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37

抑制剂 & 化合物

157

天然产物

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Cat. No. Product Name Target Signaling Pathways
T124455 Batatasin V

Others Others
Batatasin V 是一种天然产物,存在于植物Dioscorea oppositifolia L 的茎和叶中。
T7402 Meta-Topolin

3-[(9H-嘌呤-6-基氨基)甲基]苯酚,m-Topolin

Others Others
Meta-Topolin (m-Topolin) 是一种芳香细胞分裂素,具有较高的活性。
T20713 Flonicamid

UNII-9500W2Z53J,N-(cyanomethyl)-4-(trifluoromethyl)nicotinamide

Others Others
Flonicamid (N-(cyanomethyl)-4-(trifluoromethyl)nicotinamide) 是一种吡啶甲酰胺杀虫剂,在食用日本萝卜叶的过程中抑制蚜虫(M.persicae)的唾液分泌和汁液摄入。它对棉蚜、红蚜、巴迪蚜、禾谷蚜和大鼠产生毒性。
T126461 Aloenin B

Aloenin B 是一种从芦荟的叶和根中分离得到的化合物,对谷氨酸诱导的HT22细胞神经元死亡具有神经保护活性。
T19914 Chlorothalonil

DAC 2787,Daconil,Daconil M,百菌清

Antifungal Microbiology/Virology
Chlorothalonil (DAC 2787) 是一种高效低毒广谱的杀菌剂,广泛用于防治果树、蔬菜菜叶等多种害虫,对水稻、小麦、棉花等多种病害,也具有较好的防治效果。
T37742 N-hexanoyl-DL-Homoserine lactone

N-hexanoyl-DL-Homoserine lactone is a bacterial quorum sensing signaling molecule that is produced by mammalian pathogenic and rhizosphere-colonizing bacteria.1,2,3Application of N-hexanoyl-DL-homoserine lactone (60 μM) to tomato leaves suppresses the development of lesions induced by the plant pathogenic fungiB. cinerea.2It also increases root length and shoot diameter when applied toA. thalianaseedlings in a hydroponic growth system at a concentration of 10 μM.3
T9495 Haloxyfop methyl ester

Others Others
Haloxyfop methyl ester 是一种选择性除草剂,脂肪酸合成抑制剂,具有内吸作用。茎叶经处理后,迅速被杂草吸收并传递至全株,水解成酸,抑制根、茎分生组织的生长,导致死亡。
T32930 Lucyin A

Lucyin A is isolated from the leaves of Luffa cylinderica.
T33960 Phaseolotoxin

Phaseolotoxin A

Phaseolotoxin is an exotoxin from Pseudomonas sp.; cleavage of C terminal alanine and homoarginine from phaseolotoxin leaves octicidine.
T32931 Lucyoside R

Lucyoside R is isolated from the leaves of Luffa cylindrica.
T33036 Lyoniol B

LyoniolB,Lyoniol-B,Deacetyllyoniatoxin

Lyoniol B is a grayanane diterpenoids from the leaves of Craiobiodendron yunnanense.
T32566 Lantanolic acid

Lantanolic acid is a pentacyclic triterpenoid from the leaves of Lantana montevidensis.
T39734 Anthranoyllycoctonine

Anthranoyllycoctonine is a bioactive norditerpenoid alkaloid isolated from the leaves of Delphinium ajacis.
T32377 Kenposide A

Sacranoside B

Kenposide A is an aroma glycoside that is isolated from the fresh leaves of Hovenia dulsis var. tomentella.
T19285 Dithianon

Others Others
Dithianon is a broad-spectrum anthraquinone fungicide with good adhesion to the surface of leaves and fruits. Dithianon can be used to control several fungi in certain fruits and vegetables.
T31994 Grayanotoxin III

Deacylasebotoxin I,Deacetylandromedotoxin,Andromedol

Grayanotoxins are a group of closely related neurotoxins named after Leucothoe grayana, a plant native to Japan originally. Extract from leaves Leucothoe grayana (Ericaceae).
T3786L Tomatine hydrochloride

Tomatine hydrochloride is an alkaloid that occurs in the extract of leaves of wild tomato plants. It inhibits the growth of many fungi and bacteria. It is used as a precipitating agent for steroids.
T74243 Tyrosinase/elastase-IN-1

Tyrosinase/elastase-IN-1,一种来源于悬钩子叶的三萜类化合物,具有抑制酪氨酸酶和弹性蛋白酶活性的功能。
T125154 Quadranoside III

Antioxidant; Antibacterial Microbiology/Virology; oxidation-reduction
Quadranoside III 是从 Melissa officinalis 的干燥茎和叶中分离出三萜化合物,具有潜在的抗菌和抗氧化活性。
T26776 Berteroin

OR-009512,KB-47947,LP-088984,KB47947,LP088984

Berteroin is an erucin homolog and potential antioxidant. It is present in cruciferous vegetables, including rucola salad leaves, Chinese cabbage and mustard oil. It decreases the release of pro-inflammatory cytokines in LPS-stimulated macrophages. It als
T37994 16-hydroxy Hexadecanoic Acid

Juniperic acid

16-hydroxy Hexadecanoic Acid (Juniperic acid) 是从拟南芥叶和茎中分离出的化合物,可用于预防、缓解或治疗代谢性疾病。
T37865 9(S)-HOTrE

9(S)-HOTrE is a monohydroxy polyunsaturated fatty acid produced by the action of 5-lipoxygenase on α-linolenic acid. 9(S)-HOTrE is predominantly localized in cellular ester lipids of Glechoma hederacea leaves and is partially released during artificial dehydration. The biological role of 9(S)-HOTrE in G. hederacea leaves is still undetermined, but it may play a role in natural senescence. 9(S)-HOTrE is an inhibitor of spore germination and germ tube elongation of rice blast fungus with ED50 valu...
T25000 Acetylaleuritolic acid

NSC 266221,NSC-266221,NSC266221

Acetylaleuritolic acid 是一种从小花加西亚叶中分离得到的一种五环三萜类化合物,植物代谢产物。它具有抗肿瘤特性,对P-388淋巴细胞白血病测试中显示出肿瘤抑制活性。
T35705 20-hydroxy Arachidic Acid

20-hydroxy Arachidic acid is a hydroxylated fatty acid that has been found in the suberin component of silver birch (B. pendula) outer bark as well as the leaves, roots, and wood of Q. ilex from Cala Violina and Colognole, Italy. 20-hydroxy Arachidic acid was identified as a potential inhibitor of human rhinovirus coat protein in a structure-based virtual screen.
T73851 cis-β-Terpineol

Cis-β-Terpineol为一类单萜类化合物,主要从土库曼假狼紫草地上部分提取。其茎、叶、花均展现抗菌活性。
T37255 12-methyl Myristic Acid methyl ester

12-methyl Myristic acid methyl ester is a methylated fatty acid methyl ester that has been found in vermicomposts of cattle manure, carica papaya leaves, and cuticular wax of K. africana. It is a volatile compound in lipid-lowering granulated tea. Levels of 12-methyl myristic acid methyl ester are decreased in T. cruzi treated with nifurtimox compared to non-treated controls.
T73850 trans-β-Terpineol

trans-β-terpineol 为单萜类化合物,在圆叶菊叶片中可分离提取。该化合物具备抗氧化及抗菌特性,在圆叶菊中主要承担抗菌生物活性作用。
T36822 Benzovindiflupyr

Benzovindiflupyr is a fungicide.1It inhibits mitochondrial complex II, also known as succinate dehydrogenase (SDH; IC50= 5.2 nM), and mycelial growth ofS. sclerotiorum(EC50= 0.011 μg/ml). Benzovindiflupyr (60 μg/ml) completely protects eggplant leaves fromS. sclerotioruminfection. Formulations containing benzovindiflupyr have been used to control various fungal diseases in agriculture. 1.Gao, Y., He, L., Zhu, J., et al.The relationship between features enabling SDHI fungicide binding to the Sc-S...
T78931 SDH-IN-5

SDH-IN-5(化合物7d)是一种琥珀酸脱氢酶(SDH)抑制剂,IC50为3.293 μM。该化合物同时展现出对R. solani具有EC50值为0.046 μg/mL的抗真菌活性,并对水稻叶片中的茄病菌表现出显著的保护和治疗效果。
T36234 5(Z),11(Z),14(Z)-Eicosatrienoic Acid

5(Z),11(Z),14(Z)-Eicosatrienoic acid is a polyunsaturated fatty acid found in various natural sources including maritime pine (Pinus pinaster) seed oil (MPSO), gymnospermae leaves and seeds, and freshwater gastropods. A diet containing MPSO lowered high-density lipoprotein and ApoA1 levels in transgenic mice expressing human ApoA1. MPSO was found to diminish cholesterol efflux in vitro. 5(Z),11(Z),14(Z)-Eicosatrienoic acid methyl ester, when topically applied, reduces inflammatory processes, pot...
T81319 Quizalofop-P

Acetyl-CoA Carboxylase Metabolism
Quizalofop-P被杂草通过茎叶吸收,能在植株内实现向上和向下的双向运输,并在顶端和分生区域累积,通过抑制脂肪酸合成,进而导致杂草死亡。此外,Quizalofop-P对禾本科杂草与双子叶作物具有显著的选择性。
T74929 Phytoene desaturase-IN-1

Phytoene desaturase-IN-1 是高效的PDS抑制剂(Kd: 65.9 μM),通过与Phe301残基形成π-π堆叠效应。该化合物显示出广谱的芽后除草活性,并能在白化病叶片中诱导PDS mRNA水平下降及八氢番茄红素与ROS累积,适用于农业生产。
T37396 13-epi-12-oxo Phytodienoic Acid

13-epi-12-oxo Phytodienoic acid (13-epi-12-oxo PDA) is a lipoxygenase metabolite of α-linolenic acid in the leaves of green plants such as corn. ω-3 and ω-6 polyunsaturated fatty acids in plants are substrates for plant lipoxygenases. 12-oxo PDA is one of the best studied end metabolites of this enzymatic pathway. While the initial enzymatic product and major isomer of 12-oxo PDA contains side chains in the cis position, both being β to the ring, the upper side chain attached at C-13, can and fr...
T71811 Lobaric acid

Lobaric acid is a depsidone metabolite that has been isolated from Stereocaulon lichen species with antioxidant, antiproliferative, antiviral, and enzyme inhibitory activites. It scavenges superoxide radicals in a cell-free assay (IC50 = 97.9 μmol) and inhibits proliferation in a panel of leukemia, colorectal, gastric, breast, ovarian, prostate, pancreatic, and lung cancer cell lines (EC50s = 15.2-63.9 μg/ml). Lobaric acid inhibits protein tyrosine phosphatase 1B (PTP1B; IC50 = 0.87 μM for the h...
T35771 Destruxin B2

Destruxin B2 is a cyclic hexadepsipeptide mycotoxin that has been found in M. anisopliae and has antiviral, insecticidal, and phytotoxic activities.1,2,3 It inhibits secretion of hepatitis B virus surface antigen (HBsAg) by Hep3B cells expressing hepatitis B virus (HBV) DNA (IC50 = 1.3 μM).1 Destruxin B2 is toxic to Sf9 insect cells in an electric cell-substrate impedance sensing (ECIS) test with a 50% inhibitory concentration (ECIS50) value of 92 μM.4 It is also phytotoxic to B. napus leaves.3 ...
T37394 13(S)-HpOTrE

13(S)-HpOTrE is a monohydroperoxy polyunsaturated fatty acid produced in soybeans by the action of soybean LO-2 on esterified α-linolenic acid.[1] Incubation of soybean seedling biomembranes with soybean LO-2 catalyzes the formation of both 9- and 13-HpOTrE in a molar ratio of 10:1.1 In plants, 13(S)-HpOTrE can be metabolized by the hydroperoxide lyase pathway producing aldehyde and oxoacid fragments, or by the hydroperoxide dehydratase pathway producing jasmonic acid.[2],[3],[4] Treatment of to...
T37393 13(S)-HpODE

13(S)-HpODE is produced by the oxidation of linoleic acid by lipoxygenase-1 (LO-1) in many plants including soybean, flaxseed, apples, and tea leaves,1,2 and by 15-LO in mammals.3 In plants, 13(S)-HpODE is the preferred substrate for the garlic bulb divinyl ether synthase.4 In mammalian tissues, 13(S)-HpODE is generally reduced to 13(S)-HODE,a compound which exhibits many biological activities.3 A direct action for 13(S)-HpODE has been demonstrated in Syrian hamster embryo cells where it stimula...

化合物

Batatasin V
Cat.No: T124455
Synonym:
Target: Others
Meta-Topolin
Cat.No: T7402
Synonym: 3-[(9H-嘌呤-6-基氨基)甲基]苯酚,m-Topolin
Target: Others
Flonicamid
Cat.No: T20713
Synonym: UNII-9500W2Z53J,N-(cyanomethyl)-4-(trifluoromethyl)nicotinamide
Target: Others
Aloenin B
Cat.No: T126461
Synonym:
Target:
Chlorothalonil
Cat.No: T19914
Synonym: DAC 2787,Daconil,Daconil M,百菌清
Target: Antifungal
N-hexanoyl-DL-Homoserine lactone
Cat.No: T37742
Synonym:
Target:
Haloxyfop methyl ester
Cat.No: T9495
Synonym:
Target: Others
Lucyin A
Cat.No: T32930
Synonym:
Target:
Phaseolotoxin
Cat.No: T33960
Synonym: Phaseolotoxin A
Target:
Lucyoside R
Cat.No: T32931
Synonym:
Target:
Lyoniol B
Cat.No: T33036
Synonym: LyoniolB,Lyoniol-B,Deacetyllyoniatoxin
Target:
Lantanolic acid
Cat.No: T32566
Synonym:
Target:
Anthranoyllycoctonine
Cat.No: T39734
Synonym:
Target:
Kenposide A
Cat.No: T32377
Synonym: Sacranoside B
Target:
Dithianon
Cat.No: T19285
Synonym:
Target: Others
Grayanotoxin III
Cat.No: T31994
Synonym: Deacylasebotoxin I,Deacetylandromedotoxin,Andromedol
Target:
Tomatine hydrochloride
Cat.No: T3786L
Synonym:
Target:
Tyrosinase/elastase-IN-1
Cat.No: T74243
Synonym:
Target:
Quadranoside III
Cat.No: T125154
Synonym:
Target: Antioxidant, Antibacterial
Berteroin
Cat.No: T26776
Synonym: OR-009512,KB-47947,LP-088984,KB47947,LP088984
Target:
16-hydroxy Hexadecanoic Acid
Cat.No: T37994
Synonym: Juniperic acid
Target:
9(S)-HOTrE
Cat.No: T37865
Synonym:
Target:
Acetylaleuritolic acid
Cat.No: T25000
Synonym: NSC 266221,NSC-266221,NSC266221
Target:
20-hydroxy Arachidic Acid
Cat.No: T35705
Synonym:
Target:
cis-β-Terpineol
Cat.No: T73851
Synonym:
Target:
12-methyl Myristic Acid methyl ester
Cat.No: T37255
Synonym:
Target:
trans-β-Terpineol
Cat.No: T73850
Synonym:
Target:
Benzovindiflupyr
Cat.No: T36822
Synonym:
Target:
SDH-IN-5
Cat.No: T78931
Synonym:
Target:
5(Z),11(Z),14(Z)-Eicosatrienoic Acid
Cat.No: T36234
Synonym:
Target:
Quizalofop-P
Cat.No: T81319
Synonym:
Target: Acetyl-CoA Carboxylase
Phytoene desaturase-IN-1
Cat.No: T74929
Synonym:
Target:
13-epi-12-oxo Phytodienoic Acid
Cat.No: T37396
Synonym:
Target:
Lobaric acid
Cat.No: T71811
Synonym:
Target:
Destruxin B2
Cat.No: T35771
Synonym:
Target:
13(S)-HpOTrE
Cat.No: T37394
Synonym:
Target:
13(S)-HpODE
Cat.No: T37393
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN4495 Maoyerabdosin

Others Others
Maoyerabdosin 是一种提取自粳稻叶的化合物。
TN4494 Maoecrystal B

Others Others
Maoecrystal B 是一种分离自 Isodon eriocalyx var.叶子的二萜化合物。
TN4453 Lophanthoidin F

Others Others
Lophanthoidin F 是一种二萜化合物,提取自Rabdosia lophanthoides 的干叶。
TN4451 Lophanthoidin B

Others Others
Lophanthoidin B 是一种二萜类化合物,提取自从Rabdosia lophanthoides 的干叶。
TN4452 Lophanthoidin E

Others Others
Lophanthoidin E 是一种二萜化合物,分离自Rabdosia lophanthoides 的干叶。
TN4919 Rosthornin A

Others Others
Rosthornin A 是一种分离自 Rabdosia rosthornii 干叶的醚提取的 ent-kaurene diterpenoid 化合物。
TN1855 Laurolitsine

去甲异波尔定,(+)-Norboldine

Others Others
Laurolitsine ((+)-Norboldine) 是一种生物碱,从 Peumus boldusMolina 叶子中分离得到。
T4S2126 Ginkgetin

银杏双黄酮,银杏素

Apoptosis; Wnt/beta-catenin; COX; STAT; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Immunology/Inflammation; JAK/STAT signaling; Neuroscience; Stem Cells
Ginkgetin 是从银杏叶中分离得到的一种双黄酮,具有抗肿瘤、抗炎、神经保护、抗真菌的作用。它也是 Wnt 信号抑制剂,IC50值为 5.92 μM。
T6917 Oleuropein

洋橄榄苦甙,橄榄苦苷

Apoptosis; Aromatase; ROS; PPAR Apoptosis; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Oleuropein 在橄榄叶和油中发现的天然产物,通过 p53 依赖性途径以及 Bax 和 Bcl2基因的调控来诱导乳腺癌细胞凋亡,还抑制芳香化酶。它可通过直接抑制 PPARγ转录活性来发挥抗氧化,抗炎和抗动脉粥样硬化作用。
TN4920 Rosthornin B

Others Others
Rosthornin B 是分离自 Rabdosia rosthornii 干叶的醚提取物的一种ent-kaurene diterpenoid 化合物。
T13514 5-MethoxyPinocembroside

Others Others
5-MethoxyPinocembroside 是一种黄酮类天然产物,存在于辣木 Moringa oleifera 的叶子中。
T2S0967 Sennoside C

Others Others
Sennoside C 是从番泻叶和豆荚中提取的蒽醌甙,对小鼠的通便作用有辅助作用。
TN7131 1-Formyl-β-carboline

9H-pyrido[3,4-b]indole-1-carbaldehyde

Others Others
1-Formyl-β-carboline 是一种从臭椿 Ailanthus altissima 叶中提取的生物碱。
TN7083 Ternatumoside II

Others Others
Ternatumoside II 是紫荆叶的水提取物,可抑制 GIA。
TN4419 Lasiodonin

Others Others
Lasiodonin 是一种二萜化合物,提取自 Isodon lasiocarpus 中。
T37886 1-Heptadecanol

Antibacterial Microbiology/Virology
1-Heptadecanol 是分离自Solena amplexicaulis 的长链伯醇,显示出抗菌活性。
TN3847 Dihydroalpinumisoflavone

Dihydroalpinumisoflavone 是一种从 Crotalaria madurensis 的叶子和茎中提取的天然产品。
TN7110 Ginsenoside Rs2

人参皂苷Rs2

Others Others
Ginsenoside Rs2 是从人参Panax japonicus var.叶中分离得到的天然产物。
T4S2012 Dihydrosanguinarine

13,14-Dihydrosanguinarine,Dihydro Sanguinarine,二氢血根碱

Caspase; Antifungal Apoptosis; Microbiology/Virology; Proteases/Proteasome
Dihydrosanguinarine 是榕树叶片提取出的一种天然产物,具有抗真菌和抗癌活性。
T4394 Methyl Isoferulate

Others Others
Methyl Isoferulate 从毛竹叶中分离纯化。
T2S0968 Sennoside D

Others Others
Sennoside D 是一种从番泻 Cassia angustifolia 的叶子和豆荚中提取的蒽醌苷。
TN7215 Isochiisanoside

Others Others
Isochiisanoside 是一种天然产物,存在于植物刺五加Acanthopanax chiisanensis NAKAI 的叶子中。
TN2138 Rebaudioside N

Others Others
Rebaudioside N 是一种 从叶菊叶中分离得到的甜菊糖苷,是一种食品添加剂。
T2S0501 Ilexgenin A

IL Receptor; TNF Apoptosis; Immunology/Inflammation
Ilexgenin A 是一种五环三萜类化合物,提取自海南冬青,可用于研究炎症及癌症。
T67136 1-Hydroxy-2-butanone

Endogenous Metabolite; Antibiotic Metabolism; Microbiology/Virology
1-Hydroxy-2-butanone 是可从竹子汁和番茄叶中提取得到的天然产物,具有抗结核活性。
TN4325 Isorhamnetin 3-robinobioside

Antioxidant oxidation-reduction
Isorhamnetin 3-robinobioside 从白刺叶中提取,具有抗氧化和抗原毒性活性。
TN7092 Lugrandoside

Others Others
Lugrandoside 是一种新型的苯丙素苷,它已从洋地黄和 Difitalis Grandiflora Miller 的茎叶中分离得到。
T2816 7,8-Dihydroxyflavone

二羟基黄酮水合物,7,8-DHF

Apoptosis; Trk receptor Apoptosis; Tyrosine Kinase/Adaptors
7,8-Dihydroxyflavone (7,8-DHF) 是一种选择性有效的TrkB 激动剂,其模拟脑源性神经营养因子的生理作用。它有潜力研究各种神经疾病。
TN1824 Kaempferol 3-sophoroside-7-glucoside

Antioxidant oxidation-reduction
Kaempferol 3-sophoroside-7-glucoside 是一种龙脷叶中的生物活性成分,属于黄酮类,具有抗氧化和抗肥胖活性。
TN7227 3β-Acetoxyurs-12-en-11-one

11-Ketoamyrinacetate

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
3β-Acetoxyurs-12-en-11-one (11-Ketoamyrinacetate) 是一种从 Morus mesozygia 的茎皮和 Ficus hirta Vahl (桑科) 的叶中发现的熊烷三萜类天然产物。
TN4674 Nortrachelogenin-8'-O-beta-glucoside

Others Others
Nortrachelogenin-8'-O-beta-glucoside 是一种具有二芳基羟基丁内酯骨架的木脂素,其分离自 Trachelospermum jasminoides (Lindl.) Lem 的叶和茎。
TN1091 Dehydronuciferine

AChE Neuroscience
Dehydronuciferine 是一种乙酰胆碱酯酶抑制剂,其 IC50=25 μg/mL,是从 Nelumbo nucifera Gaertn 的叶子中分离得到。
TN2068 Picrinine

Lipoxygenase Metabolism
Picrinine 是一种从 Alstonia scholaris 的叶子中提取出来的 Akuammiline 生物碱。 Picrinine 具有抗炎活性,通过抑制5-脂氧合酶来发挥作用。
T7846 Aegeline

Others; Antifungal Microbiology/Virology; Others
Aegeline 是从 Aegle marmelos 的叶子中分离出来的一种生物碱酰胺,有抗高血糖和抗血脂异常的活性。
TN1126 Sakuranetin

VEGFR; NF-κB; PPAR; Antifungal Angiogenesis; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB; Tyrosine Kinase/Adaptors
Sakuranetin 是一种大米黄酮类植物抗毒素,能改善 LPS 诱导的急性肺损伤,具有抗炎、抗真菌和抗氧化作用。
T2969 Lawsone

Hennotannic acid,指甲花醌,2-hydroxy-1,4-naphthoquinone

Others; Antifungal Microbiology/Virology; Others
Lawsone (Hennotannic acid) 是一种从Lawsonia inermis 的叶片中分离得到的萘醌染料,具有抗菌和抗氧化活性。
TN2148 Retusin

5-Hydroxy-3,7,3',4'-tetramethoxyflavone,Quercetin-3,7,3',4'-tetramethyl ether

ATPase; Free radical scavengers; Tyrosinase Membrane transporter/Ion channel; oxidation-reduction; Proteases/Proteasome
Retusin 是从 Talinum triangulare 的叶子中提取的。 Retusin Retusin 可用于作为芽前和芽后除草剂的研究。
TN1917 Mauritianin

Topoisomerase DNA Damage/DNA Repair
Mauritianin 是一种从 Acalypha indica 的花和叶中分离出来的山柰酚苷,是一种拓扑异构酶 I 抑制剂。Mauritianin 具有细胞保护活性。
T2749 Ginkgolide A

银杏内酯A,BN-52020

GABA Receptor; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Neuroscience
Ginkgolide A (BN-52020) 是从银杏叶提取出来的一种天然产物,是 GABA 拮抗剂,有用于多种炎症和免疫疾病的研究潜力。
TN2324 Yuankanin

Antioxidant oxidation-reduction
Yuankanin 是一种是在百里香叶、Daphne gnidium 和Daphne feddei 中发现的天然化合物,是一种 genkwanin-5-bioside,具有抗虫和抗氧化活性并对o- 1葡萄糖苷酶、脂肪酶、胰蛋白酶和黄嘌呤氧化酶具有抑制作用。
T2835 Morin

桑色素,Toxylon pomiferum,Aurantica,Calico Yellow,Al-Morin

Others Others
Morin (Calico Yellow) 是植物性黄酮类化合物,具有较弱的抗氧化活性,是用于铝物种形成的荧光螯合剂。
T21344 1-Deoxynojirimycin hydrochloride

Moranoline,去氧野艽霉素盐酸盐,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin

PI3K; Antibacterial; Antibiotic; Glucosidase Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling
1-Deoxynojirimycin hydrochloride (Moranoline) 是一种口服有效的 α-葡萄糖苷酶抑制剂,具有降血糖、减肥和抗病毒的作用,可抑制餐后血糖,预防糖尿病。
T8202 Kaempferol 3-O-gentiobioside

Kaempferol 3-gentiobioside,山柰酚 3-龙胆双糖苷

Glucosidase Metabolism
Kaempferol 3-O-gentiobioside 是一种黄酮类化合物,从C. alata 叶中分离得到,具有抗糖尿病特性。它有抗 α-glucosidase 活性,并具有对碳水化合物酶的抑制作用,其 IC50=50.0 µM。
TN7050 Potassium 7-hydroxy-1-naphthalenesulfona

藏红花酸,2-Naphthol-8-sulfonic Acid Potassium Salt

Others Others
Potassium 7-hydroxy-1-naphthalenesulfona (2-Naphthol-8-sulfonic Acid Potassium Salt) 天然存在于茜草科栀子花的果实、鸢尾科番红花的花和玄参科玄参科的花叶中。
T2755 Rhoifolin

野漆树苷,Apigenin-7-O-rhamnoglucoside,Apigenin 7-O-neohesperidoside,Rhoifoloside

Others; p38 MAPK; NF-κB; transporter; IGF-1R; Autophagy Autophagy; MAPK; Metabolism; NF-κB; Others; Tyrosine Kinase/Adaptors
Rhoifolin (Apigenin 7-O-neohesperidoside) 是从琯溪蜜柚叶子分离的一种黄酮糖苷。它通过 RANKL 诱导的NF-κB 和MAPK 途径改善钛颗粒刺激的骨溶解并减少破骨细胞生成。它通过增强脂联素分泌,胰岛素受体-β的酪氨酸磷酸化和GLUT4易位有助于治疗糖尿病并发症。
Fr14127 Coumaran

2,3-Dihydrobenzofuran,2,3-二氢苯并呋喃

Endogenous Metabolite; AChE Metabolism; Neuroscience
Coumaran (2,3-Dihydrobenzofuran) 是一种提取自L. camara 的 (AChE) 抑制剂。2,3-Dihydrobenzofuran 能够用作生物农药。
TN2101 Primin

Antifection Microbiology/Virology
Primin 是存在于 Primula obconica 叶和茎毛状体中的天然产物,显示出抗菌和抗癌活性。
TN2296 Vinaginsenoside R4

越南参皂苷R4

Others Others
Vinaginsenoside R4 是分离自水培人参的叶子中。它能够抑制黑色素的生物合成,并增强斑马鱼的色素沉着,对 melan-a 细胞没有任何细胞毒性作用。
TN7218 Diformylphloroglucinol

2,4,6-Trihydroxyisophthalaldehyde

Antioxidant oxidation-reduction
Diformylphloroglucinol (2,4,6-Trihydroxyisophthalaldehyde) 是从蓝桉树的叶子中分离出的酰基间苯三酚,是合成具有抗氧化和抗溃疡活性间苯三酚化合物的原料。
TQ0099 20-O-Acetylingenol-3-angelate

巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1

Others Others
20-O-Acetylingenol-3-angelate (Euphorbia factor Pe1) 是一种天然化合物,存在于植物英加的叶子和茎中。它具有多种生物活性,包括抑制肿瘤生长、抗炎、抗真菌和抗氧化作用。
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天然产物

Maoyerabdosin
Cat.No: TN4495
Synonym:
Target: Others
Maoecrystal B
Cat.No: TN4494
Synonym:
Target: Others
Lophanthoidin F
Cat.No: TN4453
Synonym:
Target: Others
Lophanthoidin B
Cat.No: TN4451
Synonym:
Target: Others
Lophanthoidin E
Cat.No: TN4452
Synonym:
Target: Others
Rosthornin A
Cat.No: TN4919
Synonym:
Target: Others
Laurolitsine
Cat.No: TN1855
Synonym: 去甲异波尔定,(+)-Norboldine
Target: Others
Ginkgetin
Cat.No: T4S2126
Synonym: 银杏双黄酮,银杏素
Target: Apoptosis, Wnt/beta-catenin, COX, STAT, Autophagy
Oleuropein
Cat.No: T6917
Synonym: 洋橄榄苦甙,橄榄苦苷
Target: Apoptosis, Aromatase, ROS, PPAR
Rosthornin B
Cat.No: TN4920
Synonym:
Target: Others
5-MethoxyPinocembroside
Cat.No: T13514
Synonym:
Target: Others
Sennoside C
Cat.No: T2S0967
Synonym:
Target: Others
1-Formyl-β-carboline
Cat.No: TN7131
Synonym: 9H-pyrido[3,4-b]indole-1-carbaldehyde
Target: Others
Ternatumoside II
Cat.No: TN7083
Synonym:
Target: Others
Lasiodonin
Cat.No: TN4419
Synonym:
Target: Others
1-Heptadecanol
Cat.No: T37886
Synonym:
Target: Antibacterial
Dihydroalpinumisoflavone
Cat.No: TN3847
Synonym:
Target:
Ginsenoside Rs2
Cat.No: TN7110
Synonym: 人参皂苷Rs2
Target: Others
Dihydrosanguinarine
Cat.No: T4S2012
Synonym: 13,14-Dihydrosanguinarine,Dihydro Sanguinarine,二氢血根碱
Target: Caspase, Antifungal
Methyl Isoferulate
Cat.No: T4394
Synonym:
Target: Others
Sennoside D
Cat.No: T2S0968
Synonym:
Target: Others
Isochiisanoside
Cat.No: TN7215
Synonym:
Target: Others
Rebaudioside N
Cat.No: TN2138
Synonym:
Target: Others
Ilexgenin A
Cat.No: T2S0501
Synonym:
Target: IL Receptor, TNF
1-Hydroxy-2-butanone
Cat.No: T67136
Synonym:
Target: Endogenous Metabolite, Antibiotic
Isorhamnetin 3-robinobioside
Cat.No: TN4325
Synonym:
Target: Antioxidant
Lugrandoside
Cat.No: TN7092
Synonym:
Target: Others
7,8-Dihydroxyflavone
Cat.No: T2816
Synonym: 二羟基黄酮水合物,7,8-DHF
Target: Apoptosis, Trk receptor
Kaempferol 3-sophoroside-7-glucoside
Cat.No: TN1824
Synonym:
Target: Antioxidant
3β-Acetoxyurs-12-en-11-one
Cat.No: TN7227
Synonym: 11-Ketoamyrinacetate
Target: Antibacterial, Antibiotic, Antifungal
Nortrachelogenin-8'-O-beta-glucoside
Cat.No: TN4674
Synonym:
Target: Others
Dehydronuciferine
Cat.No: TN1091
Synonym:
Target: AChE
Picrinine
Cat.No: TN2068
Synonym:
Target: Lipoxygenase
Aegeline
Cat.No: T7846
Synonym:
Target: Others, Antifungal
Sakuranetin
Cat.No: TN1126
Synonym:
Target: VEGFR, NF-κB, PPAR, Antifungal
Lawsone
Cat.No: T2969
Synonym: Hennotannic acid,指甲花醌,2-hydroxy-1,4-naphthoquinone
Target: Others, Antifungal
Retusin
Cat.No: TN2148
Synonym: 5-Hydroxy-3,7,3',4'-tetramethoxyflavone,Quercetin-3,7,3',4'-tetramethyl ether
Target: ATPase, Free radical scavengers, Tyrosinase
Mauritianin
Cat.No: TN1917
Synonym:
Target: Topoisomerase
Ginkgolide A
Cat.No: T2749
Synonym: 银杏内酯A,BN-52020
Target: GABA Receptor, Endogenous Metabolite
Yuankanin
Cat.No: TN2324
Synonym:
Target: Antioxidant
Morin
Cat.No: T2835
Synonym: 桑色素,Toxylon pomiferum,Aurantica,Calico Yellow,Al-Morin
Target: Others
1-Deoxynojirimycin hydrochloride
Cat.No: T21344
Synonym: Moranoline,去氧野艽霉素盐酸盐,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin
Target: PI3K, Antibacterial, Antibiotic, Glucosidase
Kaempferol 3-O-gentiobioside
Cat.No: T8202
Synonym: Kaempferol 3-gentiobioside,山柰酚 3-龙胆双糖苷
Target: Glucosidase
Potassium 7-hydroxy-1-naphthalenesulfona
Cat.No: TN7050
Synonym: 藏红花酸,2-Naphthol-8-sulfonic Acid Potassium Salt
Target: Others
Rhoifolin
Cat.No: T2755
Synonym: 野漆树苷,Apigenin-7-O-rhamnoglucoside,Apigenin 7-O-neohesperidoside,Rhoifoloside
Target: Others, p38 MAPK, NF-κB, transporter, IGF-1R, Autophagy
Coumaran
Cat.No: Fr14127
Synonym: 2,3-Dihydrobenzofuran,2,3-二氢苯并呋喃
Target: Endogenous Metabolite, AChE
Primin
Cat.No: TN2101
Synonym:
Target: Antifection
Vinaginsenoside R4
Cat.No: TN2296
Synonym: 越南参皂苷R4
Target: Others
Diformylphloroglucinol
Cat.No: TN7218
Synonym: 2,4,6-Trihydroxyisophthalaldehyde
Target: Antioxidant
20-O-Acetylingenol-3-angelate
Cat.No: TQ0099
Synonym: 巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1
Target: Others
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