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Targets Recommended: Thrombin Thrombopoietin Receptor

61

抑制剂 & 化合物

13

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Cat. No. Product Name Target Signaling Pathways
TQ0223 Lusutrombopag

芦曲泊帕,鲁索曲波帕,S-888711,Mulpleta

Thrombin; Thrombopoietin Receptor Immunology/Inflammation; Proteases/Proteasome
Lusutrombopag (Mulpleta) 是一种口服生物可利用的小分子血小板生成素 (TPO) 受体激动剂,用于选择性侵入性手术前患有血小板减少症的慢性肝病的患者。
T6825 Eltrombopag Olamine

Promacta Olamine,Revolade,艾曲泊帕乙醇胺盐,Eltrombopag diethanolamine salt,SB497115,艾曲波帕乙醇胺盐,SB-497115GR

Thrombin Proteases/Proteasome
Eltrombopag Olamine (Eltrombopag diethanolamine salt) 是 Eltrombopag 的口服活性乙醇胺盐,是一种血小板生成素(TPO)受体激动剂,用于血小板减少的某些病症研究。
T4635 Ralinepag

APD811

Others; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Others
Ralinepag (APD811) 是一种可口服的非前列腺素前列环素 (IP) 受体激动剂,对人和大鼠 IP 受体以及人 DP1 受体的 EC50 分别为 8.5、530 和 850 nM。
T4460 Dapagliflozin ((2S)-1,2-propanediol, hydrate)

BMS-512148 (2S)-1,2-propanediol, hydrate,达格列净 (2S)-1,2-丙二醇水合物,Dapagliflozin propanediol monohydrate

SGLT GPCR/G Protein
Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) 是 Dapagliflozin 1,2-propanediol, hydrate 的 S 型异构体,是竞争性葡萄糖协同转运蛋白2 抑制剂,可促进尿液中葡萄糖的排泄,可用于糖尿病的研究。它诱导 HIF1表达并减轻肾脏 IR 损伤。
T2389 Dapagliflozin

达格列净,BMS-512148

SGLT; HIF Angiogenesis; Chromatin/Epigenetic; GPCR/G Protein
Dapagliflozin (BMS-512148) 竞争性的葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,可促进尿液中葡萄糖的排泄,在糖尿病 (DM) 研究中具有价值。Dapagliflozin 诱导 HIF1表达并减轻肾脏 IR 损伤。
T15273 Fedovapagon

VA483,A106483

Vasopressin Receptor GPCR/G Protein
Fedovapagon (VA106483) 是一种具有选择性和高效性的加压素 V2 受体 (V2R) 激动剂,可抑制斑马鱼节间血管的生长。Fedovapagon 可用于研究膀胱过度活动症、夜尿症和膀胱疼痛综合征。
T7417 Avatrombopag

YM477,AKR-501,1-[3-氯-5-[[[4-(4-氯-2-噻吩基)-5-(4-环己基-1-哌嗪基)-2-噻唑基]氨基]羰基]-2-吡啶基]-4-哌啶羧酸,E5501

Thrombin; Thrombopoietin Receptor Immunology/Inflammation; Proteases/Proteasome
Avatrombopag (YM477) 是一种新型口服血小板生成素 (TPO) 受体激动剂,可激活 TPO 受体并增加巨核细胞增殖/分化和血小板生成。
T20641 Propagermanium

Dipropanoic acid germanium sequioxide,SK-818,Ge 132,二羧乙基三氧化二锗,Ge132,SK 818,Ge-132

Others Others
Propagermanium (Ge132) 是一种锗的有机金属化合物,在日本已被用作治疗慢性乙型肝炎的药物。
T22870 IPAG

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
IPAG 是有效的 sigma-1 受体拮抗剂 (pKi= 4.3)。 IPAG 可诱导细胞凋亡。
T3174 Taprenepag

CP-544326

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Taprenepag (CP-544326) 是一种有效的选择性前列腺素 E2 受体激动剂,EC50为 2.8 nM,可用于研究开角治疗高眼压和青光眼的试验。
T15259 Evatanepag

CP-533536 free acid,2-[3-[N-(4-叔丁基苄基)-N-(吡啶-3-基磺酰基)氨基甲基]苯氧基]乙酸

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Evatanepag (CP-533536 free acid) 是一种 EP2 受体选择性前列腺素 E2 (PGE2) 激动剂,可诱导局部骨形成,EC50 为 0.3 nM。它在大鼠骨折愈合模型中以单剂量局部给药时表现出愈合骨折的能力。
T1766 Empagliflozin

BI 10773,恩格列净

SGLT GPCR/G Protein
Empagliflozin (BI 10773) 是一种 SGLT-2 抑制剂 (IC50=3.1 nM),具有有效的和选择性,对 SGLT-1/4/5/6 的选择性高 300 倍以上。Empagliflozin 可用于治疗二型糖尿病。
T6750 Opaganib

ABC294640

S1P Receptor GPCR/G Protein
Opaganib (ABC294640) 是选择性和竞争性的鞘氨醇激酶 2 (SK2) 抑制剂,Ki 为 9.8 μM。
T67849 O-Desethyl Dapagliflozin

Empagliflozin-4

SGLT GPCR/G Protein
O-Desethyl Dapagliflozin (Empagliflozin-4) 是一种 SGLT2 抑制剂, IC50=33nM.
T3216 Selexipag

NS-304,ACT-293987,赛乐西帕,Uptravi

Others; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Others
Selexipag (ACT-293987) 是前列环素受体激动剂,可引起肺血管舒张,用于治疗肺动脉高压。
T1088 Repaglinide

AG-EE 388 ZW,AG-EE 623ZW,瑞格列奈

Potassium Channel; PPAR DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Repaglinide (AG-EE 623ZW) 是一种能够用于2 型糖尿病的胰岛素促分泌剂。
T2562 Eltrombopag

SB-497115,SB-497115-GR,艾曲波帕

Thrombin Proteases/Proteasome
Eltrombopag (SB-497115-GR) 是一种具有巨核细胞生成刺激活性的口服活性血小板生成素受体激动剂,可结合并刺激血小板血小板生成素受体,用于血小板减少的某些病症研究。
T76822 Pagibaximab

Pagibaximab为一种嵌合IgG1抗体,针对金黄色葡萄球菌与表皮链球菌的表面脂肪酸成分具有特异性识别能力。其主要应用于预防葡萄球菌所引起的败血症。
T10957 Dapagliflozin impurity

Others Others
Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.
T124813 N-Methylsarpagine methosalt

N-Methylsarpagine methosalt 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124813。
T62864 Hetrombopag

Hetrombopag 是一种 thrombopoietin receptor 的有效激动剂。Hetrombopag 具有良好的耐受性且安全性可控。Hetrombopag 具有潜力进行免疫性血小板减少症的研究。
T126029 8-cis-Cinnamoylharpagide

8-cis-Cinnamoylharpagide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126029,CAS号为 133645-36-0。
T68888 Avatrombopag maleate

Avatrombopag, also known as AKR-501, YM477, AS 1670542 or E5501, is a novel orally-active thrombopoietin (TPO) receptor agonist. AKR-501 specifically targeted the TPO receptor and stimulated megakaryocytopoiesis throughout the development and maturation of megakaryocytes just as rhTPO did. AKR-501 may be useful in the treatment of patients with thrombocytopenia. Avatrombopag was first approved in 2018.
T27536 Hetrombopag olamine

Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.
T61876 Sipagladenant

Sipagladenant (Compound I) is an orally active inverse agonist targeting the adenosine receptor A2A [1]. It possesses potential for utilization in research pertaining to frontal lobe dysfunction [2].
T69755 Evatanepag sodium

Evatanepag, also known as CP-533536, is an EP2 receptor selective prostaglandin E2 (PGE2) agonist that induces local bone formation. CP-533536 demonstrated the ability to heal fractures when administered locally as a single dose in rat models of fracture healing.
T124431 Pagoside

TQ0285L Spaglumic acid acetate

Isospaglumic acid acetate,Spaglumic acid acetate(3106-85-2 Free base)

Endogenous Metabolite Metabolism
Spaglumic acid acetate (Isospaglumic acid acetate) 是一种在脑中以毫摩尔浓度存在的神经肽。
TMIH-0013 (S)-Empagliflozin-d4

(S)-Empagliflozin-d4 是 (S)-Empagliflozin 的氘代化合物。(S)-Empagliflozin 的 CAS 号为 864070-44-0。Empagliflozin 是有效的、选择性的钠葡萄糖协同转运蛋白-2 (SGLT-2) 抑制剂,对人 SGLT-2 的IC50为 3.1 nM。
T19548 Repaglinide D5

AG-EE 623ZW D5,瑞格列奈 D5

Others Others
Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.
T64615 EMpagliflozin iMpurity 5

(2S,3R,4R,5S,6R)-2-(4-Chloro-3-(4-hydroxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64615。
T71301 Opaganib HCl

ABC294640, also known as Opaganib, is an orally available, aryladamantane compound and selective inhibitor of sphingosine kinase-2 (SK2) with potential antineoplastic activity. Upon administration, ABC294640 competitively binds to and inhibits SK2, thereby preventing the phosphorylation of the pro-apoptotic amino alcohol sphingosine to sphingosine 1-phosphate (S1P), the lipid mediator that is pro-survival and critical for immunomodulation. This may eventually lead to the induction of apoptosis a...
T25547 Isospaglumate sodium

Isospaglumate trisodium,Sodium isospaglumate

Isospaglumate sodium is the sodium salt of isospaglumate which is an antiallergic agent.
T62865 Rafutrombopag

Rafutrombopag 是一种血小板生成素 (TPO) 激动剂。
T29708 Aganepag isopropyl

AGN-210961,AGN 210961,AGN210961

Aganepag isopropyl can be used to treat Glaucoma.
T68560 Totrombopag choline

Totrombopag, also known LGD-4665, GSK2285921 and SB559448, is an oral thromobopoietin receptor agonist, is being developed as a new generation small molecule thrombopoietin (TPO) mimetic. It is a highly selective and potent agonist of the TPO receptor and therefore induces differentiation and proliferation of megakaryocytes. The pharmacologic characteristics indicate potential therapeutic use in thrombocytopenic patients with a variety of clinical etiologies.
T67184 PeracetylEmpagliflozin

(2R,3R,4R,5S,6S)-2-(Acetoxymethyl)-6-(4-chloro-3-(4-(((S)-tetrahydrofuran-3-yl)oxy)benzyl)phenyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T67184。
T13497 3'-Hydroxy Repaglinide

Others Others
3'-Hydroxy Repaglinide is a main CYP2C8 metabolite of Repaglinide. Repaglinide is a carbamoylmethyl benzoic acid derivative and used as the treatment of type II diabetes.
T14139 Aganepag

AGN 210937

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Aganepag, a potent Prostanoid EP2 receptor agonist, exhibits remarkable selectivity with an EC50 of 0.19 nM, demonstrating no activity at the EP4 receptor. Its applications are primarily in the fields of wound healing, scar reduction, scar prevention, and the treatment and prevention of wrinkles.
TMIH-0520 Selexipag-d7

Selexipag-d7 是 Selexipag 的氘代化合物。Selexipag 的 CAS 号为 475086-01-2。Selexipag 是前列环素受体激动剂,可引起肺血管舒张,用于治疗肺动脉高压。
T64667 10× SDS-PAGE SDS Running Buffer

Others Others
10× SDS-PAGE SDS Running Buffer 是 SDS-PAGE (SDS-变性聚丙烯酰胺凝胶电泳) 10 倍浓缩的缓冲液,主要成分为三羟甲基氨基甲烷(Tris)、甘氨酸(Glycine)和十二烷基硫酸钠(SDS)。
T40654 Avatrombopag hydrochloride

AKR-501 hydrochloride,YM477hydrochloride,E5501hydrochloride

Avatrombopag hydrochloride (AKR-501) is an orally active, nonpeptide agonist of the thrombopoietin (TPO) receptor with an EC 50 of 3.3 nM. It effectively mimics the biological activities of TPO, stimulating platelet production by activating the intracellular signaling system and facilitating the generation of platelets and megakaryocytes from hemopoietic precursor cells. Additionally, Avatrombopag hydrochloride serves as a substrate for cytochrome P450 (CYP) 2C9 and CYP3A.
T16988 Taprenepag isopropyl

PF-04217329

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Taprenepag isopropyl is a highly selective agonist of the EP2 receptor.
T35619 Dapagliflozin-3-O-β-D-Glucuronide

Dapagliflozin-3-O-β-D-glucuronide is a metabolite of dapagliflozin . Dapagliflozin is a first generation selective sodium glucose cotransporter (SGLT) 2 inhibitor that blocks glucose transport.[1] Dapagliflozin is metabolized by uridine diphosphate glucuronosyltransferase (UGT) 1A9 to dapagliflozin-3-O-β-D-glucuronide, which is 2,600-fold less potent than the parent compound with regard to SGLT2 inhibition.[2]
T79850 Irpagratinib

ABSK011

FGFR Angiogenesis; Tyrosine Kinase/Adaptors
Irpagratinib (ABSK011)是一种靶向FGFR4(IC50<10 nM)的口服活性酪氨酸激酶抑制剂,可抑制FGFR4自磷酸化并阻断其信号转导至下游途径。在小鼠、大鼠和狗的PK研究中,Irpagratinib表现出高暴露量,并在皮下异种移植肿瘤模型中展示抗肿瘤活性。
T29707 Aganepag ethanediol

AGN-212409,AGN212409

Aganepag ethanediol 是一种降低眼压的抗青光眼化合物。Aganepag ethanediol 是一种选择性 EP2 受体激动剂。
TMIH-0045 3-Hydroxy Repaglinide-d5

3-Hydroxy Repaglinide-d5 是 3-Hydroxy Repaglinide 的氘代化合物。
TMIH-0519 Selexipag Active Metabolite-d7

Selexipag Active Metabolite-d7 是 Selexipag Active Metabolite 的氘代化合物。Selexipag Active Metabolite 的 CAS 号为 475085-57-5。MRE269 是一种口服的长效前列环素受体激动剂前药,是 Selexipag 的活性代谢物,用于治疗肺动脉高压。
T126028 8-O-4-Hydroxycinnamoylharpagide

8-O-4-Hydroxycinnamoylharpagide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126028,CAS号为 133645-37-1。
T34644 Simenepag isopropyl

AGN210669,AGN-210669,AGN 210669

Simenepag isopropyl can be used for the treatment of Glaucoma, Ocular Hypertension.

化合物

Lusutrombopag
Cat.No: TQ0223
Synonym: 芦曲泊帕,鲁索曲波帕,S-888711,Mulpleta
Target: Thrombin, Thrombopoietin Receptor
Eltrombopag Olamine
Cat.No: T6825
Synonym: Promacta Olamine,Revolade,艾曲泊帕乙醇胺盐,Eltrombopag diethanolamine salt,SB497115,艾曲波帕乙醇胺盐,SB-497115GR
Target: Thrombin
Ralinepag
Cat.No: T4635
Synonym: APD811
Target: Others, Prostaglandin Receptor
Dapagliflozin ((2S)-1,2-propanediol, hydrate)
Cat.No: T4460
Synonym: BMS-512148 (2S)-1,2-propanediol, hydrate,达格列净 (2S)-1,2-丙二醇水合物,Dapagliflozin propanediol monohydrate
Target: SGLT
Dapagliflozin
Cat.No: T2389
Synonym: 达格列净,BMS-512148
Target: SGLT, HIF
Fedovapagon
Cat.No: T15273
Synonym: VA483,A106483
Target: Vasopressin Receptor
Avatrombopag
Cat.No: T7417
Synonym: YM477,AKR-501,1-[3-氯-5-[[[4-(4-氯-2-噻吩基)-5-(4-环己基-1-哌嗪基)-2-噻唑基]氨基]羰基]-2-吡啶基]-4-哌啶羧酸,E5501
Target: Thrombin, Thrombopoietin Receptor
Propagermanium
Cat.No: T20641
Synonym: Dipropanoic acid germanium sequioxide,SK-818,Ge 132,二羧乙基三氧化二锗,Ge132,SK 818,Ge-132
Target: Others
IPAG
Cat.No: T22870
Synonym:
Target: Opioid Receptor
Taprenepag
Cat.No: T3174
Synonym: CP-544326
Target: Prostaglandin Receptor
Evatanepag
Cat.No: T15259
Synonym: CP-533536 free acid,2-[3-[N-(4-叔丁基苄基)-N-(吡啶-3-基磺酰基)氨基甲基]苯氧基]乙酸
Target: Prostaglandin Receptor
Empagliflozin
Cat.No: T1766
Synonym: BI 10773,恩格列净
Target: SGLT
Opaganib
Cat.No: T6750
Synonym: ABC294640
Target: S1P Receptor
O-Desethyl Dapagliflozin
Cat.No: T67849
Synonym: Empagliflozin-4
Target: SGLT
Selexipag
Cat.No: T3216
Synonym: NS-304,ACT-293987,赛乐西帕,Uptravi
Target: Others, Prostaglandin Receptor
Repaglinide
Cat.No: T1088
Synonym: AG-EE 388 ZW,AG-EE 623ZW,瑞格列奈
Target: Potassium Channel, PPAR
Eltrombopag
Cat.No: T2562
Synonym: SB-497115,SB-497115-GR,艾曲波帕
Target: Thrombin
Pagibaximab
Cat.No: T76822
Synonym:
Target:
Dapagliflozin impurity
Cat.No: T10957
Synonym:
Target: Others
N-Methylsarpagine methosalt
Cat.No: T124813
Synonym:
Target:
Hetrombopag
Cat.No: T62864
Synonym:
Target:
8-cis-Cinnamoylharpagide
Cat.No: T126029
Synonym:
Target:
Avatrombopag maleate
Cat.No: T68888
Synonym:
Target:
Hetrombopag olamine
Cat.No: T27536
Synonym:
Target:
Sipagladenant
Cat.No: T61876
Synonym:
Target:
Evatanepag sodium
Cat.No: T69755
Synonym:
Target:
Pagoside
Cat.No: T124431
Synonym:
Target:
Spaglumic acid acetate
Cat.No: TQ0285L
Synonym: Isospaglumic acid acetate,Spaglumic acid acetate(3106-85-2 Free base)
Target: Endogenous Metabolite
(S)-Empagliflozin-d4
Cat.No: TMIH-0013
Synonym:
Target:
Repaglinide D5
Cat.No: T19548
Synonym: AG-EE 623ZW D5,瑞格列奈 D5
Target: Others
EMpagliflozin iMpurity 5
Cat.No: T64615
Synonym:
Target:
Opaganib HCl
Cat.No: T71301
Synonym:
Target:
Isospaglumate sodium
Cat.No: T25547
Synonym: Isospaglumate trisodium,Sodium isospaglumate
Target:
Rafutrombopag
Cat.No: T62865
Synonym:
Target:
Aganepag isopropyl
Cat.No: T29708
Synonym: AGN-210961,AGN 210961,AGN210961
Target:
Totrombopag choline
Cat.No: T68560
Synonym:
Target:
PeracetylEmpagliflozin
Cat.No: T67184
Synonym:
Target:
3'-Hydroxy Repaglinide
Cat.No: T13497
Synonym:
Target: Others
Aganepag
Cat.No: T14139
Synonym: AGN 210937
Target: Prostaglandin Receptor
Selexipag-d7
Cat.No: TMIH-0520
Synonym:
Target:
10× SDS-PAGE SDS Running Buffer
Cat.No: T64667
Synonym:
Target: Others
Avatrombopag hydrochloride
Cat.No: T40654
Synonym: AKR-501 hydrochloride,YM477hydrochloride,E5501hydrochloride
Target:
Taprenepag isopropyl
Cat.No: T16988
Synonym: PF-04217329
Target: Prostaglandin Receptor
Dapagliflozin-3-O-β-D-Glucuronide
Cat.No: T35619
Synonym:
Target:
Irpagratinib
Cat.No: T79850
Synonym: ABSK011
Target: FGFR
Aganepag ethanediol
Cat.No: T29707
Synonym: AGN-212409,AGN212409
Target:
3-Hydroxy Repaglinide-d5
Cat.No: TMIH-0045
Synonym:
Target:
Selexipag Active Metabolite-d7
Cat.No: TMIH-0519
Synonym:
Target:
8-O-4-Hydroxycinnamoylharpagide
Cat.No: T126028
Synonym:
Target:
Simenepag isopropyl
Cat.No: T34644
Synonym: AGN210669,AGN-210669,AGN 210669
Target:
Cat. No. Product Name Target Signaling Pathways
TQ0285 Spaglumic acid

异冬谷酸,N-Acetylaspartylglutamic acid,NAAG

Endogenous Metabolite Metabolism
Spaglumic acid (N-Acetylaspartylglutamic acid) 是一种神经肽,在脑中以毫摩尔浓度存在。
T6S2025 8-​O-​Acetylharpagide

8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide

Antibacterial Microbiology/Virology
8-O-Acetylharpagide 是从 Ajuga reptans 中分离得到的一种环烯醚萜,有抗肿瘤、抗病毒、抗菌和抗炎作用。它对豚鼠的离体平滑肌有生物活性。
T6S2024 Harpagide

Antibacterial; Parasite Microbiology/Virology
Harpagide 是从Scrophularia cryptophila 中分离出来的一种鸢尾糖苷,具有抗炎和抗寄生虫活性,对T.b. rhodesiense 具有体外锥虫杀虫活性,IC50为 21 μg/mL,它对L. donovani 的IC50值为 2.0 μg/mL。
T6S2023 Harpagoside

Others; COX; NO Synthase Immunology/Inflammation; Neuroscience; Others
Harpagoside 是从爪钩草中分离出来的一种天然产物,可抑制COX-1和COX-2活性,并抑制 NO 的产生。
T74202 Hispaglabridin A

Hispaglabridin A 是一种抗氧化剂,可有效防止脂质过氧化。
TN4034 Eupaglehnin C

Others Others
Eupaglehnin C shows cytotoxic (2.19 mg/ml) against HeLa-S3.
TN3162 6-Epi-8-O-acetylharpagide

Others Others
6-Epi-8-O-acetylharpagide是一种天然产物,属于玄参科玄参属,其产品编号为 TN3162,CAS号为 97169-44-3。6-Epi-8-O-acetylharpagide可用作对照参考。
TN1321 6'-​O-​Cinnamoyl harpagide

6'-O-Cinnamoylharpagide,(1S,4AS,5R,7S,7AR)-1,4A,5,6,7,7A-六氢-4A,5,7-三羟基-7-甲基环戊二烯并[C]吡喃-1-基 BETA-D-吡喃葡萄糖苷 6-[(2E)-3-苯基-2-丙烯酸酯],6'-O-肉桂酰基哈巴苷,6'-O-肉桂酰哈巴苷

Others Others
6'-O-Cinnamoylharpagide has anti-inflammatory activity.
T20617 Sarpagine

Raupin

Sarpagine is an alkaloid with the antihypertonic effect.
TN2953 3-Hydroxysarpagine

Topoisomerase DNA Damage/DNA Repair
3-Hydroxysarpagine是一种天然产物,属于夹竹桃科萝芙木属,其产品编号为 TN2953,CAS号为 857297-90-6。3-Hydroxysarpagine可用作对照参考。
TN3167 6-Epiharpagoside

Others Others
6-Epiharpagoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3167,CAS号为 1151862-67-7。
TN3166 6-Epiharpagide

Others Others
6-Epiharpagide is a natural product from Scrophularia ningpoensis Hemsl.
T2S1749 Protogracillin

原纤细薯蓣皂甙

Others Others
Protogracillin 是一种甾体皂苷,分离自Dioscorea zingiberensisWright (DZW) 中。从 DZW 根状茎中获得的甾体皂苷具有抗血栓作用,同时由降低心血管疾病风险的潜力。

天然产物

Spaglumic acid
Cat.No: TQ0285
Synonym: 异冬谷酸,N-Acetylaspartylglutamic acid,NAAG
Target: Endogenous Metabolite
8-​O-​Acetylharpagide
Cat.No: T6S2025
Synonym: 8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide
Target: Antibacterial
Harpagide
Cat.No: T6S2024
Synonym:
Target: Antibacterial, Parasite
Harpagoside
Cat.No: T6S2023
Synonym:
Target: Others, COX, NO Synthase
Hispaglabridin A
Cat.No: T74202
Synonym:
Target:
Eupaglehnin C
Cat.No: TN4034
Synonym:
Target: Others
6-Epi-8-O-acetylharpagide
Cat.No: TN3162
Synonym:
Target: Others
6'-​O-​Cinnamoyl harpagide
Cat.No: TN1321
Synonym: 6'-O-Cinnamoylharpagide,(1S,4AS,5R,7S,7AR)-1,4A,5,6,7,7A-六氢-4A,5,7-三羟基-7-甲基环戊二烯并[C]吡喃-1-基 BETA-D-吡喃葡萄糖苷 6-[(2E)-3-苯基-2-丙烯酸酯],6'-O-肉桂酰基哈巴苷,6'-O-肉桂酰哈巴苷
Target: Others
Sarpagine
Cat.No: T20617
Synonym: Raupin
Target:
3-Hydroxysarpagine
Cat.No: TN2953
Synonym:
Target: Topoisomerase
6-Epiharpagoside
Cat.No: TN3167
Synonym:
Target: Others
6-Epiharpagide
Cat.No: TN3166
Synonym:
Target: Others
Protogracillin
Cat.No: T2S1749
Synonym: 原纤细薯蓣皂甙
Target: Others
Cat. No. Product Name Species Expression System
TMPH-00293 PAG-1 Protein, Bovine, Recombinant (His)

Bovine E. coli
Appears to be proteolytically inactive. PAG-1 Protein, Bovine, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 40.7 kDa and the accession number is Q29432.
TMPH-00295 PAG-2 Protein, Bovine, Recombinant (His)

Bovine E. coli
PAG2 or a processed derivative of this molecule might represent a factor that binds the LH receptor. PAG-2 Protein, Bovine, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 43.6 kDa and the accession number is Q28057.
TMPH-00294 PAG-1 Protein, Bovine, Recombinant (His & SUMOstar)

Bovine P. pastoris (Yeast)
Appears to be proteolytically inactive. PAG-1 Protein, Bovine, Recombinant (His & SUMOstar) is expressed in yeast with N-6xHis-sumostar tag. The predicted molecular weight is 49.8 kDa and the accession number is Q29432.
TMPY-01276 Peroxiredoxin 1 Protein, Human, Recombinant (His)

PAGA,peroxiredoxin 1,NKEFA,MSP23,PAG,TDPX2...

Human E. coli
Peroxiredoxin 1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 22.9 kDa and the accession number is A0A384NPQ2.
TMPY-02372 Peroxiredoxin 1 Protein, Mouse, Recombinant (His)

PAG,OSF-3,OSF3,Paga,PRDX1,Tdpx2,PrxI,TDX2,...

Mouse E. coli
Peroxiredoxin 1 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 23.5 kDa and the accession number is P35700.
TMPH-03081 ACE2 Protein, Paguma larvata, Recombinant (hFc)

EC:3.4.17.23,Angiotensin-converting enzyme 2,ACE-related car...

Paguma larvata HEK293 Cells
ACE2 Protein, Paguma larvata, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 112.7 kDa and the accession number is Q56NL1.
TMPH-00743 PhoP Protein, E. coli, Recombinant (HEK293, His & Myc)

E. coli HEK293 Cells
Member of the two-component regulatory system PhoP/PhoQ involved in adaptation to low Mg(2+) environments and the control of acid resistance genes. In low periplasmic Mg(2+), PhoQ phosphorylates PhoP, resulting in the expression of PhoP-activated genes (PAG) and repression of PhoP-repressed genes (PRG). In high periplasmic Mg(2+), PhoQ dephosphorylates phospho-PhoP, resulting in the repression of PAG and may lead to expression of some PRG. Mediates magnesium influx to the cytosol by activation o...
TMPK-00556 BTN3A1 Protein, Cynomolgus, Recombinant (His & Avi)

BTN3.1,CD277,BTF5,BT3.1,BTN3A1

Cynomolgus HEK293 Cells
The three butyrophilin BTN3A molecules, BTN3A1, BTN3A2, and BTN3A3, are members of the B7/butyrophilin-like group of Ig superfamily receptors, which modulate the function of T cells. BTN3A1 controls activation of human Vγ9/Vδ2 T cells by direct or indirect presentation of self and nonself phosphoantigens (pAg). BTN3A1 Protein, Cynomolgus, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 26.5 kDa and the accession number is A0A33...
TMPK-00310 BTN3A1 Protein, Human, Recombinant (His & Avi), Biotinylated

CD277,BTN3A1,BTF5,BT3.1,BTN3.1

Human HEK293 Cells
The three butyrophilin BTN3A molecules, BTN3A1, BTN3A2, and BTN3A3, are members of the B7/butyrophilin-like group of Ig superfamily receptors, which modulate the function of T cells. BTN3A1 controls activation of human Vγ9/Vδ2 T cells by direct or indirect presentation of self and nonself phosphoantigens (pAg). BTN3A1 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 27.1 kDa and the accession number...
TMPK-00557 BTN3A1 Protein, Cynomolgus, Recombinant (His & Avi), Biotinylated

BTF5,BT3.1,BTN3.1,CD277,BTN3A1

Cynomolgus HEK293 Cells
The three butyrophilin BTN3A molecules, BTN3A1, BTN3A2, and BTN3A3, are members of the B7/butyrophilin-like group of Ig superfamily receptors, which modulate the function of T cells. BTN3A1 controls activation of human Vγ9/Vδ2 T cells by direct or indirect presentation of self and nonself phosphoantigens (pAg). BTN3A1 Protein, Cynomolgus, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 26.5 kDa and the accession n...

重组蛋白

PAG-1 Protein, Bovine, Recombinant (His)
Cat.No: TMPH-00293
Species: Bovine
Expression System: E. coli
PAG-2 Protein, Bovine, Recombinant (His)
Cat.No: TMPH-00295
Species: Bovine
Expression System: E. coli
PAG-1 Protein, Bovine, Recombinant (His & SUMOstar)
Cat.No: TMPH-00294
Species: Bovine
Expression System: P. pastoris (Yeast)
Peroxiredoxin 1 Protein, Human, Recombinant (His)
Cat.No: TMPY-01276
Species: Human
Expression System: E. coli
Peroxiredoxin 1 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02372
Species: Mouse
Expression System: E. coli
ACE2 Protein, Paguma larvata, Recombinant (hFc)
Cat.No: TMPH-03081
Species: Paguma larvata
Expression System: HEK293 Cells
PhoP Protein, E. coli, Recombinant (HEK293, His & Myc)
Cat.No: TMPH-00743
Species: E. coli
Expression System: HEK293 Cells
BTN3A1 Protein, Cynomolgus, Recombinant (His & Avi)
Cat.No: TMPK-00556
Species: Cynomolgus
Expression System: HEK293 Cells
BTN3A1 Protein, Human, Recombinant (His & Avi), Biotinylated
Cat.No: TMPK-00310
Species: Human
Expression System: HEK293 Cells
BTN3A1 Protein, Cynomolgus, Recombinant (His & Avi), Biotinylated
Cat.No: TMPK-00557
Species: Cynomolgus
Expression System: HEK293 Cells
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