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Targets Recommended: Histone Demethylase MAO Monoamine Oxidase

47

抑制剂 & 化合物

2

天然产物

6

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T7942 Tranylcypromine hemisulfate

Tranylcypromine Sulfate,Tranylcypromine (hemisulfate),反苯环丙胺半硫酸盐

Histone Demethylase; MAO; Monoamine Oxidase Chromatin/Epigenetic; Metabolism; Neuroscience
Tranylcypromine hemisulfate (Tranylcypromine Sulfate) 是单胺氧化酶(MAO) 和赖氨酸特异性去甲基化酶 1 (LSD1) 的抑制剂,可用于研究抑郁症和子宫内膜异位症。
T9232 Mitochondrial fusion promoter M1

Mitochondrial Metabolism Metabolism
Mitochondrial fusion promoter M1 是一种线粒体动态调节剂,能够保持线粒体功能并促进细胞呼吸,减轻心肌缺血/再灌注大鼠的心脏损伤和大脑损伤。
T9228 Propionylpromazine hydrochloride

盐酸丙酰丙嗪,Propiopromazine hydrochloride

Dopamine Receptor GPCR/G Protein; Neuroscience
Propionylpromazine hydrochloride (Propiopromazine hydrochloride) 是多巴胺受体 D2 (DRD2) 拮抗剂,可用于研究帕金森氏病。
TQ0022 Capromorelin Tartrate

卡普瑞林酒石酸盐,CP 424391-18

GHSR GPCR/G Protein
Capromorelin Tartrate (CP 424391-18) 是口服有活性的 growth hormone secretagogue receptor 有效激动剂,能够作用于 hGHS-R1a(Ki:7 nM)。
T7778L Glypromate acetate(32302-76-4 free base)

NMDAR Neuroscience
Glypromate acetate(32302-76-4 free base) 是一种神经保护剂,是一种弱 NMDA 受体激动剂。
T1536 Promestriene

3-propyl ethyl,舒经劳,17B-methyl estradiol,Promestriano

Estrogen/progestogen Receptor Endocrinology/Hormones
Promestriene (3-propyl ethyl) 是局部有效的雌激素,是合成的雌二醇二乙醚。它对阴道萎缩有作用,但吸收量小。
T0445L Promethazine hydrochloride

盐酸异丙嗪,Promethazine HCl,Phenergan

Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Promethazine hydrochloride (Promethazine HCl) 是抗组胺药物,是 H1 受体的强拮抗剂和 mACh 受体的中度拮抗剂,对 5-HT2A、5-HT2C、D2 和 α1-肾上腺素能受体具有中等亲和力。
T0355 Valpromide

Depamide,Valpramide,丙戊酰胺,Dipropylacetamide,2-propylpentanamide

Epoxide Hydrolase; HSV Metabolism; Microbiology/Virology
Valpromide (Dipropylacetamide) 是丙戊酸的羧酰胺衍生物,用于治疗癫痫和一些情感障碍。
T0302 Triflupromazine hydrochloride

Neoprin,盐酸三氟丙嗪,Fluopromazine hydrochloride,Fluorofen,Flumazin

Dopamine Receptor; 5-HT Receptor; AChR; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Triflupromazine hydrochloride (Fluopromazine hydrochloride) 是一种抗精神病药物,是多巴胺 D1/D2 受体拮抗剂。
T68921 Impromidine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Impromidine hydrochloride 是一种非常有效和特异性的组胺H2受体激动剂,可用于进行心血管研究。
T50054 Opromazine hydrochloride

Others Others
Opromazine hydrochloride 属于吩噻嗪类抗精神病药物,通过阻断大脑中的多巴胺受体而降低多巴胺能通路的活性,主要用于治疗精神分裂症和精神病等精神疾病。
T0445 Promethazine

Proazamine,异丙嗪,Diphergan

CaMK; Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Promethazine (Proazamine) 是抗青光眼前列腺素(PG)的类似物。
T1522 Iopromide

碘普罗胺,Iopromidum,Ultravist

Others Others
Iopromide (Iopromidum) 是用于血管内的低渗透、非离子造影剂。
T19733 Prometryn

Caparol,Gesagard,Mercazin,扑草净

Others Others
Prometryn (Mercazin) 是一种除草剂,可提高棉花产量。
TP1153L Fibronectin Adhesion-promoting Peptide acetate

Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate

Others Others
Fibronectin Adhesion-promoting Peptide acetate (Heparin Binding Peptide acetate)(125720-21-0 free base) 是在纤连蛋白的羧基末端肝素结合结构域中发现的肝素结合氨基酸序列之一。
T0766 Promazine hydrochloride

Romtiazin hydrochloride,Sinophenin hydrochloride,盐酸丙嗪

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR GPCR/G Protein; Neuroscience
Promazine hydrochloride (Romtiazin hydrochloride) 是一种抗精神病药,也是一种多巴胺受体 (D2) 拮抗剂,能够抑制多巴胺能神经传递。
T1025 Tranylcypromine (2-PCPA) hydrochloride

反苯环丙胺盐酸盐,Tranylcypromine (2-PCPA) HCl,SKF-385 HCl

Histone Demethylase; MAO Chromatin/Epigenetic; Metabolism; Neuroscience
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl) 是一种单胺氧化酶抑制剂,对治疗重度抑郁症、心境恶劣障碍和非典型抑郁症有效。
T3723 Dioxopromethazine hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Dioxopromethazine hydrochloride 是一种基于目标的药物分类,在全球许多国家都有销售。
T7728 ACEPROMAZINE MALEATE

Dopamine Receptor GPCR/G Protein; Neuroscience
Acepromazine maleate 是一种 α 肾上腺素受体 (alpha-adrenoceptor) 拮抗剂,是一种吩噻嗪类促进安定的试剂。
T19368 Hypromellose

Celacol HPM 5000,HPMC,羟丙甲纤维素,(Hydroxypropyl)methyl cellulose

Others Others
Hypromellose (HPMC) 是一种水溶性的亲水性非离子纤维素醚。
T7778 Glypromate

Gly-Pro-Glu,甘氨酰-脯氨酰-谷氨酸

NMDAR Neuroscience
Glypromate (Gly-Pro-Glu) 是一种神经保护剂,是一种弱 NMDA 受体激动剂。
T71160 Levomepromazine HCl

Levomepromazine HCl is a phenothiazine with pharmacological activity similar to that of both CHLORPROMAZINE and PROMETHAZINE. It has the histamine-antagonist properties of the antihistamines together with CENTRAL NERVOUS SYSTEM effects resembling those of chlorpromazine.
T13829 Oiligodendrocyte differentiation promoter 1

Others Others
Oiligodendrocyte differentiation promoter 1 is a promoter of oiligodendrocyte differentiation .
T35015 Valdipromide

Valdipromide is a biochemical.
T34142 Promoxolane

NSC-169878,NSC169878,NSC 169878

Promoxolane is a biochemical.
T31639 Enpromate

Lilly59156,NSC 112682,59156,Lilly 59156,Lilly-59156

Enpromate 是一种合成的乙酰氨基甲酸酯,氮芥化合物。它是一种烷基化剂,具有抗肿瘤活性。
T25991 Promothiocin A

Antibiotic SF2741A,Antibiotic SF 2741A,Antibiotic SF-2741A

Promothiocin A is an antibiotic.
T24162 Impromidine

Impromidina,Impromidinum

Impromidine is a highly potent and specific agonist of the histamine H2 receptor.
T0302L Triflupromazine

Vesprin,Fluopromazine,Trifluopromazine,Adazine,Siquil

Triflupromazine is a phenothiazine drug used as an antipsychotic and antiemetic.
T13470 (±)-Levomepromazine-d6

dl-Methotrimeprazine D6,(±)-Methotrimeprazine (D6)

Adrenergic Receptor GPCR/G Protein; Neuroscience
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
T71826 (1S,2R)-Tranylcypromine hydrochloride

(1S,2R)-SKF 385 hydrochloride

(1S,2R)-Tranylcypromine ((1S,2R)-SKF 385) hydrochloride 是一种有效的抗抑郁 (antidepressant) 剂。(1S,2R)-Tranylcypromine hydrochloride 对 MAO 和 LSD1有抑制作用。
T79914 Tranylcypromine

SKF 385

Monoamine Oxidase Neuroscience
Tranylcypromine (SKF 385)为一种高效的单胺氧化酶抑制剂。
T83896 Promethazine Sulfoxide

普罗米赛因硫醚是组胺H1受体拮抗剂普罗米赛因的代谢产物,通过细胞色素P450(CYP)亚型CYP2D6作用从普罗米赛因形成。
T0445L1 Promethazine hibenzate

D-08768,D08768,D 08768

Promethazine is a neuroleptic medication and first-generation antihistamine of the phenothiazine family.
T69875 ProMMP-9 inhibitor-3c

ProMMP-9 inhibitor-3c is a potent and specific proMMP-9 inhibitor which disrupts f MMP-9 homodimerization and prevents association of proMMP-9 with both α4β1 integrin and CD44 and results in the dissociation of EGFR.
T34141 Promegestone

R5020,R-5020,普美孕酮,RU 5020,R 5020,RU-5020

Promegestone is a progestin medication used in menopausal hormone therapy and in the treatment of gynecological disorders.
T70105 Chlorpromazine Sulfone Hydrochloride

Chlorpromazine Sulfone Hydrochloride is a metabolite of Chlorpromazine -- an anti-emetic and anti-psychotic agent. It may also be used as a potential N-methyltransferase inhibitor.
TP1153 Fibronectin Adhesion-promoting Peptide

Heparin Binding Peptide

Fibronectin Adhesion-promoting Peptide (Heparin Binding Peptide) is one of the heparin-binding amino acid sequences found in the carboxy-terminal heparin-binding domain of fibronectin.
T12701 (rel)-Tranylcypromine D5 hydrochloride

2-Phenylcyclopropylamine D5 hydrochloride

Histone Demethylase Chromatin/Epigenetic
(rel)-Tranylcypromine D5 hydrochloride is a deuterium labeled (rel)-Tranylcypromine hydrochloride. (rel)-Tranylcypromine hydrochloride is an irreversible, nonselective inhibitor of monoamine oxidase (MAO) used in the treatment of depression.
T26063 Repromicin

De-epoxy rosamicin,Repromicinum

Repromicin is a chemical compound whose derivatives have strong antibacterial characteristics.
T3609 Dioxopromethazine

Prothanon,Dioxoprothazine,盐酸二氧丙嗪

Others Others
Dioxopromethazine (Dioxoprothazine) 是一种口服具有活性的抗组胺药,能够抑制哮喘症状。
T15743 Levomepromazine

Methotrimeprazine

Others Others
Methotrimeprazine is an orally available neuroleptic agent. It is commonly used to relieve nausea and vomiting in palliative care settings. Levomepromazine has antagonist actions at multiple neurotransmitter receptor sites, including cholinergic, dopamine
T60913 Aceprometazine

Aceprometazine (1664CB) 是具有口服活性的抗精神病剂。Aceprometazine 可用于精神类疾病研究,例如抑郁症。
T60944 (±)-Levomepromazine

(±)-Levomepromazine 是 Levomepromazine 的外消旋体, Levomepromazine 是具有口服活性的典型抗精神病剂。
T71773 Levomepromazine Maleate

Levomepromazine Maleate is a Tricyclic antidepressant (TCA), acting as a serotonin–norepinephrine reuptake inhibitor (SNRI) and also having other activities including antihistamine, antiadrenergic, antiserotonergic, anticholinergic, and sodium channel-blocking effects.
TP1152 Fibronectin Adhesion-promoting Peptide TFA

Heparin Binding Peptide TFA

Fibronectin Adhesion-promoting Peptide (Heparin Binding Peptide) is one of the heparin-binding amino acid sequences found in the carboxy-terminal heparin-binding domain of fibronectin. It promotes assembly of mesenchymal stem cell (MSC) spheroids into lar
T25109 ARN-6039

ARN 6039,ARN6039

ARN-6039 is an orally available inverse agonist of RORγ for Autoimmune Neuroinflammatory Demyelinating Disease. The activity of ARN-6039 against RORγ was demonstrated in a RORγ-activated IL-17A Prom/LUCPorter assay in HEK 293 cells (360 nM) and in IL-17 r

化合物

Tranylcypromine hemisulfate
Cat.No: T7942
Synonym: Tranylcypromine Sulfate,Tranylcypromine (hemisulfate),反苯环丙胺半硫酸盐
Target: Histone Demethylase, MAO, Monoamine Oxidase
Mitochondrial fusion promoter M1
Cat.No: T9232
Synonym:
Target: Mitochondrial Metabolism
Propionylpromazine hydrochloride
Cat.No: T9228
Synonym: 盐酸丙酰丙嗪,Propiopromazine hydrochloride
Target: Dopamine Receptor
Capromorelin Tartrate
Cat.No: TQ0022
Synonym: 卡普瑞林酒石酸盐,CP 424391-18
Target: GHSR
Glypromate acetate(32302-76-4 free base)
Cat.No: T7778L
Synonym:
Target: NMDAR
Promestriene
Cat.No: T1536
Synonym: 3-propyl ethyl,舒经劳,17B-methyl estradiol,Promestriano
Target: Estrogen/progestogen Receptor
Promethazine hydrochloride
Cat.No: T0445L
Synonym: 盐酸异丙嗪,Promethazine HCl,Phenergan
Target: Adrenergic Receptor, Histamine Receptor
Valpromide
Cat.No: T0355
Synonym: Depamide,Valpramide,丙戊酰胺,Dipropylacetamide,2-propylpentanamide
Target: Epoxide Hydrolase, HSV
Triflupromazine hydrochloride
Cat.No: T0302
Synonym: Neoprin,盐酸三氟丙嗪,Fluopromazine hydrochloride,Fluorofen,Flumazin
Target: Dopamine Receptor, 5-HT Receptor, AChR, Autophagy
Impromidine hydrochloride
Cat.No: T68921
Synonym:
Target: Histamine Receptor
Opromazine hydrochloride
Cat.No: T50054
Synonym:
Target: Others
Promethazine
Cat.No: T0445
Synonym: Proazamine,异丙嗪,Diphergan
Target: CaMK, Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR, Histamine Receptor
Iopromide
Cat.No: T1522
Synonym: 碘普罗胺,Iopromidum,Ultravist
Target: Others
Prometryn
Cat.No: T19733
Synonym: Caparol,Gesagard,Mercazin,扑草净
Target: Others
Fibronectin Adhesion-promoting Peptide acetate
Cat.No: TP1153L
Synonym: Fibronectin Adhesion-promoting Peptide acetate(125720-21-0 free base),Heparin Binding Peptide acetate
Target: Others
Promazine hydrochloride
Cat.No: T0766
Synonym: Romtiazin hydrochloride,Sinophenin hydrochloride,盐酸丙嗪
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR
Tranylcypromine (2-PCPA) hydrochloride
Cat.No: T1025
Synonym: 反苯环丙胺盐酸盐,Tranylcypromine (2-PCPA) HCl,SKF-385 HCl
Target: Histone Demethylase, MAO
Dioxopromethazine hydrochloride
Cat.No: T3723
Synonym:
Target: Histamine Receptor
ACEPROMAZINE MALEATE
Cat.No: T7728
Synonym:
Target: Dopamine Receptor
Hypromellose
Cat.No: T19368
Synonym: Celacol HPM 5000,HPMC,羟丙甲纤维素,(Hydroxypropyl)methyl cellulose
Target: Others
Glypromate
Cat.No: T7778
Synonym: Gly-Pro-Glu,甘氨酰-脯氨酰-谷氨酸
Target: NMDAR
Levomepromazine HCl
Cat.No: T71160
Synonym:
Target:
Oiligodendrocyte differentiation promoter 1
Cat.No: T13829
Synonym:
Target: Others
Valdipromide
Cat.No: T35015
Synonym:
Target:
Promoxolane
Cat.No: T34142
Synonym: NSC-169878,NSC169878,NSC 169878
Target:
Enpromate
Cat.No: T31639
Synonym: Lilly59156,NSC 112682,59156,Lilly 59156,Lilly-59156
Target:
Promothiocin A
Cat.No: T25991
Synonym: Antibiotic SF2741A,Antibiotic SF 2741A,Antibiotic SF-2741A
Target:
Impromidine
Cat.No: T24162
Synonym: Impromidina,Impromidinum
Target:
Triflupromazine
Cat.No: T0302L
Synonym: Vesprin,Fluopromazine,Trifluopromazine,Adazine,Siquil
Target:
(±)-Levomepromazine-d6
Cat.No: T13470
Synonym: dl-Methotrimeprazine D6,(±)-Methotrimeprazine (D6)
Target: Adrenergic Receptor
(1S,2R)-Tranylcypromine hydrochloride
Cat.No: T71826
Synonym: (1S,2R)-SKF 385 hydrochloride
Target:
Tranylcypromine
Cat.No: T79914
Synonym: SKF 385
Target: Monoamine Oxidase
Promethazine Sulfoxide
Cat.No: T83896
Synonym:
Target:
Promethazine hibenzate
Cat.No: T0445L1
Synonym: D-08768,D08768,D 08768
Target:
ProMMP-9 inhibitor-3c
Cat.No: T69875
Synonym:
Target:
Promegestone
Cat.No: T34141
Synonym: R5020,R-5020,普美孕酮,RU 5020,R 5020,RU-5020
Target:
Chlorpromazine Sulfone Hydrochloride
Cat.No: T70105
Synonym:
Target:
Fibronectin Adhesion-promoting Peptide
Cat.No: TP1153
Synonym: Heparin Binding Peptide
Target:
(rel)-Tranylcypromine D5 hydrochloride
Cat.No: T12701
Synonym: 2-Phenylcyclopropylamine D5 hydrochloride
Target: Histone Demethylase
Repromicin
Cat.No: T26063
Synonym: De-epoxy rosamicin,Repromicinum
Target:
Dioxopromethazine
Cat.No: T3609
Synonym: Prothanon,Dioxoprothazine,盐酸二氧丙嗪
Target: Others
Levomepromazine
Cat.No: T15743
Synonym: Methotrimeprazine
Target: Others
Aceprometazine
Cat.No: T60913
Synonym:
Target:
(±)-Levomepromazine
Cat.No: T60944
Synonym:
Target:
Levomepromazine Maleate
Cat.No: T71773
Synonym:
Target:
Fibronectin Adhesion-promoting Peptide TFA
Cat.No: TP1152
Synonym: Heparin Binding Peptide TFA
Target:
ARN-6039
Cat.No: T25109
Synonym: ARN 6039,ARN6039
Target:
Cat. No. Product Name Target Signaling Pathways
TN4832 Prometaphanine

Others Others
Prometaphanine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4832,CAS号为 6858-85-1。
TN6023 16-Oxoprometaphanine

16-Oxoprometaphanine是一种天然产物,属于防己科千金藤属,其产品编号为 TN6023,CAS号为 58738-31-1。16-Oxoprometaphanine可用作对照参考。

天然产物

Prometaphanine
Cat.No: TN4832
Synonym:
Target: Others
16-Oxoprometaphanine
Cat.No: TN6023
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPH-02842 CD133/PROM1 Protein, Mouse, Recombinant (His & SUMO)

CD133,Prom1,Prominin-like protein 1,Pr...

Mouse E. coli
May play a role in cell differentiation, proliferation and apoptosis. Binds cholesterol in cholesterol-containing plasma membrane microdomains and may play a role in the organization of the apical plasma membrane in epithelial cells. During early retinal development acts as a key regulator of disk morphogenesis. Involved in regulation of MAPK and Akt signaling pathways. In neuroblastoma cells suppresses cell differentiation such as neurite outgrowth in a RET-dependent manner.
TMPH-00001 CD133/PROM1 Protein-VLP, Human, Recombinant (His)

Proml1,Prom1,CD133,Prominin-like ...

Human HEK293 Cells
May play a role in cell differentiation, proliferation and apoptosis. Binds cholesterol in cholesterol-containing plasma membrane microdomains and may play a role in the organization of the apical plasma membrane in epithelial cells. During early retinal development acts as a key regulator of disk morphogenesis. Involved in regulation of MAPK and Akt signaling pathways. In neuroblastoma cells suppresses cell differentiation such as neurite outgrowth in a RET-dependent manner. CD133/PROM1 Protein...
TMPY-03690 CD133/PROM1 Protein, Rat, Recombinant (mFc)

prominin 1

Rat HEK293 Cells
CD133/PROM1 Protein, Rat, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 60 kDa and the accession number is Q7TSL4.
TMPY-03691 CD133/PROM1 Protein, Rat, Recombinant (His)

prominin 1

Rat HEK293 Cells
CD133/PROM1 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.10 kDa and the accession number is Q7TSL4.
THMH-00001 CD133/PROM1 Recombinant,Human(Yeast expression,His)

TMPH-01922 Promotilin Protein, Human, Recombinant (GST & His & Myc)

Human E. coli
Promotilin Protein, Human, Recombinant (GST & His & Myc) is expressed in E. coli.

重组蛋白

CD133/PROM1 Protein, Mouse, Recombinant (His & SUMO)
Cat.No: TMPH-02842
Species: Mouse
Expression System: E. coli
CD133/PROM1 Protein-VLP, Human, Recombinant (His)
Cat.No: TMPH-00001
Species: Human
Expression System: HEK293 Cells
CD133/PROM1 Protein, Rat, Recombinant (mFc)
Cat.No: TMPY-03690
Species: Rat
Expression System: HEK293 Cells
CD133/PROM1 Protein, Rat, Recombinant (His)
Cat.No: TMPY-03691
Species: Rat
Expression System: HEK293 Cells
CD133/PROM1 Recombinant,Human(Yeast expression,His)
Cat.No: THMH-00001
Species:
Expression System:
Promotilin Protein, Human, Recombinant (GST & His & Myc)
Cat.No: TMPH-01922
Species: Human
Expression System: E. coli
TargetMol Loading
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