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Search Results for " anti-glucocorticoid "

53

抑制剂 & 化合物

8

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Cat. No.	Product Name	Target	Signaling Pathways
T6713	Ulipristal	Estrogen/progestogen Receptor; Progesterone Receptor	Endocrinology/Hormones; Others
	Ulipristal 是性孕酮受体 (progesterone receptor) 的选择性调节剂。它能够与孕激素受体结合，抑制 PR 介导的基因表达，降低生殖系统中孕激素的活性。
T2527	Ulipristal acetate Ulipristal,醋酸乌利司他,CDB-2914	Estrogen/progestogen Receptor; Progesterone Receptor; Autophagy	Autophagy; Endocrinology/Hormones; Others
	Ulipristal acetate (CDB-2914) 是一种具有抗孕酮活性的选择性孕酮受体调节剂。它可抑制子宫平滑肌瘤病的生长。它通过抑制或延迟排卵和影响子宫内膜组织，可用作紧急避孕药。
T21404	Fluticasone furoate Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate	Glucocorticoid Receptor	Endocrinology/Hormones
	Fluticasone furoate (Avamys) 是一种合成的三氟化皮质类固醇，衍生自氟替卡松，Kd 为 0.3 nM。Fluticasone furoate 具有有效的抗炎、抗哮喘活性和低全身暴露。Fluticasone furoate 可用作过敏性鼻炎治疗研究的鼻喷雾剂。
T0094	Budesonide Entocort,Pulmicort,布地奈德,Rhinocort	Glucocorticoid Receptor	Endocrinology/Hormones
	Budesonide (Pulmicort) 是吸入型糖皮质类固醇，是一种口服具有活性的糖皮质激素受体激动剂。它能够减小肺部肿瘤的体积，逆转 DNA 低度甲基化，调节基因的 mRNA 表达。它是能够用于哮喘的抗炎药。
T1531	Mometasone furoate 糠酸莫美他松,糠酸莫米松,Sch32088	Glucocorticoid Receptor	Endocrinology/Hormones
	Mometasone furoate (Sch32088) 是糖皮质激素受体激动剂，具有抗炎和抗过敏作用。它是皮质固醇类试剂，动物模型中，可局部应用于气道炎症、慢性皮肤湿疹、哮喘。
T6503	Fluorometholone Acetate NSC 47438,Flarex,Eflone,氟米龙醋酸酯,Oxylone acetate	Glucocorticoid Receptor; Carbonic Anhydrase	Endocrinology/Hormones; Metabolism
	Fluorometholone Acetate (Oxylone acetate) 是合成的糖皮质激素皮质类固醇及皮质类固醇酯。它有效抑制碳酸酐酶 (CA) 对 hCA-I(IC50:2.18 μM)和 hCA-II(IC50:17.5 μM)。它具有抗炎活性，可用于研究外部眼部炎症。
T0188	Fluticasone (propionate) 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate	Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite	Endocrinology/Hormones; Metabolism; Microbiology/Virology
	Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂，是一种局部抗炎激素，亲和力KD 为 0.5 nM。具有抗病毒活性。
T4602	Hydrocortisone hemisuccinate Hydrocortisone 21-he,氢化可的松琥珀酸酯,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate	Glucocorticoid Receptor; Others; Interleukin	Endocrinology/Hormones; Immunology/Inflammation; Others
	Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) 是糖皮质激素，是口服有活性的甾体抗炎剂。它能够降低IL-6(IC50:6.7 μM)、IL-3(IC50:21.4 μM)的生物活性，可用于研究溃疡性结肠炎。
T15102	Dexamethasone palmitate 地塞米松棕榈酸酯,DXP	Glucocorticoid Receptor	Endocrinology/Hormones
	Dexamethasone palmitate (DXP) (DXP) 是 Dexamethasone 的前药。Dexamethasone 是糖皮质激素受体激动剂。与Dexamethasone 相比， DXP 对糖皮质激素受体的亲和力低 47 倍。DXP 显示出抗炎活性。
T0208	Prednisolone disodium phosphate 泼尼松龙21-磷酸二钠,Prednisolone phosphate sodium,Prednisolone 21-phosphate disodium,泼尼松龙磷酸钠	Glucocorticoid Receptor	Endocrinology/Hormones
	Prednisolone disodium phosphate是一种合成的糖皮质素，具有抗炎和免疫调节作用。
T9047	Fluprednisolone NSC-47439,NSC 47439,氟泼尼龙,NSC47439	Others	Others
	Fluprednisolone (NSC-47439) 是一种合成糖皮质激素，具有抗炎特性。
T22367	Methylprednisolone succinate Methylprednisolone hemisuccinate,Methylprednisolone hydrogen succinate,甲基泼尼松龙琥珀酸酯	Glucocorticoid Receptor	Endocrinology/Hormones
	Methylprednisolone succinate (Methylprednisolone hemisuccinate) 是合成的糖皮质激素，常用作抗炎剂。
T21361	Alclometasone dipropionate Vaderm,Sch 22219,Aclovate,Delonal	Others	Others
	Alclometasone dipropionate （Sch 22219）是一种人工合成的糖皮质激素，属于类固醇化合物，具有抗增生、抗炎、抗过敏、止痒和收缩血管的作用，可用于研究皮肤炎症。
T8777	Beclometasone 倍氯米松,BecloMethasone	Glucocorticoid Receptor	Endocrinology/Hormones
	Beclometasone 是糖皮质激素受体激动剂。
T6502	Fluocinonide 醋酸氟轻松,Lidex,Metosyn,氟轻松,Topsyn	Glucocorticoid Receptor	Endocrinology/Hormones
	Fluocinonide (Topsyn) 是一种糖皮质激素类固醇，具有抗炎作用，可作用于皮肤疾病的研究。
T0977	Medrysone Gimeracil,6α-Methyl-11β-hydroxyprogesterone,6A-甲基-11B-羟孕酮,甲羟松	Glucocorticoid Receptor; Others	Endocrinology/Hormones; Others
	Medrysone (6α-Methyl-11β-hydroxyprogesterone) 是局部合成的糖皮质激素，具有代谢、抗炎和抗过敏特性，有潜力用于眼科的眼炎症研究。
T2548	Diflorasone	Glucocorticoid Receptor	Endocrinology/Hormones
	Diflorasone 是一种皮质类固醇激素受体激动剂，具有抗炎和免疫抑制作用。它可通过细胞膜扩散进入细胞，并与细胞质中的糖皮质激素受体结合。它用于研究湿疹、牛皮癣等皮肤病。
T1559	Betamethasone dipropionate Diprolene AF,SCH 11460,二丙酸倍他米松,Betamethasone 17,21-dipropionate,Diprolene,倍他米松二丙酸酯,Diprosone	Glucocorticoid Receptor	Endocrinology/Hormones
	Betamethasone dipropionate (SCH 11460) 是糖皮质激素类固醇，具有免疫抑制、抗炎作用。
T8396	Prednisone acetate Prednisone 21-acetate,醋酸泼尼松	Glucocorticoid Receptor	Endocrinology/Hormones
	Prednisone acetate (Prednisone 21-acetate) 是泼尼松的醋酸盐形式，它是一种糖皮质激素受体激动剂，具有抗炎和免疫调节作用。
T15451	GW-870086	Glucocorticoid Receptor	Endocrinology/Hormones
	GW-870086 是抗炎剂，是糖皮质激素受体激动剂，在 A549 细胞中，能够降低 NFκB 报告基因活性(pIC50: 10.1)。
T1124	Flumethasone 氟米松,Flumetasone,RS-2177,NSC-54702	Glucocorticoid Receptor	Endocrinology/Hormones
	Flumethasone (RS-2177) 是皮质类固醇，可局部用药。它可与 Clioquinol 联合使用，研究外耳炎和耳真菌病。它作用于动物模型时，抗炎活性比 Cortisone 高 420 倍。
T0337	Prednisolone acetate Omnipred,醋酸泼尼松龙,Prednisolone-21-acetate	Glucocorticoid Receptor	Endocrinology/Hormones
	Prednisolone acetate (Omnipred) 是一种肾上腺皮质激素类药物，具有抗炎、抗过敏和抑制免疫等多种药理活性。
T1163	Betamethasone valerate Betnovate,倍他米松戊酸酯,Betaderm,Betamethasone 17-valerate,Luxiq	Glucocorticoid Receptor	Endocrinology/Hormones
	Betamethasone valerate (Luxiq) 的 17 戊酸酯，是一种具有抗炎活性的局部皮质类固醇。它能够抑制放射标记的糖皮质激素地塞米松与人表皮(IC50:5 nM)及小鼠皮肤(IC50:6 nM)的结合。它可用于研究复发性口疮。
T14981	Clobetasone butyrate	Glucocorticoid Receptor	Endocrinology/Hormones
	Clobetasone butyrate 是糖皮质类固醇，特别是在皮肤上，具有局部抗炎活性。它可用于改善皮质类固醇反应性症状，如特应性皮炎、牛皮癣。
T6465	Dexamethasone Sodium Phosphate Dexadreson,地塞米松磷酸钠,Dexagro,Dalalone	IL Receptor; COX	Immunology/Inflammation; Neuroscience
	Dexamethasone Sodium Phosphate (Dexadreson) 是一种白细胞介素受体调节剂，具有抗炎和免疫抑制作用。它属于类固醇合成药物的强效糖皮质激素类。
T1561	Clobetasol propionate Dermovate,Clobetasol 17-propionate,CGP9555,Temovate,丙酸氯倍他索,CCl 4725	Glucocorticoid Receptor; P450	Endocrinology/Hormones; Metabolism
	Clobetasol propionate (CGP9555) 是CYP3A5的选择性抑制剂(IC50:0.206 μM)，而对 CYP3A4 或其他主要 CYP 无抑制作用。它是皮质类固醇，对于牛皮癣和其他皮肤病具有潜在的研究价值。
T1076	Dexamethasone MK 125,Prednisolone F,NSC 34521,Hexadecadrol,地塞米松	Glucocorticoid Receptor; Mitophagy; IL Receptor; SARS-CoV; Antibacterial; Antibiotic; Autophagy; Complement System	Autophagy; Endocrinology/Hormones; Immunology/Inflammation; Microbiology/Virology
	Dexamethasone (Hexadecadrol) 是一种糖皮质激素受体激动剂和一种 IL 受体调节剂。Dexamethasone 具有抗炎和免疫抑制活性，可诱导自噬。Dexamethasone 抑制 LPS 诱导的巨噬细胞炎症反应。
T0820	Triamcinolone acetonide 曲安奈德,Aristogel,Azmacort,Aristoderm	Glucocorticoid Receptor	Endocrinology/Hormones
	Triamcinolone acetonide (Azmacort) 是皮质类固醇。它是皮质类固醇激素受体激动剂。它是抗炎糖皮质激素，局部用于治疗各种皮肤疾病。它的有效性是 prednisone 的八倍。
T1666	Fludrocortisone acetate 9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,醋酸氟氢可的松,9α-fluorocortisol acetate	Glucocorticoid Receptor; Autophagy	Autophagy; Endocrinology/Hormones
	Fludrocortisone acetate (9α-Fludrocortisone acetate) 是一种合成的盐皮质激素，可减少尿液中钠丢失量，也用于增加血压，有用于阿狄森氏病的研究潜力。
T1127	Beclometasone dipropionate Beclovent,Beclomethasone dipropionate,二丙酸倍氯米松,丙酸倍氯米松,Beconase,Vancenase	Glucocorticoid Receptor	Endocrinology/Hormones
	Beclometasone dipropionate (Vancenase) 是具有口服活性的糖皮质激素，具有抗炎和免疫抑制作用。它是Betamethasone 的前体药物，Betamethasone 是 LPS 诱导的炎症及 MMP 释放的抑制剂。
T0272	Nilutamide 尼鲁米特,RU23908	Androgen Receptor	Endocrinology/Hormones
	Nilutamide (RU23908) 是一种非甾体抗雄激素药物，有用于转移性前列腺癌的潜力。
T41303	Isoflupredone Delta-Fluorocortisone,Isoflupredona,异氟泼尼松,Isoflupredonum,9-Fluoroprednisolone	Others	Others
	Isoflupredone (Isoflupredonum) 是一种合成的皮质类固醇，通过与动物 (如马) 的糖皮质激素和矿皮质激素受体结合抑制炎症细胞和抑制炎症介质的表达在生物体内发挥作用。Isoflupredone 具有抗炎和免疫抑制作用，可应用于治疗各种肌肉骨骼、过敏性和全身炎症性疾病。
T27152	Dexamethasone Beloxil
	Dexamethasone Beloxil is a glucocorticoid, Anti-inflammatory Agent.
T21192	Diflorasone Diacetate Apexicon E,Psorcon,Maxiflor,醋酸双氟拉松,Florone E
	Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.
T13200	Triamcinolone Benetonide	Others	Others
	Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid exhibiting potent anti-inflammatory properties.
T25264	Cloprednol Novacort,Cloradryn,RS-4691,RS 4691,Syntestan
	Cloprednol is a synthetic glucocorticoid. It has an anti-inflammatory potency twice that of prednisone.
T31060	CP-472555 UNII-6T0KV7024R,CP 472555,CP472555
	CP-472555 is a selective nonsteroidal glucocorticoid receptor antagonist with anti-GR and anti-obesity activity in animal models.
T16404	ORIC-101
	ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.
T40697	Glucocorticoids receptor agonist 2
	Glucocorticoid receptor agonist 2 is a highly effective anti-inflammatory compound, derived from arylpyrazole, that actively binds to and activates the glucocorticoid receptor. This compound exhibits potent anti-inflammatory properties without disrupting insulin secretion.
T32113	Hydrocortamate Hydrochloride UNII-9QM8U7R83W,Ulcort,Hydrocortamate HCl,Magnacort,Ethamicort
	Hydrocortamate Hydrochloride is a synthetic glucocorticoid that has anti-inflammatory and immunosuppressive properties. It is used topically to treat inflammation caused by corticosteroid-responsive skin diseases.
T71346	MS4
	MS4 is a novel glucocorticoid receptor (GR) agonist with anti-inflammatory activity and displaying reduced impact on islets.
T63551	Glucocorticoid receptor-IN-1
	Glucocorticoid receptor-IN-1 是糖皮质激素受体 (glucocorticoid receptor (GR)) 对选择性调节剂，表现出抗炎活性。Glucocorticoid receptor-IN-1 具有良好的转录抑制作用，能够作用于 hMMP1 (IC50: 2.11 nM)，也具有转录激活效果，能够作用于 MMTV (EC50: 5.59 nM)。
T17291	ZK 216348 (+)-ZK 216348	Others	Others
	ZK 216348 also binds to Progesterone and mineralocorticoid receptors (IC50s: 20.4 nM and 79.9 nM, respectively). ZK 216348 is a nonsteroidal selective glucocorticoid receptor agonist (IC50: 20.3 nM). ZK 216348 has an anti-inflammatory activity similar to
T75016	Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal
	Glucocorticoid receptoragonist-1 phosphate Ala-Ala-Mal 是一种糖皮质激素受体激动剂。Glucocorticoid receptoragonist-1 phosphate Ala-Ala-Mal 可用于抗 CD40抗体偶联活性分子(ADC)。Glucocorticoid receptoragonist-1 phosphate Ala-Ala-Mal 可用于炎症和免疫调节的研究。
T74697	Glucocorticoid receptor agonist-2
	Glucocorticoid receptoragonist-2 (compound 21) 作为一种糖皮质激素受体激动剂，具有 6.6 nM 的 IC50 值，主要用于抗炎 ADC 分子的合成。同时，它也是 ABBV-3373 的活性对照物。
T33883	Paramethasone Acetate NCGC00185748-01,Monocortin,CHEBI:31963,8X50N88ZDP,UNII-8X50N88ZDP	Others	Others
	Paramethasone Acetate 是一种合成的糖皮质激素，具有抗炎和免疫抑制作用，可用于治疗系统性红斑狼疮。
T63539	Glucocorticoid receptor-IN-2
	Glucocorticoid receptor-IN-2 是糖皮质激素受体 (glucocorticoid receptor (GR)) 的选择性调节剂，表现出抗炎活性。Glucocorticoid receptor-IN-2 具有良好的转录抑制作用，能够作用于 hMMP1 (IC50: 0.171 nM)，也具有一定的转录激活作用，能够作用于 MMTV (EC50: 0.94 nM)。
T77869	Glucocorticoid receptor agonist-2 Ala-Ala-Mal
	Glucocorticoid receptor agonist-2 Ala-Ala-Mal（化合物79）是ABBV-3373的活性对照，可用于合成抗炎ADC分子。
T40808	Glucocorticoids receptor agonist 1
	Glucocorticoids receptor agonist 1 (GRA-1) is a highly effective arylpyrazole-based compound that acts as an agonist for the glucocorticoid receptor. GRA-1 exhibits strong anti-inflammatory properties while maintaining insulin secretion function.
T68877	Tetrahydrocorticosterone
	Tetrahydrocorticosterone (THB) is a glucocorticoid (GC) that has anti-inflammatory functions. For instance, 5α THB inhibits inflammatory actions by binding to GC receptor. HPLC studies in rat brains have reported that tetrahydrocorticosterone (THB) isomers are differentially distributed in males and females.

化合物

Cat.No: T6713

Target: Estrogen/progestogen Receptor, Progesterone Receptor

Ulipristal acetate

Cat.No: T2527

Synonym: Ulipristal,醋酸乌利司他,CDB-2914

Target: Estrogen/progestogen Receptor, Progesterone Receptor, Autophagy

Fluticasone furoate

Cat.No: T21404

Synonym: Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate

Target: Glucocorticoid Receptor

Cat.No: T0094

Synonym: Entocort,Pulmicort,布地奈德,Rhinocort

Target: Glucocorticoid Receptor

Mometasone furoate

Cat.No: T1531

Synonym: 糠酸莫美他松,糠酸莫米松,Sch32088

Target: Glucocorticoid Receptor

Fluorometholone Acetate

Cat.No: T6503

Synonym: NSC 47438,Flarex,Eflone,氟米龙醋酸酯,Oxylone acetate

Target: Glucocorticoid Receptor, Carbonic Anhydrase

Fluticasone (propionate)

Cat.No: T0188

Synonym: 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate

Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite

Hydrocortisone hemisuccinate

Cat.No: T4602

Synonym: Hydrocortisone 21-he,氢化可的松琥珀酸酯,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate

Target: Glucocorticoid Receptor, Others, Interleukin

Dexamethasone palmitate

Cat.No: T15102

Synonym: 地塞米松棕榈酸酯,DXP

Target: Glucocorticoid Receptor

Prednisolone disodium phosphate

Cat.No: T0208

Synonym: 泼尼松龙21-磷酸二钠,Prednisolone phosphate sodium,Prednisolone 21-phosphate disodium,泼尼松龙磷酸钠

Target: Glucocorticoid Receptor

Fluprednisolone

Cat.No: T9047

Synonym: NSC-47439,NSC 47439,氟泼尼龙,NSC47439

Target: Others

Methylprednisolone succinate

Cat.No: T22367

Synonym: Methylprednisolone hemisuccinate,Methylprednisolone hydrogen succinate,甲基泼尼松龙琥珀酸酯

Target: Glucocorticoid Receptor

Alclometasone dipropionate

Cat.No: T21361

Synonym: Vaderm,Sch 22219,Aclovate,Delonal

Target: Others

Cat.No: T8777

Synonym: 倍氯米松,BecloMethasone

Target: Glucocorticoid Receptor

Cat.No: T6502

Synonym: 醋酸氟轻松,Lidex,Metosyn,氟轻松,Topsyn

Target: Glucocorticoid Receptor

Cat.No: T0977

Synonym: Gimeracil,6α-Methyl-11β-hydroxyprogesterone,6A-甲基-11B-羟孕酮,甲羟松

Target: Glucocorticoid Receptor, Others

Cat.No: T2548

Target: Glucocorticoid Receptor

Betamethasone dipropionate

Cat.No: T1559

Synonym: Diprolene AF,SCH 11460,二丙酸倍他米松,Betamethasone 17,21-dipropionate,Diprolene,倍他米松二丙酸酯,Diprosone

Target: Glucocorticoid Receptor

Prednisone acetate

Cat.No: T8396

Synonym: Prednisone 21-acetate,醋酸泼尼松

Target: Glucocorticoid Receptor

Cat.No: T15451

Target: Glucocorticoid Receptor

Cat.No: T1124

Synonym: 氟米松,Flumetasone,RS-2177,NSC-54702

Target: Glucocorticoid Receptor

Prednisolone acetate

Cat.No: T0337

Synonym: Omnipred,醋酸泼尼松龙,Prednisolone-21-acetate

Target: Glucocorticoid Receptor

Betamethasone valerate

Cat.No: T1163

Synonym: Betnovate,倍他米松戊酸酯,Betaderm,Betamethasone 17-valerate,Luxiq

Target: Glucocorticoid Receptor

Clobetasone butyrate

Cat.No: T14981

Target: Glucocorticoid Receptor

Dexamethasone Sodium Phosphate

Cat.No: T6465

Synonym: Dexadreson,地塞米松磷酸钠,Dexagro,Dalalone

Target: IL Receptor, COX

Clobetasol propionate

Cat.No: T1561

Synonym: Dermovate,Clobetasol 17-propionate,CGP9555,Temovate,丙酸氯倍他索,CCl 4725

Target: Glucocorticoid Receptor, P450

Cat.No: T1076

Synonym: MK 125,Prednisolone F,NSC 34521,Hexadecadrol,地塞米松

Target: Glucocorticoid Receptor, Mitophagy, IL Receptor, SARS-CoV, Antibacterial, Antibiotic, Autophagy, Complement System

Triamcinolone acetonide

Cat.No: T0820

Synonym: 曲安奈德,Aristogel,Azmacort,Aristoderm

Target: Glucocorticoid Receptor

Fludrocortisone acetate

Cat.No: T1666

Synonym: 9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,醋酸氟氢可的松,9α-fluorocortisol acetate

Target: Glucocorticoid Receptor, Autophagy

Beclometasone dipropionate

Cat.No: T1127

Synonym: Beclovent,Beclomethasone dipropionate,二丙酸倍氯米松,丙酸倍氯米松,Beconase,Vancenase

Target: Glucocorticoid Receptor

Cat.No: T0272

Synonym: 尼鲁米特,RU23908

Target: Androgen Receptor

Cat.No: T41303

Synonym: Delta-Fluorocortisone,Isoflupredona,异氟泼尼松,Isoflupredonum,9-Fluoroprednisolone

Target: Others

Dexamethasone Beloxil

Cat.No: T27152

Diflorasone Diacetate

Cat.No: T21192

Synonym: Apexicon E,Psorcon,Maxiflor,醋酸双氟拉松,Florone E

Triamcinolone Benetonide

Cat.No: T13200

Target: Others

Cat.No: T25264

Synonym: Novacort,Cloradryn,RS-4691,RS 4691,Syntestan

Cat.No: T31060

Synonym: UNII-6T0KV7024R,CP 472555,CP472555

Cat.No: T16404

Glucocorticoids receptor agonist 2

Cat.No: T40697

Hydrocortamate Hydrochloride

Cat.No: T32113

Synonym: UNII-9QM8U7R83W,Ulcort,Hydrocortamate HCl,Magnacort,Ethamicort

Cat.No: T71346

Glucocorticoid receptor-IN-1

Cat.No: T63551

Cat.No: T17291

Synonym: (+)-ZK 216348

Target: Others

Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal

Cat.No: T75016

Glucocorticoid receptor agonist-2

Cat.No: T74697

Paramethasone Acetate

Cat.No: T33883

Synonym: NCGC00185748-01,Monocortin,CHEBI:31963,8X50N88ZDP,UNII-8X50N88ZDP

Target: Others

Glucocorticoid receptor-IN-2

Cat.No: T63539

Glucocorticoid receptor agonist-2 Ala-Ala-Mal

Cat.No: T77869

Glucocorticoids receptor agonist 1

Cat.No: T40808

Tetrahydrocorticosterone

Cat.No: T68877

Cat. No.	Product Name	Target	Signaling Pathways
T1560	Prednisolone 氢化泼尼松,Predonine,Hydroretrocortine,泼尼松龙,Metacortandralone	Glucocorticoid Receptor; Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Prednisolone (Hydroretrocortine) 是有口服活性的皮质类固醇和糖皮质激素。它的抗炎特性约为氢化可的松的四倍，同时减少了水和盐的保留。它能够用于眼部抗炎研究。
T2884	Cortisone Kendall's compound E,17-Hydroxy-11-dehydrocorticosterone,可的松	Glucocorticoid Receptor; Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Cortisone (17-Hydroxy-11-dehydrocorticosterone) 是 Cortisol(一种糖皮质激素)的氧化代谢产物。Cortisone 具有消炎和免疫抑制的作用。Cortisone 在高浓度下对 Glucocorticoid 与Glucocorticoid-receptor 的结合具有部分干预作用。
T0034	Cortisone acetate 醋酸可的松,Cortisone 21-acetate,NSC 49420	Glucocorticoid Receptor; Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Cortisone acetate (NSC-49420) 是 Cortisol(一种糖皮质激素)的氧化代谢产物。它在高浓度下能够部分干预 Glucocorticoid 与Glucocorticoid-receptor 的结合。它具有免疫抑制和消炎的作用。
T0269	Dichlorisone Acetate 糊状叶绿素,Diloderm,醋酸二氯松	Endogenous Metabolite; AChE	Metabolism; Neuroscience
	Dichlorisone Acetate (Diloderm) 一种是合成的糖皮质激素皮质类固醇，具有抗炎特性。
T1168	Desonide Tridesilon,地索奈德,Locapred,Prednacinolone	Glucocorticoid Receptor	Endocrinology/Hormones
	Desonide (Prednacinolone) 是一种非氟化皮质类固醇抗炎剂，能够作用于糖皮质激素受体。
T0798	Triamcinolone Fluoxyprednisolone,曲安西龙,Aristocort,Rodinolone	Glucocorticoid Receptor; COX	Endocrinology/Hormones; Immunology/Inflammation; Neuroscience
	Triamcinolone (Aristocort) 是一种皮质类固醇激素受体激动剂，也是一种合成的长效糖皮质激素，具有抗炎活性。
T2S2043	Dracorhodin perchlorate Dracorhodin perochlorate,血竭素高氯酸盐,Dracohodin perochlorate	Apoptosis; Others	Apoptosis; Others
	Dracorhodin perchlorate 是来源于中药血竭的一种天然产物。它抑制细胞生长，并以剂量和时间依赖性方式诱导成纤维细胞凋亡，将细胞周期阻滞在 G1 期，可作为抗乳腺癌的候选药物。
TN3537	Braylin	IL Receptor; TNF; NF-κB	Apoptosis; Immunology/Inflammation; NF-κB
	Braylin has anti-inflammatory, antinociceptive and immunomodulatory effects, which possibly act through the glucocorticoid receptor activation and by inhibition of the transcriptional activity of NF-ÎºB. Braylin is also a phosphodiesterase-4 inhibitor, it could represent an ideal prototype of glucocorticoid receptor ligand, able to induce synergic immunomodulatory effects.

天然产物

Cat.No: T1560

Synonym: 氢化泼尼松,Predonine,Hydroretrocortine,泼尼松龙,Metacortandralone

Target: Glucocorticoid Receptor, Endogenous Metabolite

Cat.No: T2884

Synonym: Kendall's compound E,17-Hydroxy-11-dehydrocorticosterone,可的松

Target: Glucocorticoid Receptor, Endogenous Metabolite

Cortisone acetate

Cat.No: T0034

Synonym: 醋酸可的松,Cortisone 21-acetate,NSC 49420

Target: Glucocorticoid Receptor, Endogenous Metabolite

Dichlorisone Acetate

Cat.No: T0269

Synonym: 糊状叶绿素,Diloderm,醋酸二氯松

Target: Endogenous Metabolite, AChE

Cat.No: T1168

Synonym: Tridesilon,地索奈德,Locapred,Prednacinolone

Target: Glucocorticoid Receptor

Cat.No: T0798

Synonym: Fluoxyprednisolone,曲安西龙,Aristocort,Rodinolone

Target: Glucocorticoid Receptor, COX

Dracorhodin perchlorate

Cat.No: T2S2043

Synonym: Dracorhodin perochlorate,血竭素高氯酸盐,Dracohodin perochlorate

Target: Apoptosis, Others

Cat.No: TN3537

Target: IL Receptor, TNF, NF-κB

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