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60

抑制剂 & 化合物

12

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Cat. No. Product Name Target Signaling Pathways
T73594 Chymotrypsin

Chymotrypsin A

Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism
Chymotrypsin (Chymotrypsin A) 是胰腺产生的丝氨酸蛋白酶,可切割芳香族氨基酸羧基侧的蛋白质链。
T17011 TCH-165

Proteasome Proteases/Proteasome; Ubiquitination
TCH-165 是一种蛋白酶体组装的小分子调节剂,可增加游离 20S 水平,进而增强 IDP 蛋白水解。
T21854 Proteasome inhibitor IX

PS-IX,AM114

Proteasome Proteases/Proteasome; Ubiquitination
Proteasome inhibitor IX (PS-IX) 是 Chalcone 的一种衍生物,对20S 蛋白酶体的胰凝乳蛋白酶样活性有抑制作用,IC50约为 1 μM。它抑制 HCT116 p53+/+细胞生长,IC50为 1.49 μM,显示出有效的抗癌活性。
T6027 Delanzomib

德兰佐米,CEP-18770

Apoptosis; NF-κB; Proteasome Apoptosis; NF-κB; Proteases/Proteasome; Ubiquitination
Delanzomib (CEP-18770) 是一种强效的具有口服活性的蛋白酶体的胰凝乳蛋白酶样活性抑制剂,IC50为 3.8 nM。它抑制NF-κB 活性,诱导癌细胞凋亡,具有很强的抗血管生成和抗癌活性。
T76157 Chymotrypsinogen

Chymotrypsinogen 是Chymotrypsin 的无活性前体。Chymotrypsinogen 是一种由胰腺产生的丝氨酸蛋白酶 (serine protease)。
T6941 PI-1840

PI 1840

PARP; Proteasome Chromatin/Epigenetic; DNA Damage/DNA Repair; Proteases/Proteasome; Ubiquitination
PI-1840 是一种高效的、选择性的蛋白酶体chymotrypsin-like (CT-L)抑制剂,IC50=27nM。
T23233L RETF-4NA acetate

RETF-4NA acetate(1160928-63-1 free base)

Others Others
RETF-4NA acetate 是一种敏感的、特异性的糜蛋白酶底物。
T3359 Aprotinin

抑酶肽,抑肽酶,Bovine Pancreatic Trypsin Inhibitor,Traskolan,Antilysin

Others; Serine Protease; Influenza Virus; Proteasome Microbiology/Virology; Others; Proteases/Proteasome; Ubiquitination
Aprotinin (Traskolan) 是分离自牛肺的一种广谱丝氨酸蛋白酶抑制剂,可抑制多种不同酯酶和蛋白酶的活性。
T7016 VR23

Apoptosis; Proteasome; Caspase Apoptosis; Proteases/Proteasome; Ubiquitination
VR23 是一种蛋白酶体抑制剂,对胰蛋白酶样蛋白酶体、糜蛋白酶样蛋白酶体和半胱天冬酶样蛋白酶体的 IC50 分别是1 nM、50-100 nM 和3 μM。
T6370 AEBSF hydrochloride

AEBSF HCl,Pefabloc SC

Thrombin; Serine Protease; Influenza Virus Microbiology/Virology; Proteases/Proteasome
AEBSF hydrochloride (Pefabloc SC) 是一种丝氨酸蛋白酶的不可逆抑制剂。
T2016 MLN9708

Ixazomib Citrate

Proteasome Proteases/Proteasome; Ubiquitination
MLN9708 (Ixazomib Citrate) 抑制 20S 蛋白酶体的糜蛋白酶样蛋白水解 (β5) 位点 (Ki50=0.93 nM, IC50=3.4 nM/)。 MLN9708 的生物活性形式是水溶液或血浆中的 MLN2238。
T1795 Carfilzomib

卡非佐米,PR-171

Apoptosis; Proteasome; Autophagy Apoptosis; Autophagy; Proteases/Proteasome; Ubiquitination
Carfilzomib (PR-171) 是一种蛋白酶体抑制剂,与 20S 蛋白酶体的糜蛋白酶不可逆结合。Carfilzomib 具有抗肿瘤活性,可以用于治疗多发性骨髓瘤。
T8350 TPCK

Proteasome Proteases/Proteasome; Ubiquitination
TPCK 是丝氨酸蛋白酶抑制剂,通过与 HPV-18 E7 蛋白的视网膜母细胞瘤蛋白 (RB) 结合核心发生反应,并能够消除其 RB 结合能力。将它添加到培养基内,可修饰活角质形成细胞中的 E7 蛋白。
T0372 Gabexate mesylate

甲磺酸加贝酯,FOY

Factor Xa; Serine Protease; Proteasome Metabolism; Proteases/Proteasome; Ubiquitination
Gabexate mesylate (FOY) 是一种非抗原的类胰蛋白酶丝氨酸蛋白酶抑制剂。
T21617 MG-115

Z-LL-Nva-CHO

Proteasome Proteases/Proteasome; Ubiquitination
MG-115 (Z-LL-Nva-CHO) 是一种有效且可逆的蛋白酶体抑制剂,对20S 和26S 蛋白酶体的 Ki 值分别为 21 nM 和 35 nM。MG-115 特异性抑制蛋白酶体的胰凝乳蛋白酶样活性,诱导 p53 依赖性细胞凋亡。
T63321 20S Proteasome activator 1

Proteasome Proteases/Proteasome; Ubiquitination
20S Proteasome activator 1 是一种 20S 蛋白酶激活剂,对胰蛋白酶样位点、胰凝乳蛋白酶样位点和半胱天冬酶位点的 IC50 分别为 0.3 μM、0.7 μM 和 1.8 μM。20S Proteasome activator 1 通过在细胞系统中翻译来防止致病性 α-synuclein A53T 突变体积累从而减少疾病发生的概率。20S Proteasome activator 1 可用于研究神经退行性疾病。
TP1832 Gluten Exorphin C

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Gluten exorphin C 是来源于谷朊粉的阿片肽。在 GPI 和 MVD 检测中,抑制 μ 阿片和 δ 阿片活性,IC50值分别为 40 和13.5 μM。
T2122 Ixazomib

艾沙佐米,MLN2238

Proteasome; Caspase; Autophagy Apoptosis; Autophagy; Proteases/Proteasome; Ubiquitination
Ixazomib (MLN2238) 含硼肽蛋白酶体抑制剂(PI),可抑制 20S 蛋白酶体的糜蛋白酶样蛋白水解 (β5) 位点,IC50为 3.4 nM,Ki 为 0.93 nM。它还抑制半胱天冬酶样 (β1) 和胰蛋白酶样 (β2) 蛋白水解位点,IC50值为 31和3500 nM。
T36352 Suc-Leu-Tyr-AMC

Suc-Leu-Tyr-AMC 是钙蛋白酶 I 和 II 以及木瓜蛋白酶(另一种半胱氨酸蛋白酶)的荧光底物,用于测量 20S 蛋白酶体的糜蛋白酶样肽酶活性(Ex-max:360 nm;Em-max:460 nm)。Suc-Leu-Tyr-AMC 也能被大肠杆菌的 Ti 蛋白酶裂解。
T14529 Bentiromide

Others Others
Bentiromide 是一种可被胰腺分泌的胰凝乳蛋白酶分解的多肽。Bentiromide 通过胰凝乳蛋白酶功能的体外试验确认胰腺外分泌功能。
T11290 FK-448 Free base

Others Others
FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM.
T68543 FK-386 HCl

FK-386 HCl is an inhibitor of chymotrypsin.
T26297 Tryptophanamide

S-Tryptophanamide

Tryptophanamide is a chymotrypsin inhibitor.
T68545 FK-401

FK-401 is an inhibitor of chymotrypsin.
T68647 FK-316

FK-316 is an inhibitor of chymotrypsin.
T68544 FK-375 HCl

FK-375 HCl is an inhibitor of chymotrypsin.
T25280 Cyanopeptolin 954

Cyanopeptolin-954,Cyanopeptolin954

Cyanopeptolin 954 is a chlorine-containing Microcystis aeruginosa NIVA Cya 43 chymotrypsin Inhibitor.
T26202 SP-Chymostatin B

alpha-Mapi

SP-Chymostatin B is a potent inhibitor of many proteases, including chymotrypsin, papain, chymotrypsin-like serine proteinases, chymases, and lysosomal cysteine proteinases. It weakly inhibits human leucocyte elastase. It is effective at a final concentra
T68534 FK-448 methanesulfonate

FK-448 methanesulfonate is a chymotrypsin inhibitor that has been shown to affect intestinal absorption of insulin in rats and dogs .
T74692 Ac-Phe-Gly-pNA

Ac-Phe-Gly-pNA 是一种糜蛋白酶特异性底物。
T37418 Z-LLL-AMC

Z-LLL-AMC is a fluorogenic substrate for the chymotrypsin-like activity of the 26S proteasome or 20S proteolytic core. Chymotrypsin-like activity can be quantified by fluorescent detection of free AMC (also known as 7-amino-4-methylcoumarin), which is excited at 340-360 nm and emits at 440-460 nm. Z-LLL-AMC is typically used in cell lysates after experimental treatment.
T37019 p-APMSF (hydrochloride)

p-APMSF is an irreversible inhibitor of serine proteases with Ki values of 1.02, 1.18, 1.5, and 1.54 μM for bovine trypsin, human thrombin, bovine plasmin, and bovine Factor Xa, respectively. It is selective for these proteases over bovine chymotrypsin and acetylcholinesterase.
T71198 Eglin c (60-63)

Eglin c (60-63) is a sequence of a peptide that has been studied for its inhibitory activity towards human leukocyte elastase, cathepsin G, porcine pancreatic elastase and alpha-chymotrypsin.
TP1308 Suc-Leu-Leu-Val-Tyr-AMC

Suc-Leu-Leu-Val-Tyr-AMC is a fluorescent substrate for the 20S proteasome, other chymotrypsin-like proteases.
T36962 MMP Inhibitor I (trifluoroacetate salt)

MMP inhibitor I is a peptide inhibitor of matrix metalloproteinase-1 (MMP-1), MMP-2, and MMP-3 (IC50s = 1.3, 30, and 150 μM, respectively). It is selective for MMP-1, MMP-2, and MMP-3 over the proteases thermolysin, urease, trypsin, α-chymotrypsin, plasmin, and elastase at concentrations up to 4 mM.
T80102 Z-Leu-Leu-Tyr-COCHO

Proteasome Proteases/Proteasome; Ubiquitination
Z-Leu-Leu-Tyr-COCHO为胰凝乳蛋白酶样活性抑制剂,具有Ki值为3.0 nM的高效性。
T76621 Suc-Ala-Ala-Pro-Phe-SBzl

Suc-Ala-Ala-Pro-Phe-SBzl 是一种化合物,可以作为大鼠小肠肥大细胞蛋白酶(RMCP I)、大鼠骨骼肌肥大细胞蛋白酶(RMCP II)和胰凝乳蛋白酶(Chymotrypsin)的底物。此外,Suc-Ala-Ala-Pro-Phe-SBzl 能够被甘氨酸(R208G)水解。
T36338 AAF-CMK (trifluoroacetate salt)

Tripeptidyl peptidase II (TPPII) is a serine peptidase of the subtilisin-type which removes tripeptides from the free NH2 terminus of oligopeptides. AAF-CMK is an irreversible inhibitor of TPPII commonly used at 10-100 μM. It does not significantly interfere with the chymotrypsin-like activity of the proteasome. AAF-CMK also inhibits bleomycin hydrolase and puromycin-sensitive aminopeptidase when used at 50 μM.
T14529L Bentiromide acetate

Bentiromide acetate(37106-97-1 Free base)

Others Others
Bentiromide acetate 是一种肽,用于外分泌胰腺功能不全的筛选试验和监测补充胰腺治疗的充分性。它被胰酶胰凝乳蛋白酶分解,生成对氨基苯甲酸(PABA)。
T76231 Cyclotheonellazole A

Cyclotheonellazole A为一天然大环肽类化合物,对弹性蛋白酶具显著的抑制效果(IC50=0.034 nM),且对糜蛋白酶亦有抑制作用,IC50值达0.62 nM。
T62080 GSK3494245

GSK3494245 (DDD01305143) 是一种有效的、选择性的、口服具有活力的、可在夹在 β4 和 β5 亚基之间的位点结合寄生虫蛋白酶体 (proteasome) 的糜蛋白酶样活性抑制剂,能够作用于 WTL.donovani 蛋白酶体,其 IC50 值为 0.16μM。GSK3494245 表现出良好的生物安全特性。GSK3494245 对人蛋白酶体的糜蛋白酶样活性具有适当的抑制作用 (IC50: 26S=13 μM;富集的 THP-1 提取物 IC50=40 μM)。
T78407 Suc-Ala-Ala-Phe-AMC

Suc-Ala-Ala-Phe-AMC为一荧光胰凝乳蛋白酶底物,可遭肽链内切酶所水解。该化合物适用于顶体反应的体内测定及体外酶活性分析。
T70170 Milvexian TFA

Milvexian, also known as BMS-986177 and JNJ-70033093, is a blood coagulation factor XIa inhibitor. Milvexian demonstrated good selectivity over plasma kallikreinKi = 44 nM (400-fold selective), and chymotrypsinKi = 35 nM (318-fold selective). At a dose of 1.5 mg/kg, Milvexian exhibited an overall exposure of 1215 nM/h, low clearance of 10.3 mL/min/kg, and oral bioavailability of 32%.
T62479 3CPLro-IN-1

3CPLro-IN-1 (compound A17) 是一种有效的、口服具有活力的 SARS-CoV-2 3CLpro 抑制剂 (IC50: 5.65 μM)。3-糜蛋白酶样半胱氨酸蛋白酶 (3CLpro) 是一种病毒复制中不可或缺的蛋白质,是一种有吸引力的、对抗 COVID-19 的药物靶点。
T74878 Enzyme-IN-1

Enzyme-IN-1(compound 1)为基于肽的N端亲核试剂(Ntn)水解酶抑制剂,特别针对20S蛋白酶体的糜胰蛋白酶样活性(CT-L)进行抑制,可能展现出抗炎特性。
T69297 Leupeptin HCl

Leupeptin is a naturally occurring protease inhibitor that can inhibit cysteine, serine and threonine peptidases. Leupeptin is an organic compound produced by actinomycetes. Leupeptin inhibits serine proteinases (trypsin (Ki=3.5 nM), plasmin (Ki= 3.4 nM), porcine kallikrein), and cysteine proteinases (papain, cathepsin B (Ki = 4.1 nM), endoproteinase Lys-C). It does not inhibit α-chymotrypsin or thrombin. Leupeptin is a competitive transition state inhibitor and its inhibition may be relieved by...
T81711 N-Acetyl-DL-phenylalanine β-naphthyl ester

N-Acetyl-DL-phenylalanine β-naphthyl ester 为一芳香族氨基酸酯,用作糜蛋白酶及微生物丝氨酸蛋白酶(例如枯草杆菌蛋白酶)的显色底物。
T6564L Leupeptin

Leupeptin Ac-LL,NK-381

Leupeptin is a competitive protease inhibitor produced by actinomycetes. Leupeptin can inhibit cysteine, serine and threonine peptidases. Leupeptin inhibits serine proteinases (trypsin (Ki=3.5 nM), plasmin (Ki= 3.4 nM), porcine kallikrein), and cysteine p
T78640 Z-LLF-CHO

Z-Leu-Leu-Phe-CHO

Proteasome Proteases/Proteasome; Ubiquitination
Z-LLF-CHO(Z-Leu-Leu-Phe-CHO)为垂体多催化蛋白酶复合物所具有的胰凝乳蛋白酶样活性提供有效抑制,具有Ki值为460 nM。此外,Z-LLF-CHO同样作为NF-κB核转位的抑制剂。
T81372 Proteasome-activating peptide 1

Proteasome-activating peptide 1 是一种肽,其作用是提升胰凝乳蛋白酶样蛋白酶体(proteasome)的催化活性,有效增强体外及细胞培养环境下的蛋白质降解效率。此外,该肽能阻止肌萎缩侧索硬化症(Amyotrophic Lateral Sclerosis, ALS)细胞模型中蛋白质的过度聚集。

化合物

Chymotrypsin
Cat.No: T73594
Synonym: Chymotrypsin A
Target: Serine/threonin kinase
TCH-165
Cat.No: T17011
Synonym:
Target: Proteasome
Proteasome inhibitor IX
Cat.No: T21854
Synonym: PS-IX,AM114
Target: Proteasome
Delanzomib
Cat.No: T6027
Synonym: 德兰佐米,CEP-18770
Target: Apoptosis, NF-κB, Proteasome
Chymotrypsinogen
Cat.No: T76157
Synonym:
Target:
PI-1840
Cat.No: T6941
Synonym: PI 1840
Target: PARP, Proteasome
RETF-4NA acetate
Cat.No: T23233L
Synonym: RETF-4NA acetate(1160928-63-1 free base)
Target: Others
Aprotinin
Cat.No: T3359
Synonym: 抑酶肽,抑肽酶,Bovine Pancreatic Trypsin Inhibitor,Traskolan,Antilysin
Target: Others, Serine Protease, Influenza Virus, Proteasome
VR23
Cat.No: T7016
Synonym:
Target: Apoptosis, Proteasome, Caspase
AEBSF hydrochloride
Cat.No: T6370
Synonym: AEBSF HCl,Pefabloc SC
Target: Thrombin, Serine Protease, Influenza Virus
MLN9708
Cat.No: T2016
Synonym: Ixazomib Citrate
Target: Proteasome
Carfilzomib
Cat.No: T1795
Synonym: 卡非佐米,PR-171
Target: Apoptosis, Proteasome, Autophagy
TPCK
Cat.No: T8350
Synonym:
Target: Proteasome
Gabexate mesylate
Cat.No: T0372
Synonym: 甲磺酸加贝酯,FOY
Target: Factor Xa, Serine Protease, Proteasome
MG-115
Cat.No: T21617
Synonym: Z-LL-Nva-CHO
Target: Proteasome
20S Proteasome activator 1
Cat.No: T63321
Synonym:
Target: Proteasome
Gluten Exorphin C
Cat.No: TP1832
Synonym:
Target: Opioid Receptor
Ixazomib
Cat.No: T2122
Synonym: 艾沙佐米,MLN2238
Target: Proteasome, Caspase, Autophagy
Suc-Leu-Tyr-AMC
Cat.No: T36352
Synonym:
Target:
Bentiromide
Cat.No: T14529
Synonym:
Target: Others
FK-448 Free base
Cat.No: T11290
Synonym:
Target: Others
FK-386 HCl
Cat.No: T68543
Synonym:
Target:
Tryptophanamide
Cat.No: T26297
Synonym: S-Tryptophanamide
Target:
FK-401
Cat.No: T68545
Synonym:
Target:
FK-316
Cat.No: T68647
Synonym:
Target:
FK-375 HCl
Cat.No: T68544
Synonym:
Target:
Cyanopeptolin 954
Cat.No: T25280
Synonym: Cyanopeptolin-954,Cyanopeptolin954
Target:
SP-Chymostatin B
Cat.No: T26202
Synonym: alpha-Mapi
Target:
FK-448 methanesulfonate
Cat.No: T68534
Synonym:
Target:
Ac-Phe-Gly-pNA
Cat.No: T74692
Synonym:
Target:
Z-LLL-AMC
Cat.No: T37418
Synonym:
Target:
p-APMSF (hydrochloride)
Cat.No: T37019
Synonym:
Target:
Eglin c (60-63)
Cat.No: T71198
Synonym:
Target:
Suc-Leu-Leu-Val-Tyr-AMC
Cat.No: TP1308
Synonym:
Target:
MMP Inhibitor I (trifluoroacetate salt)
Cat.No: T36962
Synonym:
Target:
Z-Leu-Leu-Tyr-COCHO
Cat.No: T80102
Synonym:
Target: Proteasome
Suc-Ala-Ala-Pro-Phe-SBzl
Cat.No: T76621
Synonym:
Target:
AAF-CMK (trifluoroacetate salt)
Cat.No: T36338
Synonym:
Target:
Bentiromide acetate
Cat.No: T14529L
Synonym: Bentiromide acetate(37106-97-1 Free base)
Target: Others
Cyclotheonellazole A
Cat.No: T76231
Synonym:
Target:
GSK3494245
Cat.No: T62080
Synonym:
Target:
Suc-Ala-Ala-Phe-AMC
Cat.No: T78407
Synonym:
Target:
Milvexian TFA
Cat.No: T70170
Synonym:
Target:
3CPLro-IN-1
Cat.No: T62479
Synonym:
Target:
Enzyme-IN-1
Cat.No: T74878
Synonym:
Target:
Leupeptin HCl
Cat.No: T69297
Synonym:
Target:
N-Acetyl-DL-phenylalanine β-naphthyl ester
Cat.No: T81711
Synonym:
Target:
Leupeptin
Cat.No: T6564L
Synonym: Leupeptin Ac-LL,NK-381
Target:
Z-LLF-CHO
Cat.No: T78640
Synonym: Z-Leu-Leu-Phe-CHO
Target: Proteasome
Proteasome-activating peptide 1
Cat.No: T81372
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1372 Alpha-Amyrin

alpha-Amyrenol,α-Amyrin,alpha-Amyrine,Viminalol,α-香树脂醇

P450; Serine Protease; ROS Immunology/Inflammation; Metabolism; Proteases/Proteasome
Alpha-Amyrin (alpha-Amyrine) 是一种具有抗肿瘤作用的胰蛋白酶和糜蛋白酶抑制剂。 alpha-Amyrin 可用于作为肝调节剂的研究。
T2O2730 L-Serine

(S)-Serine,L-丝氨酸,丝氨酸,serine,(-)-Serine,(S)-2-Amino-3-hydroxypropanoic acid

Endogenous Metabolite Metabolism
L-Serine (serine) 是一种人体非必需氨基酸,它存在于许多蛋白质中,并且在功能上很重要。L-Serine 也存在于丝氨酸蛋白酶类的活性位点,包括胰蛋白酶和凝乳胰蛋白酶。
TN3228 7-Hydroxy-3-(4-hydroxybenzyl)chroman

Others Others
7-Hydroxy-3-(4-hydroxybenzyl)chroman shows moderate inhibitory activity against a chymotrypsin-like activity of the proteasome.
T15638 K-252c

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a cell-permeable PKC inhibitor (IC50: 2.45 μM). K-252c also inhibits β-lactamase, chymotrypsin, and malate dehydrogenase. K-252c causes apoptosis in human chronic myelogenous leukemia cancer cells.
T75648 Rivulariapeptolides 1155

Rivulariapeptolides 1155 是一种有效的丝氨酸蛋白酶 (serine protease) 抑制剂,对糜蛋白酶、弹性蛋白酶、蛋白蛋白酶 K 的 IC50分别为 41.84、4.94、56.54 nM。
T10238 Aclacinomycin A hydrochloride

盐酸阿柔比星,Aclarubicin hydrochloride

Proteasome Proteases/Proteasome; Ubiquitination
Aclacinomycin A (Aclarubicin) hydrochloride is a fluorescent molecule and the first described non-peptidic inhibitor showing discrete specificity for the CTRL (chymotrypsin-like) activity of the 20S proteasome. Aclacinomycin A hydrochloride is also a dual inhibitor of topoisomerase I and II.
TN3383 α-Amyrin palmitate

alpha-Amyrin palmitate

PKA Tyrosine Kinase/Adaptors
alpha-Amyrin palmitate is antiarthritic in the adjuvant model of arthritis in rats. alpha-Amyrin palmitate is a potent non-competitive inhibitor of chymotrypsin (Ki=6 microM), it also shows weak cytotoxicity against the A2780 human ovarian cancer cell line.
T75649 Rivulariapeptolides 1185

Rivulariapeptolides 1185 是一种高效的选择性丝氨酸蛋白酶抑制剂,其对胰凝蛋白酶、弹性蛋白酶和蛋白酶 K 的 IC50分别为 13.17 nM、23.59 nM 和 55.26 nM。
TN5655 Broussonin B

Broussonins A and B, new phytoalexins from diseased paper mulberry. Broussonin B can induce neurite outgrowth in PC-12 cells at concentration of 50 microg/ml, and show moderate inhibitory activities against a chymotrypsin-like activity of the proteasome.B
T75651 Rivulariapeptolides 988

Rivulariapeptolides 988作为一种高效选择性丝氨酸蛋白酶抑制剂,对胰凝蛋白酶、弹性蛋白酶和蛋白酶K的IC50分别为95.46 nM、15.29 nM和85.50 nM。
T75652 Molassamide B

Molassamide B,丝氨酸蛋白酶抑制剂,对胰凝乳蛋白酶、弹性蛋白酶及蛋白酶 K 具有显著抑制活性,其IC50值分别为24.65、11.69和5.42 nM。
T75650 Rivulariapeptolides 1121

Rivulariapeptolides 1121,作为一种高效的选择性丝氨酸蛋白酶抑制剂,对胰凝蛋白酶、弹性蛋白酶和蛋白酶K展示出了显著的抑制活性,其IC50值分别为35.52 nM、13.24 nM和48.05 nM。

天然产物

Alpha-Amyrin
Cat.No: TN1372
Synonym: alpha-Amyrenol,α-Amyrin,alpha-Amyrine,Viminalol,α-香树脂醇
Target: P450, Serine Protease, ROS
L-Serine
Cat.No: T2O2730
Synonym: (S)-Serine,L-丝氨酸,丝氨酸,serine,(-)-Serine,(S)-2-Amino-3-hydroxypropanoic acid
Target: Endogenous Metabolite
7-Hydroxy-3-(4-hydroxybenzyl)chroman
Cat.No: TN3228
Synonym:
Target: Others
K-252c
Cat.No: T15638
Synonym:
Target: PKC
Rivulariapeptolides 1155
Cat.No: T75648
Synonym:
Target:
Aclacinomycin A hydrochloride
Cat.No: T10238
Synonym: 盐酸阿柔比星,Aclarubicin hydrochloride
Target: Proteasome
α-Amyrin palmitate
Cat.No: TN3383
Synonym: alpha-Amyrin palmitate
Target: PKA
Rivulariapeptolides 1185
Cat.No: T75649
Synonym:
Target:
Broussonin B
Cat.No: TN5655
Synonym:
Target:
Rivulariapeptolides 988
Cat.No: T75651
Synonym:
Target:
Molassamide B
Cat.No: T75652
Synonym:
Target:
Rivulariapeptolides 1121
Cat.No: T75650
Synonym:
Target:
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