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30

抑制剂 & 化合物

2

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T1167	Cyproterone acetate Androcur,醋酸环丙氯地孕酮,Cyproterone 17-O-acetate,醋酸环丙孕酮	Androgen Receptor	Endocrinology/Hormones
	Cyproterone acetate (Cyproterone 17-O-acetate) 是能够抗雄激素(IC50=7.1 nM) 和孕激素合成的类固醇。它与 progesteron 和糖皮质激素受体有亲和力。
T4102	Goserelin acetate 醋酸戈舍瑞林,Fertilan,ICI-118630 acetate,Zoladex	Apoptosis; GNRH Receptor	Apoptosis; GPCR/G Protein
	Goserelin acetate (Fertilan) 是一种促性腺激素释放激素 (GnRH/LHRH) 十肽类似物，能作为GnRH 激动剂。它可研究乳腺癌、上皮性卵巢癌和前列腺癌。
T1490	Gestodene SHB 331,WL 70,孕二烯酮	Estrogen/progestogen Receptor; Progesterone Receptor	Endocrinology/Hormones; Others
	Gestodene (WL 70) 是一种孕激素类避孕药。
T9035	Testosterone undecanoate	Others; Androgen Receptor	Endocrinology/Hormones; Others
	Testosterone undecanoate 是一种睾酮酯，是睾酮的代谢产物，睾酮是很有前途的男性激素避孕雄激素。
T72058L	CDD-1102 HCl CDD-1102 HCl(2757619-84-2 Free base)	Epigenetic Reader Domain	Chromatin/Epigenetic
	CDD-1102 HCl 是一种新型BRDT-BD4 / BRD2-BD1302选择性抑制剂，在体内外实验中显示出非激素避孕潜力。
T2567	Etonogestrel 3-Oxodesogestrel,3-keto-Desogestrel,依托孕烯,Nexplanon,Implanon	Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Progesterone Receptor; Endogenous Metabolite	Endocrinology/Hormones; Metabolism; Others
	Etonogestrel (Implanon) 是孕激素去氧孕烯的生物活性代谢物，与靶器官中的孕酮受体和雌激素受体高亲和力地结合，可诱导FKBP51mRNA 和蛋白表达。它是一种甾体孕激素，用作激素避孕药。
TP1705	Gastrin I (1-14), human	Others	Others
	Gastrin I (1-14), human 是人胃泌素 I 肽的 1-14 片段。其中Gastrin I 是内源性胃肠肽激素。Gastrin 是胃酸分泌的主要激素调节剂。
T24415	Lotrifen Privaprol,L-12717,DL 717-IT,L 12717,L12717,Canocenta	Others	Others
	Lotrifen (Privaprol) 是一种非激素抗生育药物，Lotrifen 引起妊娠停止和复旧。在胚泡着床后，它直接作用于受精卵，受精卵经历一个缓慢而逐渐的退化过程，并以受精卵的再吸收或排出而结束。
T17217	Vamorolone 地塞米松EP杂质E,VBP15	Glucocorticoid Receptor; NF-κB	Endocrinology/Hormones; NF-κB
	Vamorolone (VBP15) 是一种首创的，具有口服活性的解离性类固醇 (dissociative steroidal) 抗炎药和膜稳定剂。它抑制 (NF-κB) 抑制作用，并降低了激素的影响。它改善肌营养不良，无副作用。
T0272	Nilutamide 尼鲁米特,RU23908	Androgen Receptor	Endocrinology/Hormones
	Nilutamide (RU23908) 是一种非甾体抗雄激素药物，有用于转移性前列腺癌的潜力。
T11847L	Liarozole R75251 dihydrochloride,利阿唑	P450; Retinoid Receptor	Metabolism
	Liarozole (R75251 dihydrochloride) 是一种咪唑衍生物，是一种具有口服活性的维甲酸 (RA) 代谢阻断剂(RAMBA)，具有抗肿瘤作用。它能够抑制维甲酸依赖的细胞色素P450(CYP26) 4- 羟基化 (IC50=7 μM)，导致组织维甲酸水平增加。
T0824	4-Nonylphenol polyethoxylate Nonoxynol,Nonoxinol-9,壬苯醇醚	COX	Immunology/Inflammation; Neuroscience
	4-Nonylphenol polyethoxylate (Nonoxinol-9) 是一种表面活性剂，普遍用作避孕药中的杀精剂。
T68775	Etamestrol
	Etamestrol is a synthetic, steroidal estrogen described as an ovulation inhibitor or hormonal contraceptive
T31108	CTP-347 CTP347,CTP 347
	CTP-347, a deuterated version of paroxetine, is potentially the best non-hormonal drug in its class for the treatment of hot flashes.
T19811	Nomegestrol
	Nomegestrol is a progestin. It is used in the treatment of gynecological disorders, in menopausal hormone therapy for the treatment of menopausal symptoms, and in hormonal contraceptives.
T34107	Polythiazide P2525,NSC-108161,NSC 108161,P-2525,NSC108161
	Polythiazide (NSC-108161, P-2525) is used to treat fluid retention (edema) caused by a variety of causes, including congestive heart failure, severe liver disease (cirrhosis), kidney disease, or steroid or hormonal medication.
T68551	Cabergoline diphosphate
	Cabergoline diphosphate is a dopamine D2 receptor agonist used for prolactinoma treatment. Cabergoline permits rapid and effective hormonal and tumor control by normalizing prolactin-producing pituitary adenomas levels.
TP1694	Thymus peptide C
	Thymus peptide C, a hormonal drug derived from the thymus glands of young calves, acts as a substitute for the physiological functions of the thymus.
T82803	Butylparaben sodium Butyl parahydroxybenzoate sodium,Butyl 4-hydroxybenzoate sodium	DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	Butylparaben sodium 可通过干扰激素控制和/或破坏 RNA 及蛋白质合成来显著影响睾丸中的精子发生晚期。
TP1827L	Neuronostatin-13 human acetate Neuronostatin-13 human acetate(1096485-24-3 free base)	Others	Others
	Neuronostatin-13 human acetate(1096485-24-3 free base) 是一种 13 个氨基酸的肽类激素，在调节激素和心脏功能中起重要作用。
T83243	7'-Hydroxy ABA 7'-OH ABA
	7'-Hydroxy ABA (7'-OH ABA) 是由 Abscisic acid (Abscisic acid) 通过羟基化其7'-碳原子形成的代谢产物，具备显著的激素活性。
T11847	Liarozole dihydrochloride R75251 dihydrochloride	Others	Others
	Liarozole dihydrochloride is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase).Liarozole dihydrochloride is an imidazole derivative; it is being investigated as a non-hormonal agent in prostate cancer and in the treatment of various other cancers and skin disorders.
T74995	8′-Hydroxy ABA
	8′-Hydroxy ABA (8'-OH-ABA) 为脱落酸 (ABA) 的主要分解产物，该化合物具备激素活性，能促进油合成。然而，8′-Hydroxy ABA 是一种不稳定的化合物。
T82162	Human follicular gonadotropin releasing peptide hF-GRP
	Human follicular gonadotropin releasing peptide (hF-GRP)是一种刺激垂体分泌促黄体激素(LH)及促卵泡激素(FSH)的激素类多肽，其作用可在体外实现。
TP1552	TLQP-30
	Chronic intracerebroventricular (ICV) injection of a VGF peptide named TLQP-21 increased resting energy expenditure and temperature in mice. Furthermore, in mice fed a high-fat diet, the same peptide prevented the increase in body and white adipose tissue
T35839	3-Iodothyronamine (hydrochloride)
	3-Iodothyronamine is derived from the deiodination and decarboxylation of endogenous thyroxine. It activates the G protein-coupled receptor known as trace amine-associated receptor 1 at nanomolar concentrations whereupon it rapidly influences thyroid hormone actions including body temperature, heart rate, and cardiac output. It has also been reported to function in controlling lipid and glucose utilization, hormonal secretion, and neuronal function, and has been considered for use in chemically-...
T27289	Etacstil GW 5638,GW-5638,GW5638,DPC974,DPC 974,DPC-974
	GW5638 is a estrogen receptor ligand. GW5638 is a prodrug of its active metabolite GW7604. GW5638 appears to act as an antagonist in these in vitro systems, although in a manner distinct from other known ER modulators. GW5638 is also classified as a pseud
T71578	Endoxifen mesylate
	Endoxifen, also known as N-desmethyl-4-hydroxytamoxifen, is a chemical that is under development for estrogen receptor-positive breast cancer. It is also being evaluated as an antipsychotic for treatment of mania and other psychotic disorders. Endoxifen is a nonsteroidal selective estrogen receptor modulator (SERM) of the triphenylethylene group. It is an active metabolite of tamoxifen and has been found to be effective in patients that have failed previous hormonal therapies (tamoxifen, aromat...
T19228	Calcitriol Impurities D 24-Homo Calcitriol,24-Homo-1,25-dihydroxyvitamin D3	Antiviral	Immunology/Inflammation
	Calcitriol Impurities D (24-Homo Calcitriol) 是维生素的一种激素形式，可促进HL-60人早幼粒细胞白血病细胞分化为单核细胞。Calcitriol Impurities D 具有骨吸收活性，抑制人类免疫缺陷病毒在人体细胞中的复制。Calcitriol Impurities D 具有抗病毒活性们可以用于治疗艾滋病和病毒感染。
T65994	(6S)-N-Benzyl-6-(4-hydroxybenzyl)-8-(naphthalen-1-ylmethyl)-4,7-dioxohexahydro-2H-pyrazino[1,2-a]pyrimidine-1(6H)-carboxamide
	Wnt signaling is required for direct multiple biological processes and also plays key roles in the pathogenesis of various diseases. Cyclic AMP response element-binding protein (CREB) is a transcription factor that is a member of the leucine zipper family of DNA binding proteins. This protein binds as a homodimer to the cAMP-responsive element, an octameric palindrome. The protein is phosphorylated by several protein kinases, and induces transcription of genes in response to hormonal stimulation...

化合物

Cyproterone acetate

Cat.No: T1167

Synonym: Androcur,醋酸环丙氯地孕酮,Cyproterone 17-O-acetate,醋酸环丙孕酮

Target: Androgen Receptor

Goserelin acetate

Cat.No: T4102

Synonym: 醋酸戈舍瑞林,Fertilan,ICI-118630 acetate,Zoladex

Target: Apoptosis, GNRH Receptor

Cat.No: T1490

Synonym: SHB 331,WL 70,孕二烯酮

Target: Estrogen/progestogen Receptor, Progesterone Receptor

Testosterone undecanoate

Cat.No: T9035

Target: Others, Androgen Receptor

Cat.No: T72058L

Synonym: CDD-1102 HCl(2757619-84-2 Free base)

Target: Epigenetic Reader Domain

Cat.No: T2567

Synonym: 3-Oxodesogestrel,3-keto-Desogestrel,依托孕烯,Nexplanon,Implanon

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite

Gastrin I (1-14), human

Cat.No: TP1705

Target: Others

Cat.No: T24415

Synonym: Privaprol,L-12717,DL 717-IT,L 12717,L12717,Canocenta

Target: Others

Cat.No: T17217

Synonym: 地塞米松EP杂质E,VBP15

Target: Glucocorticoid Receptor, NF-κB

Cat.No: T0272

Synonym: 尼鲁米特,RU23908

Target: Androgen Receptor

Cat.No: T11847L

Synonym: R75251 dihydrochloride,利阿唑

Target: P450, Retinoid Receptor

4-Nonylphenol polyethoxylate

Cat.No: T0824

Synonym: Nonoxynol,Nonoxinol-9,壬苯醇醚

Target: COX

Cat.No: T68775

Cat.No: T31108

Synonym: CTP347,CTP 347

Cat.No: T19811

Cat.No: T34107

Synonym: P2525,NSC-108161,NSC 108161,P-2525,NSC108161

Cabergoline diphosphate

Cat.No: T68551

Thymus peptide C

Cat.No: TP1694

Butylparaben sodium

Cat.No: T82803

Synonym: Butyl parahydroxybenzoate sodium,Butyl 4-hydroxybenzoate sodium

Target: DNA/RNA Synthesis

Neuronostatin-13 human acetate

Cat.No: TP1827L

Synonym: Neuronostatin-13 human acetate(1096485-24-3 free base)

Target: Others

Cat.No: T83243

Synonym: 7'-OH ABA

Liarozole dihydrochloride

Cat.No: T11847

Synonym: R75251 dihydrochloride

Target: Others

8′-Hydroxy ABA

Cat.No: T74995

Human follicular gonadotropin releasing peptide

Cat.No: T82162

Synonym: hF-GRP

Cat.No: TP1552

3-Iodothyronamine (hydrochloride)

Cat.No: T35839

Cat.No: T27289

Synonym: GW 5638,GW-5638,GW5638,DPC974,DPC 974,DPC-974

Endoxifen mesylate

Cat.No: T71578

Calcitriol Impurities D

Cat.No: T19228

Synonym: 24-Homo Calcitriol,24-Homo-1,25-dihydroxyvitamin D3

Target: Antiviral

(6S)-N-Benzyl-6-(4-hydroxybenzyl)-8-(naphthalen-1-ylmethyl)-4,7-dioxohexahydro-2H-pyrazino[1,2-a]pyrimidine-1(6H)-carboxamide

Cat.No: T65994

Cat. No.	Product Name	Target	Signaling Pathways
T14853	Cabergoline FCE-21336,卡麦角林	Dopamine Receptor; 5-HT Receptor; Autophagy	Autophagy; GPCR/G Protein; Neuroscience
	Cabergoline (FCE-21336) 是一种麦角衍生的多巴胺 D2亚类受体激动剂，高亲和力作用于D2、D3和5-HT2B 受体，Ki 分别为 0.7、1.5 和 1.2。
T38515	Ascr#7
	Ascr#7, an ascaroside-based hormonal compound, plays a significant role in nematode physiology. It is specifically expressed throughout the various stages of nematode development. Notably, ascarosides exhibit the capability to initiate the formation of dauer larvae, which are characterized by their long lifespan and exceptional stress resistance.

天然产物

Cat.No: T14853

Synonym: FCE-21336,卡麦角林

Target: Dopamine Receptor, 5-HT Receptor, Autophagy

Cat.No: T38515

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