购物车

搜索结果

Search Results for " dlk "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T11056 DLK-IN-1

DNA Alkylation DNA Damage/DNA Repair
DLK-IN-1 is a selective oral active inhibitor of bisleucine zipper kinase (DLK, MAP3K12) with Ki of 3 nM. DLK-IN-1 is active in the Alzheimer's disease model, retains excellent CNS permeability, and after multiple days of administration, its concentration
T3707 GNE-3511

GNE3511

DNA Alkylation; MAPK DNA Damage/DNA Repair; MAPK
GNE-3511是双亮氨酸拉链激酶 (DLK)抑制剂(Ki:0.5 nM)。
T6057 URMC-099

ROCK; MLK; VEGFR; SGK; DNA Alkylation; Trk receptor; c-Met/HGFR; LRRK2; MEK; IGF-1R; Syk; Bcr-Abl; CDK; Src; Aurora Kinase; Autophagy Angiogenesis; Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; MAPK; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
URMC-099 是一种具有优异的血脑屏障穿透性的,可口服的混合谱系激酶 3 抑制剂,IC50为14 nM。
T73457 DN-1289

DNA Alkylation DNA Damage/DNA Repair
DN-1289 是一种可口服可通过血脑屏障且具有选择性高效性的抑制剂,对双亮氨酸拉链激酶 (DLK)的 IC50 值为17 nM,对 亮氨酸拉链轴承激酶 (LZK)的 IC50 值为 40 nM。DN-1289 对小鼠模型中视神经挤压 (ONC) 诱导的 p-c-Jun 有显著的抑制作用。
T11440 GNE-8505

DNA Alkylation DNA Damage/DNA Repair
GNE-8505 is an orally available inhibitor of Dual leucine zipper kinase (DLK).
T79303 IACS-52825

IACS-52825是一种选择性DLK抑制剂,具有1.3 nM的Kd值,适用于研究化疗引起的周围神经病变。

化合物

DLK-IN-1
Cat.No: T11056
Synonym:
Target: DNA Alkylation
GNE-3511
Cat.No: T3707
Synonym: GNE3511
Target: DNA Alkylation, MAPK
URMC-099
Cat.No: T6057
Synonym:
Target: ROCK, MLK, VEGFR, SGK, DNA Alkylation, Trk receptor, c-Met/HGFR, LRRK2, MEK, IGF-1R, Syk, Bcr-Abl, CDK, Src, Aurora Kinase, Autophagy
DN-1289
Cat.No: T73457
Synonym:
Target: DNA Alkylation
GNE-8505
Cat.No: T11440
Synonym:
Target: DNA Alkylation
IACS-52825
Cat.No: T79303
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼