Grepafloxacin
Cat.No: T38586
Synonym: dl-Grepafloxacin,OPC-17116
Target:
AMY-101
Cat.No: TP2139
Synonym: Cp40
Target: Others
TP-271
Cat.No: T28997
Synonym: TP271
Target:
Moxifloxacin N-Sulfate (sodium salt)
Cat.No: T36993
Synonym:
Target:
Acorafloxacin HCl
Cat.No: T23622
Synonym: JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl
Target:
Avarofloxacin
Cat.No: T10420
Synonym: JNJ-Q2
Target: Others
Cefaloridine
Cat.No: T19678
Synonym: Cephaloridine,Sch 11527
Target:
AMY-101 TFA
Cat.No: TP2139L
Synonym: Cp40 TFA
Target: Others
Trimethoprim lactate
Cat.No: T39862
Synonym:
Target:
meplazumab
Cat.No: T9931
Synonym:
Target: Others
Antibacterial agent 111
Cat.No: T61123
Synonym:
Target:
Sulfametrole
Cat.No: T60569
Synonym:
Target:
Dehydroandrographolide succinate potassium sodium salt
Cat.No: T40971
Synonym:
Target:
Efmarodocokin alfa
Cat.No: T77174
Synonym:
Target:
Acloproxalap
Cat.No: T60238
Synonym:
Target:
Lanopepden camsylate
Cat.No: T70642
Synonym:
Target:
Omadacycline HCl
Cat.No: T71266
Synonym:
Target:
FIZZ-1 (32-51) (mouse)
Cat.No: T76320
Synonym:
Target:
Nemonoxacin
Cat.No: T74821
Synonym:
Target:
1-Palmitoyl Lysophosphatidic Acid (sodium salt)
Cat.No: T37283
Synonym:
Target:
Suvratoxumab
Cat.No: T76990
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3381 Lysionotin

岩豆素

Others Others
Lysionotin (Nevadensin) 是一种类黄酮,分离自黄花草药中。它可抑制 α-Toxin (一种成孔蛋白) 的表达,并在体内和体外针对金黄色葡萄球菌显示出显著的保护作用。它可用于研究由金黄色葡萄球菌引起的肺炎。
T37101 1-Hydroxyanthraquinone

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
1-Hydroxyanthraquinone 是口服有效的天然产物,来源于植物 Tabebuia avellanedae,显示出致癌活性。
T8065 Tiamulin

Thiamutilin,泰妙菌素

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Tiamulin (Thiamutilin) 是一类二萜,广泛用于控制猪的传染疾病,包括猪痢疾和地方性肺炎等。
T0793 Kanamycin sulfate

硫酸卡那霉素,Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Kanamycin sulfate (Kanamycin monosulfate) 是氨基糖苷类杀菌抗生素,它通过与细菌30S 核糖体结合起作用。
T3907 Tenuigenin

Senegenin,Senegin,远志皂苷元

NF-κB; Caspase; Antibacterial Apoptosis; Microbiology/Virology; NF-κB; Proteases/Proteasome
Tenuigenin (Senegenin) 是从中草药远志根中分离出来的主要活性成分,用于中药,具有抗氧化和抗炎活性。它抑制 NF-κB 活化,预防金黄色葡萄球菌诱导的肺炎。
T1262 Tazobactam

Tazobactamum,Tazobactam acid,他唑巴坦酸,YTR-830H,CL-298741,他唑巴坦

Antibacterial; Antibiotic Microbiology/Virology
Tazobactam (YTR-830H) acid 是一种具有抗菌活性的β-内酰胺酶抑制剂。
T1153 Trimethoprim

NIH 204,BW 56-72,甲氧苄啶,NSC-106568

DHFR; DNA/RNA Synthesis; Antifolate; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Trimethoprim (NSC-106568) 是抑菌抗生素,也是具有口服活性的二氢叶酸还原酶抑制剂。它对多种革兰氏阳性和革兰氏阴性需氧细菌具有活性,可用于尿路感染,肺孢子菌肺炎和志贺氏菌病的研究。
T0971 Dirithromycin

Dirithromycinum,地红霉素,ASE 136,LY237216,Diritromicina,Dirithromycine

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Dirithromycin (LY237216) 是一种红霉素衍生物,是一种具有口服活性的半合成大环内酯类抗生素。它用于治疗许多不同类型的细菌感染。
T2S0257 Dehydroandrographolide succinate

Others; Influenza Virus Microbiology/Virology; Others
Dehydroandrographolide succinate 是从中药穿心莲中提取的一种天然产物,具有免疫刺激、抗感染和抗炎作用,有潜力研究病毒性肺炎和病毒性上呼吸道感染。
T5041 Faropenem sodium

法罗培南,法罗培南钠

Antibacterial; Antibiotic Microbiology/Virology
Faropenem sodium 是一种口服生物可利用的青霉烯类抗生素,能有效杀灭结核分枝杆菌,治疗结核病和社区获得性肺炎。
TN5284 Sodium Houttuyfonate

Houttuynin sodium bisulfite,新鱼腥草素钠

NF-κB; Antibacterial; Antifungal Microbiology/Virology; NF-κB
Sodium Houttuyfonate (Houttuynin sodium bisulfite) 是亚硫酸氢钠与鱼腥草结合而成的活性化合物,具有抗真菌、抗菌、抗炎和心血管保护活性,主要用于治疗化脓性皮肤感染、呼吸道感染,包括老年患者的肺炎和慢性支气管炎。
T38016 Hirsutide

Hirsutide is a cyclotetrapeptide fungal metabolite produced by the entomopathogenic fungus Hirsutella. It has antibacterial activity against C. pyogenes, S. aureus, P. aeruginosa, and K. pneumonia (MICs = 25, 13, 6, and 21 μg/cm3, respectively). Hirsutide also has antifungal activity against C. albicans, M. audouinii, A. niger, and Ganoderma (MICs = 13, 6, 25, and 6 μg/cm3, respectively).

天然产物

Lysionotin
Cat.No: T3381
Synonym: 岩豆素
Target: Others
1-Hydroxyanthraquinone
Cat.No: T37101
Synonym:
Target: DNA/RNA Synthesis
Tiamulin
Cat.No: T8065
Synonym: Thiamutilin,泰妙菌素
Target: Others, Antibacterial, Antibiotic
Kanamycin sulfate
Cat.No: T0793
Synonym: 硫酸卡那霉素,Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan
Target: ribosome, Antibacterial, Antibiotic
Tenuigenin
Cat.No: T3907
Synonym: Senegenin,Senegin,远志皂苷元
Target: NF-κB, Caspase, Antibacterial
Tazobactam
Cat.No: T1262
Synonym: Tazobactamum,Tazobactam acid,他唑巴坦酸,YTR-830H,CL-298741,他唑巴坦
Target: Antibacterial, Antibiotic
Trimethoprim
Cat.No: T1153
Synonym: NIH 204,BW 56-72,甲氧苄啶,NSC-106568
Target: DHFR, DNA/RNA Synthesis, Antifolate, Antibacterial, Antibiotic
Dirithromycin
Cat.No: T0971
Synonym: Dirithromycinum,地红霉素,ASE 136,LY237216,Diritromicina,Dirithromycine
Target: ribosome, Antibacterial, Antibiotic
Dehydroandrographolide succinate
Cat.No: T2S0257
Synonym:
Target: Others, Influenza Virus
Faropenem sodium
Cat.No: T5041
Synonym: 法罗培南,法罗培南钠
Target: Antibacterial, Antibiotic
Sodium Houttuyfonate
Cat.No: TN5284
Synonym: Houttuynin sodium bisulfite,新鱼腥草素钠
Target: NF-κB, Antibacterial, Antifungal
Hirsutide
Cat.No: T38016
Synonym:
Target:
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