187
22
Cat. No. | Product Name | Target | Signaling Pathways |
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T22831 |
Protein kinase inhibitor H-7 dihydrochloride
H-7 dihydrochloride |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride0) 是一种有效的蛋白激酶 C(PKC)抑制剂。Protein kinase inhibitor H-7 dihydrochloride(100 μM)显著抑制 TPA (皮肤肿瘤启动子,12-O-tetradecanoylphorbol-13-acetate) 和磷脂酶 C 促使的 ODC (鸟氨酸脱羧酶),抑制 PMA 诱导的混杂细胞溶解活性。 | |||
T41267 |
PROTAC(H-PGDS)-7
|
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PROTAC(H-PGDS)-7 是一种有选择性的、有效的小分子造血前列腺素 D 合酶 (H-PGDS)PROTAC 降解剂,在 KU812细胞中展现出降解活性,DC50为 17.3 pM。PROTAC(H-PGDS)-7是一种类药化合物,能有效抑制前列腺素 D2 (PGD2)的产生,抑制炎症因子重生作用。PROTAC(H-PGDS)-7是治疗 DMD 和其他H-PGDS 相关疾病的候选化合物。 | |||
T60109 |
Protein kinase inhibitor H-7
5-(2-methylpiperazine-1-sulfonyl)isoquinoline,蛋白激酶抑制剂H-7,1-(5-Isoquinolinylsulfonyl)-2-methylpiperazine |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
Protein kinase inhibitor H-7 (5-(2-methylpiperazine-1-sulfonyl)isoquinoline) 是有效的蛋白激酶 C (PKC) 和环核苷酸依赖性蛋白激酶抑制剂,抑制 PKC 的 Ki 值为 6 μM。 | |||
T9308 |
AzoMethine-H Monosodium salt hydrate
Sodium 5-hydroxy-4-((2-hydroxybenzylidene)amino)-7-sulfonaphthalene-2-sulfonate hydrate,偶氮甲碱-H 单钠盐 水合物 |
Others | Others |
AzoMethine-H Monosodium salt hydrate (Sodium 5-hydroxy-4-((2-hydroxybenzylidene)amino)-7-sulfonaphthalene-2-sulfonate hydrate) 是一种试剂,用于比色测定土壤、植物、堆肥、肥料、水和营养液中的硼。 | |||
T15458 |
H2DCFDA
2',7'-二氯荧光素二乙酸酯,2',7'-Dichlorodihydrofluorescein diacetate,DCFH-DA |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
H2DCFDA (DCFH-DA) 属于绿色荧光染料,是一种检测细胞内活性氧 (ROS) 的探针 (Ex/Em=488/525 nm),具有细胞膜渗透性。 | |||
T38766L |
Histone H3 (1-35) acetate
|
Others | Others |
Histone H3 (1-35) acetate 是组蛋白 H3 的 35 个残基肽。组蛋白 H3 是一种重要的蛋白质,在基因的动态和长期调控中发挥作用。 | |||
T7501 |
Iso-H7 dihydrochloride
1-(5-硫代异喹啉)-3-甲基哌嗪二盐酸盐 |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
与 H-7 相比,Iso-H7 dihydrochloride 是一种较弱的磷酸激酶 C 抑制剂。 | |||
T77692 |
F7H
|
Wnt/beta-catenin; Antibacterial | Cytoskeletal Signaling; Microbiology/Virology; Stem Cells |
F7H 是一种有效的卷曲蛋白受体 (Frizzled receptor) FZD7 拮抗剂,IC50 值为 1.25 μM。F7H 是一种有效的 FZD7 跨膜结构域 (TMD) 的配体,具有潜在的抗肿瘤和抑菌活性。 | |||
T68950 | Hepta-histidine | ||
Hepta-histidine is a novel inhibitor of Tau aggregation against Tau-related neurodegenerative diseases including Alzheimer's disease (AD). | |||
T18998 |
H-L-Photo-lysine hydrochloride
H-L-Photo-lysine hydrochloride (1253643-88-7 free base) |
Others | Others |
H-L-Photo-lysine hydrochloride, a photo-cross-linker, is a diazirine-containing lysine amino acid. It can site-selective incorporated into proteins and is used to crosslink protein-protein interactions in vitro and in living cells. | |||
T6928 |
Pantoprazole
SKF96022,泮托拉唑,BY1023 |
Apoptosis; Proton pump; Autophagy | Apoptosis; Autophagy; Membrane transporter/Ion channel |
Pantoprazole (BY1023) 是一种质子泵抑制剂,用于短期治疗由胃食管反流病引起的食管糜烂和溃疡。它联合阿霉素可显著增加肿瘤生长延迟。它是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。 | |||
T5887 |
7-Hydroxy-3,4-dihydro-2(1H)-quinolinone
3,4-Dihydro-7-hydroxy-2(1H)-quinolinone,3,4-二氢-7-羟基-2(1H)-喹啉酮 |
MAO; Monoamine Oxidase | Metabolism; Neuroscience |
7-Hydroxy-3,4-dihydro-2(1H)-quinolinone 是弱MAO-A 抑制剂,IC50=183 μM,对 MAO-B 无作用。 | |||
T9571 |
2,4,5-Trichloro-7H-pyrrolo[2,3-d]pyrimid
|
Others | Others |
2,4,5-Trichloro-7H-pyrrolo[2,3-d]pyrimid 是一种化学试剂。 | |||
TD0076 |
AMCA-H N-succinimidyl ester
7-Hydroxy-4-methylcoumarin-3-acetic acid, succinimidyl ester,7-羟基-4-甲基香豆素-3-乙酸琥珀酰亚胺酯 |
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The amine-reactive AMCA, SE (7-amino-4-methylcoumarin-3-acetic acid, succinimidyl ester) and its conjugates yield blue-fluorescence (approximate excitation/emission maxima ~353/442) that can be used as a contrasting color in multicolor applications. | |||
T1909 |
L-701324
7-氯-4-羟基-3-(3-苯氧基)苯基-2(1H)-喹啉,L701324 |
NMDAR; iGluR | Membrane transporter/Ion channel; Neuroscience |
L-701324 是一种 NMDA 受体,对甘氨酸位点具有高亲和力和选择性,用作口服活性和长效抗惊厥药。 | |||
T0161 |
Pantoprazole Sodium Hydrate
SKF96022 sodium hydrate,泮托拉唑钠水合物,BY1023 (sodium hydrate),SKF96022 (sodium hydrate) |
Apoptosis; Potassium Channel; Proton pump; Autophagy | Apoptosis; Autophagy; Membrane transporter/Ion channel |
Pantoprazole Sodium Hydrate (BY1023 (sodium hydrate)) 是一种具有口服活性的质子泵抑制剂。它是取代的苯并咪唑,是H+/K+-ATPase 抑制剂。它可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。 | |||
T36260 | NR 7h | ||
Potent and selective p38α and p38β degrader (DC50 < 50 nM). Displays no significant degradation of p38γ, p38δ, JNK1/2 or ERK1/2. Inhibits phosphorylation of MK2 in UV-treated cancer cells and LPS-stimulated bone marrow-derived macrophages (BMDM). Exhibits similar effect to p38α gene knockout in BBL358 cells. Active in vivo. | |||
T6929 |
Pantoprazole sodium
Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc |
Apoptosis; Others; Proton pump; HIF; Autophagy | Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Others |
Pantoprazole sodium (Pantecta) 是一种具有口服活性的质子泵抑制剂,是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,IC50为 6.8 μM。它可以改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。 | |||
T11760 |
KIN101
3-(4-Bromophenyl)-7-[(methylsulfonyl)oxy]-4-oxo-4H-chromene,3-(4-溴苯基)-4-氧代-7-[(甲磺酰基)氧基]-4H-色烯 |
HCV Protease; Influenza Virus; RSV; Antifection | Microbiology/Virology; Proteases/Proteasome |
KIN101 (3-(4-Bromophenyl)-7-[(methylsulfonyl)oxy]-4-oxo-4H-chromene) 是 IRF-3 依赖性信号传导的异黄酮激动剂,可诱导 IRF-3 核易位。 它对 RNA 病毒、HCV 和 RSV 具有抗病毒活性。 | |||
T82246 |
H7
|
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H7为第二型近红外(NIR-II)荧光团。 | |||
T21527 |
HBX 41108
HBX-41108,7-氯-9-氧代-9H-茚并[1,2-B]吡嗪-2,3-二甲腈 |
DUB; p53 | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination |
HBX 41108 (HBX-41108) 是一种泛素特异性蛋白酶 7 的非竞争性抑制剂,IC50为 424 nM。它诱导 p53 依赖的凋亡,抑制 USP7 介导的 p53 去泛素化以稳定 p53 并抑制癌细胞生长。 | |||
T76381 |
H1-7 (histone H1 phosphorylation site), PKA Substrate
|
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H1-7 (histone H1 phosphorylation site),PKASubstrate 是一种合成多肽,可作为PKA 底物。 | |||
T124870 | 2H-1-Benzopyran-7-yloxy | ||
2H-1-Benzopyran-7-yloxy 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124870。 | |||
T65517 | 4-Chloro-7-tosyl-7H-pyrrolo[2,3-d]pyrimidine | ||
4-Chloro-7-tosyl-7H-pyrrolo[2,3-d]pyrimidine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65517,CAS号为 479633-63-1。 | |||
T65626 |
8-Bromo-3-methyl-1H-purine-2,6(3H,7H)-dione
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8-Bromo-3-methyl-1H-purine-2,6(3H,7H)-dione 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65626,CAS号为 93703-24-3。 | |||
T64948 | 7-Amino-2H-chromen-2-one | ||
7-Amino-2H-chromen-2-one 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64948。 | |||
T125949 |
7-[(7-Methoxy-3,7-dimethyl-2,5-octadienyl)oxy]-2H-
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7-[(7-Methoxy-3,7-dimethyl-2,5-octadienyl)oxy]-2H- 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125949,CAS号为 1388140-07-5。 | |||
TNU1027 | 7-Deaza-2’-deoxyguanosine; 2-Amino-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidin-4(3H)-one | ||
Nucleoside Derivatives - 7-Deaza-purine nucleoside | |||
T64449 | rel-(3aR,4S,7R,7aS)-3a,4,7,7a-Tetrahydro-1H-4,7-methanoisoindole-1,3(2H)-dione | ||
rel-(3aR,4S,7R,7aS)-3a,4,7,7a-Tetrahydro-1H-4,7-methanoisoindole-1,3(2H)-dione 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64449,CAS号为 6265-30-1。 | |||
TNU1026 |
7-(2-Deoxy-β-D-erythro-pentofuranosyl)-5-fluoro-7H-pyrrolo[2,3-d]pyrimidin-4-amine
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Nucleoside Derivatives - Fluoro-modified nucleosides, 7-Deaza-purine nucleosides | |||
T60186 |
(S)-4-methyl-N-(3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-2-(pyrimidin-5-yl)-1,2,3,4-tetrahydroisoquinoline-7-carboxamide
|
Discoidin Domain Receptor (DDR) | Tyrosine Kinase/Adaptors |
MitoBloCK-6 是一种有效的 Erv1/ALR 抑制剂,IC50 分别为 900 nM 和 700 nM。MitoBloCK-6 还抑制 Erv2 (IC50=1.4 μM)。MitoBloCK-6 可通过细胞色素 c 的释放诱导 hESCs 细胞凋亡。 | |||
T66320 |
8-Bromo-7-(but-2-yn-1-yl)-3-methyl-1-((4-methylquinazolin-2-yl)methyl)-1H-purine-2,6(3H,7H)-dione
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8-Bromo-7-(but-2-yn-1-yl)-3-methyl-1-((4-methylquinazolin-2-yl)methyl)-1H-purine-2,6(3H,7H)-dione 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66320,CAS号为 853029-57-9。 | |||
TNU1032 |
7-(2-Deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine
|
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Nucleoside Derivatives - 7-Deaza-purine nucleosides; 6-De-aminopurine nucleosides | |||
T75332 |
7-Hydroxy-4-methyl-2(1H)-quinolone
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7-Hydroxy-4-methyl-2(1H)-quinolone (compound 2b) 是一种荧光产物,主要用于检测 DNA 损伤的羟基自由基。储存时需避光。 | |||
T126216 |
1α,7α,10αH-Guaia-4,11-dien-3-one
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1α,7α,10αH-Guaia-4,11-dien-3-one 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126216。 | |||
TNU1022 |
4-Chloro-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]-pyrimidine
|
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4-Chloro-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]-pyrimidine is a Nucleoside Derivative - Halo-nucleoside, 7-Deaza-purine nucleoside. | |||
T66262 |
7-(Diethylamino)-4-methyl-2H-chromen-2-one
|
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7-(Diethylamino)-4-methyl-2H-chromen-2-one 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66262,CAS号为 91-44-1。 | |||
T131535 | 3-formyl-4-oxo-4H-chromen-7-yl acetate | ||
3-formyl-4-oxo-4H-chromen-7-yl acetate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131535。 | |||
T67616 |
4-(Chloromethyl)-7-hydroxy-2H-chromen-2-one
|
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4-(Chloromethyl)-7-hydroxy-2H-chromen-2-one 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67616,CAS号为 25392-41-0。 | |||
T65771 |
1,7'-Dimethyl-2'-propyl-1H,1'H-2,5'-bibenzo[d]imidazole
|
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1,7'-Dimethyl-2'-propyl-1H,1'H-2,5'-bibenzo[d]imidazole 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65771,CAS号为 152628-02-9。 | |||
T66608 |
2,4-Dichloro-7H-pyrrolo[2,3-d]pyrimidine
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2,4-Dichloro-7H-pyrrolo[2,3-d]pyrimidine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66608,CAS号为 90213-66-4。 | |||
TNU1262 |
1H-Imidazo[4,5-d]pyridazin-7-amine
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1H-Imidazo[4,5-d]pyridazin-7-amine belongs to Heterocyclic Compounds - Purines; Intermediates and Building Blocks - Nucleoside bases. | |||
TNU0055 |
6-Chloro-7-deazapurine-2F-β-D-arabinofuranose
|
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6-Chloro-7-deazapurine-2F-β-D-arabinofuranose is a Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, halo nucleoside; Arabino-nucleoside. | |||
TNU0056 | 2’-Deoxy-2’-fluoro-arabino-tubercidine | ||
Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, Arabino-nucleoside | |||
TNU1069 |
4-Chloro-7-(2,3-O-isopropylidene-β-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine
|
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Nucleoside Derivatives - 7-Deaza-purine nucleoside; Halo-nucleoside, Protected nucleosides with NH2/OH open; Scaffolds and Template | |||
TNU1025 |
4-Chloro-5-iodo-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine
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4-Chloro-5-iodo-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine is a Nucleoside Derivative - Halo-nucleoside, 7-Deaza-purine nucleoside. | |||
TNU0102 |
4-Chloro-7-(2-b-C-methyl-β-D-ribofuranosyl)-7H-pyrrolo[2,3-d] pyrimidine
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4-Chloro-7-(2-b-C-methyl-β-D-ribofuranosyl)-7H-pyrrolo[2,3-d] pyrimidine is a Nucleoside Derivative - 7-Deaza-purine nucleoside; 2'-Modified nucleoside; Halo-nucleoside; Scaffold and Template. | |||
TNU0717 |
4-Chloro-5-iodo-7H-pyrrol[2,3-d]pyrimidine
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Heterocyclic compound - purine; Intermediate and building blocks– electrophile and nucleophile; Nucleoside base | |||
T125498 |
7-Methoxy-8-(3-methyl-2-oxobutoxy)-2H-1-benzopyran
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7-Methoxy-8-(3-methyl-2-oxobutoxy)-2H-1-benzopyran 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125498,CAS号为 188426-72-4。 | |||
T65919 |
7-(4-Bromobutoxy)-3,4-dihydroquinolin-2(1H)-one
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7-(4-Bromobutoxy)-3,4-dihydroquinolin-2(1H)-one 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65919,CAS号为 129722-34-5。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T1116 |
Biotin
Vitamin B7,生物素,D-Biotin,Vitamin H,D-生物素(维生素H) |
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Biotin (Vitamin H) 是一种水溶性B族维生素,是细胞生长、脂肪酸产生以及脂肪和氨基酸代谢所必需的。 | |||
T3798 |
Ziyuglycoside I
Gouguside 7,Ziyu-glycoside I,3-O-alpha-L-Arabinopyranosylpomolic acid beta-D-glucopyranosyl ester,地榆皂苷 I,苦丁冬青甙 H,Zigu-glucoside I,Kudinoside H |
Apoptosis; Others | Apoptosis; Others |
Ziyuglycoside I (Gouguside 7) 是从地榆根中分离的一种天然产物。它可用作化妆品的有效成分,具有抗皱活性,并增加 I 型胶原蛋白的表达。它引发p53介导的细胞周期阻滞和凋亡,可用于三阴乳腺癌的相关研究。 | |||
T81845 | Maximin H7 | ||
Maximin H7为源自Bombina maxima蟾蜍的抗菌肽。 | |||
T80357 |
Bombinin H7
|
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Bombinin H7 是一种抗菌肽,提取自铃蟾Bombina的皮肤分泌物。该化合物对Bacillus megateriumBm11显示出高效活性,其致死浓度达到25.2 μM。 | |||
TN2388 |
Cleroindicin C
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Others | Others |
Cleroindicin C is a natural product from plants | |||
T75697 | 1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone | ||
1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone,为喹诺酮类生物碱,作用为二酰基甘油酰基转移酶抑制剂与血管紧张素II受体阻断剂,其IC50值依次为20.1 μM与34.1 μM。此化合物亦展现对幽门螺杆菌的有效抗活性,MIC值达10 μg/mL。 | |||
TN2035 |
Paeonilactone A
(3R,3AR,6S,7AR)-四氢-6-羟基-3,6-二甲基-2,5(3H,4H)-苯并呋喃二酮,芍药内苷A |
Others | Others |
Paeonilactone A是一种天然产物,属于芍药科芍药属,其产品编号为 TN2035,CAS号为 98751-79-2。Paeonilactone A可用作对照参考。 | |||
TN2037 |
Paeonilactone C
(3S,3AR,6S,7AR)-3-[(苯甲酰基氧基)甲基]四氢-6-羟基-6-甲基-2,5(3H,4H)-苯并呋喃二酮,芍药内苷 C |
Others | Others |
Paeonilactone C significantly protects primary cultures of rat cortical cells against H2O2-induced neurotoxicity. | |||
T83385 |
2H-1-Benzopyran-2-one, 6-[(1R,2S)-2,3-dihydroxy-1-methoxy-3-methylbutyl]-7-methoxy-
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2H-1-Benzopyran-2-one, 6-[(1R,2S)-2,3-dihydroxy-1-methoxy-3-methylbutyl]-7-methoxy-是一种香豆素类化合物,首次分离自白芷(Angelica dahurica)的茎部。 | |||
TN2413 |
Diacetylpiptocarphol
|
Others | Others |
Diacetylpiptocarphol has antiplasmodial activity | |||
T83558 | (3S,4aS,10aS)-3-(Acetyloxy)-2,3,4,4a,10,10a-hexahydro-6-hydroxy-1,1,4a-trimethyl-7-(1-methylethyl)-9(1H)-phenanthrenone | ||
(3S,4aS,10aS)-3-(Acetyloxy)-2,3,4,4a,10,10a-hexahydro-6-hydroxy-1,1,4a-trimethyl-7-(1-methylethyl)-9(1H)-phenanthrenone(化合物3)是从丹参(Salvia miltiorrhiza)根提取的棕榈酸盐。该化合物展现出抗癌活性,对于不同的人类癌症细胞系具有显著的抑制效果,其DC50值分别为:HeLa细胞系25.5 μg/mL、HepG2细胞系37.5 μg/mL以及OVCAR-3细胞系30.2 μg/mL。 | |||
TN3049 |
4-Methoxycinnamyl alcohol
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Others | Others |
4-Methoxycinnamyl alcohol 对MCF-7、HeLa 和DU145癌症细胞系显示出毒性,IC50值分别为14.24、7.82和22.10μg/mL。4-methoxycinnamyl alcohol 是从Foeniculum vulgare 中分离出来的。4-Methoxycinnamyl alcohol 没有显示出凋亡作用,却在10μg/mL DNA 碎片研究显示48小时后发生了坏死。 | |||
T2S0843 |
Negletein
黄芩素-7-甲醚,7-O-Methylbaicalein,Baicalein-7-methylether |
IL Receptor; TNF; NOS; Interleukin | Apoptosis; Immunology/Inflammation |
Negletein (7-O-Methylbaicalein) 一种神经保护剂,可增强神经生长因子的作用并诱导 PC12 细胞中的神经突生长。它通过抑制TNF-α和IL-1β表现出抗炎活性,其 IC50值分别为 16.4 和 10.8 μM。它还具有抗菌、抗缺氧和抗阿尔茨海默病活性。 | |||
T2S1865 |
Octyl gallate
Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯 |
Antioxidant; Influenza Virus; Reactive Oxygen Species; Antibacterial; Antifungal; HSV | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction |
Octyl gallate (Octyl 3,4,5-trihydroxybenzoate) 具有抗菌、抗氧化作用,有选择性和敏感性的荧光特性,广泛用作食品添加剂。它对 HSV-1,水泡性口炎病毒和脊髓灰质炎病毒有显著的抗病毒作用。 | |||
T3S2344 |
β,β-Dimethylacrylshikonin
β,β-二甲基丙烯酰紫草素,Dimethylacrylshikonin,β, β-Dimethylacrylshikonin |
ERK; HIF/HIF Prolyl-Hydroxylase | Chromatin/Epigenetic; MAPK; Metabolism |
β,β-Dimethylacrylshikonin (Dimethylacrylshikonin) 是一种萘醌衍生物,从 Arnebia nobilis 中提取得到。它利用 PI3K 通路诱导 eNOS、VEGF 和 HIF-1α 的表达,促进血管生成,具有抗肿瘤活性。 | |||
T6S1684 |
8-Gingerol
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Antioxidant; Antibacterial; TRP/TRPV Channel | Membrane transporter/Ion channel; Microbiology/Virology; oxidation-reduction |
8-Gingerol 分离自姜的根状茎,是口服有效的 TRPV1激活剂,EC50值为5.0 µM。8-Gingerol 抑制 COX-2,还能抑制体外 H. pylori 的生长。 | |||
TN5009 | Shizukanolide H | Others | Others |
Shizukanolide H是一种天然产物,属于金粟兰科金粟兰属,其产品编号为 TN5009,CAS号为 1136932-34-7。Shizukanolide H可用作对照参考。 | |||
TN4142 |
Glochidonol
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Others | Others |
Glochidonol exhibits strong inhibitory effects against three human tumor cell lines, MCF-7, NCI-H-460 and SF-268, the GI(50) values of 9.0 +/- 3.7, 4.9 +/- 0.2 and 9.8 +/- 0.5, respectively; it also exerts its antiproliferative activity through the involv | |||
TN4140 |
Glochidiol
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Others | Others |
Glochidiol exhibits strong inhibitory effects against all three human tumor cell lines (MCF-7, NCI-H-460 and SF-268), it exerts its antiproliferative activity through the involvement of apoptosis. It exhibits a strong inhibitory effect on mouse skin tumor | |||
TN5657 | Goniotriol | ||
Goniotriol shows antimycobacterial activity against Mycobacterium tuberculosis (MIC =100 microg/mL). It exhibits antiplasmodial activity against Plasmodium falciparum (IC50=2.6 microg/mL). Goniotriol shows cytotoxicity against cancer cells, KB, BC1, NCI-H | |||
T35752 |
Xanthoquinodin A1
Xanthoquinodin A1 |
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Xanthoquinodin A1 is a fungal metabolite that has been found inHumicolaand has diverse biological activities.1,2It inhibitsE. tenellaschizont formation in BHK-21 cells with a minimum effective concentration (MEC) value of 0.02 μg/ml.1Xanthoquinodin A1 is active againstB. subtilis,M. luteus,S. aureus,A. laidlawii, andB. fragilisin a disc assay when used at a concentration of 1 mg/ml. It is also active againstB. cereus(MIC = 0.44 μM).2Xanthoquinodin A1 is cytotoxic to KB, MCF-7, and NCI H187 cance... | |||
T36448 |
(E)-Ajoene
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(E)-Ajoene is a disulfide that has been found inA. sativumand has diverse biological activities.1,2,3,4It is active against Gram-positive and Gram-negative bacteria (MICs = 10-250 and 150->500 μg/ml, respectively) and fungi (MICs = 15-50 μg/ml).1(E)-Ajoene inhibits proliferation of a variety of cancer cells, including MDA-MB-231 breast, HeLa cervical, and WHCO1 esophageal cancer cells (IC50s = 18.6, 61, and 39.2 μM, respectively).2It also inhibits human glutathione reductase andT. cruzitrypanoth... |