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78

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T0138 Cefpiramide acid

Cefpiramidum,头孢匹胺,Cefpiramido

Antibacterial Microbiology/Virology
Cefpiramide acid (Cefpiramidum) 是第三代头孢菌素类抗生素。
T6231 Tebipenem Pivoxil

ME1211,Orapenem,替​比​培​南​匹​酯

Antibacterial; Antibiotic Microbiology/Virology
Tebipenem Pivoxil (Orapenem) 是一种碳青霉烯类新型口服抗生素。
T5189 Omadacycline

PTK 0796,Amadacycline

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Omadacycline (Amadacycline) 是一种具有口服活性的氨基甲基环素抗菌剂,是四环素类抗生素。它与 30S 核糖体亚基结合,抑制细菌蛋白质合成。它可用于研究急性细菌性皮肤和皮肤结构感染,感染性肺炎和尿路感染。
T1114 Ciclopirox olamine

环吡酮乙醇胺盐,环吡司胺,Ciclopirox ethanolamine

ATPase; Others; Ferroptosis; Antibacterial; Antifungal Apoptosis; Membrane transporter/Ion channel; Microbiology/Virology; Others
Ciclopirox olamine 是一种合成的抗真菌剂,可研究浅表真菌病。
T11227L1 Eravacycline HCl

Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl

Antibiotic Microbiology/Virology
Eravacycline HCl (TP-434 HCl) 是一种具有广谱抗菌活性的强效抗生素。
T4270 Cefquinome sulfate

硫酸头孢喹肟,硫酸头孢喹诺

Antibacterial; Antibiotic Microbiology/Virology
Cefquinome sulfate 是一种半合成的头孢烯广谱抗生素,具有抗菌活性。
T16789 Rosoxacin

罗索沙星,Acrosoxacin

Antibacterial; Antibiotic Microbiology/Virology
Rosoxacin (Acrosoxacin) 是具有口服活性的喹诺酮类抗生素,具有广谱的抗菌活性,抑制革兰氏阴性菌,包括淋病奈瑟氏球菌(MIC90=0.03 mg/ml)。它在尿路感染中有应用的潜能。
T11007L Levofloxacin Hydrochloride Impurity A

Levofloxacin Hydrochloride Impurity A(117707-40-1 Free base),左氧氟沙星杂质A(盐酸盐)

Antibacterial Microbiology/Virology
Levofloxacin Hydrochloride Impurity A 是一种喹诺酮类药物,具有广谱抗菌作用。
T1444 Lomefloxacin

洛美沙星,SC47111A

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin (SC47111A) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T8390 Cefazolin

头孢唑林,头孢唑啉

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazolin 是一种头孢类抗生素, 用于多种细菌感染的研究。
T19858 Brodimoprim

DHFR; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Brodimoprim 是甲氧苄啶的一种类似物,是口服有效的二氢叶酸还原酶抑制剂,对广谱革兰氏阴性和革兰氏阳性细菌具有高度的抑制作用。
T4991 Ertapenem sodium

厄他培南钠,MK-826,L-749345,尔他培南钠

Antibacterial; Antibiotic Microbiology/Virology
Ertapenem sodium (MK-826) 是碳青霉烯,是一种 β-内酰胺抗生素,具有广谱抗菌活性。
T0425 Pefloxacin Mesylate

Pefloxacinium mesylate,甲磺酸培氟沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。
T11227L Eravacycline dihydrochloride

TP-434-046,TP-434 dihydrochloride

Antibacterial Microbiology/Virology
Eravacycline dihydrochloride (TP-434-046) 是一种有效的广谱抗菌剂,可对抗六种大肠杆菌(MIC:0.125-0.25 mg/L)。
T8142 Difloxacin hydrochloride

Difloxacin HCl,盐酸二氟沙星

Antibacterial; Antibiotic Microbiology/Virology
Difloxacin hydrochloride (Difloxacin HCl) 是一种广谱抗菌药物。它干扰 DNA 促旋酶和拓扑异构酶 IV 的活性,抑制细菌 DNA 促旋酶并显示出浓度依赖性的杀菌作用。
T38359 Dup-721

Antibacterial Microbiology/Virology
DuP-721 是广谱的口服有效的抗菌剂,可以抑制多种临床敏感和耐药细菌,特别是结核杆菌M. tuberculosis。
T6268 Ceftiofur hydrochloride

头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur hydrochloride (U-67279A) 是头孢噻呋的盐酸盐形式,是一种β-内酰胺酶稳定的半合成广谱头孢菌素,具有抗菌活性。
T0717 Enoxacin hydrate

CI-919 hydrate,Enoxacin Sesquihydrate,依诺沙星半水合物,AT-2266 hydrate,依诺沙星倍半水合物

DNA gyrase; DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Enoxacin hydrate (AT-2266 hydrate) 是氟喹诺酮,可干扰DNA 复制,抑制细菌 DNA 促旋酶 (IC50=126 µg/ml) 和拓扑异构酶 IV (IC50=26.5 µg/ml)。它是特异性癌症生长抑制剂,抑制革兰氏阳性和阴性细菌。
TN6672 Cyclo(L-Phe-L-Pro)

Free radical scavengers; COX; Antibacterial; Antifungal Immunology/Inflammation; Microbiology/Virology; Neuroscience; oxidation-reduction
Cyclo(L-Phe-L-Pro) 具有广谱抗菌和抗真菌活性。 Cyclo(L-Phe-L-Pro) 对耐甲氧西林金黄色葡萄球菌和棉子肠球菌具有活性。
T12004 Meropenem trihydrate

美罗培南三水合物,SM 7338 trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Meropenem trihydrate (SM 7338 trihydrate) 是一种碳青霉烯抗生素,具有广谱抗菌活性。它对敏感和耐药的杜克氏杆菌 (MIC 值为 0.015-0.12 mg/mL), 淋病奈瑟氏球菌 (MIC 值为 0.02-0.06 mg/mL)和流感嗜血杆菌 (MIC 值为 0.03-0.12 mg/mL) 具有活性。
T0717L Enoxacin

依诺沙星,NSC 629661,AT 2266,Pd107779,CI 919

DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Enoxacin (NSC-629661) 是一种可干扰DNA 复制的氟喹诺酮,抑制细菌 DNA 促旋酶 (IC50=126 µg/ml) 和拓扑异构酶 IV (IC50=26.5 µg/ml)。它是特异性癌症生长抑制剂,可有效抑制革兰氏阳性和阴性细菌。
T1492 Gemifloxacin mesylate

LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。
T1451 Levofloxacin hydrate

左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin hydrate (Cravit hydrate) 是抗生素化合物,抑制细菌DNA 旋转酶活性。
T66175 Ceftriaxone Sodium

GSK-3; Antibiotic; Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Microbiology/Virology; PI3K/Akt/mTOR signaling; Stem Cells
Ceftriaxone Sodium 是一种广谱 β-内酰胺类三代头孢菌素类抗生素 (antibiotic),具有抗炎、抗肿瘤、抗菌和抗氧化活性。Ceftriaxone Sodium 是一种共价 GSK3β和 Aurora B 抑制剂, 可用于研究败血症和感染性心内膜炎。
T1625 Lomefloxacin hydrochloride

Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin hydrochloride (Okacyn) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T4501 Ceftizoxime

头孢唑肟,Epocelin

Antibacterial; Antibiotic Microbiology/Virology
Ceftizoxime (Epocelin) 是一种强效抗菌剂,它通过干扰细菌细胞壁合成和抑制肽聚糖的交联起作用。它对广谱的 β-内酰胺酶具有高度抗性,并且对多种需氧和厌氧的革兰氏阳性和革兰氏阴性微生物均有效。
T1482 Ciclopirox

环吡酮,HOE296b,环吡酮胺

ATPase; Ferroptosis; Antibacterial; Autophagy; Antifungal Apoptosis; Autophagy; Membrane transporter/Ion channel; Microbiology/Virology
Ciclopirox (HOE296b) 是一种合成的抗真菌剂,可研究浅表真菌病。
T0932 Cefixime

FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635

Antibacterial; Antibiotic Microbiology/Virology
Cefixime (FR-17027) 是一种头孢菌素类抗生素, 可研究一些细菌感染。
T8747 Levofloxacin hydrochloride

DNA gyrase; Topoisomerase DNA Damage/DNA Repair
Levofloxacin hydrochloride 是一种广谱的第三代氟喹诺酮类抗生素,是氧氟沙星的光学活性 L-异构体,具有抗菌活性。左氧氟沙星通过细菌细胞壁扩散并通过抑制 DNA 促旋酶(细菌拓扑异构酶 II)起作用,这是一种 DNA 复制、RNA 转录和细菌 DNA 修复所需的酶。 DNA 促旋酶活性的抑制导致细菌细胞生长受阻。
T24525 Negamycin

Negamycin is an agent of broad-spectrum antibacterial that acts by inhibiting protein synthesis.
T25095 Antibiotic LB 10517

LB 10517,LB10517,Antibiotic LB10517,LB-10517,Antibiotic LB-10517

Antibiotic LB 10517 is a catechol-substituted cephalosporin with a broad spectrum of antibacterial.
T14923 Cefpiramide sodium

头孢匹胺钠,SM-1652,Wy-44635

Others Others
Cefpiramide sodium (SM-1652; Wy-44635) is a Pseudomonas-active cephalosporin. It has a broad spectrum of antibacterial activity.
T26612 AM-8191 HCl

AM-8191,AM 8191,AM8191

AM-8191, a bacterial topoisomerase inhibitors, has broad-spectrum antibacterial activity.
T25461 Grepafloxacin, (S)-

L-Grepafloxacin

Grepafloxacin, (S)- is an oral broad-spectrum fluoroquinolone antibacterial used for the treatment of bacterial infections.
T13026 Sulfadimethoxypyrimidine D4

Others Others
Sulfadimethoxypyrimidine D4, a deuterium-labeled version of Sulfadimethoxypyrimidine, is a sulfonamide antibiotic characterized by its broad-spectrum antibacterial effectiveness.
T38867 Antibacterial agent 42

Antibacterial Agent 42 demonstrates potent antibacterial activity by effectively reducing the Minimum Inhibitory Concentration (MIC) of the broad-spectrum antibacterial agent Ceftazidime.
T11227 Eravacycline

TP-434

Antibacterial Microbiology/Virology
Eravacycline (TP-434) 是一种有效的广谱抗菌剂。
T31025 CP 65207

CP65207;CP 81054,CP-65207,CP65207,CP 81054

CP 65207 is a new broad-spectrum penicillin antibacterial agent, which is a mixture of two stereoisomers (1:1).
T23622 Acorafloxacin HCl

JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl

Acorafloxacin is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and skin structure infections and community-acquired pneumonia.
T16513 PF 03709270

ulopenem etzadroxil

Others Others
PF 03709270 is an orally available ester prodrug form of sulopenem. It has broad-spectrum antibacterial activity against most gram-positive and gram-negative bacteria.
T10420 Avarofloxacin

JNJ-Q2

Others Others
Avarofloxacin (JNJ-Q2) is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and community-acquired pneumonia and skin structure infections.
T61493 Olanexidine

Olanexidine is a broad-spectrum antibacterial agent and antiseptic, effective against both Gram-positive and Gram-negative bacteria. It is commonly utilized in the research of infection and inflammation [1] [2] [3].
T72093 Thiamphenicol glycinate hydrochloride

甲砜霉素甘氨酸酯盐酸盐

Thiamphenicol glycinate hydrochloride 是一种广谱抗菌剂,可用于呼吸道感染的研究。
T75322 Cephaloridine hydrate

Cephaloridine hydrate,一种广谱性抗菌抗生素(antibiotic),具有剂量相关的肾毒性。
T83594 (+)-Thienamycin

(+)-Thienamycin是一种从Streptomyces cattleya中提取的有效的广谱抗菌剂和β-内酰胺酶抑制剂。
T68149 tacapenem

Tacapenem 是一种β-内酰胺类抗菌剂。它具有广谱抗菌活性,对β-内酰胺酶具有很高的稳定性。
T76260 Tet-213 TFA

Tet-213 TFA为具有广谱抗菌活性的抗菌肽,能促进被感染伤口的修复。
T39172 SMAP-29

SMAP-29 is a broad spectrum antibacterial and antifungal α-helical cathelicidin-derived peptide with strong potential as an antiinfective agent. It effectively permeabilizes bacterial membranes and induces significant alterations in the surface morphology of susceptible microorganisms.
T76259 Tet-213

Tet-213为一种具有广谱抗菌活性的抗菌肽,能促进被感染伤口的修复。

化合物

Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Cefpiramide acid
Cat.No: T0138
Synonym: Cefpiramidum,头孢匹胺,Cefpiramido
Target: Antibacterial
Tebipenem Pivoxil
Cat.No: T6231
Synonym: ME1211,Orapenem,替​比​培​南​匹​酯
Target: Antibacterial, Antibiotic
Omadacycline
Cat.No: T5189
Synonym: PTK 0796,Amadacycline
Target: ribosome, Antibacterial, Antibiotic
Ciclopirox olamine
Cat.No: T1114
Synonym: 环吡酮乙醇胺盐,环吡司胺,Ciclopirox ethanolamine
Target: ATPase, Others, Ferroptosis, Antibacterial, Antifungal
Eravacycline HCl
Cat.No: T11227L1
Synonym: Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl
Target: Antibiotic
Cefquinome sulfate
Cat.No: T4270
Synonym: 硫酸头孢喹肟,硫酸头孢喹诺
Target: Antibacterial, Antibiotic
Rosoxacin
Cat.No: T16789
Synonym: 罗索沙星,Acrosoxacin
Target: Antibacterial, Antibiotic
Levofloxacin Hydrochloride Impurity A
Cat.No: T11007L
Synonym: Levofloxacin Hydrochloride Impurity A(117707-40-1 Free base),左氧氟沙星杂质A(盐酸盐)
Target: Antibacterial
Lomefloxacin
Cat.No: T1444
Synonym: 洛美沙星,SC47111A
Target: Topoisomerase, Antibacterial, Antibiotic
Cefazolin
Cat.No: T8390
Synonym: 头孢唑林,头孢唑啉
Target: Others, Antibacterial, Antibiotic
Brodimoprim
Cat.No: T19858
Synonym:
Target: DHFR, Antibacterial
Ertapenem sodium
Cat.No: T4991
Synonym: 厄他培南钠,MK-826,L-749345,尔他培南钠
Target: Antibacterial, Antibiotic
Pefloxacin Mesylate
Cat.No: T0425
Synonym: Pefloxacinium mesylate,甲磺酸培氟沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Eravacycline dihydrochloride
Cat.No: T11227L
Synonym: TP-434-046,TP-434 dihydrochloride
Target: Antibacterial
Difloxacin hydrochloride
Cat.No: T8142
Synonym: Difloxacin HCl,盐酸二氟沙星
Target: Antibacterial, Antibiotic
Dup-721
Cat.No: T38359
Synonym:
Target: Antibacterial
Ceftiofur hydrochloride
Cat.No: T6268
Synonym: 头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride
Target: Antibacterial, Antibiotic
Enoxacin hydrate
Cat.No: T0717
Synonym: CI-919 hydrate,Enoxacin Sesquihydrate,依诺沙星半水合物,AT-2266 hydrate,依诺沙星倍半水合物
Target: DNA gyrase, DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic
Cyclo(L-Phe-L-Pro)
Cat.No: TN6672
Synonym:
Target: Free radical scavengers, COX, Antibacterial, Antifungal
Meropenem trihydrate
Cat.No: T12004
Synonym: 美罗培南三水合物,SM 7338 trihydrate
Target: Antibacterial, Antibiotic
Enoxacin
Cat.No: T0717L
Synonym: 依诺沙星,NSC 629661,AT 2266,Pd107779,CI 919
Target: DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic
Gemifloxacin mesylate
Cat.No: T1492
Synonym: LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate
Target: DNA gyrase, Topoisomerase, Antibacterial
Levofloxacin hydrate
Cat.No: T1451
Synonym: 左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Ceftriaxone Sodium
Cat.No: T66175
Synonym:
Target: GSK-3, Antibiotic, Aurora Kinase
Lomefloxacin hydrochloride
Cat.No: T1625
Synonym: Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin
Target: Topoisomerase, Antibacterial, Antibiotic
Ceftizoxime
Cat.No: T4501
Synonym: 头孢唑肟,Epocelin
Target: Antibacterial, Antibiotic
Ciclopirox
Cat.No: T1482
Synonym: 环吡酮,HOE296b,环吡酮胺
Target: ATPase, Ferroptosis, Antibacterial, Autophagy, Antifungal
Cefixime
Cat.No: T0932
Synonym: FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635
Target: Antibacterial, Antibiotic
Levofloxacin hydrochloride
Cat.No: T8747
Synonym:
Target: DNA gyrase, Topoisomerase
Negamycin
Cat.No: T24525
Synonym:
Target:
Antibiotic LB 10517
Cat.No: T25095
Synonym: LB 10517,LB10517,Antibiotic LB10517,LB-10517,Antibiotic LB-10517
Target:
Cefpiramide sodium
Cat.No: T14923
Synonym: 头孢匹胺钠,SM-1652,Wy-44635
Target: Others
AM-8191 HCl
Cat.No: T26612
Synonym: AM-8191,AM 8191,AM8191
Target:
Grepafloxacin, (S)-
Cat.No: T25461
Synonym: L-Grepafloxacin
Target:
Sulfadimethoxypyrimidine D4
Cat.No: T13026
Synonym:
Target: Others
Antibacterial agent 42
Cat.No: T38867
Synonym:
Target:
Eravacycline
Cat.No: T11227
Synonym: TP-434
Target: Antibacterial
CP 65207
Cat.No: T31025
Synonym: CP65207;CP 81054,CP-65207,CP65207,CP 81054
Target:
Acorafloxacin HCl
Cat.No: T23622
Synonym: JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl
Target:
PF 03709270
Cat.No: T16513
Synonym: ulopenem etzadroxil
Target: Others
Avarofloxacin
Cat.No: T10420
Synonym: JNJ-Q2
Target: Others
Olanexidine
Cat.No: T61493
Synonym:
Target:
Thiamphenicol glycinate hydrochloride
Cat.No: T72093
Synonym: 甲砜霉素甘氨酸酯盐酸盐
Target:
Cephaloridine hydrate
Cat.No: T75322
Synonym:
Target:
(+)-Thienamycin
Cat.No: T83594
Synonym:
Target:
tacapenem
Cat.No: T68149
Synonym:
Target:
Tet-213 TFA
Cat.No: T76260
Synonym:
Target:
SMAP-29
Cat.No: T39172
Synonym:
Target:
Tet-213
Cat.No: T76259
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2010 Ombuin

商陆黄素,商陆素

Antibacterial Microbiology/Virology
Ombuin 是一种从花椒中分离出的广谱抗菌剂,MIC 为 125 至 500 μg/mL。
T8063 Cephapirin Benzathine

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cephapirin Benzathine 是头孢哌啶的苄硫醚盐形式,是一种广谱抗生素。
T8258 Chloramphenicol succinate sodium

Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Chloramphenicol succinate sodium 是 Chloramphenicol 的前药,具有血液学毒性。它是琥珀酸脱氢酶的竞争底物和抑制剂。
T10164 5,6-Dihydroxyindole

Dopamine lutine

Endogenous Metabolite Metabolism
5,6-Dihydroxyindole (Dopamine lutine) 是黑色素的前体,显示出广谱的抗菌,抗真菌,抗病毒,抗寄生虫活性。5,6-Dihydroxyindole 也显示出细胞毒性作用。
T1687L Doxycycline (hyclate)

Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate

MMP; ribosome; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hyclate (WC2031) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline hyclate 具有抗菌活性和抗肿瘤活性。
T1687 Doxycycline

Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素

MMP; ribosome; Antibacterial; Antibiotic; Parasite Microbiology/Virology; Proteases/Proteasome
Doxycycline (Doxiciclina) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline 具有抗菌活性和抗肿瘤活性。
T1304 Chlortetracycline hydrochloride

Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。
TN6683 Cyclo(Pro-Trp)

Cyclo(Pro-Trp) and cyclo(Phe-Pro) show broad spectrum antibacterial properties.
T14347 Aureothricin

Antibacterial Microbiology/Virology
Aureothricin, a dithiolopyrrolone (DTP) antibiotic originally derived from Streptomyces, demonstrates a broad-spectrum of antibacterial effectiveness. Additionally, it inhibits the adhesion of human umbilical vein endothelial cells (HUVECs) to vitronectin[1].
T10825 Citrinin

NSC 186,桔霉素

Others Others
Citrinin is a mycotoxin that causes contamination in the food and is associated with different toxic effects. Citrinin also possesses a broad spectrum of bioactivities, including antifungal, antibacterial, and potential anticancer and neuroprotective effe
T8261 Ceftazidime Pentahydrate

头孢他啶五水合物,头孢他啶

Antibacterial; Antibiotic Microbiology/Virology
Ceftazidime pentahydrate 是一种β-内酰胺类抗菌剂,对革兰氏阳性和革兰氏阴性需氧细菌有广谱活性,可静脉内或肌肉给药。它对肠杆菌科特别有效,对大多数 β-内酰胺酶具有抗水解作用。
T79948 Kadsurenin B

Kadsurenin B为PAF(platelet-activating factor)拮抗剂,展现出神经保护作用。该化合物在药理学领域显示出广泛的研究潜力,包括抗菌、抗炎、神经保护、抗氧化、抗血小板聚集、细胞毒性和抗寄生虫等效能。
T80019 17-Hydroxyneomatrine

17-Hydroxyneomatrine 是一种从苦参 (Sophora flavescens) 提取的化合物,有效抑制人宫颈癌Hela细胞生长,并展现抗菌、抗过敏、抗肿瘤、抗心律失常、消肿、利尿、免疫调节等多种生物活性。
T80403 Nv-CATH

Nv-CATH是一种具有广谱抗菌活性的蛙源抗菌肽,有效针对革兰氏阳性菌和革兰氏阴性菌。它能显著提供保护,防止小鼠遭受金黄色葡萄球菌致命感染,并且通过免疫调节和抗微生物机制双重作用抵御细菌感染。

天然产物

Ombuin
Cat.No: TN2010
Synonym: 商陆黄素,商陆素
Target: Antibacterial
Cephapirin Benzathine
Cat.No: T8063
Synonym:
Target: Others, Antibacterial, Antibiotic
Chloramphenicol succinate sodium
Cat.No: T8258
Synonym: Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠
Target: Others, Antibacterial, Antibiotic
5,6-Dihydroxyindole
Cat.No: T10164
Synonym: Dopamine lutine
Target: Endogenous Metabolite
Doxycycline (hyclate)
Cat.No: T1687L
Synonym: Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate
Target: MMP, ribosome, Antibacterial, Antibiotic
Doxycycline
Cat.No: T1687
Synonym: Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素
Target: MMP, ribosome, Antibacterial, Antibiotic, Parasite
Chlortetracycline hydrochloride
Cat.No: T1304
Synonym: Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素
Target: ribosome, Antibacterial, Antibiotic
Cyclo(Pro-Trp)
Cat.No: TN6683
Synonym:
Target:
Aureothricin
Cat.No: T14347
Synonym:
Target: Antibacterial
Citrinin
Cat.No: T10825
Synonym: NSC 186,桔霉素
Target: Others
Ceftazidime Pentahydrate
Cat.No: T8261
Synonym: 头孢他啶五水合物,头孢他啶
Target: Antibacterial, Antibiotic
Kadsurenin B
Cat.No: T79948
Synonym:
Target:
17-Hydroxyneomatrine
Cat.No: T80019
Synonym:
Target:
Nv-CATH
Cat.No: T80403
Synonym:
Target:
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