1
40
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T34560 |
Scammonin II
|
||
Scammonin II is a resin glycoside of radix scammoniae from Convolvulus scammonia. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5S1895 |
Norisoboldine
Laurelliptine,去甲异波尔定,(+)-Laurelliptine |
MAPK; Adenosine Receptor | GPCR/G Protein; MAPK; Neuroscience |
Norisoboldine ((+)-Laurelliptine) 是一种可口服的芳基烃受体激动剂,是乌药中主要的异喹啉类生物碱,可用于类风湿性关节炎和溃疡性结肠炎的研究。 | |||
T4587 |
Mirificin
BCP10902,Puerarin Apioside,葛根素芹菜糖苷,芹糖葛根素苷 |
Tyrosinase | Proteases/Proteasome |
Mirificin (BCP10902) 是一种葛根中的异黄酮。它能够抑制酪氨酸酶(Tyrosinase),IC50=12.66 μM。 | |||
T3848 |
7,2′-Dihydroxy-3′,4′-dimethoxyisoflavan 7-O-β-D-glucoside
Isomucronulatol 7-O-glucoside,7,2'-dihydroxy-3',4'-dimethoxyisoflavane-7-O-glucoside,黄芪异黄烷苷 |
Others | Others |
7,2′-Dihydroxy-3′,4′-dimethoxyisoflavan 7-O-β-D-glucoside (Isomucronulatol 7-O-glucoside) 是一种具有生物活性的异黄酮,分离自黄芪中。 | |||
TCS2170 |
2,5-Dihydroxyacetophenone
Quinacetophenone,2-Acetylhydroquinone,2-5-dihydroxyacetophenone,2 ',5'-二羟基苯乙酮,Acetylhydroquinone,2,5-二羟基苯乙酮,DHAP |
ERK; NF-κB; Tyrosinase | MAPK; NF-κB; Proteases/Proteasome |
2,5-Dihydroxyacetophenone (Quinacetophenone) 是从熟地黄中分离出的一种天然产物,通过阻断 ERK1/2和 NF-κB 信号通路,抑制活化巨噬细胞中炎症介质的产生。 | |||
T3S1896 |
Lindenenol
Linderene,Lindeneol,乌药醇 |
Others; Antibacterial | Microbiology/Virology; Others |
Lindenenol (Linderene) 是从Radix linderae 中分离得到的,有抗氧化和抗菌作用。 | |||
TN7243 |
Fallaxsaponin A
|
||
Fallaxsaponin A 是从远志中总皂苷的碱性水解产物中分离出来的。 | |||
T4961 |
9''-Methyl salvianolate B
9'-Methyl lithospermate B,9’-丹酚酸B单甲酯,9''-丹酚酸B单甲酯 |
Others | Others |
9'-Methyl lithospermate B 是一种酚类化合物,提取自 RadixSalvia miltiorrhizae。 | |||
T3773 |
Oxypaeoniflorin
氧化芍药苷,Oxypaeoniflora |
Others | Others |
Oxypaeoniflorin (Oxypaeoniflora) 从 Paeoniae 中分离得到的单萜糖苷化合物,是一种抗氧化剂,是具有神经保护和抗炎作用。 | |||
TN1927 |
Methyl Kakuol
1-(6-methoxy-1,3-benzodioxol-5-yl)propan-1-one |
TRP/TRPV Channel | Membrane transporter/Ion channel |
Methyl Kakuol 是 TRPA1 的激动剂,EC50 为 0.27 µM,可用于作为 MBST 成分 Asiasari Radix 的活性成分的研究。 | |||
TN3273 | 8-Deacetylyunaconitine | Others | Others |
8-Deacetylyunaconitine 是一种源自乌头的二萜生物碱。 | |||
TN7027 |
Benzoylalbiflorin
Paeonivayin,苯甲酰芍药内酯苷 |
Others | Others |
Benzoylalbiflorin (Paeonivayin) 是一种分离自 Radix Paeoniae Alba 的单萜。其中 Radix Paeoniae Alba 是传统中药,已用于研究类风湿关节炎,能够缓解炎症,闭经,鼻出血,腹痛和其他症状。 | |||
T2986 |
Jatrorrhizine hydrochloride
|
Others | Others |
Jatrorrhizine hydrochloride 是从小檗、根中提取的。 | |||
T3018 |
Protocatechualdehyde
Protocatechuic aldehyde,3,4-Dihydroxybenzaldehyde,Rancinamycin IV,Catechaldehyde,原儿茶醛 |
Reactive Oxygen Species; Antibacterial | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB |
Protocatechualdehyde (3,4-Dihydroxybenzaldehyde), a natural polyphenol compound derived from radix Salviae Miltiorrhizae roots, exhibits diverse biological activities and finds extensive medicinal applications as an antioxidant, anti-aging, antibacterial, and anti-inflammatory agent. | |||
TN7111 | Hydroxyisogermafurenolide | Others | Others |
Hydroxyisogermafurenolide 是来自姜黄的天然产物。 | |||
TN1782 |
(+)-Isolariciresinol
(+)-Cyclolariciresinol,Isolariciresinol |
Immunology/Inflammation related | Immunology/Inflammation |
(+)-Isolariciresinol ((+)-Cyclolariciresinol) 从板蓝根中提取,具有抗氧化和抗炎活性,可用于风湿病研究。 | |||
T2S0473 |
Rehmannioside C
|
Others | Others |
Rehmannioside C is an iridoid glucoside. Rehmannioside C has been isolated from Radix Rehmanniae Praeparata[1]. | |||
T3S0012 |
coniferyl ferulate
|
P-gp; GST | Membrane transporter/Ion channel; Neuroscience; oxidation-reduction |
Coniferyl ferulate 是从川芎中提取的一种天然产物,是强效的谷胱甘肽 S-转移酶抑制剂,强抑制人胎盘型谷胱甘肽 S-转移酶,IC50为 0.3 μM。它还可逆转多药耐药性并下调 P-糖蛋白。 | |||
T3387 |
Phytolaccagenin
|
Others; Antibacterial | Microbiology/Virology; Others |
Phytolaccagenin 是一种三萜类皂苷,是商陆的活性成分,有抗真菌活性,抗炎活性和较低的毒性。在东亚国家广泛用于治疗炎症相关疾病。 | |||
T6S1880 |
Benzoylaconine
苯甲酰乌头原碱,Pikraconitin,Isaconitine,Benzoylaconitine |
Others | Others |
Benzoylaconine (Isaconitine) 是一种中药附子生物碱。 | |||
T0036 |
18β-Glycyrrhetinic acid
Enoxolone,甘草次酸,18β-甘草次酸,Glycyrrhetin |
Dehydrogenase; Endogenous Metabolite | Metabolism |
18β-Glycyrrhetinic acid (Enoxolone) 是甘草的主要生物活性成分,具有抗炎,抗增殖和抗溃疡的特性。 | |||
T5S2195 |
Sibiricose A5
西伯利亚远志糖A5 |
Dehydrogenase | Metabolism |
Sibiricose A5 是一种寡糖酯,分离自Polygalae Radix,具有抗氧化作用。 | |||
T10383 |
Asatone
|
NF-κB | NF-κB |
Asatone 是一种从细辛中分离到的活性成分,通过活化 NF-κB 及下调 p-MAPK (ERK,JNK 和 p38) 通路起作用,具有抗炎作用。 | |||
T2983 |
3,4,5-Trimethoxycinnamic acid
3-(3,4,5-Trimethoxyphenyl)acrylic Acid,O-Methylsinapic acid,3,4,5-三甲氧基肉桂酸 |
GABA Receptor; Endogenous Metabolite | Membrane transporter/Ion channel; Metabolism; Neuroscience |
3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) 是从远志中分离得到的苯丙素类天然产物,可延长动物的睡眠时间,增强 GAD65 和 GABAA 受体 γ 亚基,具有抗应激作用。 | |||
T3019 |
Physcion
大黄素甲醚,Physcione,Parietin,Rheochrysidin |
Dehydrogenase; Antibacterial | Metabolism; Microbiology/Virology |
Physcion (Physcione) 是一种从中药大黄中分离的蒽醌,作为 6-磷酸葡萄糖酸脱氢酶的抑制剂,IC50和 Kd 值分别为 38.5 μM 和 26.0 μM。它具有通便、保肝、抗炎、抗菌、抗增殖、抗肿瘤作用。 | |||
T3860 |
Isoliquiritin apioside
|
MMP; p38 MAPK; NF-κB | MAPK; NF-κB; Proteases/Proteasome |
Isoliquiritin apioside 可抑制癌细胞和内皮细胞的侵袭和血管生成,显著降低 PMA 诱导的MMP9活性增加,并抑制 PMA 诱导的MAPK 和NF-κB 活化。 | |||
T5S2204 |
Sibiricose A6
西伯利亚远志糖A6 |
Antioxidant | oxidation-reduction |
Sibiricose A6 是一种寡糖酯,分离自Polygalae Radix,具有抗氧化作用。 | |||
T3903 |
Angoroside C
安格洛甙C,安格洛苷C |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Angoroside C 是一种苯丙苷,从 Radix Scrophulariae 中提取到,有益于心室重构。 | |||
TN1683 |
Gentisin
龙胆根素,龍膽根素 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Gentisin 是一种提取于 Gentianae radix (Gentianaceae) 的天然化合物,具有诱变活性。 | |||
T6S1653 |
Albiflorin
Alibiflorin,芍药内酯苷 |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Albiflorin (Alibiflorin) 是一种牡丹根中的主要成分,是一种单萜糖苷。它具有神经保护、抗炎、抗氧化和缓解疼痛作用。 | |||
T7090 |
Jionoside A1
焦地黄苯乙醇甙A1,焦地黄苯乙醇苷A1 |
Others | Others |
Jionoside A1 分离自Radix Rehmanniae Praeparata 中,具有剂量依赖性免疫增强作用,并对 H2O2处理的 SH-SY5Y 细胞具有中等保护活性。 | |||
T3891 |
Oroxylin A-7-O-glucuronide
Oroxylin A Glucoronide,千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Oroxyloside,Oroxylin A 7-O-beta-D-glucuronide |
Others | Others |
Oroxylin A-7-O-glucuronide (Oroxylin A Glucoronide) 是一种类黄酮葡糖苷酸,提取自 Scutellaria baicalensis 干燥的根中,具有脯氨酰寡肽酶(POP)抑制作用。 | |||
T5702 |
Tenuifoliside B
|
Dehydrogenase | Metabolism |
Tenuifoliside B 是一种分离自Polygalae Radix 中的成分,能够抑制氰化钾引起的缺氧和东莨菪碱引起的记忆障碍。它有成为 AD 先导化合物的潜力。它具有潜在的认知改善和脑保护作用。 | |||
T38524 |
Paeoniflorin sulfite
|
||
During the sulfur-fumigation process of Paeoniae Radix Alba, Paeoniflorin, which serves as a principal constituent, can be converted into Paeoniflorin sulfite. | |||
TN1447 |
L-Borneol 7-O-[β-D-apiofuranosyl-(1→6)]-β-D-glucopyranoside
FT-0775891,Borneol 7-O-[beta-D-apiofuranosyl-(1->6)]-beta-D-glucopyranoside,龙脑 7-O-[Β-D-呋喃芹菜糖基-(1→6)]-Β-D-吡喃葡萄糖苷 |
Others | Others |
Borneol 7-O-[beta-D-apiofuranosyl-(1->6)]-beta-D-glucopyranoside is a natural product from Radix ophiopogonis. | |||
T83365 |
3′-O-Angeloylhamaudol
|
||
3′-O-Angeloylhamaudol为香豆素类化合物,源自Radix Saposhnikoviae的提取分离。 | |||
T81020 |
Tenaxin I
|
||
Tenaxin I,一种从黄芩提取物中鉴定出的成分,具有神经氨酸酶抑制活性。 | |||
T83593 |
(+)-trans-3'-Acetyl-4'-isobutyrylkhellactone
|
||
(+)-trans-3'-Acetyl-4'-isobutyrylkhellactone,这种角型吡喃香豆素类化合物是从Peucedani Radix中分离出的一种天然产物。 | |||
TN5094 |
Tangshenoside I
|
Glucokinase | Metabolism |
Tangshenoside I might be a potential bioactive marker related to the hematopoietic and immunologic functions of Codonopsis Radix, which could be recommended as the index compound. It has α-glucosidase inhibition activity. | |||
T75433 | Norisoboldine hydrochloride | ||
Norisoboldine hydrochloride是一种口服活性天然芳基烃受体(AhR)激动剂,作为林参中的主要异喹啉类生物碱,适用于类风湿性关节炎和溃疡性结肠炎的研究。 | |||
TN1440 |
Beta-Hydroxyisovalerylshikonin
|
EGFR; Tyrosine Kinases; Prostaglandin Receptor; Src; AMPK; Fatty Acid Synthase | Angiogenesis; Chromatin/Epigenetic; GPCR/G Protein; Immunology/Inflammation; JAK/STAT signaling; Metabolism; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors |
Beta-hydroxyisovalerylshikonin 是分离自Lithospermium radix 的天然产物,具有抑制PTK 的作用, 对 EGFR 和 v-Src 受体作用的IC50分别为 0.7 μM 和 1 μM。它对多种肿瘤细胞系均有抑制作用,可以高效诱导 NCI-H522 和 DMS114 细胞的死亡。 |