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45

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T10979 DCPIB

Potassium Channel; Chloride channel Membrane transporter/Ion channel
DCPIB 是选择性可逆体积调节性阴离子通道抑制剂,抑制肿胀激活氯电流,在 CPAE 细胞中,IC50值为 4.1 μM。它能够电压依赖性激活钾离子通道 TREK1 和 TRAAK,抑制 TRESK、TASK1 和 TASK3的 IC50值分别为 0.14、0.95 和 50.72 μM。
T16347 NS3623

Potassium Channel Membrane transporter/Ion channel
NS3623 是 hERG1 (KV11.1)钾通道激活剂,激活IKr 和Ito 电流,具有抗心律失常作用。NS3623也是 hERG1 通道抑制剂。
T16420 P-1075

Potassium Channel Membrane transporter/Ion channel
P-1075 是磺酰脲受体2相关的 ATP 敏感性的钾通道(SUR2-KIR6)的激活剂,EC50为 45 nM。它在兔子中通过打开线粒体 K (ATP) 通道产生活性氧,产生保护心脏的功效。
T14186 17-ODYA

17-十八炔酸,Alkynyl Stearic Acid

Others; PROTAC Linker Others; PROTAC
17-ODYA (Alkynyl Stearic Acid) 是 CYP450 ω-羟化酶抑制剂。它能够抑制与花生四烯酸孵育的大鼠肾皮质微粒体形成 20-HETE 、dihydroxyeicosatrienoic acids、epoxyeicosatrienoic acids。它可以改善异丙肾上腺素诱导的培养心肌细胞凋亡和坏死。
T7714 Temocapil

Tyrosinase Proteases/Proteasome
Temocapil 是一种酪氨酸激酶抑制剂。
T6698 Temocapril hydrochloride

CS-622 HCl,Acecol,Temocapril HCl,CS-622,盐酸替莫普利

RAAS Endocrinology/Hormones
Temocapril hydrochloride (CS-622 HCl) 是血管紧张素转化酶 (ACE) 抑制剂。Temocapril HCl 能够用于充血性心力衰竭、急性心肌梗死、高血压、胰岛素抵抗和肾脏疾病的研究。
T26016 R 56865

R-56865,R56865

Sodium Channel Membrane transporter/Ion channel
R 56865 是一种弱电位操作通道抑制剂,抑制人分离心肌细胞的晚期钠电流。
T8005 Cardiogenol C hydrochloride

2-[[2-[(4-甲氧基苯基)氨基]-4-嘧啶基]氨基]乙醇盐酸盐,Cardiogenol C HCl,Cardiogenol C

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
Cardiogenol C hydrochloride (Cardiogenol C) 是一种细胞渗透性嘧啶诱导剂,能够促使 ESCs 分化为心肌细胞。在有限的可塑性范围内,它可以对已经沿袭的祖细胞类型产生心肌生成效应,是一种心肌生成试剂,在动物模型中可以用作细胞移植研究中提高心脏修复的工具。
T29670 ADR-925

ICRF198,ICRF-198,ADR 925,ICRF 198,ADR925

Endogenous Metabolite Metabolism
ADR-925 (ICRF 198) 是右雷佐生的一种活性螯合铁代谢物,具有使新生大鼠心肌细胞免受阿霉素诱导的损伤的能力。
T8786 VUT-MK142

Others Others
VUT-MK142 是强效心肌合成剂,能够诱导心脏前中胚层向心肌细胞分化,促进干细胞向心肌细胞分化进行的心脏修复。
T2052 KY02111

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
KY02111 是典型的 WNT 信号抑制剂,能够促进人多潜能干细胞向心肌细胞分化,可用于研究人类心肌细胞再生。
T69760 TT-10

TAZ-K

YAP Stem Cells
TT-10 (TAZ-K) 作为YES相关蛋白(YAP)-转录增强因子结构域(TEAD)活性的激活剂,适用于心肌细胞丢失伴随心脏病研究。
T4100 AS8351

NSC51355,AS-8351,AS 8351

Histone Demethylase Chromatin/Epigenetic
AS8351 (NSC51355) 是一种组蛋白去甲基化酶抑制剂,可以诱导人胎儿肺成纤维细胞重编程为功能性心肌细胞。
T27064 CP-312

CP312,Cardioprotectant 312

Reactive Oxygen Species; Autophagy Autophagy; Immunology/Inflammation; Metabolism; NF-κB
CP-312 (Cardioprotectant 312)是一种抗氧化防御反应激活剂,它通过诱导血红素加氧酶-1发挥作用,通过诱导 HMOX1 表达来靶向抗氧化反应网络,从而保护 hiPSC-CM 的活力。CP-312 保护人 iPSC 衍生的心肌细胞免受氧化应激。
T2301 SB 202190

FHPI,SB202190

Apoptosis; p38 MAPK; Autophagy Apoptosis; Autophagy; MAPK
SB 202190 (FHPI) 是一种 p38 MAPK 抑制剂,可以抑制 p38α 和 p38β2 (IC50=50/100 nM),具有选择性和细胞渗透性。SB 202190 具有抗肿瘤活性,还可以诱导人胚胎干细胞向心肌细胞分化。
T21871 MMPSI

Caspase-3/7 Inhibitor I

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
MMPSI (Caspase-3/7 Inhibitor I) 是一种新型的、非肽类的小分子 caspase 3 和 caspase 7 抑制剂,可减少离体兔心脏或心肌细胞缺血性损伤的作用,以浓度依赖性方式抑制 H16c2 细胞凋亡 。MMPSI 可用于研究心脏保护和心肌损伤。
T30251 AZD-1305

UNII-CZO834LXQM,AZD 1305

Others Others
AZD-1305是一种新型抗心律失常化合物,主要阻断哺乳动物细胞和心室心肌细胞中 IKr 的快速组分、l 型钙电流和病房内钠电流,可用于研究逆转心律失常。
T3230 NLRP3-IN-2

5-Chloro-N-(p-sulfamoylphenethyl)-o-anisamide,4-[2-(5-氯-2-甲氧基苯甲酰氨基)乙基]苯磺酰胺,NLRP3 Inflammasome Inhibitor I

NOD-like Receptor (NLR); NOD Immunology/Inflammation; NF-κB
NLRP3-IN-2 (5-Chloro-N-(p-sulfamoylphenethyl)-o-anisamide) 是一种能够合成格列本脲的中间物,对心肌细胞中NLRP3炎症小体的形成具有抑制作用,在小鼠心肌缺血/再灌注后限制梗死面积,且对代谢无影响。
T7284 Argipressin acetate (113-79-1(free base))

Others Others
Vasopressin acetate (113-79-1(free base)) 是一种具有血管收缩和抗利尿活性的肽激素,可与血管精氨酸加压素受体 V1 结合,在 A7r5 大鼠主动脉平滑肌细胞和新生大鼠心肌细胞中的 Kd 值分别为 1.31 和 1.44 nM。
T37807 JTV 519 fumarate

Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo. Hunt et al (2007) K201 (JTV519) suppresses spontaneous Ca2+ release and [3H]ryanodine binding to RyR2 irrespective of FKBP12.6 association. Biochem.J. 404 431 PMID:17313373 |Chen et al (2008) Effect of K201, a novel antiarrhythmic drug on calcium handling and arrhythmogenic activity of pulmonary vein cardiomyocytes. Br.J.Pharmacol. 153 915 PMID:17994112 |...
T0005 Aspirin

阿司匹林,Acetylsalicylate,Acetylsalicylic Acid,邻乙酰水杨酸,ASA

Mitophagy; Virus Protease; COX; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Aspirin (Acetylsalicylic Acid) 是一种选择性 COX 抑制剂,具有多种药理活性。它是组蛋白去乙酰化酶抑制剂,可上调细胞周期阻滞蛋白 p21,抑制携带 COX-1 的卵巢 Y 细胞。 它还抑制 HUVEC 和新生大鼠心室心肌细胞中 COX-2 的表达,分别减少 PG 的产生和 ERK 和 NF-KB 的下调。
TP1219 Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate

ANP (1-28), human, porcineANP(1-28)

Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate 是颗粒鸟苷酸环化酶的刺激剂,已被发现通过增加环鸟苷单磷酸的合成来保护分离的心肌细胞免受复氧诱导的高收缩。Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate 也有助于在反复运动期间刺激脂解,并在运动期间控制脂解。
T35832 Brain Natriuretic Peptide (1-32), rat acetate

Brain Natriuretic Peptide (1-32), rat acetate (BNP (1-32), rat acetate) is a 32 amino acid polypeptide hormone synthesized by ventricular cardiomyocytes as a result of myocardial cell stretching (cardiomyocyte distension)[1].
T38354 Lactosylsphingosine (d18:1)

Lactosylsphingosine (d18:1)

Lactosylsphingosine is a bioactive sphingolipid and a form of lactosylceramide that is lacking the fatty acyl group. Lyso-lactosylceramide (1-50 μM) reduces viability of human neutrophils in a concentration-dependent manner. Unlike lactosylceramide,lactosylsphingosine has no effect on protein synthesis and cell proliferation in cardiomyocytes. Lactosylsphingosine is a precursor in the synthesis of lyso-ganglioside GM3.
T71579 GOE-5438

GOE-5438 is a calcium antagonist that has been shown to inhibit the excitation and contraction of single cardiomyocytes.
T76438 QEQLERALNSS TFA

QEQLERALNSS TFA 是一种衍生自促红细胞生成素的HBSP,具有组织保护活性,能够保护心肌细胞免受凋亡(apoptosis)。
T7434 Argipressin

Arg8-vasopressin,Vasopressin,醋酸精氨酸加压素,精氨加压素,AVP

Vasopressin Receptor GPCR/G Protein
Argipressin (Vasopressin) 是一种具有血管收缩和抗利尿活性的肽激素,可与血管精氨酸加压素受体 V1 结合,在 A7r5 大鼠主动脉平滑肌细胞和新生大鼠心肌细胞中的 Kd 值分别为 1.31 和 1.44 nM。
TP1940 Ac-RYYRIK-NH2

High affinity ligand for the NOP site (Ki = 1.5 nM). Antagonizes nociceptin-stimulated GTP binding in rat brain and the chronotropic effect of nociceptin on rat cardiomyocytes. However, displays potent agonist properties in vivo, inhibiting locomotor acti
T41232 GSK 2833503A

GSK 2833503A is a potent and selective TRPC6 and TRPC3 antagonist (IC50 = 3-16 nM and 21-100 nM, respectively). GSK 2833503A exhibits >63-fold selectivity over other ion channels, including other TRP channels, CaV1.2, hERG and NaV1.5. GSK 2833503A suppresses angiotensin II or endothelin-1-induced cardiac hypertrophy signaling in HEK293 cellsin vitroand in cardiomyocytes.
T72248 MRS2768 tetrasodium salt

MRS2768 tetrasodium salt,作为一种具有中等效力和选择性的P2Y2受体激动剂,能够保护心肌细胞免受缺血损伤。
T78377 CTP

CTP为一种具心脏靶向性的肽。它在体外能够转导心肌细胞,并能有效特异性地转导小鼠心脏组织。CTP可专门用于将治疗性肽、蛋白质及核酸传递至心脏。
TP1756 Brain Natriuretic Peptide (1-32), rat

Brain Natriuretic Peptide (BNP) (1-32), rat

Brain Natriuretic Peptide (BNP) (1-32), rat is a 32 amino acid polypeptide secreted by the ventricles of the heart in response to excessive stretching of heart muscle cells (cardiomyocytes).Brain natriuretic peptide (type B natriuretic peptide) was origin
T63452 Benidipine

Benidipine 是一种有效的、口服具有活力的钙通道拮抗剂。Benidipine 能够提高内皮细胞型一氧化氮合酶的活性,改善高血压大鼠冠状动脉循环。Benidipine 能够抗缺血/再灌注心肌细胞的凋亡。
T36218 19R(20S)-EpDPA

19R(20S)-EpDPA is an oxylipin and a metabolite of docosahexaenoic acid .1,2It is formed from DHA by various cytochrome P450 (CYP) isoforms in a stereoselective manner.219R(20S)-EpDPA (30 nM) prevents calcium-induced increases in the spontaneous beating of isolated neonatal rat cardiomyocytes (NRCMs).3 1.Cinelli, M.A., Yang, J., Scharmen, A., et al.Enzymatic synthesis and chemical inversion provide both enantiomers of bioactive epoxydocosapentaenoic acidsJ. Lipid Res.59(11)2237-2252(2018) 2.Lucas...
T76252L WLSEAGPVVTVRALRGTGSW TFA

WLSEAGPVVTVTVRALGTGSW TFA 为心肌细胞特异性肽。该化合物通过表达外泌体,提高心肌细胞的特定摄取能力,降低心肌细胞凋亡率,并在体内心肌内注射后提升心脏潴留能力。
T35592 SB 202190 hydrochloride

SB 202190 hydrochloride 是一种 p38 MAPK 抑制剂,可以抑制 p38α 和 p38β2 (IC50=50/100 nM),具有选择性和细胞渗透性。SB 202190 hydrochloride 具有抗肿瘤活性,还可以诱导人胚胎干细胞向心肌细胞分化。
T79179 GLX481304

GLX481304是一种针对Nox-2和-4的特异性抑制剂,具有1.25 μM的半抑制浓度(IC50)。它能减少离体小鼠心肌细胞中活性氧(ROS)的生成,并增强心肌收缩功能。此化合物适用于心脏缺血性损伤研究。
T80975 TMDJ-035

Calcium Channel Membrane transporter/Ion channel; Metabolism
TMDJ-035为选择性RyR2抑制剂。该化合物能够抑制携带ryr2突变的小鼠心肌细胞中异常的Ca2+波动和瞬态现象。作为研究RyR2通道开闭机制及其动力学的实验工具,TMDJ-035的应用十分关键。
T64266 KR-39038

KR-39038 是一种口服具有活力的 GRK5 (G 蛋白偶联受体激酶 5) 抑制剂 (IC50: 0.02 μM)。KR-39038 能够抑制新生儿心肌细胞的 HDAC5 通路,明显抑制血管紧张素 II 诱导的细胞肥大,具有显著的抗心肌肥厚和改善心功能作用。KR-39038 能够用于进行心力衰竭的研究。
T83043 Anti-MI/R injury agent 1

Anti-MI/R injury agent 1 (compound 18) 是一种口服有效的人参三醇衍生物,专用于抗心肌缺血/再灌注 (MI/R) 损伤。该化合物能增强经氧-葡萄糖剥夺和再灌注 (OGD/R) 诱导心肌细胞损伤模型中的细胞活力,显着缩小大鼠心肌梗死面积,减少循环心肌肌钙蛋白 I (cTnI) 的释放,并减轻心脏组织损害。
T37297 Ru360

Ru360, an oxygen-bridged dinuclear ruthenium amine complex, is a selective mitochondrial calcium uptake inhibitor. Ru360 potently inhibits Ca2+ uptake into mitochondria with an IC50 of 0.184 nM. Ru360 binds to mitochondria with high affinity (Kd of 0.34 nM). Ru360 has antiarrhythmic and cardioprotective effects[1][2]. Ru360 permeates slowly into the cell, and specifically inhibits mitochondrial calcium uptake in intact cardiomyocytes and in isolated heart. 1 μm Ru360 is taken up by myocardial ce...
T36215 17R(18S)-EpETE

17R(18S)-EpETE is an oxylipin and a cytochrome P450 metabolite of eicosapentaenoic acid .1,217R(18S)-EpETE is an activator of large-conductance calcium-activated potassium (BKCa) channels, increasing the potassium current amplitude by 15-fold in isolated rat cerebral artery vascular smooth muscle cells (VSMCs) at +60 mV when used at a concentration of 50 nM.2It has negative chronotropic effects in isolated neonatal rat cardiomyocytes (NRCMs; EC50= ~1-2 nM) and prevents calcium-induced increases ...
T35712 Debutyldronedarone hydrochloride

SR35021 hydrochloride

N-Desbutyl dronedarone is an active metabolite of the antiarrhythmic agent dronedarone .1,2,3It is formed from dronedarone by cytochrome P450s (CYPs) and monoamine oxidase (MAO) in human hepatocyte preparations.4N-Desbutyl dronedarone inhibits the binding of 3,3’,5-triiodo-L-thyronine to the thyroid hormone receptors TRα1and TRβ1(IC50s = 59 and 280 μM for the chicken and human receptors, respectively).1It inhibits CYP2J2-mediated formation of 14,15-EET from arachidonic acid and soluble epoxide h...
T37475 Cyclic ADP-Ribose (ammonium salt)

cADP-Ribose,cADPR,Cyclic ADP-Ribose (ammonium salt)

Cyclic ADP-ribose (cADP-ribose) is an endogenous metabolite of NAD+ that mobilizes the release of stored Ca2+ in the endoplasmic reticulum via ryanodine receptors in various cell types.[1],[2],[3],[4],[5] This second messenger is generated via the cADP-ribose synthases CD38 and CD157.[6],[5],[7] cADP-Ribose may also trigger the cell surface Ca2+ influx channel TRPM2 in a temperature-dependent manner.[8] In vitro, cADP-ribose modulates Ca2+ signaling in rat and mouse cardiomyocytes treated with i...
T2161 Cardiogenol C

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
Cardiogenol C 是一种细胞渗透性嘧啶诱导剂,能够诱导 ESCs 分化为心肌细胞(EC50:100 nM)。在有限的可塑性范围内,它可以对已经沿袭的祖细胞类型产生心肌病,是一种心肌发生剂。

化合物

DCPIB
Cat.No: T10979
Synonym:
Target: Potassium Channel, Chloride channel
NS3623
Cat.No: T16347
Synonym:
Target: Potassium Channel
P-1075
Cat.No: T16420
Synonym:
Target: Potassium Channel
17-ODYA
Cat.No: T14186
Synonym: 17-十八炔酸,Alkynyl Stearic Acid
Target: Others, PROTAC Linker
Temocapil
Cat.No: T7714
Synonym:
Target: Tyrosinase
Temocapril hydrochloride
Cat.No: T6698
Synonym: CS-622 HCl,Acecol,Temocapril HCl,CS-622,盐酸替莫普利
Target: RAAS
R 56865
Cat.No: T26016
Synonym: R-56865,R56865
Target: Sodium Channel
Cardiogenol C hydrochloride
Cat.No: T8005
Synonym: 2-[[2-[(4-甲氧基苯基)氨基]-4-嘧啶基]氨基]乙醇盐酸盐,Cardiogenol C HCl,Cardiogenol C
Target: Wnt/beta-catenin
ADR-925
Cat.No: T29670
Synonym: ICRF198,ICRF-198,ADR 925,ICRF 198,ADR925
Target: Endogenous Metabolite
VUT-MK142
Cat.No: T8786
Synonym:
Target: Others
KY02111
Cat.No: T2052
Synonym:
Target: Wnt/beta-catenin
TT-10
Cat.No: T69760
Synonym: TAZ-K
Target: YAP
AS8351
Cat.No: T4100
Synonym: NSC51355,AS-8351,AS 8351
Target: Histone Demethylase
CP-312
Cat.No: T27064
Synonym: CP312,Cardioprotectant 312
Target: Reactive Oxygen Species, Autophagy
SB 202190
Cat.No: T2301
Synonym: FHPI,SB202190
Target: Apoptosis, p38 MAPK, Autophagy
MMPSI
Cat.No: T21871
Synonym: Caspase-3/7 Inhibitor I
Target: Apoptosis, Caspase
AZD-1305
Cat.No: T30251
Synonym: UNII-CZO834LXQM,AZD 1305
Target: Others
NLRP3-IN-2
Cat.No: T3230
Synonym: 5-Chloro-N-(p-sulfamoylphenethyl)-o-anisamide,4-[2-(5-氯-2-甲氧基苯甲酰氨基)乙基]苯磺酰胺,NLRP3 Inflammasome Inhibitor I
Target: NOD-like Receptor (NLR), NOD
Argipressin acetate (113-79-1(free base))
Cat.No: T7284
Synonym:
Target: Others
JTV 519 fumarate
Cat.No: T37807
Synonym:
Target:
Aspirin
Cat.No: T0005
Synonym: 阿司匹林,Acetylsalicylate,Acetylsalicylic Acid,邻乙酰水杨酸,ASA
Target: Mitophagy, Virus Protease, COX, Autophagy
Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
Cat.No: TP1219
Synonym: ANP (1-28), human, porcineANP(1-28)
Target:
Brain Natriuretic Peptide (1-32), rat acetate
Cat.No: T35832
Synonym:
Target:
Lactosylsphingosine (d18:1)
Cat.No: T38354
Synonym: Lactosylsphingosine (d18:1)
Target:
GOE-5438
Cat.No: T71579
Synonym:
Target:
QEQLERALNSS TFA
Cat.No: T76438
Synonym:
Target:
Argipressin
Cat.No: T7434
Synonym: Arg8-vasopressin,Vasopressin,醋酸精氨酸加压素,精氨加压素,AVP
Target: Vasopressin Receptor
Ac-RYYRIK-NH2
Cat.No: TP1940
Synonym:
Target:
GSK 2833503A
Cat.No: T41232
Synonym:
Target:
MRS2768 tetrasodium salt
Cat.No: T72248
Synonym:
Target:
CTP
Cat.No: T78377
Synonym:
Target:
Brain Natriuretic Peptide (1-32), rat
Cat.No: TP1756
Synonym: Brain Natriuretic Peptide (BNP) (1-32), rat
Target:
Benidipine
Cat.No: T63452
Synonym:
Target:
19R(20S)-EpDPA
Cat.No: T36218
Synonym:
Target:
WLSEAGPVVTVRALRGTGSW TFA
Cat.No: T76252L
Synonym:
Target:
SB 202190 hydrochloride
Cat.No: T35592
Synonym:
Target:
GLX481304
Cat.No: T79179
Synonym:
Target:
TMDJ-035
Cat.No: T80975
Synonym:
Target: Calcium Channel
KR-39038
Cat.No: T64266
Synonym:
Target:
Anti-MI/R injury agent 1
Cat.No: T83043
Synonym:
Target:
Ru360
Cat.No: T37297
Synonym:
Target:
17R(18S)-EpETE
Cat.No: T36215
Synonym:
Target:
Debutyldronedarone hydrochloride
Cat.No: T35712
Synonym: SR35021 hydrochloride
Target:
Cyclic ADP-Ribose (ammonium salt)
Cat.No: T37475
Synonym: cADP-Ribose,cADPR,Cyclic ADP-Ribose (ammonium salt)
Target:
Cardiogenol C
Cat.No: T2161
Synonym:
Target: Wnt/beta-catenin
Cat. No. Product Name Target Signaling Pathways
T20793 Magnesium Lithospermate B

丹參酸B鎂,Monomethyl lithospermate B,丹参酸 B 镁,Lithospermate B

Others Others
Magnesium Lithospermate B 是一种咖啡酸四聚体的衍生物,从Salviae miltiorrhizae 中提取得到。它能够抑制神经炎症并减轻神经变性。它被广泛用于心血管疾病的研究,并且可以防止葡萄糖引起的细胞内氧化损伤。
TN3612 Caulophine

Others Others
Caulophine has the ability to protect cardiomyocytes from oxidative and ischemic injury through an antioxidative mechanism.
TMA0153 Safflor Yellow A

藏红花

BCL; Caspase Apoptosis; Proteases/Proteasome
Safflor Yellow A protects cultured rat cardiomyocytes against A/R injury, maybe via inhibiting cellular oxidative stress and apoptosis.
T13582 Bisandrographolide C

Others Others
Bisandrographolide C is identified from Andrographis paniculata. Bisandrographolide C activates TRPV1 and TRPV3 channels (Kds: 289 and 341 μM) and protects cardiomyocytes from hypoxia-reoxygenation injury.
TN6453 Nardoaristolone B

Nardoaristolone B, a nor-sesquiterpenoid with an unusual fused ring system and having protective effects on the injury of neonatal rat cardiomyocytes. The novel mosquito-repellentsynthetic hydrindanesbased on noreremophilanes and nardoaristolone B which s
T16885 Simvastatin acid ammonium

辛伐他汀铵盐,Tenivastatin ammonium

Others Others
Simvastatin ammonium is an active metabolite of simvastatin lactone mediated. Simvastatin ammonium reduces indoxyl sulfate-mediated reactive oxygen species and modulates OATP3A1 expression in cardiomyocytes and HEK293 cells transfected with the OATP3A1 ge
T81532 Pedaliin 6''-acetate

Pedaliin 6''-acetate (compound 10) 为甘青青兰中分离得到的天然产物,具有抗氧化活性,并能对抗DOX诱导的H9c2心肌细胞毒性,表现出细胞保护效应,其EC50为19.1 μM。
TN5639 Rocaglaol

Ferrugin,Aglaiastatin A

Rocaglaol is a potent anticancer drug that induces apoptosis of LNCaP cells through the mitochondrial pathway and its G2/M-phase cell cycle arrest is associated with the down-regulation of Cdc25C and the dephosphorylation of Cdc2. Rocaglaol can reduce tis

天然产物

Magnesium Lithospermate B
Cat.No: T20793
Synonym: 丹參酸B鎂,Monomethyl lithospermate B,丹参酸 B 镁,Lithospermate B
Target: Others
Caulophine
Cat.No: TN3612
Synonym:
Target: Others
Safflor Yellow A
Cat.No: TMA0153
Synonym: 藏红花
Target: BCL, Caspase
Bisandrographolide C
Cat.No: T13582
Synonym:
Target: Others
Nardoaristolone B
Cat.No: TN6453
Synonym:
Target:
Simvastatin acid ammonium
Cat.No: T16885
Synonym: 辛伐他汀铵盐,Tenivastatin ammonium
Target: Others
Pedaliin 6''-acetate
Cat.No: T81532
Synonym:
Target:
Rocaglaol
Cat.No: TN5639
Synonym: Ferrugin,Aglaiastatin A
Target:
TargetMol Loading
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