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Search Results for " bronchial asthma "

25

抑制剂 & 化合物

1

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Cat. No.	Product Name	Target	Signaling Pathways
T8239	Cromoglicic acid	Others	Others
	Cromoglicic acid 可防止肥大细胞释放炎性化学物质，例如组胺。
T3965	Fevipiprant QAW039,NVP-QAW039,非维匹仑	GPR; Prostaglandin Receptor	Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation
	Fevipiprant (NVP-QAW039) 是一种选择性、强效、可逆的竞争性 CRTh2 拮抗剂，KD 值为1.1 nM，IC50为0.44 nM，能够引发人体嗜酸性粒细胞的形状变化。
T0188	Fluticasone (propionate) 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate	Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite	Endocrinology/Hormones; Metabolism; Microbiology/Virology
	Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂，是一种局部抗炎激素，亲和力KD 为 0.5 nM。具有抗病毒活性。
T2270	Trans-Tranilast Tranilast trans-,反式-曲尼司特,反-曲尼司特	RAAS	Endocrinology/Hormones
	Trans-Tranilast 是抗过敏剂，可用于过敏性鼻炎、支气管哮喘和特应性皮炎的研究。
T0277	Metaproterenol hemisulfate Orciprenaline sulfate,Metaproterenol Sulfate,硫酸奥西那林	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Metaproterenol hemisulfate (Orciprenaline sulfate) 是一种 β2-肾上腺素能受体 (β2AR) 激动剂(IC50=68 nM)，是一种直接作用的拟交感神经药，具有抗炎活性。
T0477	Zileuton Abbott 64077,齐留通,A 64077	Ferroptosis; Lipoxygenase; COX	Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
	Zileuton (A 64077) 是羟基脲的合成衍生物，是一种选择性的5-脂氧合酶抑制剂，具有平喘特性。
T4195	Betahistine PT 9 base,倍他司汀,Vasomotal,Serc base	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Betahistine (Vasomotal) 是可口服的组胺 H1 受体激动剂和 H3 受体的拮抗剂，可用作血管扩张剂，用于类风湿性关节炎的研究。
T1682	Methacholine Chloride 醋甲胆碱,Mecholyl chloride,氯化乙酰甲胆碱,Acetyl-β-methylcholine chloride	AChR	Neuroscience
	Methacholine Chloride (Acetyl-β-methylcholine chloride) 是副交感神经系统中的毒蕈碱-3 受体激动剂。它可用于测量气道高反应性，作为评估哮喘样症状和正常静息呼气流速的诊断辅助手段。它直接作用于平滑肌上的乙酰胆碱受体，引起收缩和气道狭窄。
T30141L	Arpenal HCl Arpenal hydrochloride
	Arpenal HCl is a ganglionic blocking agent which may be useful in the treatment of bronchial asthma.
T28651	S-5751 S 5751
	S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.
T23472	Tranilast Sodium	Others	Others
	Tranilast Sodium has been used for the treatment of bronchial asthma. Tranilast is also used to autoimmune diseases, atopic and fibrotic pat.
T30141	Arpenal
	Arpenal is a ganglionic blocking agent which may be useful in the treatment of bronchial asthma.
T70294	KAA-276 free base
	KAA-276 free base is a novel potent and long-lasting histamine HI-receptor antagonist with less-topical irritation, and can be topically administered by inhalation for the treatment of bronchial asthma.
T70293	KAA-276 HCl
	KAA-276 HCl is the salt form of KAA-276 free base, a novel potent and long-lasting histamine HI-receptor antagonist with less-topical irritation, and can be topically administered by inhalation for the treatment of bronchial asthma.
T61075	Piperilate
	Piperilate, also known as Pipethanate, is a hetrazepine derivative PAF antagonist and anticholinergic mixture, commonly utilized in bronchial asthma research. This compound exhibits hypotensive properties and has been found to effectively counteract the toxic effects of organophosphates in mice [1] [2] [3].
T26628	Andolast CR2039,CR-2039,CR 2039
	Andolast, also known as CR-2039, an anti-allergic agent for the treatment of bronchial asthma, chronic obstructive pulmonary disease (COPD). Andolast acts at different cellular levels to inhibit immunoglobulin E synthesis. Andolast proved to be significan
T121458	8011-6561
	1,1-Diphenyl-4-(pyrrolidin-1-yl)but-2-yn-1-ol 是一种抗胆碱能药物，具有用于支气管哮喘研究的潜力。
T21411	Isoproterenol Norisodrine,Isoprenaline,Novodrin,Isuprel,Medihaler-Iso	Endogenous Metabolite; Adrenergic Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Isoproterenol (Norisodrine) 是一种非选择性且具有口服活性的 β-肾上腺素受体激动剂。Isoproterenol 是有效的外周血管扩张剂和支气管扩张剂。Isoproterenol 可用于研究心动过缓和支气管哮喘，用于治疗心脏传导阻滞、心动过缓。
T60289	Pemirolast
	Pemirolast 是一种具有口服活性的抗过敏剂。Pemirolast 通过抑制感觉神经肽的释放来减轻紫杉醇超敏反应，可用于对支气管哮喘和结膜炎的研究。
T71329	Theophylline-d6
	Theophylline-d6 is intended for use as an internal standard for the quantification of theophylline by GC- or LC-MS. Theophylline is an inhibitor of phosphodiesterase. It is also an adenosine A1 and A2 receptor antagonist. Theophylline induces relaxation of isolated cat bronchial smooth muscle segments precontracted with acetylcholine. It inhibits ovalbumin-induced increases in bronchoalveolar lavage fluid (BALF) eosinophil infiltration in an ovalbumin-sensitized mouse model of allergic asthma. F...
T60590	Chloropyramine
	Chloropyramine 是竞争性可逆 H1 受体拮抗剂，可用于过敏性疾病的研究，例如结膜炎和支气管哮喘。Chloropyramine 表现出抗乳腺癌活性。
T22189	APC 366
	APC 366 是肥大细胞类胰蛋白酶 (tryptase) 的选择性抑制剂，Ki 值为7.1 μM。在羊过敏性哮喘模型中，APC 366 抑制抗原诱导的早期哮喘反应 (EAR)、晚期哮喘反应 (LAR) 和支气管高反应性 (BHR)。
T0246L	Betahistine mesylate Extovyl,甲磺酸倍他司汀,Melopat,Meginalisk	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Betahistine mesylate (Extovyl) 是可口服的组胺 H1 受体激动剂和 H3 受体的拮抗剂，可用作血管扩张剂，用于类风湿性关节炎的研究。
T80891	Urodilatin
	Urodilatin为ANF-(99-126)的同类物，属于利尿钠调节肽。该化合物主要应用于急性肾功能衰竭、充血性心力衰竭、支气管哮喘等疾病的研究领域。
T60332	Methacholine bromide
	Methacholine (Acetyl-β-methylcholine) bromide 是一种有效的muscarinic-3 (M3)激动剂。Methacholine bromide 直接作用于平滑肌上的乙酰胆碱受体，导致支气管收缩和气道变窄。Methacholine bromide 对识别支气管高反应性 (BHR) 显示出高灵敏度，BHR 是哮喘的重要特征。Methacholine bromide 可用于测量气道高反应性 (AHR)，作为评估具有哮喘样症状和正常静息呼气流速的个体的诊断辅助[2]。

化合物

Cromoglicic acid

Cat.No: T8239

Target: Others

Cat.No: T3965

Synonym: QAW039,NVP-QAW039,非维匹仑

Target: GPR, Prostaglandin Receptor

Fluticasone (propionate)

Cat.No: T0188

Synonym: 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate

Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite

Trans-Tranilast

Cat.No: T2270

Synonym: Tranilast trans-,反式-曲尼司特,反-曲尼司特

Target: RAAS

Metaproterenol hemisulfate

Cat.No: T0277

Synonym: Orciprenaline sulfate,Metaproterenol Sulfate,硫酸奥西那林

Target: Adrenergic Receptor

Cat.No: T0477

Synonym: Abbott 64077,齐留通,A 64077

Target: Ferroptosis, Lipoxygenase, COX

Cat.No: T4195

Synonym: PT 9 base,倍他司汀,Vasomotal,Serc base

Target: Histamine Receptor

Methacholine Chloride

Cat.No: T1682

Synonym: 醋甲胆碱,Mecholyl chloride,氯化乙酰甲胆碱,Acetyl-β-methylcholine chloride

Target: AChR

Cat.No: T30141L

Synonym: Arpenal hydrochloride

Cat.No: T28651

Synonym: S 5751

Tranilast Sodium

Cat.No: T23472

Target: Others

Cat.No: T30141

KAA-276 free base

Cat.No: T70294

Cat.No: T70293

Cat.No: T61075

Cat.No: T26628

Synonym: CR2039,CR-2039,CR 2039

Cat.No: T121458

Cat.No: T21411

Synonym: Norisodrine,Isoprenaline,Novodrin,Isuprel,Medihaler-Iso

Target: Endogenous Metabolite, Adrenergic Receptor

Cat.No: T60289

Theophylline-d6

Cat.No: T71329

Cat.No: T60590

Cat.No: T22189

Betahistine mesylate

Cat.No: T0246L

Synonym: Extovyl,甲磺酸倍他司汀,Melopat,Meginalisk

Target: Histamine Receptor

Cat.No: T80891

Methacholine bromide

Cat.No: T60332

Cat. No.	Product Name	Target	Signaling Pathways
T0892	Diphylline 二羟丙茶碱,Dyphylline,Diprophylline	PDE; Adenosine Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Diphylline (Diprophylline) 是一种A1/A2腺苷受体拮抗剂，也是环状核苷酸磷酸二酯酶抑制剂。它是一种黄嘌呤衍生物，具有支气管扩张和血管扩张作用，有用于治疗慢性支气管炎和肺气肿的潜力。

天然产物

Cat.No: T0892

Synonym: 二羟丙茶碱,Dyphylline,Diprophylline

Target: PDE, Adenosine Receptor

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