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抑制剂 & 化合物

11

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Cat. No. Product Name Target Signaling Pathways
T1883 Des(benzylpyridyl) Atazanavi

HIV Protease Microbiology/Virology; Proteases/Proteasome
Des(benzylpyridyl) Atazanavi 是 Atazanavir 的 N-脱烷基代谢物 (M1),一种 HIV 蛋白酶抑制剂。
T7779 Nelfinavir

AG1341,甲磺酸萘非那韦

HIV Protease Microbiology/Virology; Proteases/Proteasome
Nelfinavir (AG1341) 是一种口服活性的 HIV-1 蛋白酶抑制剂,用于抑制 HIV 感染,是一种广谱抗癌剂。
T7903 Saquinavir

Ro 31-8959,沙奎那韦

SARS-CoV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Saquinavir (Ro 31-8959) 是一种 HIV 蛋白酶抑制剂,可研究逆转录病毒。它也是 SARS-CoV 3CLpro 抑制剂,IC50为 1.36 μM。
T1623 Lopinavir

ABT-378,洛匹那韦

SARS-CoV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Lopinavir (ABT-378) 是一种选择性肽模拟 HIV-1 蛋白酶的高效抑制剂。它通过阻止 HIV-1 的成熟而起作用,从而阻断其感染性。它也是 SARS-CoV 3CLpro 的抑制剂。
T9854 HIV-1 inhibitor-6 

3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) 是一种有效的HIV-1 pre-mRNA 选择性剪接抑制剂,可以阻断HIV 复制。
T2324 Darunavir

地瑞那韦,达芦那韦,TMC114

HIV Protease Microbiology/Virology; Proteases/Proteasome
Darunavir (TMC114) 是一种 HIV 蛋白酶抑制剂,用于治疗艾滋病和 HIV 感染。 由于单独使用时会出现抗病毒药物耐药性,因此与其他抗 HIV 药物联合使用。
T6001 Nelfinavir Mesylate

Viracept,Nelfin,AG1343,AG 1343 Mesylate,甲磺酸奈非那韦

HIV Protease Microbiology/Virology; Proteases/Proteasome
Nelfinavir Mesylate (Viracept) 是一种口服活性的 HIV-1蛋白酶抑制剂,用于抑制 HIV 感染,是一种广谱抗癌剂。
T3695 Pepstatin

抑肽素,Pepstatin A,Pepsin Inhibitor S 735A,Ahpatinin C

Amino Acids and Derivatives; Proteasome; HIV Protease; Autophagy Autophagy; Metabolism; Microbiology/Virology; Proteases/Proteasome; Ubiquitination
Pepstatin (Pepsin Inhibitor S 735A) 是由放线菌类产生的特异性天冬氨酸蛋白酶抑制剂,可抑制 HIV 蛋白酶的活性。
T6388 Amprenavir

141W94,安普那韦,Prozei,KVX-478,VX-478,安瑞那韦

SARS-CoV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Amprenavir (KVX-478) 是一种 HIV 蛋白酶抑制剂,Ki 为0.6 nM。它也是 SARS-CoV 3CLpro 抑制剂,IC50为 1.09 μM。
T1525 Ritonavir

RTV,利托那韦,Abbott 84538,A 84538,ABT 538

Apoptosis; SARS-CoV; HIV Protease Apoptosis; Microbiology/Virology; Proteases/Proteasome
Ritonavir (ABT 538) 是一种 HIV 蛋白酶抑制剂,可研究 HIV 感染和 AIDS 。它也是 SARS-CoV 3CLpro 的抑制剂,IC50为 1.61 μM。
T3335 Darunavir Ethanolate

地瑞那韦乙醇盐,UIC 94017,Darunavir Ethanolate,TMC114,达芦那韦乙醇

HIV Protease Microbiology/Virology; Proteases/Proteasome
Darunavir Ethanolate (UIC 94017) 是一种HIV 蛋白酶抑制剂,可以用于 HIV/AIDS 的相关研究。对野生型 HIV-1 蛋白酶的Ki 值为1 nM。
T0100L Atazanavir

Zrivada,Reyataz,Latazanavir,阿扎那韦,BMS-232632

P450; SARS-CoV; HIV Protease; P-gp Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Atazanavir (BMS-232632) 是一种高选择性的HIV-1蛋白酶抑制剂,可研究艾滋病毒感染。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 3.49 μM。它是CYP3A4的底物和抑制剂,也是P-糖蛋白的抑制剂和诱导剂。
T5863 Indinavir sulfate

L735524 sulfate,MK-639 sulfate,硫酸茚地那韦

SARS-CoV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Indinavir sulfate (L735524 sulfate) 是一种 HIV 蛋白酶抑制剂。它抑制 HIV-1 蛋白酶,IC50 值为 0.41 nM,Ki 值为 0.24 nM。它也是SARS-CoV 3CLpro 抑制剂,IC50为 1.71 μM。
T0100 Atazanavir sulfate

阿扎那韦硫酸盐,BMS-232632,BMS-232632 sulfate,硫酸阿扎那韦

P450; SARS-CoV; HIV Protease; P-gp Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Atazanavir sulfate (BMS-232632 sulfate) 是一种氮杂肽和 HIV 蛋白酶抑制剂,与其他抗 HIV 药物联合用于治疗 HIV 感染和艾滋病。它也是SARS-CoV 3CLpro 抑制剂,IC50为 3.49 μM。
T0825 Ebselen

SPI-1005,PZ-51,依布硒,CCG-39161

Phosphatase; Virus Protease; Calcium Channel; COX; HIV Protease Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ebselen (CCG-39161) 是一种谷胱甘肽过氧化物酶模拟物,是电压依赖性钙通道阻断剂。它抑制Mpro 和COVID-19病毒,是HIV-1衣壳 CTD 二聚化的抑制剂,具有抗炎、抗癌和抗氧化活性。
T8156 Saquinavir mesylate

沙奎拉韦,沙奎那韦甲磺酸盐,Ro 31-8959/003

HIV Protease; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Saquinavir mesylate (Ro 31-8959/003) 是一种 HIV 蛋白酶抑制剂,可研究逆转录病毒。
T1776L Plerixafor octahydrochloride

盐酸普乐沙福,JM3100 octahydrochloride,Plerixafor 8HCl (AMD3100 8HCl),Plerixafor 8HCl,SID791 octahydrochloride,AMD 3100 octahydrochloride,JM 3100 8HCl

Virus Protease; HIV Protease; CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Plerixafor octahydrochloride (JM3100 octahydrochloride) 是一种选择性的CXCR4拮抗剂,IC50为 44 nM。Plerixafor 是一种具有造血干细胞动员活性的双环霉素。
T4578 Tipranavir

PNU-140690

SARS-CoV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Tipranavir 是一种蛋白酶抑制剂,对1种以上蛋白酶抑制剂耐药的HIV-1具有抑制作用 。Tipranavir 可有效抑制 HIV-1 蛋白酶 酶活性和二聚化,对抗多种蛋白酶抑制剂(PI)的HIV-1分离株具有有效的活性(IC50 为 66-410 nM)。Tipranavir 对SARS-CoV-2 3CLpro 活性有抑制作用。
T8238 Fosamprenavir Calcium Salt

福沙那伟钙,Diallyl Trisulfide,GW433908G

HIV Protease Microbiology/Virology; Proteases/Proteasome
Fosamprenavir Calcium Salt (GW433908G) 是抗逆转录病毒蛋白酶抑制剂 Amprenavir 的磷酸酯前药,具有改善的溶解性和抗HIV 感染作用。
T24362 L 756423

L756423,MK-944a,MK944a,L-756,423,L-756423,MK 944a

HIV Protease Microbiology/Virology; Proteases/Proteasome
L 756423 (L756423) 是一种新型有效且具有选择性和竞争性的HIV蛋白酶抑制剂,对 HIV-1 PR 的 Ki 值为0.049 nM。L 756423 能阻止HIV(IIIb)感染的 MT25 淋巴细胞在0.50-0.1nM处的扩散,可用于研究获得性免疫缺陷综合征(AIDS)。
T26552 Acetylpepstatin

Ac-Val-Val-Sta-Ala-Sta-OH,Acetyl-pepstatin

Acetylpepstatin is an inhibitor of HIV-1 protease, HIV-2 protease, aspartyl protease.
T24536 NIT

NIT is an HIV-1 protease inhibitor.
T26446 A 77003

A-77003,Abbott 77003,A77003

A 77003 is a HIV-1 protease inhibitor. A77003 impairs HIV-1 protease-mediated Gag processing.
T26445 A 76889

A76889,A-76889

A 76889 is an inhibitor of HIV-1 protease.
T24331 L 682679

L-682679,L-682,679,L682,679,L 682,679,L682679

L 682679 is an inhibitor of HIV protease.
T28442 PPL-100

PL 461,PL461,PL-461,PPL100

PPL-100, a HIV protease inhibitor, is used potentially for the treatment of HIV infection.
T16555 PNU-103017

HIV Protease Microbiology/Virology; Proteases/Proteasome
PNU-103017 is an inhibitor of HIV protease.
T24336 L 687908

L687908,L-687,908,L 687,908,L-687908,L687,908

L 687908 is a potent inhibitor of hydroxyethylene-containing HIV protease.
T24199 JG 365

JG-365,JG365

JG 365 is an HIV protease inhibitor.
T24343 L 694746

L 694,746,L694746,L-694,746,L694,746,L-694746

L 694746 is an inhibitor of HIV-1 protease.
T15683 L-689502

HIV Protease Microbiology/Virology; Proteases/Proteasome
L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM).
T24266 KNI-1657

KNI-1657 is a potent and selective HIV-1 protease inhibitor (Anti-HIV-1 pNL4-3, EC50: 3 nM). KNI-1657 is a highly potent HIV-1 Protease Inhibitor against Lopinavir.
T24008 DMP 323

JCR424,DMP-323,JCR-424,JCR 424,DMP323

DMP 323 is a potent inhibitor of HIV-1 protease.
T69423 GRL-98065

GRL-98065 is an HIV protease inhibitor.
T24361 L 754394

L754394,L-754,394,L 754,394,L-754394,L754,394

L 754394 is an effective and specific inhibitor of the HIV-1 protease.
T26451 A 80987

A80987,A-80987

A 80987 is an inhibitor of HIV-1 protease.
T24355 L 739594

L739,594,L-739,594,L 739,594,L-739594,L739594

L 739594 is an inhibitor of HIV-1 protease.
T26571 AG-1859

AG 001859,AG 1859,AG-001859,AG001859

AG-1859, an HIV protease inhibitor, is used potentially for the treatment of HIV infection.
T30839 Cgp 53820

Cgp53820,Cgp-53820

CGP 53820 is a pseudosymmetric inhibitor of HIV-1 Protease.
T25352 Droxinavir HCl

SC-55389A,SC 55389A,SC55389A,Droxinavir hydrochloride

Droxinavir HCl is an antiviral agent and HIV protease inhibitor.
T26024 R 87366

R87366,R-87366

R 87366 is used as a water-soluble HIV protease inhibitor.
T68277 KNI 10033

KNI 10033 is a potent inhibitor of HIV protease
T64112 HIV-1 protease-IN-5

HIV-1 protease-IN-5 是一种 HIV-1 protease 抑制剂 (IC50: 1.64 nM)。HIV-1 protease-IN-5 对野生型和 DRV 耐药型 HIV-1 表现出明显的作用。
T69236 P-1946

P-1946 is an HIV-1 protease inhibitor.
T30924 CI-1029

CI1029,PD 178390,UNII-VDH375TRL9,PD178390

CI-1029 is an HIV protease inhibitor that is effective against mutant HIV proteases and drug-resistant HIV strains. It has excellent protease activity, good antiviral efficacy in cell tests, and has good bioavailability in a variety of animal species.
T70422 MDL-104168

MDL-104168 is a macrocyclic HIV-protease inhibitor.
T27097 CTP518

CTP 518,Deuterated Atazanivir-D3-1,CTP-518

CTP518, a deuterated Atazanivir derivative, is a HIV protease inhibitor.
T27737 KNI-272

NSC-651714,Kynostatin-272,Kynostatin272,KNI272,Kynostatin 272

Kynostatin-272 is a HIV protease inhibitor. KNI-272 blocked the maturation of viral particles.
T15163 DPC-681

DPH-153893

Others Others
DPC-681 is a potent and selective HIV protease inhibitor (IC90s: 4 to 40 nM for wild-type HIV-1).
T70204 XM 412

XM 412, also known as DMP 450, is an HIV protease inhibitor.

化合物

Des(benzylpyridyl) Atazanavi
Cat.No: T1883
Synonym:
Target: HIV Protease
Nelfinavir
Cat.No: T7779
Synonym: AG1341,甲磺酸萘非那韦
Target: HIV Protease
Saquinavir
Cat.No: T7903
Synonym: Ro 31-8959,沙奎那韦
Target: SARS-CoV, HIV Protease
Lopinavir
Cat.No: T1623
Synonym: ABT-378,洛匹那韦
Target: SARS-CoV, HIV Protease
HIV-1 inhibitor-6 
Cat.No: T9854
Synonym: 3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-
Target: HIV Protease
Darunavir
Cat.No: T2324
Synonym: 地瑞那韦,达芦那韦,TMC114
Target: HIV Protease
Nelfinavir Mesylate
Cat.No: T6001
Synonym: Viracept,Nelfin,AG1343,AG 1343 Mesylate,甲磺酸奈非那韦
Target: HIV Protease
Pepstatin
Cat.No: T3695
Synonym: 抑肽素,Pepstatin A,Pepsin Inhibitor S 735A,Ahpatinin C
Target: Amino Acids and Derivatives, Proteasome, HIV Protease, Autophagy
Amprenavir
Cat.No: T6388
Synonym: 141W94,安普那韦,Prozei,KVX-478,VX-478,安瑞那韦
Target: SARS-CoV, HIV Protease
Ritonavir
Cat.No: T1525
Synonym: RTV,利托那韦,Abbott 84538,A 84538,ABT 538
Target: Apoptosis, SARS-CoV, HIV Protease
Darunavir Ethanolate
Cat.No: T3335
Synonym: 地瑞那韦乙醇盐,UIC 94017,Darunavir Ethanolate,TMC114,达芦那韦乙醇
Target: HIV Protease
Atazanavir
Cat.No: T0100L
Synonym: Zrivada,Reyataz,Latazanavir,阿扎那韦,BMS-232632
Target: P450, SARS-CoV, HIV Protease, P-gp
Indinavir sulfate
Cat.No: T5863
Synonym: L735524 sulfate,MK-639 sulfate,硫酸茚地那韦
Target: SARS-CoV, HIV Protease
Atazanavir sulfate
Cat.No: T0100
Synonym: 阿扎那韦硫酸盐,BMS-232632,BMS-232632 sulfate,硫酸阿扎那韦
Target: P450, SARS-CoV, HIV Protease, P-gp
Ebselen
Cat.No: T0825
Synonym: SPI-1005,PZ-51,依布硒,CCG-39161
Target: Phosphatase, Virus Protease, Calcium Channel, COX, HIV Protease
Saquinavir mesylate
Cat.No: T8156
Synonym: 沙奎拉韦,沙奎那韦甲磺酸盐,Ro 31-8959/003
Target: HIV Protease, Autophagy
Plerixafor octahydrochloride
Cat.No: T1776L
Synonym: 盐酸普乐沙福,JM3100 octahydrochloride,Plerixafor 8HCl (AMD3100 8HCl),Plerixafor 8HCl,SID791 octahydrochloride,AMD 3100 octahydrochloride,JM 3100 8HCl
Target: Virus Protease, HIV Protease, CXCR
Tipranavir
Cat.No: T4578
Synonym: PNU-140690
Target: SARS-CoV, HIV Protease
Fosamprenavir Calcium Salt
Cat.No: T8238
Synonym: 福沙那伟钙,Diallyl Trisulfide,GW433908G
Target: HIV Protease
L 756423
Cat.No: T24362
Synonym: L756423,MK-944a,MK944a,L-756,423,L-756423,MK 944a
Target: HIV Protease
Acetylpepstatin
Cat.No: T26552
Synonym: Ac-Val-Val-Sta-Ala-Sta-OH,Acetyl-pepstatin
Target:
NIT
Cat.No: T24536
Synonym:
Target:
A 77003
Cat.No: T26446
Synonym: A-77003,Abbott 77003,A77003
Target:
A 76889
Cat.No: T26445
Synonym: A76889,A-76889
Target:
L 682679
Cat.No: T24331
Synonym: L-682679,L-682,679,L682,679,L 682,679,L682679
Target:
PPL-100
Cat.No: T28442
Synonym: PL 461,PL461,PL-461,PPL100
Target:
PNU-103017
Cat.No: T16555
Synonym:
Target: HIV Protease
L 687908
Cat.No: T24336
Synonym: L687908,L-687,908,L 687,908,L-687908,L687,908
Target:
JG 365
Cat.No: T24199
Synonym: JG-365,JG365
Target:
L 694746
Cat.No: T24343
Synonym: L 694,746,L694746,L-694,746,L694,746,L-694746
Target:
L-689502
Cat.No: T15683
Synonym:
Target: HIV Protease
KNI-1657
Cat.No: T24266
Synonym:
Target:
DMP 323
Cat.No: T24008
Synonym: JCR424,DMP-323,JCR-424,JCR 424,DMP323
Target:
GRL-98065
Cat.No: T69423
Synonym:
Target:
L 754394
Cat.No: T24361
Synonym: L754394,L-754,394,L 754,394,L-754394,L754,394
Target:
A 80987
Cat.No: T26451
Synonym: A80987,A-80987
Target:
L 739594
Cat.No: T24355
Synonym: L739,594,L-739,594,L 739,594,L-739594,L739594
Target:
AG-1859
Cat.No: T26571
Synonym: AG 001859,AG 1859,AG-001859,AG001859
Target:
Cgp 53820
Cat.No: T30839
Synonym: Cgp53820,Cgp-53820
Target:
Droxinavir HCl
Cat.No: T25352
Synonym: SC-55389A,SC 55389A,SC55389A,Droxinavir hydrochloride
Target:
R 87366
Cat.No: T26024
Synonym: R87366,R-87366
Target:
KNI 10033
Cat.No: T68277
Synonym:
Target:
HIV-1 protease-IN-5
Cat.No: T64112
Synonym:
Target:
P-1946
Cat.No: T69236
Synonym:
Target:
CI-1029
Cat.No: T30924
Synonym: CI1029,PD 178390,UNII-VDH375TRL9,PD178390
Target:
MDL-104168
Cat.No: T70422
Synonym:
Target:
CTP518
Cat.No: T27097
Synonym: CTP 518,Deuterated Atazanivir-D3-1,CTP-518
Target:
KNI-272
Cat.No: T27737
Synonym: NSC-651714,Kynostatin-272,Kynostatin272,KNI272,Kynostatin 272
Target:
DPC-681
Cat.No: T15163
Synonym: DPH-153893
Target: Others
XM 412
Cat.No: T70204
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5783 Rosamultin

野蔷薇苷,罗莎白素

Antioxidant; HIV Protease Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Rosamultin 是从Potentilla anserina L 分离的 19 α-羟基型三萜。它抑制 HIV-1 蛋白酶,具有抗氧化、抗炎和镇痛作用。
TN1059 Ganoderic acid B

IL Receptor; HIV Protease; JAK; STAT Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Microbiology/Virology; Proteases/Proteasome; Stem Cells
Ganoderic acid B 是从灵芝中分离的一种三萜类天然产物。它是端粒酶抑制剂,抑制 Epstein-Barr 病毒抗原的活化。它是 HIV-1 蛋白酶抑制剂。
T4S1383 Escin IA

Aescin IA,Escin IA;Aescin IA,Escin IA

HIV Protease Microbiology/Virology; Proteases/Proteasome
Escin IA (Escin IA;Aescin IA);Aescin IA 是从马蹄中七叶树分离出的一种三萜皂苷,抑制HIV-1蛋白酶,IC50值为 35 μM。它具有抗 TNBC 转移活性,其作用机制涉及通过下调 LOXL2 表达抑制上皮-间质转化过程。
T4S1387 Isoescin IA

七叶皂苷C,异七叶皂苷 IA

HIV Protease Microbiology/Virology; Proteases/Proteasome
Isoescin IA 是一种从七叶树种子中分离出来的三萜皂苷。它具有抗HIV-1蛋白酶活性。
T5429 Theaflavin 3,3'-digallate

茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG

Virus Protease; Antioxidant; HIV Protease; HSV Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Theaflavin 3,3'-digallate (8-Gingerol) 是一种寨卡病毒蛋白酶抑制剂,IC50为 2.3 μM。它直接与 ZIKVpro 结合并抑制 ZIKV 复制,可抑制 gp41 和 NS2B-3 蛋白酶的活性,并具有抗 HSV 和 HIV-1病毒活性。它是红茶中的主要多酚,有抗肿瘤作用。
T3323 Ursonic Acid

CCRIS 7123,NSC4060,熊果酮酸,Prunol,3-Ketoursolic acid,Malol,TOS-BB-0966

Apoptosis; HIV Protease; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology; Proteases/Proteasome
Ursonic Acid (TOS-BB-0966) 是一种天然三萜酸,属于熊果烷三萜类,其结构基于五环熊果烷骨架。 它具有作为 HIV-1 蛋白酶抑制剂的潜力。
T5S0983 Absinthin

Absinthiin,Absynthin,洋艾素

HIV Protease Microbiology/Virology; Proteases/Proteasome
Absinthin (Absynthin) 是结构独特的三萜类化合物,是艾草苦味高的原因。它是苦味受体hTAS2R46的激动剂,它利用 hTAS2R46 介导的受体特异性机制抑制组胺诱导的细胞内 Ca2+升高。
TN4347 Jacoumaric acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
Jacoumaric acid is a lead molecule from the library or database of natural compounds as a HIV-1 protease inhibitor.
T10928 Cytochalasin A

HIV Protease Microbiology/Virology; Proteases/Proteasome
Cytochalasin A is a cell-permeable fungal toxin and is an oxidized derivative of cytochalasin B. Cytochalasin A is an inhibitor of HIV-1 protease (IC50 = 3 μM), inhibits actin polymerization and interferes with microtubule assembly by reacting with sulfhy
T75705 Pepstatin Trifluoroacetate

Pepstatin (Pepstatin A) Trifluoroacetate 是一种由放线菌产生的特异性天冬氨酸蛋白酶(aspartic proteases)抑制剂,口服活性强。该化合物能有效抑制hemoglobin-pepsin、hemoglobin-proctase、casein-pepsin、casein-proctase、casein-acid protease和hemoglobin-acid protease的活性,其IC50值分别为4.5 nM、6.2 nM、150 nM、290 nM、520 nM和260 nM。此外,对HIV protease也有抑制作用。
TMA1012 Ganoderiol F

Androgen Receptor; HIV Protease; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology; Proteases/Proteasome
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency virus-1 protease with IC(50) values of 20-40 microM. It induced HO-1 expression, activation of the mitogen-activated protein kinase EKR and up-regulation of cyclin-dependent kinase inhibitor p16 and suppressed lipopolysaccharide (LPS)-induced nitric oxide (NO) production.

天然产物

Rosamultin
Cat.No: T5783
Synonym: 野蔷薇苷,罗莎白素
Target: Antioxidant, HIV Protease
Ganoderic acid B
Cat.No: TN1059
Synonym:
Target: IL Receptor, HIV Protease, JAK, STAT
Escin IA
Cat.No: T4S1383
Synonym: Aescin IA,Escin IA;Aescin IA,Escin IA
Target: HIV Protease
Isoescin IA
Cat.No: T4S1387
Synonym: 七叶皂苷C,异七叶皂苷 IA
Target: HIV Protease
Theaflavin 3,3'-digallate
Cat.No: T5429
Synonym: 茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG
Target: Virus Protease, Antioxidant, HIV Protease, HSV
Ursonic Acid
Cat.No: T3323
Synonym: CCRIS 7123,NSC4060,熊果酮酸,Prunol,3-Ketoursolic acid,Malol,TOS-BB-0966
Target: Apoptosis, HIV Protease, Endogenous Metabolite
Absinthin
Cat.No: T5S0983
Synonym: Absinthiin,Absynthin,洋艾素
Target: HIV Protease
Jacoumaric acid
Cat.No: TN4347
Synonym:
Target: HIV Protease
Cytochalasin A
Cat.No: T10928
Synonym:
Target: HIV Protease
Pepstatin Trifluoroacetate
Cat.No: T75705
Synonym:
Target:
Ganoderiol F
Cat.No: TMA1012
Synonym:
Target: Androgen Receptor, HIV Protease, Autophagy
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