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35

抑制剂 & 化合物

20

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T77439	Glembatumumab	Others	Others
	Glembatumumab 是一种靶向在人类乳腺癌和黑色素瘤中表达的 GPNMB 细胞外结构域的完全人类 IgG2 单克隆抗体。Glembatumumab 是 Glembatumumab vedotin 的裸抗，可用于研究抗体-活性分子偶联物（Glembatumumab vedotin ）。
T2711	Chembridge-5861528 TCS 5861528	TRP/TRPV Channel	Membrane transporter/Ion channel
	Chembridge-5861528 (TCS 5861528) 是有效的 TRPA1离子通道阻断剂。
T67988	Embeconazole R 120758,CS 758	Antifungal	Microbiology/Virology
	Embeconazole (R 120758) 是一种三唑类抗真菌剂。Embeconazole 对念珠菌、曲霉菌、新型隐球菌等临床重要真菌具有较强的体外活性。
T74178	Glembatumumab vedotin CR011-vcMMAE,CR 011 ADC,CDX-011	Microtubule Associated	Cytoskeletal Signaling
	Glembatumumab vedotin (CDX-011) 是一种抗体活性小分子偶联物，Glembatumumab vedotin 具有强大的抗癌作用，可用于研究三阴性乳腺癌(TNBC)。
T60092	CHEMBL1276927 N-[3-(1H-benzimidazol-2-yl)phenyl]-3-methylbenzamide,N-(3-(1H-benzo[d]imidazol-2-yl)phenyl)-3-methylbenzamide,N-[3-(1H-苯并[d]咪唑-2-基)苯基]-3-甲基苯甲酰胺	Antibacterial; Parasite	Microbiology/Virology
	CHEMBL1276927 (N-(3-(1H-benzo[d]imidazol-2-yl)phenyl)-3-methylbenzamide) 对肺炎衣原体和多诺瓦尼利什曼原虫具有抗菌和抗寄生虫活性。
TP1286	Carcinoembryonic Antigen CEA 癌胚抗原	Others	Others
	Carcinoembryonic Antigen CEA 是一种广谱性肿瘤标志物，是大肠癌组织产生的一种糖蛋白，作为抗原可引起患者的免疫反应。
TP2417	Tidembersat	Others	Others
	Tidembersat 是一种小分子化合物，可用于治疗和/或预防退行性疾病，如亨廷顿舞蹈病、精神分裂症、神经。
T9908	Pembrolizumab	PD-1/PD-L1	Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation
	Pembrolizumab 是一种抑制 PD-1 受体的人源化单克隆抗体，是一个 HER2 二聚化抑制剂类，它会削弱 HER2 与 HER 家族其他成员结合的能力。
T2429	Olverembatinib dimesylate GZD824 Dimesylate,HQP1351	Bcr-Abl	Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	Olverembatinib dimesylate (GZD824 Dimesylate) 是一种高效的、口服具有活性的pan-Bcr-Abl 抑制剂，具有抗肿瘤活性。它能广泛而有效地抑制突变型 Bcr-Abl。它对天然的 Bcr-Abl 和 Bcr-AblT315I 作用的IC50值分别为 0.34 nM 和 0.68 nM。
T28750	Sembragiline RG-1577,EVT-302,RO-4602522,RO4602522,RG1577,EVT302	MAO	Metabolism; Neuroscience
	Sembragiline (EVT-302) 是一种具有选择性的 MAO-B 抑制剂，可用于研究阿尔茨海默病（AD）。
T60093	CHEMBL1380345 N,N'-(Ethane-1,2-diyl)bis(3-methylbenzenesulfonamide)	Antibacterial	Microbiology/Virology
	CHEMBL1380345 对金黄色葡萄球菌、蜡状芽孢杆菌和大肠杆菌具有抗菌活性，pMIC 值分别为 3.64、3.56 和 3.70。
T8598	CHEMBL241987 2-PHENYL-2,5-DIHYDRO-4H-PYRAZOLO[3,4-C]QUINOLIN-4-ONE	Adenosine Receptor	GPCR/G Protein; Neuroscience
	CHEMBL241987 靶向腺苷受体 A3（人）。
T27112	Cytembena	DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	Cytembena 是一种细胞抑制剂，是一种致癌化合物，可之间纤维腺瘤发生的几率。Cytembena 广泛地抑制 DNA 的生物合成。
T3071	Olverembatinib GZD 824	Bcr-Abl	Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	Olverembatinib (GZD 824) 是一种高效的、口服具有活性的pan-Bcr-Abl 抑制剂，具有抗肿瘤活性。它能广泛而有效地抑制突变型 Bcr-Abl。它对天然的 Bcr-Abl 和 Bcr-AblT315I 作用的IC50值分别为 0.34 nM 和 0.68 nM。
T131083	Cembratetraene-16,2:19,6-diolide
	Cembratetraene-16,2:19,6-diolide 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T131083。
T69405	Metformin embonate
	Metformin embonate is an AMP-activated protein kinase (AMPK) activator that improves glycemic control by improving insulin sensitivity and decreasing intestinal absorption of glucose.
T81824	Membrane-Permeable Sequence, MPS
	Membrane-Permeable Sequence（MPS）是一种CPP，常用于研究跨膜机制。
T70261	Amitriptyline Embonate
	Amitriptyline Embonate is an inhibitor of the re-uptake of norepinephrine and serotonin, thereby inhibiting N-methyl-D-aspartate (NMDA) receptors.
T124625	α-Cembrenediol
	α-Cembrenediol 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T124625。
T28749	SEMBL
	SEMBL, a novel inhibitor of DNA binding of NF-kappaB component p65 in vitro, inhibits NF-kappaB and cellular invasion in ovarian carcinoma ES-2 cells.
T124052	Calophymembranside B
	Calophymembranside B 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T124052，CAS号为 869285-60-9。
T82476	Embramine hydrochloride
	Embramine (hydrochloride) 为具有抗组胺及抗胆碱能特性的单乙醇胺类化合物。
T68384	SCHEMBL12616233
	SCHEMBL12616233 is a novel inhibitor of SARS-CoV-2 main protease (MPro).
T70054	Novembichin
	Novembichin is a nitrogen mustard agent that crosslinks with DNA, causing inhibition of DNA synthesis.
T80209	Human membrane-bound PD-L1 polypeptide	PD-1/PD-L1	Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation
	Human membrane-bound PD-L1 polypeptide 作为抗原，可诱导生成相应的PD-L1抗体。
T124967	D7-Mesembrenone
	D7-Mesembrenone 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T124967，CAS号为 35714-44-4。
TP2198	Platelet Membrane Glycoprotein IIB Peptide (296-306)	Others	Others
	GPllb is composed of a 125 Kd heavy chain that is disulfide-linked to a 23 Kd light chain. Hydropathicity analysis of the cDNA sequence indicates that GPllb is anchored to the platelet through a single transmembrane domain located within 20 amino acids of
T31619	Embusartan UNII-4MY73645XA,Bay 10-6734
	Embusartan (BAY 10-6734) is a potent, orally active angiotensin II receptor antagonist used as an antihypertensive agent.
T131462	Embelin Dimethyl ether
	Embelin Dimethyl ether 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T131462。
T11180	Embramine	Others	Others
	Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.
T35434	β-Cembrenediol
	β-Cembrenediol (β-CBT) is a natural product from tobacco plants that is found in cigarette smoke condensate. β-CBT inhibits induction of the early antigen of Epstein-Barr virus (EA-EBV) by 12-O-tetradecanoylphorbol-13-acetate (TPA) in vitro (IC50 = 21.9 μM). It inhibits tumor promoting effects of TPA on 7,12-demethylbenz[a]anthracene-induced papilloma formation in vivo. β-CBT is also released into soil by flue-cured tobacco plants and exerts autotoxicity as well as phytotoxic activity against L....
T71902	CHEMBL94431
	CHEMBL94431 is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase.
T31373	Dembrexine HCl Dembroxol
	Dembrexine is a bioactive agent.
T76916	Bafisontamab
	Bafisontamab (EMB-01) 是一种靶向EGFR 和cMET 的双特异性抗体，具有抗肿瘤活性。
T37880	OPC-167832
	OPC-167832 is a potent and orally active dprE1 Inhibitor with an IC50 of 0.258 μM. OPC-167832 has antituberculosis activity and can be used for the research of tuberculosis caused by Mycobacterium tuberculosis[1]. OPC-167832 exhibits very low MICs against laboratory strains of M. tuberculosis H37Rv (MIC: 0.0005 μg/ml) and Kurono (MIC: 0.0005 μg/ml) and strains with monoresistance to rifampin (RIF), isoniazid (INH), ethambutol (EMB), streptomycin (STR), and pyrazinamide (PZA) (MIC: 0.00024-0.001 ...

化合物

Cat.No: T77439

Target: Others

Chembridge-5861528

Cat.No: T2711

Synonym: TCS 5861528

Target: TRP/TRPV Channel

Cat.No: T67988

Synonym: R 120758,CS 758

Target: Antifungal

Glembatumumab vedotin

Cat.No: T74178

Synonym: CR011-vcMMAE,CR 011 ADC,CDX-011

Target: Microtubule Associated

Cat.No: T60092

Synonym: N-[3-(1H-benzimidazol-2-yl)phenyl]-3-methylbenzamide,N-(3-(1H-benzo[d]imidazol-2-yl)phenyl)-3-methylbenzamide,N-[3-(1H-苯并[d]咪唑-2-基)苯基]-3-甲基苯甲酰胺

Target: Antibacterial, Parasite

Carcinoembryonic Antigen CEA

Cat.No: TP1286

Synonym: 癌胚抗原

Target: Others

Cat.No: TP2417

Target: Others

Cat.No: T9908

Target: PD-1/PD-L1

Olverembatinib dimesylate

Cat.No: T2429

Synonym: GZD824 Dimesylate,HQP1351

Target: Bcr-Abl

Cat.No: T28750

Synonym: RG-1577,EVT-302,RO-4602522,RO4602522,RG1577,EVT302

Target: MAO

Cat.No: T60093

Synonym: N,N'-(Ethane-1,2-diyl)bis(3-methylbenzenesulfonamide)

Target: Antibacterial

Cat.No: T8598

Synonym: 2-PHENYL-2,5-DIHYDRO-4H-PYRAZOLO[3,4-C]QUINOLIN-4-ONE

Target: Adenosine Receptor

Cat.No: T27112

Target: DNA/RNA Synthesis

Cat.No: T3071

Synonym: GZD 824

Target: Bcr-Abl

Cembratetraene-16,2:19,6-diolide

Cat.No: T131083

Metformin embonate

Cat.No: T69405

Membrane-Permeable Sequence, MPS

Cat.No: T81824

Amitriptyline Embonate

Cat.No: T70261

α-Cembrenediol

Cat.No: T124625

Cat.No: T28749

Calophymembranside B

Cat.No: T124052

Embramine hydrochloride

Cat.No: T82476

SCHEMBL12616233

Cat.No: T68384

Cat.No: T70054

Human membrane-bound PD-L1 polypeptide

Cat.No: T80209

Target: PD-1/PD-L1

D7-Mesembrenone

Cat.No: T124967

Platelet Membrane Glycoprotein IIB Peptide (296-306)

Cat.No: TP2198

Target: Others

Cat.No: T31619

Synonym: UNII-4MY73645XA,Bay 10-6734

Embelin Dimethyl ether

Cat.No: T131462

Cat.No: T11180

Target: Others

β-Cembrenediol

Cat.No: T35434

Cat.No: T71902

Cat.No: T31373

Synonym: Dembroxol

Cat.No: T76916

Cat.No: T37880

Cat. No.	Product Name	Target	Signaling Pathways
T0810	Ethambutol dihydrochloride Ethambutol 2HCl,盐酸乙胺丁醇,Emb dihydrochloride,CL40881	Antibacterial; Antibiotic; Antifungal	Microbiology/Virology
	Ethambutol dihydrochloride (CL40881) 能抗分枝杆菌，可抑制阿拉伯糖基转移酶活性来阻止细胞壁形成。
T2S1682	Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside Pinocembrin 7-O-(3''-galloyl-4'',6''-(S)-hexahydroxydiphenoyl)-beta-D-glucose,pinocembrin-7-o-3-o-galloyl-4-6-hexahydroxydiphenoyl-beta-d-glucoside	Amylase	Metabolism
	Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside 可抑制 α-淀粉酶活性，IC50值为0.03 umol/ml。
T2992	Pinocembrin 乔松素,5,7-Dihydroxyflavanone,Dihydrochrysin,Galangin flavanone,松属素	NF-κB; Reactive Oxygen Species; Antibacterial; Autophagy	Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
	Pinocembrin (5,7-Dihydroxyflavanone) 是从蜂胶中得到的黄酮类物质，是一种竞争性组氨酸脱羧酶抑制剂，也是抗过敏剂，具有抗氧化、抗菌、抗炎的作用。
T13514	5-MethoxyPinocembroside	Others	Others
	5-MethoxyPinocembroside 是一种黄酮类天然产物，存在于辣木 Moringa oleifera 的叶子中。
TN2078	Pinocembrin chalcone 2',4',6'-Trihydroxychalcone,Pinocembrinchalcone	Calcium Channel; Tyrosinase; Antibacterial; Antifection	Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Proteases/Proteasome
	Pinocembrin chalcone 是一种具有抗诱变作用的酪氨酸酶抑制剂。 Pinocembrin 查尔酮可用于预防胃溃疡的研究。
T5710	Pinocembrin-7-O-β-D-glucopyranoside Pinocembrin 7-O-beta-D-glucoside,乔松素7-O-Β-D葡萄糖苷,乔松苷	Others	Others
	Pinocembrin-7-O-β-D-glucopyranoside (Pinocembrin 7-O-beta-D-glucoside) 是黄酮类化合物，能够提高脂质过氧化。
TN4221	Homoembelin 2,5-dihydroxy-3-nonyl-1,4-benzoquinone	Antibacterial	Microbiology/Virology
	Homoembelin (2,5-dihydroxy-3-nonyl-1,4-benzoquinone) 是来自 E. ribes 和 C. monocarpus 的色素，具有抗菌效果，可用于耐多药细菌感染的研究。
T6485	Embelin NSC 91874,恩贝酸,恩贝酸/恩贝灵,Emberine,Embelic acid	Apoptosis; NF-κB; Lipoxygenase; IAP; Prostaglandin Receptor; Autophagy	Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; Metabolism; NF-κB
	Embelin (Embelic acid) 是从日本 Ardisia 草药中分离出来的一种非肽类细胞渗透性XIAP 抑制剂，诱导口腔鳞癌细胞自噬和凋亡。它阻断 NF-kappaB 信号通路，从而抑制 NF-kappaB 调节的抗凋亡和转移基因产物。在高水平 XIAP 的前列腺癌细胞中抑制细胞生长，诱导凋亡，并激活 caspase-9。
TN2077	(+/-)-Pinocembrin NSC 43318,(±)-5,7-Dihydroxyflavanone	GPR; Others	Endocrinology/Hormones; GPCR/G Protein; Others
	(+/-)-Pinocembrin (NSC-43318) 是一种来自腋松的天然产物，它是一种 GPR120 配体，能促进 HaCaT 细胞系的伤口愈合。
TN5509	(2S)-Pinocembrin 7-O-[2''-O-(5'''-O-trans-cinnamoyl)-β-D-apiofuranosyl]-β-D-glucoside (2S)-Pinocembrin 7-O-[cinnamoyl(1→5)-β-D-apiosyl(1→2)]-β-D-glucoside
	(2S)-Pinocembrin 7-O-[2''-O-(5'''-O-trans-cinnamoyl)-β-D-apiofuranosyl]-β-D-glucoside 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN5509，CAS号为 773899-29-9。
T77289	5-O-Methylembelin
	5-O-Methylembelin 是一种天然异香豆素，可抑制PCSK9、低密度脂蛋白受体 (IDOL) 和甾醇调节元件结合蛋白 2 (SREBP2) mRNA 的表达。
TN6319	Embinin
	Embinin 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN6319，CAS号为 52589-13-6。
T28019	(-)-Mesembrine Mesembrin,Mesembrine,Mesembranone
	Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).
T83379	2-Hydroxypinocembrin
	2-Hydroxypinocembrin 是一种具有 C-糖基转移酶活性的2-羟基黄烷酮类黄酮底物。
TN4792	Pinocembrin diacetate	Others	Others
	Pinocembrin diacetate 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN4792，CAS号为 111441-88-4。
T73857	Mesembrine
	Mesembrine ((+)-Mesembrine) 一种主要的生物碱，具有芳基八氢吲哚骨架。Mesembrine 是一种5-HT 转运蛋白抑制剂，Ki 为 1.4 nM。Mesembrine 还抑制磷酸二酯酶 4B (PDE4B)，IC50为 7.8 μM。
T72856	(+)-Cembrene A
	(+)-Cembrene A 是一种α-glucosidase 抑制剂，IC50为 30.31 μM。(+)-Cembrene A 对人正常肝细胞 (LO2) 无毒性。
TN4791	Pinocembrin 7-acetate	Others	Others
	Pinocembrin 7-acetate has antitumor activity.
T72742	(-)-Pinocembrin (-)-乔松素
	(-)-Pinocembrin 对 H37Ra 结核分枝杆菌展示了抗菌活性，无论是休眠还是活跃期，其 IC50 值分别为1.11 mg/mL 和 1.21 mg/mL。作为一种抗增殖剂，(-)-Pinocembrin 对于 THP-1、A549、Panc-1、HeLa 和 MCF7 细胞系，IC50 值范围为 1.88 至 11.00 mg/mL。
T19772	Mesembrenone (+)-Mesembrenone
	Mesembrenone is a selective the serotonin transporter (SERT) inhibitor. Mesembrenone is the main alkaloid of Sceletium tortuosum.

天然产物

Ethambutol dihydrochloride

Cat.No: T0810

Synonym: Ethambutol 2HCl,盐酸乙胺丁醇,Emb dihydrochloride,CL40881

Target: Antibacterial, Antibiotic, Antifungal

Pinocembrin 7-O-[3''-O-galloyl-4'',6''-hexahydroxydiphenoyl]-β-D-glucoside

Cat.No: T2S1682

Synonym: Pinocembrin 7-O-(3''-galloyl-4'',6''-(S)-hexahydroxydiphenoyl)-beta-D-glucose,pinocembrin-7-o-3-o-galloyl-4-6-hexahydroxydiphenoyl-beta-d-glucoside

Target: Amylase

Cat.No: T2992

Synonym: 乔松素,5,7-Dihydroxyflavanone,Dihydrochrysin,Galangin flavanone,松属素

Target: NF-κB, Reactive Oxygen Species, Antibacterial, Autophagy

5-MethoxyPinocembroside

Cat.No: T13514

Target: Others

Pinocembrin chalcone

Cat.No: TN2078

Synonym: 2',4',6'-Trihydroxychalcone,Pinocembrinchalcone

Target: Calcium Channel, Tyrosinase, Antibacterial, Antifection

Pinocembrin-7-O-β-D-glucopyranoside

Cat.No: T5710

Synonym: Pinocembrin 7-O-beta-D-glucoside,乔松素7-O-Β-D葡萄糖苷,乔松苷

Target: Others

Cat.No: TN4221

Synonym: 2,5-dihydroxy-3-nonyl-1,4-benzoquinone

Target: Antibacterial

Cat.No: T6485

Synonym: NSC 91874,恩贝酸,恩贝酸/恩贝灵,Emberine,Embelic acid

Target: Apoptosis, NF-κB, Lipoxygenase, IAP, Prostaglandin Receptor, Autophagy

(+/-)-Pinocembrin

Cat.No: TN2077

Synonym: NSC 43318,(±)-5,7-Dihydroxyflavanone

Target: GPR, Others

(2S)-Pinocembrin 7-O-[2''-O-(5'''-O-trans-cinnamoyl)-β-D-apiofuranosyl]-β-D-glucoside

Cat.No: TN5509

Synonym: (2S)-Pinocembrin 7-O-[cinnamoyl(1→5)-β-D-apiosyl(1→2)]-β-D-glucoside

5-O-Methylembelin

Cat.No: T77289

Cat.No: TN6319

Cat.No: T28019

Synonym: Mesembrin,Mesembrine,Mesembranone

2-Hydroxypinocembrin

Cat.No: T83379

Pinocembrin diacetate

Cat.No: TN4792

Target: Others

Cat.No: T73857

Cat.No: T72856

Pinocembrin 7-acetate

Cat.No: TN4791

Target: Others

(-)-Pinocembrin

Cat.No: T72742

Synonym: (-)-乔松素

Cat.No: T19772

Synonym: (+)-Mesembrenone

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