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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T1674	Nateglinide 那格列奈,A4166,Senaglinide	Potassium Channel; Proteasome; PPAR	DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Proteases/Proteasome; Ubiquitination
	Nateglinide (Senaglinide) 是 D-苯丙氨酸的一种衍生物，是口服有效的、短效促胰岛素释放化合物，也是 DPP IV 抑制剂。 Nateglinide 抑制胰岛 β 细胞中 ATP 敏感的 K+通道。Nateglinide 在 2 型糖尿病中具有研究价值。
T4548	Procaterol hydrochloride	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Procaterol hydrochloride 用于治疗哮喘的短效β2-肾上腺素受体激动剂。
T4551	Acrivastine Acrivastin,阿伐斯汀,BW825C,Semprex	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Acrivastine (Acrivastin) 是一种短效组胺 1 受体拮抗剂，可用于研究过敏性鼻炎。
T0747	Sulfathiazole 2-Sulfanilamidothiazole,磺胺噻唑	Antibacterial; Antibiotic; Autophagy	Autophagy; Microbiology/Virology
	Sulfathiazole (2-Sulfanilamidothiazole) 是一种短效磺胺类抗生素。
T0015	Mephenesin Cresoxydiol,甲酚甘油醚,Memphenesin,Mephedan,Decontractyl	NMDAR; iGluR	Membrane transporter/Ion channel; Neuroscience
	Mephenesin (Cresoxydiol) 是 NMDA 受体拮抗剂，也是中枢性肌松弛剂。
T3288	Sulfisomidin Sulfisomidine,Sulfadimetine,磺胺二甲基异嘧啶,sulfamethin,磺胺二甲异嘧啶,Sulfaisodimidine	Antibacterial; Antibiotic	Microbiology/Virology
	Sulfisomidin (Sulfaisodimidine) 是一种具有口服活性的短效磺酰胺类抗菌剂。它可研究下尿路感染。
T6652	Salbutamol hemisulfate Ventolin Sulfate,沙丁胺醇半硫酸盐,Albuterol,Salbutamol Sulfate,硫酸沙丁胺醇,Bronchospray,Albuterol Sulfate	Adrenergic Receptor; Autophagy	Autophagy; GPCR/G Protein; Neuroscience
	Salbutamol hemisulfate (Albuterol Sulfate) 是一种短效的β2肾上腺素受体激动剂，IC50 为 8.93 μM。
T5028	Landiolol hydrochloride ONO-1101 hydrochloride,盐酸兰地洛尔	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Landiolol hydrochloride (ONO-1101 hydrochloride) 是一种肾上腺素能受体拮抗剂，是一种 beta1 高选择性的超短作用β- 阻断剂(β1 /β2 选择性 = 255:1, 半衰期 4 分钟)。
T6461	Dapoxetine hydrochloride LY-210448,LY-210448 hydrochloride,Dapoxetine HCl,盐酸达泊西汀,Priligy	5-HT Receptor; Serotonin Transporter	GPCR/G Protein; Neuroscience
	Dapoxetine hydrochloride (LY-210448 hydrochloride) 是一种具有口服活性的、选择性的血清素再摄取 (serotonin reuptake) 抑制剂 (SSRI)，可用于研究早泄 (PE) 。
T0767	Sulfapyridine 磺胺吡啶,Sulfidine,Sulfidin,2-Sulfapyridine	Antibacterial; Antibiotic; Autophagy	Autophagy; Microbiology/Virology
	Sulfapyridine (2-Sulfapyridine) 是一种磺酰胺类抗生素，是 Sulfasalazine 的代谢产物。它抑制重组 P. carinii 二氢蝶呤合成酶，IC50为 0.18 μM。它具有抗菌，抗炎和抗风湿作用。
T0750	Sulfisoxazole NU-445,磺胺二甲异唑,Sulfafurazole,磺胺异恶唑	Endothelin Receptor; Antibacterial; Antibiotic; Autophagy	Autophagy; GPCR/G Protein; Microbiology/Virology
	Sulfisoxazole (Sulfafurazole) 是一种内皮素受体拮抗剂，是磺胺类抗生素。它靶向内皮素受体 A，抑制乳腺癌外显子释放。
T1603	Glipizide CP 28720,K 4024,格列吡嗪	Potassium Channel; PPAR; ABC	DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
	Glipizide (CP 28720) 是一种有效的、具有口服活性的磺酰脲类抗糖尿病试剂 (anti-diabetic agent)，在 2 型糖尿病的研究中具有价值，但不适用于1 型糖尿病。Glipizide 是通过部分阻断郎格汉斯胰岛细胞中 ATP 敏感钾通道 (KATP)发挥活性。
T0930	Sulfadiazine Sulphadiazine,磺胺嘧啶	Antibacterial; Antibiotic; Parasite; Autophagy	Autophagy; Microbiology/Virology
	Sulfadiazine (Sulphadiazine) 是一种磺胺类抗生素具有抗疟活性，可研究弓形虫病。
T9516	Binodenoson WRC 0470,MRE-0470,比诺地松,2-(cyclohexylmethylidenehydrazino)adenos	Adenosine Receptor	GPCR/G Protein; Neuroscience
	Binodenoson (WRC 0470) 是一种选择性A2A 腺苷受体激动剂，KD 为270 nM。它是一种短效冠状动脉血管扩张剂，作为放射性示踪剂的辅助剂，用于心肌应激成像。
T11174	(R)-Elagolix 恶拉戈利,NBI-56418	GNRH Receptor	GPCR/G Protein
	(R)-Elagolix (NBI-56418) 是口服具有活性的、选择性高的非肽类促性腺激素释放激素受体短期有效拮抗剂 (KD = 54 pM)。
T0114	Trichlormethiazide Naqua,Metahydrin,三氯噻嗪,Trichlormetazid	ATPase; Carbonic Anhydrase	Membrane transporter/Ion channel; Metabolism
	Trichlormethiazide (Naqua) 是一种口服具有活力的噻嗪类利尿剂，具有降压作用。它能够提高急性肾功能衰竭大鼠的尿量、Na 和 K 排泄，并有改善降低的肌酐清除率。
T15257	Etripamil MSP-2017,(-)-MSP-2017	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Etripamil (MSP-2017) 是一种短效L 型钙通道拮抗剂，可用于治疗阵发性室上性心动过速的研究。它通过抑制房室结细胞中钙慢通道的钙离子流入，显示房室结传导并延长房室结不应期
T0999	Clevidipine Clevidipine butyrate,丁酸氯维地平,氯维地平,Cleviprex	Calcium Channel; AChR	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Clevidipine (Clevidipine butyrate) butyrate 是一种二氢吡啶 L 型钙通道阻滞剂，IC50为7.1 nM。它对血管平滑肌有选择性，可用于降低血压。
T1139	Salbutamol Albuterol,沙丁胺醇,AH-3365	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Salbutamol (Albuterol) 是短效的 β2 肾上腺素受体激动剂，用于哮喘和慢性阻塞性肺疾病(COPD) 引发的支气管痉挛的研究。
T29005	Trefentanil hydrochloride
	Trefentanil hydrochloride is a short-acting analgesic.
T30623	Buthalital sodium baytinal
	Buthalital sodium is a short-acting anesthetic derived from barbiturates.
T5028L	Landiolol ONO1101,ONO 1101,ONO-1101
	Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.
T69394	Carbuterol hydrochloride
	Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.
T28383	PF-4455242
	PF-4455242 is a selective, short-acting antagonist of the κ-opioid receptor.
T27543	HIE-124
	HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.
T26919	BU09059 BU 09059,BU-09059
	BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).
T28421	Pirbuterol Pirbuterolum,CP-24,314-14
	Pirbuterol, a short-acting β2 adrenoreceptor agonist, has bronchodilating action used in the treatment of asthma.
T23402	Sulfathiazole sodium	Others	Others
	Sulfathiazole Sodium is an organosulfur compound. It also has been used as a short-acting sulfa drug.
T34079	Pirbuterol Acetate pirbuterol sulfate,EINECS 265-862-4,Maxair,Pirbuterol acetate (USAN)
	Pibuterol Acetate is a short-acting beta-2 adrenergic receptor agonist with bronchiectasis and is used as a respiratory activated quantitative inhaler in the treatment of asthma.
T12780L	RP-001 hydrochloride	Others	Others
	RP-001 hydrochloride is a selective agonist of picomolar short-acting S1P1 (EDG1)(EC50 of 9 pM), has little activity on S1P2-S1P4 and only moderate affinity for S1P5.
T34740	Sulfacytine Renoquid,CI636,CI-636,CI 636,磺胺西汀,Sulfacitinum
	Sulfacytine is a short-acting sulfonamides antibiotic that is taken orally to treat bacterial infections. Sulfonamides, a group of antibiotics, work by inhibiting bacterial production of folic acid.
T12780	RP-001	Others	Others
	RP-001 is a selective agonist of picomolar short-acting S1P1 (EDG1)(EC50 of 9 pM), has little activity on S1P2-S1P4 and only moderate affinity for S1P5.
T13035	Sulfathiazole-d4	Others	Others
	Sulfathiazole D4 is a deuterium labeled Sulfathiazole. Sulfathiazole used as a short-acting sulfonamide antibiotic.
T70089	Colterol (free base)
	Colterol (free base) is a short-acting β2-adrenoreceptor agonist. Bitolterol, a prodrug for colterol, is used in the management of bronchospasm in asthma and chronic obstructive pulmonary disease.
T10241	Acrivastine D7 BW825C D7	Others	Others
	Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.
T39820	Dapiglutide ZP7570
	Dapiglutide (ZP7570) is a long-acting dual agonist of glucagon-like peptide-1 receptor (GLP-1R) and glucagon-like peptide-2 receptor (GLP-2R) that holds potential for short bowel syndrome (SBS) research.
T25030	Albuterol stearate
	Albuterol stearate is a salt of Albuterol. Albuterol is a short-acting, selective beta2-adrenergic receptor agonist used in the treatment of asthma and COPD. It is 29 times more selective for beta2 receptors than beta1 receptors.
T69472	Edrophonium
	Edrophonium is a rapid-onset, short-acting cholinesterase inhibitor used in cardiac arrhythmias and in the diagnosis of myasthenia gravis. It has also been used as an antidote to curare principles.
T69148	Colterol HCl
	Colterol HCl is the salt form of Colterol (free base), a short-acting β2-adrenoreceptor agonist. Bitolterol, a prodrug for colterol, is used in the management of bronchospasm in asthma and chronic obstructive pulmonary disease.
T10436L	AZD4573 HCl (2057509-72-3 free base) AZD4573 hydrochloride,AZD4573,AZD4573 HCl,AZD-4573,AZD 4573
	AZD-4573 is a selective and short-acting inhibitor of the serine/threonine cyclin-dependent kinase 9, the catalytic subunit of the RNA polymerase II elongation factor positive transcription elongation factor b. It also has a potential antineoplastic activ
T37378	Propofol β-D-Glucuronide
	Propofol β-D-glucuronide is a metabolite of propofol sulfate , a short-acting anesthetic agent. [1] [2] The metabolite is generated through the glucuronidation of propofol by uridine diphosphate glucuronosyltransferases. Propofol metabolism appears to occur more rapidly in women than men. [1]
T69144	Hexylcaine HCl
	Hexylcaine HCl also called cyclaine or osmocaine, is a short-acting local anesthetic. It acts by inhibiting sodium channel conduction. Overdose can lead to headache, tinnitus, numbness and tingling around the mouth and tongue, convulsions, inability to breathe, and decreased heart function.
TP1473	Velmupressin c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively.
TP1560	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm a highly efficient, selective and short-acting peptide V2 receptor agonist (V2R), with EC50s of hV2R and rV2R being 0.25 and 0.05 nM, respectively.
TP1205	Velmupressin acetate V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively.
TP1171	Apraglutide TFA (1295353-98-8 free base) Apraglutide TFA,FE 203799e (TFA)
	Apraglutide TFA (FE 203799 TFA), a synthetic 33-amino-acid peptide and a long-acting GLP-2 analogue, enhances adaptation and linear intestinal growth in a neonatal piglet model of short bowel syndrome with total resection of the ileum.
T70551	Albuterol adipate
	Albuterol adipate is a salt of Albuterol -- β2-AR agonist. Albuterol is a short-acting, selective beta2-adrenergic receptor agonist used in the treatment of asthma and COPD. It is 29 times more selective for beta2 receptors than beta1 receptors giving it higher specificity for pulmonary beta receptors versus beta1-adrenergic receptors located in the heart.
T68811	Trimetaphan camsilate
	Trimetaphan camsilate is a drug that counteracts cholinergic transmission at the ganglion type of nicotinic receptors of the autonomic ganglia and therefore blocks both the sympathetic nervous system and the parasympathetic nervous system. It acts as a non-depolarizing competitive antagonist at the nicotinic acetylcholine receptor, is short-acting, and is given intravenously.
T60502	Isoetharine hydrochloride
	Isoetharine (hydrochloride) (compound I) 是一种选择性和口服活性的短效β-肾上腺能受体激动剂，广泛用作吸入治疗研究中的支气管扩张剂。
T76001	Apraglutide TFA
	Apraglutide TFA (FE 203799 TFA) 是一种合成的、含33个氨基酸的肽类药物，为长效GLP-2类似物。它能在全回肠切除后导致的新生短肠综合征小猪中增强适应性和线性肠生长。

化合物

Cat.No: T1674

Synonym: 那格列奈,A4166,Senaglinide

Target: Potassium Channel, Proteasome, PPAR

Procaterol hydrochloride

Cat.No: T4548

Target: Adrenergic Receptor

Cat.No: T4551

Synonym: Acrivastin,阿伐斯汀,BW825C,Semprex

Target: Histamine Receptor

Cat.No: T0747

Synonym: 2-Sulfanilamidothiazole,磺胺噻唑

Target: Antibacterial, Antibiotic, Autophagy

Cat.No: T0015

Synonym: Cresoxydiol,甲酚甘油醚,Memphenesin,Mephedan,Decontractyl

Target: NMDAR, iGluR

Cat.No: T3288

Synonym: Sulfisomidine,Sulfadimetine,磺胺二甲基异嘧啶,sulfamethin,磺胺二甲异嘧啶,Sulfaisodimidine

Target: Antibacterial, Antibiotic

Salbutamol hemisulfate

Cat.No: T6652

Synonym: Ventolin Sulfate,沙丁胺醇半硫酸盐,Albuterol,Salbutamol Sulfate,硫酸沙丁胺醇,Bronchospray,Albuterol Sulfate

Target: Adrenergic Receptor, Autophagy

Landiolol hydrochloride

Cat.No: T5028

Synonym: ONO-1101 hydrochloride,盐酸兰地洛尔

Target: Adrenergic Receptor

Dapoxetine hydrochloride

Cat.No: T6461

Synonym: LY-210448,LY-210448 hydrochloride,Dapoxetine HCl,盐酸达泊西汀,Priligy

Target: 5-HT Receptor, Serotonin Transporter

Cat.No: T0767

Synonym: 磺胺吡啶,Sulfidine,Sulfidin,2-Sulfapyridine

Target: Antibacterial, Antibiotic, Autophagy

Cat.No: T0750

Synonym: NU-445,磺胺二甲异唑,Sulfafurazole,磺胺异恶唑

Target: Endothelin Receptor, Antibacterial, Antibiotic, Autophagy

Cat.No: T1603

Synonym: CP 28720,K 4024,格列吡嗪

Target: Potassium Channel, PPAR, ABC

Cat.No: T0930

Synonym: Sulphadiazine,磺胺嘧啶

Target: Antibacterial, Antibiotic, Parasite, Autophagy

Cat.No: T9516

Synonym: WRC 0470,MRE-0470,比诺地松,2-(cyclohexylmethylidenehydrazino)adenos

Target: Adenosine Receptor

Cat.No: T11174

Synonym: 恶拉戈利,NBI-56418

Target: GNRH Receptor

Trichlormethiazide

Cat.No: T0114

Synonym: Naqua,Metahydrin,三氯噻嗪,Trichlormetazid

Target: ATPase, Carbonic Anhydrase

Cat.No: T15257

Synonym: MSP-2017,(-)-MSP-2017

Target: Calcium Channel

Cat.No: T0999

Synonym: Clevidipine butyrate,丁酸氯维地平,氯维地平,Cleviprex

Target: Calcium Channel, AChR

Cat.No: T1139

Synonym: Albuterol,沙丁胺醇,AH-3365

Target: Adrenergic Receptor

Trefentanil hydrochloride

Cat.No: T29005

Buthalital sodium

Cat.No: T30623

Synonym: baytinal

Cat.No: T5028L

Synonym: ONO1101,ONO 1101,ONO-1101

Carbuterol hydrochloride

Cat.No: T69394

Cat.No: T28383

Cat.No: T27543

Cat.No: T26919

Synonym: BU 09059,BU-09059

Cat.No: T28421

Synonym: Pirbuterolum,CP-24,314-14

Sulfathiazole sodium

Cat.No: T23402

Target: Others

Pirbuterol Acetate

Cat.No: T34079

Synonym: pirbuterol sulfate,EINECS 265-862-4,Maxair,Pirbuterol acetate (USAN)

RP-001 hydrochloride

Cat.No: T12780L

Target: Others

Cat.No: T34740

Synonym: Renoquid,CI636,CI-636,CI 636,磺胺西汀,Sulfacitinum

Cat.No: T12780

Target: Others

Sulfathiazole-d4

Cat.No: T13035

Target: Others

Colterol (free base)

Cat.No: T70089

Cat.No: T10241

Synonym: BW825C D7

Target: Others

Cat.No: T39820

Synonym: ZP7570

Albuterol stearate

Cat.No: T25030

Cat.No: T69472

Cat.No: T69148

AZD4573 HCl (2057509-72-3 free base)

Cat.No: T10436L

Synonym: AZD4573 hydrochloride,AZD4573,AZD4573 HCl,AZD-4573,AZD 4573

Propofol β-D-Glucuronide

Cat.No: T37378

Cat.No: T69144

Cat.No: TP1473

Synonym: c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm

Cat.No: TP1560

Velmupressin acetate

Cat.No: TP1205

Synonym: V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate

Apraglutide TFA (1295353-98-8 free base)

Cat.No: TP1171

Synonym: Apraglutide TFA,FE 203799e (TFA)

Albuterol adipate

Cat.No: T70551

Trimetaphan camsilate

Cat.No: T68811

Isoetharine hydrochloride

Cat.No: T60502

Apraglutide TFA

Cat.No: T76001

Cat. No.	Product Name	Target	Signaling Pathways
T0419	Testosterone propionate	Others; Androgen Receptor; Transferase	Endocrinology/Hormones; Metabolism; Others
	Testosterone Propionate is a short acting oil-based injectable formulation of testosterone. Testosterone inhibits gonadotropin secretion from the pituitary gland and ablates estrogen production in the ovaries, thereby decreasing endogenous estrogen levels.

天然产物

Testosterone propionate

Cat.No: T0419

Target: Others, Androgen Receptor, Transferase

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