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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7942 |
Tranylcypromine hemisulfate
Tranylcypromine Sulfate,Tranylcypromine (hemisulfate),反苯环丙胺半硫酸盐 |
Histone Demethylase; MAO; Monoamine Oxidase | Chromatin/Epigenetic; Metabolism; Neuroscience |
Tranylcypromine hemisulfate (Tranylcypromine Sulfate) 是单胺氧化酶(MAO) 和赖氨酸特异性去甲基化酶 1 (LSD1) 的抑制剂,可用于研究抑郁症和子宫内膜异位症。 | |||
T9232 |
Mitochondrial fusion promoter M1
|
Mitochondrial Metabolism | Metabolism |
Mitochondrial fusion promoter M1 是一种线粒体动态调节剂,能够保持线粒体功能并促进细胞呼吸,减轻心肌缺血/再灌注大鼠的心脏损伤和大脑损伤。 | |||
T9228 |
Propionylpromazine hydrochloride
盐酸丙酰丙嗪,Propiopromazine hydrochloride |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Propionylpromazine hydrochloride (Propiopromazine hydrochloride) 是多巴胺受体 D2 (DRD2) 拮抗剂,可用于研究帕金森氏病。 | |||
TQ0022 |
Capromorelin Tartrate
卡普瑞林酒石酸盐,CP 424391-18 |
GHSR | GPCR/G Protein |
Capromorelin Tartrate (CP 424391-18) 是口服有活性的 growth hormone secretagogue receptor 有效激动剂,能够作用于 hGHS-R1a(Ki:7 nM)。 | |||
T7778L |
Glypromate acetate(32302-76-4 free base)
|
NMDAR | Neuroscience |
Glypromate acetate(32302-76-4 free base) 是一种神经保护剂,是一种弱 NMDA 受体激动剂。 | |||
T1536 |
Promestriene
3-propyl ethyl,舒经劳,17B-methyl estradiol,Promestriano |
Estrogen/progestogen Receptor | Endocrinology/Hormones |
Promestriene (3-propyl ethyl) 是局部有效的雌激素,是合成的雌二醇二乙醚。它对阴道萎缩有作用,但吸收量小。 | |||
T0445L |
Promethazine hydrochloride
盐酸异丙嗪,Promethazine HCl,Phenergan |
Adrenergic Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Promethazine hydrochloride (Promethazine HCl) 是抗组胺药物,是 H1 受体的强拮抗剂和 mACh 受体的中度拮抗剂,对 5-HT2A、5-HT2C、D2 和 α1-肾上腺素能受体具有中等亲和力。 | |||
T0355 |
Valpromide
Depamide,Valpramide,丙戊酰胺,Dipropylacetamide,2-propylpentanamide |
Epoxide Hydrolase; HSV | Metabolism; Microbiology/Virology |
Valpromide (Dipropylacetamide) 是丙戊酸的羧酰胺衍生物,用于治疗癫痫和一些情感障碍。 | |||
T0302 |
Triflupromazine hydrochloride
Neoprin,盐酸三氟丙嗪,Fluopromazine hydrochloride,Fluorofen,Flumazin |
Dopamine Receptor; 5-HT Receptor; AChR; Autophagy | Autophagy; GPCR/G Protein; Neuroscience |
Triflupromazine hydrochloride (Fluopromazine hydrochloride) 是一种抗精神病药物,是多巴胺 D1/D2 受体拮抗剂。 | |||
T68921 |
Impromidine hydrochloride
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Impromidine hydrochloride 是一种非常有效和特异性的组胺H2受体激动剂,可用于进行心血管研究。 | |||
T50054 |
Opromazine hydrochloride
|
Others | Others |
Opromazine hydrochloride 属于吩噻嗪类抗精神病药物,通过阻断大脑中的多巴胺受体而降低多巴胺能通路的活性,主要用于治疗精神分裂症和精神病等精神疾病。 | |||
T0445 |
Promethazine
Proazamine,异丙嗪,Diphergan |
CaMK; Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Promethazine (Proazamine) 是抗青光眼前列腺素(PG)的类似物。 | |||
T1522 |
Iopromide
碘普罗胺,Iopromidum,Ultravist |
Others | Others |
Iopromide (Iopromidum) 是用于血管内的低渗透、非离子造影剂。 | |||
T19733 |
Prometryn
Caparol,Gesagard,Mercazin,扑草净 |
Others | Others |
Prometryn (Mercazin) 是一种除草剂,可提高棉花产量。 | |||
TP1153L |
Fibronectin Adhesion-promoting Peptide acetate
Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate |
Others | Others |
Fibronectin Adhesion-promoting Peptide acetate (Heparin Binding Peptide acetate)(125720-21-0 free base) 是在纤连蛋白的羧基末端肝素结合结构域中发现的肝素结合氨基酸序列之一。 | |||
T0766 |
Promazine hydrochloride
Romtiazin hydrochloride,Sinophenin hydrochloride,盐酸丙嗪 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR | GPCR/G Protein; Neuroscience |
Promazine hydrochloride (Romtiazin hydrochloride) 是一种抗精神病药,也是一种多巴胺受体 (D2) 拮抗剂,能够抑制多巴胺能神经传递。 | |||
T1025 |
Tranylcypromine (2-PCPA) hydrochloride
反苯环丙胺盐酸盐,Tranylcypromine (2-PCPA) HCl,SKF-385 HCl |
Histone Demethylase; MAO | Chromatin/Epigenetic; Metabolism; Neuroscience |
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl) 是一种单胺氧化酶抑制剂,对治疗重度抑郁症、心境恶劣障碍和非典型抑郁症有效。 | |||
T3723 |
Dioxopromethazine hydrochloride
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Dioxopromethazine hydrochloride 是一种基于目标的药物分类,在全球许多国家都有销售。 | |||
T7728 |
ACEPROMAZINE MALEATE
|
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Acepromazine maleate 是一种 α 肾上腺素受体 (alpha-adrenoceptor) 拮抗剂,是一种吩噻嗪类促进安定的试剂。 | |||
T19368 |
Hypromellose
Celacol HPM 5000,HPMC,羟丙甲纤维素,(Hydroxypropyl)methyl cellulose |
Others | Others |
Hypromellose (HPMC) 是一种水溶性的亲水性非离子纤维素醚。 | |||
T7778 |
Glypromate
Gly-Pro-Glu,甘氨酰-脯氨酰-谷氨酸 |
NMDAR | Neuroscience |
Glypromate (Gly-Pro-Glu) 是一种神经保护剂,是一种弱 NMDA 受体激动剂。 | |||
T71160 |
Levomepromazine HCl
|
||
Levomepromazine HCl is a phenothiazine with pharmacological activity similar to that of both CHLORPROMAZINE and PROMETHAZINE. It has the histamine-antagonist properties of the antihistamines together with CENTRAL NERVOUS SYSTEM effects resembling those of chlorpromazine. | |||
T13829 |
Oiligodendrocyte differentiation promoter 1
|
Others | Others |
Oiligodendrocyte differentiation promoter 1 is a promoter of oiligodendrocyte differentiation . | |||
T35015 |
Valdipromide
|
||
Valdipromide is a biochemical. | |||
T34142 |
Promoxolane
NSC-169878,NSC169878,NSC 169878 |
||
Promoxolane is a biochemical. | |||
T31639 |
Enpromate
Lilly59156,NSC 112682,59156,Lilly 59156,Lilly-59156 |
||
Enpromate 是一种合成的乙酰氨基甲酸酯,氮芥化合物。它是一种烷基化剂,具有抗肿瘤活性。 | |||
T25991 |
Promothiocin A
Antibiotic SF2741A,Antibiotic SF 2741A,Antibiotic SF-2741A |
||
Promothiocin A is an antibiotic. | |||
T24162 |
Impromidine
Impromidina,Impromidinum |
||
Impromidine is a highly potent and specific agonist of the histamine H2 receptor. | |||
T0302L |
Triflupromazine
Vesprin,Fluopromazine,Trifluopromazine,Adazine,Siquil |
||
Triflupromazine is a phenothiazine drug used as an antipsychotic and antiemetic. | |||
T13470 |
(±)-Levomepromazine-d6
dl-Methotrimeprazine D6,(±)-Methotrimeprazine (D6) |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor. | |||
T71826 |
(1S,2R)-Tranylcypromine hydrochloride
(1S,2R)-SKF 385 hydrochloride |
||
(1S,2R)-Tranylcypromine ((1S,2R)-SKF 385) hydrochloride 是一种有效的抗抑郁 (antidepressant) 剂。(1S,2R)-Tranylcypromine hydrochloride 对 MAO 和 LSD1有抑制作用。 | |||
T79914 |
Tranylcypromine
SKF 385 |
Monoamine Oxidase | Neuroscience |
Tranylcypromine (SKF 385)为一种高效的单胺氧化酶抑制剂。 | |||
T83896 |
Promethazine Sulfoxide
|
||
普罗米赛因硫醚是组胺H1受体拮抗剂普罗米赛因的代谢产物,通过细胞色素P450(CYP)亚型CYP2D6作用从普罗米赛因形成。 | |||
T0445L1 |
Promethazine hibenzate
D-08768,D08768,D 08768 |
||
Promethazine is a neuroleptic medication and first-generation antihistamine of the phenothiazine family. | |||
T69875 | ProMMP-9 inhibitor-3c | ||
ProMMP-9 inhibitor-3c is a potent and specific proMMP-9 inhibitor which disrupts f MMP-9 homodimerization and prevents association of proMMP-9 with both α4β1 integrin and CD44 and results in the dissociation of EGFR. | |||
T34141 |
Promegestone
R5020,R-5020,普美孕酮,RU 5020,R 5020,RU-5020 |
||
Promegestone is a progestin medication used in menopausal hormone therapy and in the treatment of gynecological disorders. | |||
T70105 |
Chlorpromazine Sulfone Hydrochloride
|
||
Chlorpromazine Sulfone Hydrochloride is a metabolite of Chlorpromazine -- an anti-emetic and anti-psychotic agent. It may also be used as a potential N-methyltransferase inhibitor. | |||
TP1153 |
Fibronectin Adhesion-promoting Peptide
Heparin Binding Peptide |
||
Fibronectin Adhesion-promoting Peptide (Heparin Binding Peptide) is one of the heparin-binding amino acid sequences found in the carboxy-terminal heparin-binding domain of fibronectin. | |||
T12701 |
(rel)-Tranylcypromine D5 hydrochloride
2-Phenylcyclopropylamine D5 hydrochloride |
Histone Demethylase | Chromatin/Epigenetic |
(rel)-Tranylcypromine D5 hydrochloride is a deuterium labeled (rel)-Tranylcypromine hydrochloride. (rel)-Tranylcypromine hydrochloride is an irreversible, nonselective inhibitor of monoamine oxidase (MAO) used in the treatment of depression. | |||
T26063 |
Repromicin
De-epoxy rosamicin,Repromicinum |
||
Repromicin is a chemical compound whose derivatives have strong antibacterial characteristics. | |||
T3609 |
Dioxopromethazine
Prothanon,Dioxoprothazine,盐酸二氧丙嗪 |
Others | Others |
Dioxopromethazine (Dioxoprothazine) 是一种口服具有活性的抗组胺药,能够抑制哮喘症状。 | |||
T15743 |
Levomepromazine
Methotrimeprazine |
Others | Others |
Methotrimeprazine is an orally available neuroleptic agent. It is commonly used to relieve nausea and vomiting in palliative care settings. Levomepromazine has antagonist actions at multiple neurotransmitter receptor sites, including cholinergic, dopamine | |||
T60913 |
Aceprometazine
|
||
Aceprometazine (1664CB) 是具有口服活性的抗精神病剂。Aceprometazine 可用于精神类疾病研究,例如抑郁症。 | |||
T60944 |
(±)-Levomepromazine
|
||
(±)-Levomepromazine 是 Levomepromazine 的外消旋体, Levomepromazine 是具有口服活性的典型抗精神病剂。 | |||
T71773 |
Levomepromazine Maleate
|
||
Levomepromazine Maleate is a Tricyclic antidepressant (TCA), acting as a serotonin–norepinephrine reuptake inhibitor (SNRI) and also having other activities including antihistamine, antiadrenergic, antiserotonergic, anticholinergic, and sodium channel-blocking effects. | |||
TP1152 |
Fibronectin Adhesion-promoting Peptide TFA
Heparin Binding Peptide TFA |
||
Fibronectin Adhesion-promoting Peptide (Heparin Binding Peptide) is one of the heparin-binding amino acid sequences found in the carboxy-terminal heparin-binding domain of fibronectin. It promotes assembly of mesenchymal stem cell (MSC) spheroids into lar | |||
T25109 |
ARN-6039
ARN 6039,ARN6039 |
||
ARN-6039 is an orally available inverse agonist of RORγ for Autoimmune Neuroinflammatory Demyelinating Disease. The activity of ARN-6039 against RORγ was demonstrated in a RORγ-activated IL-17A Prom/LUCPorter assay in HEK 293 cells (360 nM) and in IL-17 r |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN4832 | Prometaphanine | Others | Others |
Prometaphanine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4832,CAS号为 6858-85-1。 | |||
TN6023 |
16-Oxoprometaphanine
|
||
16-Oxoprometaphanine是一种天然产物,属于防己科千金藤属,其产品编号为 TN6023,CAS号为 58738-31-1。16-Oxoprometaphanine可用作对照参考。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02842 |
CD133/PROM1 Protein, Mouse, Recombinant (His & SUMO)
CD133,Prom1,Prominin-like protein 1,Pr... |
Mouse | E. coli |
May play a role in cell differentiation, proliferation and apoptosis. Binds cholesterol in cholesterol-containing plasma membrane microdomains and may play a role in the organization of the apical plasma membrane in epithelial cells. During early retinal development acts as a key regulator of disk morphogenesis. Involved in regulation of MAPK and Akt signaling pathways. In neuroblastoma cells suppresses cell differentiation such as neurite outgrowth in a RET-dependent manner. | |||
TMPH-00001 |
CD133/PROM1 Protein-VLP, Human, Recombinant (His)
Proml1,Prom1,CD133,Prominin-like ... |
Human | HEK293 Cells |
May play a role in cell differentiation, proliferation and apoptosis. Binds cholesterol in cholesterol-containing plasma membrane microdomains and may play a role in the organization of the apical plasma membrane in epithelial cells. During early retinal development acts as a key regulator of disk morphogenesis. Involved in regulation of MAPK and Akt signaling pathways. In neuroblastoma cells suppresses cell differentiation such as neurite outgrowth in a RET-dependent manner. CD133/PROM1 Protein... | |||
TMPY-03690 |
CD133/PROM1 Protein, Rat, Recombinant (mFc)
prominin 1 |
Rat | HEK293 Cells |
CD133/PROM1 Protein, Rat, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 60 kDa and the accession number is Q7TSL4. | |||
TMPY-03691 |
CD133/PROM1 Protein, Rat, Recombinant (His)
prominin 1 |
Rat | HEK293 Cells |
CD133/PROM1 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.10 kDa and the accession number is Q7TSL4. | |||
THMH-00001 |
CD133/PROM1 Recombinant,Human(Yeast expression,His)
|
||
TMPH-01922 |
Promotilin Protein, Human, Recombinant (GST & His & Myc)
|
Human | E. coli |
Promotilin Protein, Human, Recombinant (GST & His & Myc) is expressed in E. coli. |