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57

抑制剂 & 化合物

19

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Cat. No. Product Name Target Signaling Pathways
T1070 Cefmetazole sodium

头孢美唑钠,Sodium cefmetazole

Antibacterial; Antibiotic Microbiology/Virology
Cefmetazole sodium (Sodium cefmetazole) 是具有广谱抗菌活性的半合成头孢霉素抗生素。它通过与青霉素结合蛋白结合,阻止肽聚糖的交联,导致细胞壁完整性的丧失。它可研究妇科、腹腔内、尿道、呼吸道和皮肤和软组织感染。
T8620 piperacillin

Pipril,Pipracil,哌拉西林,Pipercillin

Antibacterial Microbiology/Virology
Piperacillin (Pipercillin) 是半合成青霉素,可以作用于革兰氏阳性和革兰氏阴性需氧和厌氧菌。与其他青霉素相比,它对产生 β-内酰胺酶的菌类表现出更强的活性。
T21358 Dalbavancin

BI 397,BI-397,VER 001,A-A 1,BI397,VER-001,Dalbavancin HCl,达巴万星

Antibacterial; Antibiotic Microbiology/Virology
Dalbavancin (BI-397) HCl 是一种半合成的脂糖肽抗生素,对革兰氏阳性细菌有杀菌活性。Dalbavancin 抑制金黄色葡萄球菌和炭疽芽孢杆菌的 MIC90分别为 0.06 μg/mL 和 0.25 μg/mL。
T60163 Lurtotecan

GI147211,OSI-211

Topoisomerase DNA Damage/DNA Repair
Lurtotecan (GI147211) 是一种半合成的喜树碱类似物。Lurtotecan 是一种具有抗癌作用的拓扑异构酶I 抑制剂。
T6268 Ceftiofur hydrochloride

头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur hydrochloride (U-67279A) 是头孢噻呋的盐酸盐形式,是一种β-内酰胺酶稳定的半合成广谱头孢菌素,具有抗菌活性。
T35346 Tiamulin fumarate

Thiamutilin fumarate

Antibacterial Microbiology/Virology
Tiamulin fumarate (Thiamutilin fumarate)是一种半合成的二萜类抗生素,具有抗菌活性,抑制蛋白质合成,可用于研究气囊炎。
T4270 Cefquinome sulfate

硫酸头孢喹肟,硫酸头孢喹诺

Antibacterial; Antibiotic Microbiology/Virology
Cefquinome sulfate 是一种半合成的头孢烯广谱抗生素,具有抗菌活性。
T7666 Valorphin TFA(144313-54-2(free base))

Valorphin TFA(144313-54-2(free bas))

Others Others
Valorphin TFA(144313-54-2(free base)) 是具有 opioid 类镇痛活性的二氢戊酸的半合成衍生物。
T1031 Cloxacillin sodium monohydrate

Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物

Antibacterial; Antibiotic Microbiology/Virology
Cloxacillin sodium monohydrate (Cloxacillin Sodium) 有抗菌作用,对Staphylococcus aureus25923 的最小抑菌浓度为256 mg/L。
T0234 Methicillin sodium salt

Methicillin sodium,Meticillin sodium,甲氧西林钠

Antibacterial; Antibiotic Microbiology/Virology
Methicillin sodium salt 是β-内酰胺抗生素,抑制参与肽聚糖合成的青霉素结合蛋白。
T67964 Terflavoxate

Microtubule Associated Cytoskeletal Signaling
Terflavoxate 是一种新型的、具有口服活性的半合成的他汀类微管抑制剂,常与卡培他滨一起联合使用。Terflavoxate 用于癌症的研究。
T13038 Sultamicillin

Antibacterial; Antibiotic Microbiology/Virology
Sultamicillin 是一种具有口服活性的氨苄西林/舒巴坦双前药。它是一种半合成 β-内酰胺酶抑制剂。
T6706 Ticarcillin sodium

Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Ticarcillin sodium (Aerugipen hydrate) 主要用于抗革兰氏阴性菌, 也能用于研究嗜麦芽感染。
T1523 Teniposide

替尼泊苷,NSC 122819,替尼泊甙,VM26

Topoisomerase DNA Damage/DNA Repair
Teniposide (VM26) 是鬼臼毒素的半合成衍生物,具有抗肿瘤活性,通过与拓扑异构酶 II 和 DNA 形成复合物来抑制 DNA 合成。
T0967 Teicoplanin

Antibiotic MDL-507,MDL-507,替考拉宁,Teichomycin

Antibacterial; Antibiotic Microbiology/Virology
Teicoplanin (MDL-507) 是一种半合成的糖肽抗生素, 可用于由革兰氏阳性菌引起的严重感染的相关研究。
T2691 Oritavancin diphosphate

奥利万星二磷酸盐,LY333328 diphosphate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Oritavancin diphosphate (LY333328 diphosphate) 是一种新型半合成的糖肽抗生素, 可研究革兰氏阳性菌感染。
T6386 Ampicillin sodium

氨苄西林钠,Domicillin,D-(-)-α-Aminobenzylpenicillin sodium salt,Penialmen,Citteral

Antibacterial; Antibiotic Microbiology/Virology
Ampicillin sodium (Domicillin) 是Ampicillin 的钠盐形式,是Ampicillin 的广谱半合成衍生物。它通过与青霉素结合蛋白结合来抑制细菌细胞壁的合成,从而抑制肽聚糖的合成,肽聚糖是细菌细胞壁的关键成分。
T1501 Rifabutin

LM-427,Ansamycin,利福布汀,利福布丁

HSP; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Rifabutin (LM-427) 是半合成的安莎霉素抗生素,抑制 DNA 依赖性 RNA 聚合酶,有抗分枝杆菌作用。
T1579 Mestranol

Devocin,Norquen,美雌醇,Menophase

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Mestranol (Devocin) 是一种雌激素受体激动剂,是一种非活性的前药,在转化为炔雌醇时具有生物活性。动物实验中,它可以与黄体酮联合使用,它可用于更年期激素或月经紊乱的研究。
T2577 Dienogest

地诺孕素,STS 557

Apoptosis; Estrogen/progestogen Receptor; Progesterone Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; Others
Dienogest (STS 557) 是一种孕酮受体激动剂,作用于子宫内膜异位,有口服的子宫内膜活性。
T1213 Piperacillin sodium

哌拉西林钠,Sodium piperacillin,CL227193,Piperacillin sodium salt

Antibacterial; Antibiotic Microbiology/Virology
Piperacillin sodium salt(CL227193) )是一种β-内酰胺类广谱抗生素。
T1122 Cephalothin sodium

头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin

Antibacterial; Antibiotic Microbiology/Virology
Cephalothin sodium (Cefalotin) 是一种头孢类抗生素, 具有广泛的抗菌活性,抑制革兰氏阳性和阴性菌。
T1005L Amoxicillin trihydrate

Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin trihydrate (Moxaline trihydrate) 是一种中谱β内酰胺抗菌素。
T24297 L 640876

L640,876,L-640876,L-640,876,L640876,L 640,876

L 640876 is a semisynthetic antibiotic.
T10496 Bencianol

ZY15051,苯西阿诺

Others Others
Bencianol is a semisynthetic flavonoid with anti-spasmogenic activities.
T32388 Ketocillin sodium

Ketocillin sodium is a semisynthetic penicillin.
T33352 Methylepoxyproscillaridin

Methylepoxyproscillaridin is a semisynthetic cardiac glycoside.
T25223 Cefpimizole sodium

AC 1370 sodium,AC 1370,AC1370,AC-1370

Cefpimizole sodium is a Semisynthetic cephalosporin with antibacterial activity.
T21105 Azlocillin

Azlocilline,Azlin

Azlocillin is a semisynthetic ampicillin-derived penicillin belonging to acylureido.
T20196 Cefamandole

头孢孟多,Compound 83405,L-Cefamandole,Mancef,Mandol

Cefamandole is a semisynthetic wide-spectrum cephalosporin with prolonged action. It is used also as the nafate.
T32476 L 705589

L705589,L-705589

L 705589 is a semisynthetic pneumocandin Bo derivative that is water-soluble.
T30555 BO 1341

BO1341,BO-1341

BO 1341 is a semisynthetic cephalosporin.
T37271 9(E)-Erythromycin A oxime

(9E)-Erythromycin A oxime is a metabolite of the semisynthetic antibiotic roxithromycin .
T32749 Liga 20

Liga-20,Liga20

Liga 20 is a semisynthetic GM1 ganglioside with N-dichloroacetylsphingosine that protecting neurons in culture against glutamate toxicity.
T33695 NK 611

NK611,NK-611

NK 611 is a new semisynthetic analogue of etoposide and has been found to be more potent against several cancer cell lines in vitro than etoposide.
T20164 Lymecycline

Limeciclina,Mucomycin,Tetralisal

Lymecycline is a semisynthetic antibiotic. It is related to TETRACYCLINE.
T39811 D-4-Hydroxyphenylglycine

4-Hydroxy-D-phenylglycine,D-(-)-4-Hydroxyphenylglycine,D-4-Hydroxyphenylglycine

D-4-Hydroxyphenylglycine (D-(-)-4-Hydroxyphenylglycine) is a crucial raw material in the synthesis of semisynthetic β-lactam antibiotics, including Amoxicillin and Cefadroxil .
T68475 AO-1535

AO-1535 is a semisynthetic monoglycosylceramide derived from O-glycosilated sphingosine. It has been shown to inhibit superoxide production by macrophages suggesting a potential clinical application of AO 1535 in the treatment of inflammatory dermatoses.
T1023 Cefoxitin sodium

Cenomycin,MK-306,头孢西丁钠,Betacef,Merxin

Antibacterial; Antibiotic Microbiology/Virology
Cefoxitin sodium (Betacef) 是一种头霉素类抗生素。Cefoxitin 干扰细胞壁合成。它对革兰氏阴性和革兰氏阳性菌有活性。
T34996 Ukrain

NSC631570,NSC 631570,NSC-631570

Ukrain, also known as NSC-631570, is claimed to be a semisynthetic compound of thiophosphoric acid (triaziridide) and the alkaloid chelidonine derived from the common weed, Chelidonium majus (greater celandine), which grows primarily in Europe and Asia.
T37881 Oritavancin(LY-333328)

Oritavancin is a novel semisynthetic glycopeptide antibiotics. On August 6, 2014, the FDA approved oritavancin for treatment of skin infections. Oritavancin possesses potent and rapid bactericidal activity in vitro against a broad spectrum of both resistant and susceptible Gram-positive bacteria, including Staphylococcus aureus, MRSA, enterococci, and streptococci.
T71521 NK-611 free acid

NK-611 free acid is a new semisynthetic analogue of etoposide, which presumably also acts through inhibition of topoisomerase II, and has been found to be more potent against several cancer cell lines in vitro than etoposide.
T19678 Cefaloridine

Cephaloridine,Sch 11527

Cefaloridine is a first-generation semisynthetic derivative of cephalosporin C. It is unique among cephalosporins in that it exists as a zwitterion. Cephaloridine was very effective to cure pneumococcal pneumonia. It has a high clinical and bacteriologica
T70250 Demeclocycline calcium

Demeclocycline calcium is a semisynthetic tetracycline antibiotic which was derived from a strain of Streptomyces aureofaciens. Demeclocycline binds to bacterial 30S ribosomal subunit and prevents binding of aminoacyl-tRNA to the mRNA-ribosome complex, thereby inhibiting protein synthesis. Demeclocycline also inhibits the effect of vasopressin on the renal tubules, thereby causing diuresis.
T74378 Temocillin

Temocillin为6-α-甲氧基青霉素衍生物,为半合成β-内酰胺类抗生素,对多数需氧革兰氏阴性菌展现特定抗菌活性。
T69093 Epirubicin

IMI-28,表柔比星,4-epi DX,4'-Epidoxorubicin,IMI 28,4-epidoxorubicin,epi DX,4-epiadriamycin

Epirubicin (4'-Epidoxorubicin) 是阿霉素的半合成的 L-阿拉伯糖衍生物,能够抑制 Topoisomerase,起到抗肿瘤的作用。Epirubicin 抑制 DNA 和 RNA 合成。Epirubicin 是一种 Forkhead box 蛋白 p3 (Foxp3) 抑制剂,可抑制调节性 T 细胞活性。
T75253 Dalbavancin hydrochloride

Dalbavancin hydrochloride (MDL-63397 hydrochloride)为半合成脂糖肽类抗生素,有效对抗革兰氏阳性菌。其对金黄色葡萄球菌与炭疽芽孢杆菌的MIC90分别为0.06 μg/mL与0.25 μg/mL。
T83858 Tauro-Obeticholic Acid sodium

Tauro-6-Ethylchenodeoxycholic Acid,Tauro-6-Ethyl-CDCA,Obeticholic Acid Taurine Conjugate,Tauro-OCA,T-ECDCA

陶氏奥贝胆酸是奥贝胆酸的活性代谢物,属于法尼索德X受体(FXR)激动剂并且是熊脱氧胆酸的半合成衍生物。陶氏奥贝胆酸通过在肝脏中与牛磺酸结合形成,但可以通过肠道微生物被再次转换回奥贝胆酸。
T1005 Amoxicillin

Amoxycillin,阿莫西林

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin (Amoxycillin) 是一种具有广谱抗菌活性和良好口服吸收的抗生素。
T36671 C2 Phytoceramide (t18:0/2:0)

C2 Phytoceramide is a bioactive semisynthetic sphingolipid that inhibits formyl peptide-induced oxidant release (IC50 = 0.38 μM) in suspended polymorphonuclear cells. It increases COX-2 protein levels 15-fold through ERK signaling. It induces death of keratinocytes (20% viability) with an ED50 value of 30 μM, the same concentration at which 35% of cells in a TUNEL assay are apoptotic. C2 Phytoceramide also has antiproliferative effects in CHO cells, with greater than 80% cytotoxicity achieved at...

化合物

Cefmetazole sodium
Cat.No: T1070
Synonym: 头孢美唑钠,Sodium cefmetazole
Target: Antibacterial, Antibiotic
piperacillin
Cat.No: T8620
Synonym: Pipril,Pipracil,哌拉西林,Pipercillin
Target: Antibacterial
Dalbavancin
Cat.No: T21358
Synonym: BI 397,BI-397,VER 001,A-A 1,BI397,VER-001,Dalbavancin HCl,达巴万星
Target: Antibacterial, Antibiotic
Lurtotecan
Cat.No: T60163
Synonym: GI147211,OSI-211
Target: Topoisomerase
Ceftiofur hydrochloride
Cat.No: T6268
Synonym: 头孢噻呋盐酸盐,Ceftiofur HCl,U-67279A,Excenel hydrochloride
Target: Antibacterial, Antibiotic
Tiamulin fumarate
Cat.No: T35346
Synonym: Thiamutilin fumarate
Target: Antibacterial
Cefquinome sulfate
Cat.No: T4270
Synonym: 硫酸头孢喹肟,硫酸头孢喹诺
Target: Antibacterial, Antibiotic
Valorphin TFA(144313-54-2(free base))
Cat.No: T7666
Synonym: Valorphin TFA(144313-54-2(free bas))
Target: Others
Cloxacillin sodium monohydrate
Cat.No: T1031
Synonym: Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物
Target: Antibacterial, Antibiotic
Methicillin sodium salt
Cat.No: T0234
Synonym: Methicillin sodium,Meticillin sodium,甲氧西林钠
Target: Antibacterial, Antibiotic
Terflavoxate
Cat.No: T67964
Synonym:
Target: Microtubule Associated
Sultamicillin
Cat.No: T13038
Synonym:
Target: Antibacterial, Antibiotic
Ticarcillin sodium
Cat.No: T6706
Synonym: Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen
Target: Others, Antibacterial, Antibiotic
Teniposide
Cat.No: T1523
Synonym: 替尼泊苷,NSC 122819,替尼泊甙,VM26
Target: Topoisomerase
Teicoplanin
Cat.No: T0967
Synonym: Antibiotic MDL-507,MDL-507,替考拉宁,Teichomycin
Target: Antibacterial, Antibiotic
Oritavancin diphosphate
Cat.No: T2691
Synonym: 奥利万星二磷酸盐,LY333328 diphosphate
Target: Others, Antibacterial, Antibiotic
Ampicillin sodium
Cat.No: T6386
Synonym: 氨苄西林钠,Domicillin,D-(-)-α-Aminobenzylpenicillin sodium salt,Penialmen,Citteral
Target: Antibacterial, Antibiotic
Rifabutin
Cat.No: T1501
Synonym: LM-427,Ansamycin,利福布汀,利福布丁
Target: HSP, DNA/RNA Synthesis, Antibacterial, Antibiotic
Mestranol
Cat.No: T1579
Synonym: Devocin,Norquen,美雌醇,Menophase
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Dienogest
Cat.No: T2577
Synonym: 地诺孕素,STS 557
Target: Apoptosis, Estrogen/progestogen Receptor, Progesterone Receptor, Autophagy
Piperacillin sodium
Cat.No: T1213
Synonym: 哌拉西林钠,Sodium piperacillin,CL227193,Piperacillin sodium salt
Target: Antibacterial, Antibiotic
Cephalothin sodium
Cat.No: T1122
Synonym: 头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin
Target: Antibacterial, Antibiotic
Amoxicillin trihydrate
Cat.No: T1005L
Synonym: Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate
Target: Antibacterial, Antibiotic
L 640876
Cat.No: T24297
Synonym: L640,876,L-640876,L-640,876,L640876,L 640,876
Target:
Bencianol
Cat.No: T10496
Synonym: ZY15051,苯西阿诺
Target: Others
Ketocillin sodium
Cat.No: T32388
Synonym:
Target:
Methylepoxyproscillaridin
Cat.No: T33352
Synonym:
Target:
Cefpimizole sodium
Cat.No: T25223
Synonym: AC 1370 sodium,AC 1370,AC1370,AC-1370
Target:
Azlocillin
Cat.No: T21105
Synonym: Azlocilline,Azlin
Target:
Cefamandole
Cat.No: T20196
Synonym: 头孢孟多,Compound 83405,L-Cefamandole,Mancef,Mandol
Target:
L 705589
Cat.No: T32476
Synonym: L705589,L-705589
Target:
BO 1341
Cat.No: T30555
Synonym: BO1341,BO-1341
Target:
9(E)-Erythromycin A oxime
Cat.No: T37271
Synonym:
Target:
Liga 20
Cat.No: T32749
Synonym: Liga-20,Liga20
Target:
NK 611
Cat.No: T33695
Synonym: NK611,NK-611
Target:
Lymecycline
Cat.No: T20164
Synonym: Limeciclina,Mucomycin,Tetralisal
Target:
D-4-Hydroxyphenylglycine
Cat.No: T39811
Synonym: 4-Hydroxy-D-phenylglycine,D-(-)-4-Hydroxyphenylglycine,D-4-Hydroxyphenylglycine
Target:
AO-1535
Cat.No: T68475
Synonym:
Target:
Cefoxitin sodium
Cat.No: T1023
Synonym: Cenomycin,MK-306,头孢西丁钠,Betacef,Merxin
Target: Antibacterial, Antibiotic
Ukrain
Cat.No: T34996
Synonym: NSC631570,NSC 631570,NSC-631570
Target:
Oritavancin(LY-333328)
Cat.No: T37881
Synonym:
Target:
NK-611 free acid
Cat.No: T71521
Synonym:
Target:
Cefaloridine
Cat.No: T19678
Synonym: Cephaloridine,Sch 11527
Target:
Demeclocycline calcium
Cat.No: T70250
Synonym:
Target:
Temocillin
Cat.No: T74378
Synonym:
Target:
Epirubicin
Cat.No: T69093
Synonym: IMI-28,表柔比星,4-epi DX,4'-Epidoxorubicin,IMI 28,4-epidoxorubicin,epi DX,4-epiadriamycin
Target:
Dalbavancin hydrochloride
Cat.No: T75253
Synonym:
Target:
Tauro-Obeticholic Acid sodium
Cat.No: T83858
Synonym: Tauro-6-Ethylchenodeoxycholic Acid,Tauro-6-Ethyl-CDCA,Obeticholic Acid Taurine Conjugate,Tauro-OCA,T-ECDCA
Target:
Amoxicillin
Cat.No: T1005
Synonym: Amoxycillin,阿莫西林
Target: Antibacterial, Antibiotic
C2 Phytoceramide (t18:0/2:0)
Cat.No: T36671
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1424 Ethynyl estradiol

乙炔基雌二醇,17α-Ethynylestradiol,Ethinyl Estradiol,炔雌醇

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Ethynyl estradio 是一种高效的生物活性雌激素。
T8065 Tiamulin

Thiamutilin,泰妙菌素

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Tiamulin (Thiamutilin) 是一类二萜,广泛用于控制猪的传染疾病,包括猪痢疾和地方性肺炎等。
T8063 Cephapirin Benzathine

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cephapirin Benzathine 是头孢哌啶的苄硫醚盐形式,是一种广谱抗生素。
T5647 6-Methylcoumarin

Toncarine,6-甲基香豆素

Others Others
6-Methylcoumarin (Toncarine) 是一种合成香料,广泛用于化妆品中。
T0190 Vinorelbine

长春瑞宾,KW-2307 base

Microtubule Associated Cytoskeletal Signaling
Vinorelbine (KW-2307 base) 是一种半合成的长春花生物碱。它与微管蛋白结合并阻止有丝分裂纺锤体的形成,导致中期肿瘤细胞生长停滞。
T8062 Cefazedone

Refosporen,头孢西酮

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazedone (Refosporen) 是一种具有抗革兰氏阳性和革兰氏阴性菌活性的时间依赖性头孢菌素抗生素。
T0814 Ampicillin Trihydrate

NCI-C56086,氨苄青霉素三水合物

Antibacterial; Antibiotic Microbiology/Virology
Ampicillin Trihydrate (NCI-C56086) 是一种 β-内酰胺类广谱抗生素,可对抗多种革兰氏阳性和革兰氏阴性细菌。
T8302 Ceftiofur

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur 是一种半合成抗生素,对家畜的各种革兰氏阳性和革兰氏阴性菌、好氧菌和厌氧菌均有抗菌活性。
T6447 Clindamycin

Clinimycin,Sobelin,Chlolincocin,克林霉素

Antibacterial; Antibiotic Microbiology/Virology
Clindamycin (Sobelin) 从细菌核糖体中解离肽基-tRNA,破坏细菌蛋白质合成。 它是一种半合成广谱抗生素,由母体化合物林可霉素化学修饰而成。
T0518 Methacycline hydrochloride

Rondomycin,盐酸甲烯土霉素,盐酸美他环素,Methacycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Methacycline hydrochloride (Rondomycin) 是四环素抗生素,可抑制细菌蛋白质的合成。它是上皮-间质转化 (EMT) 抑制剂。它在体外可阻断 EMT,体内抑制纤维发生,不会直接影响 TGF-β1 Smad 信号传导。它是抗菌剂,有潜力研究肺纤维化。
T6194 Fidaxomicin

非达米星,Tiacumicin B,OPT-80,Clostomicin B1,PAR-101

Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Fidaxomicin (Tiacumicin B) 是一种大环RNA 聚合酶抑制剂,具有窄谱活性。它选择性地根除致病性艰难梭菌,对构成正常健康肠道菌群的多种细菌影响很小。
T5853 Rubitecan

RFS 2000,鲁比特康,9-Nitrocamptothecin

Topoisomerase DNA Damage/DNA Repair
Rubitecan (9-Nitrocamptothecin) 是一种与喜树碱相关的半合成药物,具有有效的抗肿瘤和抗病毒特性。它是一种 DNA 拓扑异构酶 I 抑制剂,以浓度依赖性方式抑制 DNA 拓扑异构酶 I 并在无细胞试验中增加超螺旋 DNA 的比例。
T3524 Halofuginone hydrobromide

卤夫酮溴氢酸盐,Tempostatin,RU-19110 (hydrobromide),Stenorol,常山酮溴酸盐

Others; Calcium Channel; DNA/RNA Synthesis; Sodium Channel; Parasite; TGF-beta/Smad Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Others; Stem Cells
Halofuginone hydrobromid 是Febrifugine 的衍生物,是竞争性脯氨酰-tRNA 合成酶抑制剂。它是 I 型胶原合成的特异性抑制剂,并通过抑制TGF-β活性可减轻骨关节炎。它具有抗疟疾、抗炎、抗癌、抗纤维化作用。
T0034 Cortisone acetate

醋酸可的松,Cortisone 21-acetate,NSC 49420

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Cortisone acetate (NSC-49420) 是 Cortisol(一种糖皮质激素)的氧化代谢产物。它在高浓度下能够部分干预 Glucocorticoid 与Glucocorticoid-receptor 的结合。它具有免疫抑制和消炎的作用。
T0486L Irinotecan Hydrochloride

盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan Hydrochloride (CPT-11 hydrochloride) 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。
T1607 Hydrastinine hydrochloride

北美黄连碱分碱盐酸盐,北美黄连碱分碱

Others Others
Hydrastinine hydrochloride 是金印草中的一种主要生物碱成分,可用作止血剂。
T33492 Methyl pyropheophorbide-a

MPPa (Methyl pyropheophorbide-a),NSC267052,Pyropheophorbidea,MPPa,NSC-267052,NSC 267052

Pyropheophorbide-a methyl ester (MPPa) is a PDT photosensitizer, and is also a semisynthetic natural product derived from chlorophyll a. The absorption peak of MPPa in organic solvent and in cells was at 667 and 674 nm, respectively. 3-(4,5-Dimethylthiazo
T82277 GM1a Ganglioside oligosaccharide

GM1a Ganglioside oligosaccharide为ganglioside GM1的半合成形式,后者作为霍乱毒素的天然受体,在生长调节及激素诱导反应的耦合中具有关键功能。
T1521 (±)-10-Hydroxycamptothecin

Hydroxy Camptothecine,10-羟基喜树碱,10-Hydroxycamptothecin

Topoisomerase DNA Damage/DNA Repair
(±)-10-Hydroxycamptothecin (Hydroxy Camptothecine) 是一种从喜树茎木中分离出来的生物碱,抑制拓扑异构酶 I 活性,具有广谱抗肿瘤活性。

天然产物

Ethynyl estradiol
Cat.No: T1424
Synonym: 乙炔基雌二醇,17α-Ethynylestradiol,Ethinyl Estradiol,炔雌醇
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Tiamulin
Cat.No: T8065
Synonym: Thiamutilin,泰妙菌素
Target: Others, Antibacterial, Antibiotic
Cephapirin Benzathine
Cat.No: T8063
Synonym:
Target: Others, Antibacterial, Antibiotic
6-Methylcoumarin
Cat.No: T5647
Synonym: Toncarine,6-甲基香豆素
Target: Others
Vinorelbine
Cat.No: T0190
Synonym: 长春瑞宾,KW-2307 base
Target: Microtubule Associated
Cefazedone
Cat.No: T8062
Synonym: Refosporen,头孢西酮
Target: Others, Antibacterial, Antibiotic
Ampicillin Trihydrate
Cat.No: T0814
Synonym: NCI-C56086,氨苄青霉素三水合物
Target: Antibacterial, Antibiotic
Ceftiofur
Cat.No: T8302
Synonym:
Target: Antibacterial, Antibiotic
Clindamycin
Cat.No: T6447
Synonym: Clinimycin,Sobelin,Chlolincocin,克林霉素
Target: Antibacterial, Antibiotic
Methacycline hydrochloride
Cat.No: T0518
Synonym: Rondomycin,盐酸甲烯土霉素,盐酸美他环素,Methacycline HCl
Target: ribosome, Antibacterial, Antibiotic
Fidaxomicin
Cat.No: T6194
Synonym: 非达米星,Tiacumicin B,OPT-80,Clostomicin B1,PAR-101
Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic
Rubitecan
Cat.No: T5853
Synonym: RFS 2000,鲁比特康,9-Nitrocamptothecin
Target: Topoisomerase
Halofuginone hydrobromide
Cat.No: T3524
Synonym: 卤夫酮溴氢酸盐,Tempostatin,RU-19110 (hydrobromide),Stenorol,常山酮溴酸盐
Target: Others, Calcium Channel, DNA/RNA Synthesis, Sodium Channel, Parasite, TGF-beta/Smad
Cortisone acetate
Cat.No: T0034
Synonym: 醋酸可的松,Cortisone 21-acetate,NSC 49420
Target: Glucocorticoid Receptor, Endogenous Metabolite
Irinotecan Hydrochloride
Cat.No: T0486L
Synonym: 盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride
Target: Topoisomerase, Autophagy
Hydrastinine hydrochloride
Cat.No: T1607
Synonym: 北美黄连碱分碱盐酸盐,北美黄连碱分碱
Target: Others
Methyl pyropheophorbide-a
Cat.No: T33492
Synonym: MPPa (Methyl pyropheophorbide-a),NSC267052,Pyropheophorbidea,MPPa,NSC-267052,NSC 267052
Target:
GM1a Ganglioside oligosaccharide
Cat.No: T82277
Synonym:
Target:
(±)-10-Hydroxycamptothecin
Cat.No: T1521
Synonym: Hydroxy Camptothecine,10-羟基喜树碱,10-Hydroxycamptothecin
Target: Topoisomerase
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