88
11
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1883 |
Des(benzylpyridyl) Atazanavi
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Des(benzylpyridyl) Atazanavi 是 Atazanavir 的 N-脱烷基代谢物 (M1),一种 HIV 蛋白酶抑制剂。 | |||
T7779 |
Nelfinavir
AG1341,甲磺酸萘非那韦 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Nelfinavir (AG1341) 是一种口服活性的 HIV-1 蛋白酶抑制剂,用于抑制 HIV 感染,是一种广谱抗癌剂。 | |||
T7903 |
Saquinavir
Ro 31-8959,沙奎那韦 |
SARS-CoV; HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Saquinavir (Ro 31-8959) 是一种 HIV 蛋白酶抑制剂,可研究逆转录病毒。它也是 SARS-CoV 3CLpro 抑制剂,IC50为 1.36 μM。 | |||
T1623 |
Lopinavir
ABT-378,洛匹那韦 |
SARS-CoV; HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Lopinavir (ABT-378) 是一种选择性肽模拟 HIV-1 蛋白酶的高效抑制剂。它通过阻止 HIV-1 的成熟而起作用,从而阻断其感染性。它也是 SARS-CoV 3CLpro 的抑制剂。 | |||
T9854 |
HIV-1 inhibitor-6
3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo- |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) 是一种有效的HIV-1 pre-mRNA 选择性剪接抑制剂,可以阻断HIV 复制。 | |||
T2324 |
Darunavir
地瑞那韦,达芦那韦,TMC114 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Darunavir (TMC114) 是一种 HIV 蛋白酶抑制剂,用于治疗艾滋病和 HIV 感染。 由于单独使用时会出现抗病毒药物耐药性,因此与其他抗 HIV 药物联合使用。 | |||
T6001 |
Nelfinavir Mesylate
Viracept,Nelfin,AG1343,AG 1343 Mesylate,甲磺酸奈非那韦 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Nelfinavir Mesylate (Viracept) 是一种口服活性的 HIV-1蛋白酶抑制剂,用于抑制 HIV 感染,是一种广谱抗癌剂。 | |||
T3695 |
Pepstatin
抑肽素,Pepstatin A,Pepsin Inhibitor S 735A,Ahpatinin C |
Amino Acids and Derivatives; Proteasome; HIV Protease; Autophagy | Autophagy; Metabolism; Microbiology/Virology; Proteases/Proteasome; Ubiquitination |
Pepstatin (Pepsin Inhibitor S 735A) 是由放线菌类产生的特异性天冬氨酸蛋白酶抑制剂,可抑制 HIV 蛋白酶的活性。 | |||
T6388 |
Amprenavir
141W94,安普那韦,Prozei,KVX-478,VX-478,安瑞那韦 |
SARS-CoV; HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Amprenavir (KVX-478) 是一种 HIV 蛋白酶抑制剂,Ki 为0.6 nM。它也是 SARS-CoV 3CLpro 抑制剂,IC50为 1.09 μM。 | |||
T1525 |
Ritonavir
RTV,利托那韦,Abbott 84538,A 84538,ABT 538 |
Apoptosis; SARS-CoV; HIV Protease | Apoptosis; Microbiology/Virology; Proteases/Proteasome |
Ritonavir (ABT 538) 是一种 HIV 蛋白酶抑制剂,可研究 HIV 感染和 AIDS 。它也是 SARS-CoV 3CLpro 的抑制剂,IC50为 1.61 μM。 | |||
T3335 |
Darunavir Ethanolate
地瑞那韦乙醇盐,UIC 94017,Darunavir Ethanolate,TMC114,达芦那韦乙醇 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Darunavir Ethanolate (UIC 94017) 是一种HIV 蛋白酶抑制剂,可以用于 HIV/AIDS 的相关研究。对野生型 HIV-1 蛋白酶的Ki 值为1 nM。 | |||
T0100L |
Atazanavir
Zrivada,Reyataz,Latazanavir,阿扎那韦,BMS-232632 |
P450; SARS-CoV; HIV Protease; P-gp | Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome |
Atazanavir (BMS-232632) 是一种高选择性的HIV-1蛋白酶抑制剂,可研究艾滋病毒感染。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 3.49 μM。它是CYP3A4的底物和抑制剂,也是P-糖蛋白的抑制剂和诱导剂。 | |||
T5863 |
Indinavir sulfate
L735524 sulfate,MK-639 sulfate,硫酸茚地那韦 |
SARS-CoV; HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Indinavir sulfate (L735524 sulfate) 是一种 HIV 蛋白酶抑制剂。它抑制 HIV-1 蛋白酶,IC50 值为 0.41 nM,Ki 值为 0.24 nM。它也是SARS-CoV 3CLpro 抑制剂,IC50为 1.71 μM。 | |||
T0100 |
Atazanavir sulfate
阿扎那韦硫酸盐,BMS-232632,BMS-232632 sulfate,硫酸阿扎那韦 |
P450; SARS-CoV; HIV Protease; P-gp | Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome |
Atazanavir sulfate (BMS-232632 sulfate) 是一种氮杂肽和 HIV 蛋白酶抑制剂,与其他抗 HIV 药物联合用于治疗 HIV 感染和艾滋病。它也是SARS-CoV 3CLpro 抑制剂,IC50为 3.49 μM。 | |||
T0825 |
Ebselen
SPI-1005,PZ-51,依布硒,CCG-39161 |
Phosphatase; Virus Protease; Calcium Channel; COX; HIV Protease | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome |
Ebselen (CCG-39161) 是一种谷胱甘肽过氧化物酶模拟物,是电压依赖性钙通道阻断剂。它抑制Mpro 和COVID-19病毒,是HIV-1衣壳 CTD 二聚化的抑制剂,具有抗炎、抗癌和抗氧化活性。 | |||
T8156 |
Saquinavir mesylate
沙奎拉韦,沙奎那韦甲磺酸盐,Ro 31-8959/003 |
HIV Protease; Autophagy | Autophagy; Microbiology/Virology; Proteases/Proteasome |
Saquinavir mesylate (Ro 31-8959/003) 是一种 HIV 蛋白酶抑制剂,可研究逆转录病毒。 | |||
T1776L |
Plerixafor octahydrochloride
盐酸普乐沙福,JM3100 octahydrochloride,Plerixafor 8HCl (AMD3100 8HCl),Plerixafor 8HCl,SID791 octahydrochloride,AMD 3100 octahydrochloride,JM 3100 8HCl |
Virus Protease; HIV Protease; CXCR | Autophagy; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome |
Plerixafor octahydrochloride (JM3100 octahydrochloride) 是一种选择性的CXCR4拮抗剂,IC50为 44 nM。Plerixafor 是一种具有造血干细胞动员活性的双环霉素。 | |||
T4578 |
Tipranavir
PNU-140690 |
SARS-CoV; HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Tipranavir 是一种蛋白酶抑制剂,对1种以上蛋白酶抑制剂耐药的HIV-1具有抑制作用 。Tipranavir 可有效抑制 HIV-1 蛋白酶 酶活性和二聚化,对抗多种蛋白酶抑制剂(PI)的HIV-1分离株具有有效的活性(IC50 为 66-410 nM)。Tipranavir 对SARS-CoV-2 3CLpro 活性有抑制作用。 | |||
T8238 |
Fosamprenavir Calcium Salt
福沙那伟钙,Diallyl Trisulfide,GW433908G |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Fosamprenavir Calcium Salt (GW433908G) 是抗逆转录病毒蛋白酶抑制剂 Amprenavir 的磷酸酯前药,具有改善的溶解性和抗HIV 感染作用。 | |||
T24362 |
L 756423
L756423,MK-944a,MK944a,L-756,423,L-756423,MK 944a |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
L 756423 (L756423) 是一种新型有效且具有选择性和竞争性的HIV蛋白酶抑制剂,对 HIV-1 PR 的 Ki 值为0.049 nM。L 756423 能阻止HIV(IIIb)感染的 MT25 淋巴细胞在0.50-0.1nM处的扩散,可用于研究获得性免疫缺陷综合征(AIDS)。 | |||
T26552 |
Acetylpepstatin
Ac-Val-Val-Sta-Ala-Sta-OH,Acetyl-pepstatin |
||
Acetylpepstatin is an inhibitor of HIV-1 protease, HIV-2 protease, aspartyl protease. | |||
T24536 | NIT | ||
NIT is an HIV-1 protease inhibitor. | |||
T26446 |
A 77003
A-77003,Abbott 77003,A77003 |
||
A 77003 is a HIV-1 protease inhibitor. A77003 impairs HIV-1 protease-mediated Gag processing. | |||
T26445 |
A 76889
A76889,A-76889 |
||
A 76889 is an inhibitor of HIV-1 protease. | |||
T24331 |
L 682679
L-682679,L-682,679,L682,679,L 682,679,L682679 |
||
L 682679 is an inhibitor of HIV protease. | |||
T28442 |
PPL-100
PL 461,PL461,PL-461,PPL100 |
||
PPL-100, a HIV protease inhibitor, is used potentially for the treatment of HIV infection. | |||
T16555 |
PNU-103017
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
PNU-103017 is an inhibitor of HIV protease. | |||
T24336 |
L 687908
L687908,L-687,908,L 687,908,L-687908,L687,908 |
||
L 687908 is a potent inhibitor of hydroxyethylene-containing HIV protease. | |||
T24199 |
JG 365
JG-365,JG365 |
||
JG 365 is an HIV protease inhibitor. | |||
T24343 |
L 694746
L 694,746,L694746,L-694,746,L694,746,L-694746 |
||
L 694746 is an inhibitor of HIV-1 protease. | |||
T15683 | L-689502 | HIV Protease | Microbiology/Virology; Proteases/Proteasome |
L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM). | |||
T24266 | KNI-1657 | ||
KNI-1657 is a potent and selective HIV-1 protease inhibitor (Anti-HIV-1 pNL4-3, EC50: 3 nM). KNI-1657 is a highly potent HIV-1 Protease Inhibitor against Lopinavir. | |||
T24008 |
DMP 323
JCR424,DMP-323,JCR-424,JCR 424,DMP323 |
||
DMP 323 is a potent inhibitor of HIV-1 protease. | |||
T69423 |
GRL-98065
|
||
GRL-98065 is an HIV protease inhibitor. | |||
T24361 |
L 754394
L754394,L-754,394,L 754,394,L-754394,L754,394 |
||
L 754394 is an effective and specific inhibitor of the HIV-1 protease. | |||
T26451 |
A 80987
A80987,A-80987 |
||
A 80987 is an inhibitor of HIV-1 protease. | |||
T24355 |
L 739594
L739,594,L-739,594,L 739,594,L-739594,L739594 |
||
L 739594 is an inhibitor of HIV-1 protease. | |||
T26571 |
AG-1859
AG 001859,AG 1859,AG-001859,AG001859 |
||
AG-1859, an HIV protease inhibitor, is used potentially for the treatment of HIV infection. | |||
T30839 |
Cgp 53820
Cgp53820,Cgp-53820 |
||
CGP 53820 is a pseudosymmetric inhibitor of HIV-1 Protease. | |||
T25352 |
Droxinavir HCl
SC-55389A,SC 55389A,SC55389A,Droxinavir hydrochloride |
||
Droxinavir HCl is an antiviral agent and HIV protease inhibitor. | |||
T26024 |
R 87366
R87366,R-87366 |
||
R 87366 is used as a water-soluble HIV protease inhibitor. | |||
T68277 | KNI 10033 | ||
KNI 10033 is a potent inhibitor of HIV protease | |||
T64112 | HIV-1 protease-IN-5 | ||
HIV-1 protease-IN-5 是一种 HIV-1 protease 抑制剂 (IC50: 1.64 nM)。HIV-1 protease-IN-5 对野生型和 DRV 耐药型 HIV-1 表现出明显的作用。 | |||
T69236 |
P-1946
|
||
P-1946 is an HIV-1 protease inhibitor. | |||
T30924 |
CI-1029
CI1029,PD 178390,UNII-VDH375TRL9,PD178390 |
||
CI-1029 is an HIV protease inhibitor that is effective against mutant HIV proteases and drug-resistant HIV strains. It has excellent protease activity, good antiviral efficacy in cell tests, and has good bioavailability in a variety of animal species. | |||
T70422 |
MDL-104168
|
||
MDL-104168 is a macrocyclic HIV-protease inhibitor. | |||
T27097 |
CTP518
CTP 518,Deuterated Atazanivir-D3-1,CTP-518 |
||
CTP518, a deuterated Atazanivir derivative, is a HIV protease inhibitor. | |||
T27737 |
KNI-272
NSC-651714,Kynostatin-272,Kynostatin272,KNI272,Kynostatin 272 |
||
Kynostatin-272 is a HIV protease inhibitor. KNI-272 blocked the maturation of viral particles. | |||
T15163 |
DPC-681
DPH-153893 |
Others | Others |
DPC-681 is a potent and selective HIV protease inhibitor (IC90s: 4 to 40 nM for wild-type HIV-1). | |||
T70204 |
XM 412
|
||
XM 412, also known as DMP 450, is an HIV protease inhibitor. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5783 |
Rosamultin
野蔷薇苷,罗莎白素 |
Antioxidant; HIV Protease | Microbiology/Virology; oxidation-reduction; Proteases/Proteasome |
Rosamultin 是从Potentilla anserina L 分离的 19 α-羟基型三萜。它抑制 HIV-1 蛋白酶,具有抗氧化、抗炎和镇痛作用。 | |||
TN1059 |
Ganoderic acid B
|
IL Receptor; HIV Protease; JAK; STAT | Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Microbiology/Virology; Proteases/Proteasome; Stem Cells |
Ganoderic acid B 是从灵芝中分离的一种三萜类天然产物。它是端粒酶抑制剂,抑制 Epstein-Barr 病毒抗原的活化。它是 HIV-1 蛋白酶抑制剂。 | |||
T4S1383 |
Escin IA
Aescin IA,Escin IA;Aescin IA,Escin IA |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Escin IA (Escin IA;Aescin IA);Aescin IA 是从马蹄中七叶树分离出的一种三萜皂苷,抑制HIV-1蛋白酶,IC50值为 35 μM。它具有抗 TNBC 转移活性,其作用机制涉及通过下调 LOXL2 表达抑制上皮-间质转化过程。 | |||
T4S1387 |
Isoescin IA
七叶皂苷C,异七叶皂苷 IA |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Isoescin IA 是一种从七叶树种子中分离出来的三萜皂苷。它具有抗HIV-1蛋白酶活性。 | |||
T5429 |
Theaflavin 3,3'-digallate
茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG |
Virus Protease; Antioxidant; HIV Protease; HSV | Microbiology/Virology; oxidation-reduction; Proteases/Proteasome |
Theaflavin 3,3'-digallate (8-Gingerol) 是一种寨卡病毒蛋白酶抑制剂,IC50为 2.3 μM。它直接与 ZIKVpro 结合并抑制 ZIKV 复制,可抑制 gp41 和 NS2B-3 蛋白酶的活性,并具有抗 HSV 和 HIV-1病毒活性。它是红茶中的主要多酚,有抗肿瘤作用。 | |||
T3323 |
Ursonic Acid
CCRIS 7123,NSC4060,熊果酮酸,Prunol,3-Ketoursolic acid,Malol,TOS-BB-0966 |
Apoptosis; HIV Protease; Endogenous Metabolite | Apoptosis; Metabolism; Microbiology/Virology; Proteases/Proteasome |
Ursonic Acid (TOS-BB-0966) 是一种天然三萜酸,属于熊果烷三萜类,其结构基于五环熊果烷骨架。 它具有作为 HIV-1 蛋白酶抑制剂的潜力。 | |||
T5S0983 |
Absinthin
Absinthiin,Absynthin,洋艾素 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Absinthin (Absynthin) 是结构独特的三萜类化合物,是艾草苦味高的原因。它是苦味受体hTAS2R46的激动剂,它利用 hTAS2R46 介导的受体特异性机制抑制组胺诱导的细胞内 Ca2+升高。 | |||
TN4347 |
Jacoumaric acid
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Jacoumaric acid is a lead molecule from the library or database of natural compounds as a HIV-1 protease inhibitor. | |||
T10928 |
Cytochalasin A
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Cytochalasin A is a cell-permeable fungal toxin and is an oxidized derivative of cytochalasin B. Cytochalasin A is an inhibitor of HIV-1 protease (IC50 = 3 μM), inhibits actin polymerization and interferes with microtubule assembly by reacting with sulfhy | |||
T75705 | Pepstatin Trifluoroacetate | ||
Pepstatin (Pepstatin A) Trifluoroacetate 是一种由放线菌产生的特异性天冬氨酸蛋白酶(aspartic proteases)抑制剂,口服活性强。该化合物能有效抑制hemoglobin-pepsin、hemoglobin-proctase、casein-pepsin、casein-proctase、casein-acid protease和hemoglobin-acid protease的活性,其IC50值分别为4.5 nM、6.2 nM、150 nM、290 nM、520 nM和260 nM。此外,对HIV protease也有抑制作用。 | |||
TMA1012 |
Ganoderiol F
|
Androgen Receptor; HIV Protease; Autophagy | Autophagy; Endocrinology/Hormones; Microbiology/Virology; Proteases/Proteasome |
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency virus-1 protease with IC(50) values of 20-40 microM. It induced HO-1 expression, activation of the mitogen-activated protein kinase EKR and up-regulation of cyclin-dependent kinase inhibitor p16 and suppressed lipopolysaccharide (LPS)-induced nitric oxide (NO) production. |