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78

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T0138 Cefpiramide acid

Cefpiramidum,头孢匹胺,Cefpiramido

Antibacterial Microbiology/Virology
Cefpiramide acid (Cefpiramidum) 是第三代头孢菌素类抗生素。
T5189 Omadacycline

PTK 0796,Amadacycline

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Omadacycline (Amadacycline) 是一种具有口服活性的氨基甲基环素抗菌剂,是四环素类抗生素。它与 30S 核糖体亚基结合,抑制细菌蛋白质合成。它可用于研究急性细菌性皮肤和皮肤结构感染,感染性肺炎和尿路感染。
T6231 Tebipenem Pivoxil

ME1211,Orapenem,替​比​培​南​匹​酯

Antibacterial; Antibiotic Microbiology/Virology
Tebipenem Pivoxil (Orapenem) 是一种碳青霉烯类新型口服抗生素。
T1114 Ciclopirox olamine

环吡酮乙醇胺盐,环吡司胺,Ciclopirox ethanolamine

ATPase; Others; Ferroptosis; Antibacterial; Antifungal Apoptosis; Membrane transporter/Ion channel; Microbiology/Virology; Others
Ciclopirox olamine 是一种合成的抗真菌剂,可研究浅表真菌病。
T16789 Rosoxacin

罗索沙星,Acrosoxacin

Antibacterial; Antibiotic Microbiology/Virology
Rosoxacin (Acrosoxacin) 是具有口服活性的喹诺酮类抗生素,具有广谱的抗菌活性,抑制革兰氏阴性菌,包括淋病奈瑟氏球菌(MIC90=0.03 mg/ml)。它在尿路感染中有应用的潜能。
T11227L1 Eravacycline HCl

Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl

Antibiotic Microbiology/Virology
Eravacycline HCl (TP-434 HCl) 是一种具有广谱抗菌活性的强效抗生素。
T4270 Cefquinome sulfate

硫酸头孢喹肟,硫酸头孢喹诺

Antibacterial; Antibiotic Microbiology/Virology
Cefquinome sulfate 是一种半合成的头孢烯广谱抗生素,具有抗菌活性。
T1444 Lomefloxacin

洛美沙星,SC47111A

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin (SC47111A) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T8390 Cefazolin

头孢唑林,头孢唑啉

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazolin 是一种头孢类抗生素, 用于多种细菌感染的研究。
T11007L Levofloxacin Hydrochloride Impurity A

Levofloxacin Hydrochloride Impurity A(117707-40-1 Free base),左氧氟沙星杂质A(盐酸盐)

Antibacterial Microbiology/Virology
Levofloxacin Hydrochloride Impurity A 是一种喹诺酮类药物,具有广谱抗菌作用。
T4991 Ertapenem sodium

厄他培南钠,MK-826,L-749345,尔他培南钠

Antibacterial; Antibiotic Microbiology/Virology
Ertapenem sodium (MK-826) 是碳青霉烯,是一种 β-内酰胺抗生素,具有广谱抗菌活性。
T19858 Brodimoprim

DHFR; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Brodimoprim 是甲氧苄啶的一种类似物,是口服有效的二氢叶酸还原酶抑制剂,对广谱革兰氏阴性和革兰氏阳性细菌具有高度的抑制作用。
T0425 Pefloxacin Mesylate

Pefloxacinium mesylate,甲磺酸培氟沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。
T11227L Eravacycline dihydrochloride

TP-434-046,TP-434 dihydrochloride

Antibacterial Microbiology/Virology
Eravacycline dihydrochloride (TP-434-046) 是一种有效的广谱抗菌剂,可对抗六种大肠杆菌(MIC:0.125-0.25 mg/L)。
T8142 Difloxacin hydrochloride

Difloxacin HCl,盐酸二氟沙星

Antibacterial; Antibiotic Microbiology/Virology
Difloxacin hydrochloride (Difloxacin HCl) 是一种广谱抗菌药物。它干扰 DNA 促旋酶和拓扑异构酶 IV 的活性,抑制细菌 DNA 促旋酶并显示出浓度依赖性的杀菌作用。
T0717 Enoxacin hydrate

CI-919 hydrate,Enoxacin Sesquihydrate,依诺沙星半水合物,AT-2266 hydrate,依诺沙星倍半水合物

DNA gyrase; DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Enoxacin hydrate (AT-2266 hydrate) 是氟喹诺酮,可干扰DNA 复制,抑制细菌 DNA 促旋酶 (IC50=126 µg/ml) 和拓扑异构酶 IV (IC50=26.5 µg/ml)。它是特异性癌症生长抑制剂,抑制革兰氏阳性和阴性细菌。
T6268 Ceftiofur hydrochloride

头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur hydrochloride (U-67279A) 是头孢噻呋的盐酸盐形式,是一种β-内酰胺酶稳定的半合成广谱头孢菌素,具有抗菌活性。
T38359 Dup-721

Antibacterial Microbiology/Virology
DuP-721 是广谱的口服有效的抗菌剂,可以抑制多种临床敏感和耐药细菌,特别是结核杆菌M. tuberculosis。
TN6672 Cyclo(L-Phe-L-Pro)

Free radical scavengers; COX; Antibacterial; Antifungal Immunology/Inflammation; Microbiology/Virology; Neuroscience; oxidation-reduction
Cyclo(L-Phe-L-Pro) 具有广谱抗菌和抗真菌活性。 Cyclo(L-Phe-L-Pro) 对耐甲氧西林金黄色葡萄球菌和棉子肠球菌具有活性。
T12004 Meropenem trihydrate

美罗培南三水合物,SM 7338 trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Meropenem trihydrate (SM 7338 trihydrate) 是一种碳青霉烯抗生素,具有广谱抗菌活性。它对敏感和耐药的杜克氏杆菌 (MIC 值为 0.015-0.12 mg/mL), 淋病奈瑟氏球菌 (MIC 值为 0.02-0.06 mg/mL)和流感嗜血杆菌 (MIC 值为 0.03-0.12 mg/mL) 具有活性。
T0717L Enoxacin

依诺沙星,NSC 629661,AT 2266,Pd107779,CI 919

DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Enoxacin (NSC-629661) 是一种可干扰DNA 复制的氟喹诺酮,抑制细菌 DNA 促旋酶 (IC50=126 µg/ml) 和拓扑异构酶 IV (IC50=26.5 µg/ml)。它是特异性癌症生长抑制剂,可有效抑制革兰氏阳性和阴性细菌。
T1492 Gemifloxacin mesylate

LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。
T1451 Levofloxacin hydrate

左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin hydrate (Cravit hydrate) 是抗生素化合物,抑制细菌DNA 旋转酶活性。
T66175 Ceftriaxone Sodium

GSK-3; Antibiotic; Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Microbiology/Virology; PI3K/Akt/mTOR signaling; Stem Cells
Ceftriaxone Sodium 是一种广谱 β-内酰胺类三代头孢菌素类抗生素 (antibiotic),具有抗炎、抗肿瘤、抗菌和抗氧化活性。Ceftriaxone Sodium 是一种共价 GSK3β和 Aurora B 抑制剂, 可用于研究败血症和感染性心内膜炎。
T1625 Lomefloxacin hydrochloride

Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Lomefloxacin hydrochloride (Okacyn) 是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
T4501 Ceftizoxime

头孢唑肟,Epocelin

Antibacterial; Antibiotic Microbiology/Virology
Ceftizoxime (Epocelin) 是一种强效抗菌剂,它通过干扰细菌细胞壁合成和抑制肽聚糖的交联起作用。它对广谱的 β-内酰胺酶具有高度抗性,并且对多种需氧和厌氧的革兰氏阳性和革兰氏阴性微生物均有效。
T1482 Ciclopirox

环吡酮,HOE296b,环吡酮胺

ATPase; Ferroptosis; Antibacterial; Autophagy; Antifungal Apoptosis; Autophagy; Membrane transporter/Ion channel; Microbiology/Virology
Ciclopirox (HOE296b) 是一种合成的抗真菌剂,可研究浅表真菌病。
T0932 Cefixime

FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635

Antibacterial; Antibiotic Microbiology/Virology
Cefixime (FR-17027) 是一种头孢菌素类抗生素, 可研究一些细菌感染。
T8747 Levofloxacin hydrochloride

DNA gyrase; Topoisomerase DNA Damage/DNA Repair
Levofloxacin hydrochloride 是一种广谱的第三代氟喹诺酮类抗生素,是氧氟沙星的光学活性 L-异构体,具有抗菌活性。左氧氟沙星通过细菌细胞壁扩散并通过抑制 DNA 促旋酶(细菌拓扑异构酶 II)起作用,这是一种 DNA 复制、RNA 转录和细菌 DNA 修复所需的酶。 DNA 促旋酶活性的抑制导致细菌细胞生长受阻。
T24525 Negamycin

Negamycin is an agent of broad-spectrum antibacterial that acts by inhibiting protein synthesis.
T26612 AM-8191 HCl

AM-8191,AM 8191,AM8191

AM-8191, a bacterial topoisomerase inhibitors, has broad-spectrum antibacterial activity.
T14923 Cefpiramide sodium

头孢匹胺钠,SM-1652,Wy-44635

Others Others
Cefpiramide sodium (SM-1652; Wy-44635) is a Pseudomonas-active cephalosporin. It has a broad spectrum of antibacterial activity.
T25095 Antibiotic LB 10517

LB 10517,LB10517,Antibiotic LB10517,LB-10517,Antibiotic LB-10517

Antibiotic LB 10517 is a catechol-substituted cephalosporin with a broad spectrum of antibacterial.
T25461 Grepafloxacin, (S)-

L-Grepafloxacin

Grepafloxacin, (S)- is an oral broad-spectrum fluoroquinolone antibacterial used for the treatment of bacterial infections.
T38867 Antibacterial agent 42

Antibacterial Agent 42 demonstrates potent antibacterial activity by effectively reducing the Minimum Inhibitory Concentration (MIC) of the broad-spectrum antibacterial agent Ceftazidime.
T13026 Sulfadimethoxypyrimidine D4

Others Others
Sulfadimethoxypyrimidine D4, a deuterium-labeled version of Sulfadimethoxypyrimidine, is a sulfonamide antibiotic characterized by its broad-spectrum antibacterial effectiveness.
T31025 CP 65207

CP65207;CP 81054,CP-65207,CP65207,CP 81054

CP 65207 is a new broad-spectrum penicillin antibacterial agent, which is a mixture of two stereoisomers (1:1).
T23622 Acorafloxacin HCl

JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl

Acorafloxacin is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and skin structure infections and community-acquired pneumonia.
T16513 PF 03709270

ulopenem etzadroxil

Others Others
PF 03709270 is an orally available ester prodrug form of sulopenem. It has broad-spectrum antibacterial activity against most gram-positive and gram-negative bacteria.
T11227 Eravacycline

TP-434

Antibacterial Microbiology/Virology
Eravacycline (TP-434) 是一种有效的广谱抗菌剂。
T10420 Avarofloxacin

JNJ-Q2

Others Others
Avarofloxacin (JNJ-Q2) is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and community-acquired pneumonia and skin structure infections.
T61493 Olanexidine

Olanexidine is a broad-spectrum antibacterial agent and antiseptic, effective against both Gram-positive and Gram-negative bacteria. It is commonly utilized in the research of infection and inflammation [1] [2] [3].
T75322 Cephaloridine hydrate

Cephaloridine hydrate,一种广谱性抗菌抗生素(antibiotic),具有剂量相关的肾毒性。
T72093 Thiamphenicol glycinate hydrochloride

甲砜霉素甘氨酸酯盐酸盐

Thiamphenicol glycinate hydrochloride 是一种广谱抗菌剂,可用于呼吸道感染的研究。
T68149 tacapenem

Tacapenem 是一种β-内酰胺类抗菌剂。它具有广谱抗菌活性,对β-内酰胺酶具有很高的稳定性。
T83594 (+)-Thienamycin

(+)-Thienamycin是一种从Streptomyces cattleya中提取的有效的广谱抗菌剂和β-内酰胺酶抑制剂。
T39172 SMAP-29

SMAP-29 is a broad spectrum antibacterial and antifungal α-helical cathelicidin-derived peptide with strong potential as an antiinfective agent. It effectively permeabilizes bacterial membranes and induces significant alterations in the surface morphology of susceptible microorganisms.
T76260 Tet-213 TFA

Tet-213 TFA为具有广谱抗菌活性的抗菌肽,能促进被感染伤口的修复。
T75246 Cyclacillin

Cyclacillin (Wy-4508),一种口服氨基青霉素类抗生素,展示对革兰氏阳性及阴性病原体的广泛抗菌活性。

化合物

Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Cefpiramide acid
Cat.No: T0138
Synonym: Cefpiramidum,头孢匹胺,Cefpiramido
Target: Antibacterial
Omadacycline
Cat.No: T5189
Synonym: PTK 0796,Amadacycline
Target: ribosome, Antibacterial, Antibiotic
Tebipenem Pivoxil
Cat.No: T6231
Synonym: ME1211,Orapenem,替​比​培​南​匹​酯
Target: Antibacterial, Antibiotic
Ciclopirox olamine
Cat.No: T1114
Synonym: 环吡酮乙醇胺盐,环吡司胺,Ciclopirox ethanolamine
Target: ATPase, Others, Ferroptosis, Antibacterial, Antifungal
Rosoxacin
Cat.No: T16789
Synonym: 罗索沙星,Acrosoxacin
Target: Antibacterial, Antibiotic
Eravacycline HCl
Cat.No: T11227L1
Synonym: Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl
Target: Antibiotic
Cefquinome sulfate
Cat.No: T4270
Synonym: 硫酸头孢喹肟,硫酸头孢喹诺
Target: Antibacterial, Antibiotic
Lomefloxacin
Cat.No: T1444
Synonym: 洛美沙星,SC47111A
Target: Topoisomerase, Antibacterial, Antibiotic
Cefazolin
Cat.No: T8390
Synonym: 头孢唑林,头孢唑啉
Target: Others, Antibacterial, Antibiotic
Levofloxacin Hydrochloride Impurity A
Cat.No: T11007L
Synonym: Levofloxacin Hydrochloride Impurity A(117707-40-1 Free base),左氧氟沙星杂质A(盐酸盐)
Target: Antibacterial
Ertapenem sodium
Cat.No: T4991
Synonym: 厄他培南钠,MK-826,L-749345,尔他培南钠
Target: Antibacterial, Antibiotic
Brodimoprim
Cat.No: T19858
Synonym:
Target: DHFR, Antibacterial
Pefloxacin Mesylate
Cat.No: T0425
Synonym: Pefloxacinium mesylate,甲磺酸培氟沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Eravacycline dihydrochloride
Cat.No: T11227L
Synonym: TP-434-046,TP-434 dihydrochloride
Target: Antibacterial
Difloxacin hydrochloride
Cat.No: T8142
Synonym: Difloxacin HCl,盐酸二氟沙星
Target: Antibacterial, Antibiotic
Enoxacin hydrate
Cat.No: T0717
Synonym: CI-919 hydrate,Enoxacin Sesquihydrate,依诺沙星半水合物,AT-2266 hydrate,依诺沙星倍半水合物
Target: DNA gyrase, DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic
Ceftiofur hydrochloride
Cat.No: T6268
Synonym: 头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride
Target: Antibacterial, Antibiotic
Dup-721
Cat.No: T38359
Synonym:
Target: Antibacterial
Cyclo(L-Phe-L-Pro)
Cat.No: TN6672
Synonym:
Target: Free radical scavengers, COX, Antibacterial, Antifungal
Meropenem trihydrate
Cat.No: T12004
Synonym: 美罗培南三水合物,SM 7338 trihydrate
Target: Antibacterial, Antibiotic
Enoxacin
Cat.No: T0717L
Synonym: 依诺沙星,NSC 629661,AT 2266,Pd107779,CI 919
Target: DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic
Gemifloxacin mesylate
Cat.No: T1492
Synonym: LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate
Target: DNA gyrase, Topoisomerase, Antibacterial
Levofloxacin hydrate
Cat.No: T1451
Synonym: 左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Ceftriaxone Sodium
Cat.No: T66175
Synonym:
Target: GSK-3, Antibiotic, Aurora Kinase
Lomefloxacin hydrochloride
Cat.No: T1625
Synonym: Lomefloxacin HCl,盐酸洛美沙星,Okacyn,Maxaquin
Target: Topoisomerase, Antibacterial, Antibiotic
Ceftizoxime
Cat.No: T4501
Synonym: 头孢唑肟,Epocelin
Target: Antibacterial, Antibiotic
Ciclopirox
Cat.No: T1482
Synonym: 环吡酮,HOE296b,环吡酮胺
Target: ATPase, Ferroptosis, Antibacterial, Autophagy, Antifungal
Cefixime
Cat.No: T0932
Synonym: FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635
Target: Antibacterial, Antibiotic
Levofloxacin hydrochloride
Cat.No: T8747
Synonym:
Target: DNA gyrase, Topoisomerase
Negamycin
Cat.No: T24525
Synonym:
Target:
AM-8191 HCl
Cat.No: T26612
Synonym: AM-8191,AM 8191,AM8191
Target:
Cefpiramide sodium
Cat.No: T14923
Synonym: 头孢匹胺钠,SM-1652,Wy-44635
Target: Others
Antibiotic LB 10517
Cat.No: T25095
Synonym: LB 10517,LB10517,Antibiotic LB10517,LB-10517,Antibiotic LB-10517
Target:
Grepafloxacin, (S)-
Cat.No: T25461
Synonym: L-Grepafloxacin
Target:
Antibacterial agent 42
Cat.No: T38867
Synonym:
Target:
Sulfadimethoxypyrimidine D4
Cat.No: T13026
Synonym:
Target: Others
CP 65207
Cat.No: T31025
Synonym: CP65207;CP 81054,CP-65207,CP65207,CP 81054
Target:
Acorafloxacin HCl
Cat.No: T23622
Synonym: JNJ-32729463,JNJ-Q2 hydrochloride,Acorafloxacin hydrochloride,JNJ 32729463,JNJ-Q2 HCl
Target:
PF 03709270
Cat.No: T16513
Synonym: ulopenem etzadroxil
Target: Others
Eravacycline
Cat.No: T11227
Synonym: TP-434
Target: Antibacterial
Avarofloxacin
Cat.No: T10420
Synonym: JNJ-Q2
Target: Others
Olanexidine
Cat.No: T61493
Synonym:
Target:
Cephaloridine hydrate
Cat.No: T75322
Synonym:
Target:
Thiamphenicol glycinate hydrochloride
Cat.No: T72093
Synonym: 甲砜霉素甘氨酸酯盐酸盐
Target:
tacapenem
Cat.No: T68149
Synonym:
Target:
(+)-Thienamycin
Cat.No: T83594
Synonym:
Target:
SMAP-29
Cat.No: T39172
Synonym:
Target:
Tet-213 TFA
Cat.No: T76260
Synonym:
Target:
Cyclacillin
Cat.No: T75246
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2010 Ombuin

商陆黄素,商陆素

Antibacterial Microbiology/Virology
Ombuin 是一种从花椒中分离出的广谱抗菌剂,MIC 为 125 至 500 μg/mL。
T8063 Cephapirin Benzathine

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cephapirin Benzathine 是头孢哌啶的苄硫醚盐形式,是一种广谱抗生素。
T8258 Chloramphenicol succinate sodium

Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Chloramphenicol succinate sodium 是 Chloramphenicol 的前药,具有血液学毒性。它是琥珀酸脱氢酶的竞争底物和抑制剂。
T1687 Doxycycline

Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素

MMP; ribosome; Antibacterial; Antibiotic; Parasite Microbiology/Virology; Proteases/Proteasome
Doxycycline (Doxiciclina) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline 具有抗菌活性和抗肿瘤活性。
T10164 5,6-Dihydroxyindole

Dopamine lutine

Endogenous Metabolite Metabolism
5,6-Dihydroxyindole (Dopamine lutine) 是黑色素的前体,显示出广谱的抗菌,抗真菌,抗病毒,抗寄生虫活性。5,6-Dihydroxyindole 也显示出细胞毒性作用。
T1687L Doxycycline (hyclate)

Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate

MMP; ribosome; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hyclate (WC2031) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline hyclate 具有抗菌活性和抗肿瘤活性。
T1304 Chlortetracycline hydrochloride

Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。
TN6683 Cyclo(Pro-Trp)

Cyclo(Pro-Trp) and cyclo(Phe-Pro) show broad spectrum antibacterial properties.
T14347 Aureothricin

Antibacterial Microbiology/Virology
Aureothricin, a dithiolopyrrolone (DTP) antibiotic originally derived from Streptomyces, demonstrates a broad-spectrum of antibacterial effectiveness. Additionally, it inhibits the adhesion of human umbilical vein endothelial cells (HUVECs) to vitronectin[1].
T10825 Citrinin

NSC 186,桔霉素

Others Others
Citrinin is a mycotoxin that causes contamination in the food and is associated with different toxic effects. Citrinin also possesses a broad spectrum of bioactivities, including antifungal, antibacterial, and potential anticancer and neuroprotective effe
T8261 Ceftazidime Pentahydrate

头孢他啶五水合物,头孢他啶

Antibacterial; Antibiotic Microbiology/Virology
Ceftazidime pentahydrate 是一种β-内酰胺类抗菌剂,对革兰氏阳性和革兰氏阴性需氧细菌有广谱活性,可静脉内或肌肉给药。它对肠杆菌科特别有效,对大多数 β-内酰胺酶具有抗水解作用。
T79948 Kadsurenin B

Kadsurenin B为PAF(platelet-activating factor)拮抗剂,展现出神经保护作用。该化合物在药理学领域显示出广泛的研究潜力,包括抗菌、抗炎、神经保护、抗氧化、抗血小板聚集、细胞毒性和抗寄生虫等效能。
T80019 17-Hydroxyneomatrine

17-Hydroxyneomatrine 是一种从苦参 (Sophora flavescens) 提取的化合物,有效抑制人宫颈癌Hela细胞生长,并展现抗菌、抗过敏、抗肿瘤、抗心律失常、消肿、利尿、免疫调节等多种生物活性。
T80403 Nv-CATH

Nv-CATH是一种具有广谱抗菌活性的蛙源抗菌肽,有效针对革兰氏阳性菌和革兰氏阴性菌。它能显著提供保护,防止小鼠遭受金黄色葡萄球菌致命感染,并且通过免疫调节和抗微生物机制双重作用抵御细菌感染。

天然产物

Ombuin
Cat.No: TN2010
Synonym: 商陆黄素,商陆素
Target: Antibacterial
Cephapirin Benzathine
Cat.No: T8063
Synonym:
Target: Others, Antibacterial, Antibiotic
Chloramphenicol succinate sodium
Cat.No: T8258
Synonym: Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠
Target: Others, Antibacterial, Antibiotic
Doxycycline
Cat.No: T1687
Synonym: Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素
Target: MMP, ribosome, Antibacterial, Antibiotic, Parasite
5,6-Dihydroxyindole
Cat.No: T10164
Synonym: Dopamine lutine
Target: Endogenous Metabolite
Doxycycline (hyclate)
Cat.No: T1687L
Synonym: Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate
Target: MMP, ribosome, Antibacterial, Antibiotic
Chlortetracycline hydrochloride
Cat.No: T1304
Synonym: Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素
Target: ribosome, Antibacterial, Antibiotic
Cyclo(Pro-Trp)
Cat.No: TN6683
Synonym:
Target:
Aureothricin
Cat.No: T14347
Synonym:
Target: Antibacterial
Citrinin
Cat.No: T10825
Synonym: NSC 186,桔霉素
Target: Others
Ceftazidime Pentahydrate
Cat.No: T8261
Synonym: 头孢他啶五水合物,头孢他啶
Target: Antibacterial, Antibiotic
Kadsurenin B
Cat.No: T79948
Synonym:
Target:
17-Hydroxyneomatrine
Cat.No: T80019
Synonym:
Target:
Nv-CATH
Cat.No: T80403
Synonym:
Target:
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