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5

抑制剂 & 化合物

44

天然产物

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Cat. No. Product Name Target Signaling Pathways
T124040 Bijaponicaxanthone C

Bijaponicaxanthone C 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124040。
T25278 Cucumarioside A2-2

Cucumarioside A2-2 is a triterpene glycoside isolated from the Far-Eastern sea cucumber Cucumaria japonica, that exhibits antitumor activity.
T34320 Rhodexin A

Rhodexin A is a cardetonic agent of the plant Rhodea japonica.
T33335 Methyl adenophorate

Methyl adenophorate is a triterpenoid of Adenophora triphylla var. japonica roots.
T35686 3-Acetyl Betulinaldehyde

3-Acetyl betulinaldehyde is a triterpene and derivative of the cholesterol biosynthesis inhibitor betulin that has been found inA. japonica.1It is an intermediate in the synthesis of 3-acetylbetulinic acid, as well as various lupine and germanicane triterpenes and saponins with anticancer activity.2 1.Tung, N.H., Kwon, H.-J., Kim, J.-H., et al.An anti-influenza component of the bark of Alnus japonicaArch. Pharm. Res.33(3)363-367(2010) 2.Thibeault, D., Gauthier, C., Legault, J., et al.Synthesis a...

化合物

Bijaponicaxanthone C
Cat.No: T124040
Synonym:
Target:
Cucumarioside A2-2
Cat.No: T25278
Synonym:
Target:
Rhodexin A
Cat.No: T34320
Synonym:
Target:
Methyl adenophorate
Cat.No: T33335
Synonym:
Target:
3-Acetyl Betulinaldehyde
Cat.No: T35686
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN4495 Maoyerabdosin

Others Others
Maoyerabdosin 是一种提取自粳稻叶的化合物。
T5S0055 Chelidonine

Helidonine,Khelidonin,白屈菜碱,Stylophorin

Apoptosis; Others; Influenza Virus Apoptosis; Microbiology/Virology; Others
Chelidonine (Stylophorin) 是白屈菜中的一种异喹啉生物碱,有抗肿瘤和抗病毒作用。它可导致细胞周期 G2/M 停滞,诱导 caspase 依赖和非依赖性的细胞凋亡。
T3S1534 Secoxyloganin

断氧化马钱苷,幼枝含断氧化马钱子甙,金银花

Anti-infection Microbiology/Virology
Secoxyloganin 是从Lonicera japonicaThunb 提取得到,能够抑制血流量减少,具有抗过敏活性。
TN6774 Emodin 6-O-β-D-glucoside

大黄素-6-O-β-D-葡萄糖苷,Glucoemodin

Others Others
Emodin 6-O-β-D-glucoside (Glucoemodin) 是一种从 Reynoutria japonica 中提取的活性化合物。它具有显著的抗炎和屏障保护活性,可用于研究动脉粥样硬化及糖尿病并发症。
T10117 3'-​O-​Acetylhamaudol

Others Others
3'-O-Acetylhamaudol 是提取于 Angelica japonica 根部,能够抗血管生成和激活肠上皮淋巴细胞,具有抗肿瘤活性。
TN2241 Styraxlignolide F

Others Others
Styraxlignolide F 是一种分离自 Styrax japonica 天然产物。
TN6726 methyl chlorogenate

NF-κB NF-κB
methyl chlorogenate 是从 Eriobotrya japonica 中分离得到的,它是 NFkappaB 的抑制剂。
TN1129 Protostemotinine

Others Others
Protostemotinine 是一种分离自 Stemona sessilifolia 的生物碱。
T13768 (+)-Medicarpin

Estrogen/progestogen Receptor Endocrinology/Hormones
(+)-Medicarpin, a pterocarpan, is an isoflavonoid compound derived from multiple medicinal plant species such as Sophora japonica, Zollernia paraensis, Platymiscium yucatamun, Machaerium aristulatum, and Platymiscium floribundum. It exhibits potent inhibition of osteoclastogenesis and facilitates bone healing and increased bone mass through osteoblast differentiation, which is mediated by the estrogen receptor (ER) β.
TN2079 (-)-Pinoresinol

Others; TNF; NF-κB; COX Apoptosis; Immunology/Inflammation; Neuroscience; NF-κB; Others
(-)-Pinoresinol 是从 Serissa japonica (Thunb.) Thunb 的全植物中分离得到的天然产物。
TN7230 Butyl chlorogenate

Others Others
Butylchlorogenate 是一种忍冬、Urceola rosea 中分离出的天然化合物。
TN3689 Comanthoside A

Comanthosid A

Others Others
Comanthoside A (Comanthosid A) 是一种可从 Comanthosphace japonica 中分离的天然黄酮苷。Comanthoside A 也 是合成 Linaroside和 Comanthoside B 的关键中间体。
TQ0309 Glaucocalyxin B

蓝萼乙素 B,蓝萼乙素

Autophagy Autophagy
Glaucocalyxin B 是从碎米桠中分离出来的二萜类天然产物,可降低 HL-60 细胞的生长,IC50为 5.86 μM,具有抗癌和抗肿瘤活性。
T4S0675 Polygalasaponin V

瓜子金皂苷V,瓜子金皂苷 V

Others Others
Polygalasaponin V 是一种三萜皂苷,分离自Polygala japonica 的地上部分。其中Polygala japonica 是民间的药用植物,在中国南方用作祛痰、抗菌、抗炎、抗抑郁药。
TN6967 (R)-Isomucronulatol

(-)-Isomucronulatol,2H-1-Benzopyran-7-ol

Apoptosis Apoptosis
(R)-Isomucronulatol (2H-1-Benzopyran-7-ol) 是一种可从黄芪、刺槐、虎杖和甘草叶片中提取得到的类黄酮,抑制BMSCs 在TNF-α微环境中的增殖和凋亡。(R)-Isomucronulatol 具有潜在的抗炎活性。
TN7225 2'-Hydroxy-3,4-dimethoxychalcone

Antioxidant; Parasite Microbiology/Virology; oxidation-reduction
2'-Hydroxy-3,4-dimethoxychalcone 是从槐树根分离除的查耳酮化合物,具有抗氧化活性,抑制了多诺瓦尼乳杆菌寄生虫 EC 的细胞内存活50值介于 0.39 和 0.41 μg/mL 之间,可用于研究糖尿病,治疗血吸虫病、疟疾和其它感染。
T6S2252 Sweroside

Others Others
Sweroside 是分离自Lonicera japonica 中,具有细胞保护、抗骨质疏松和保护肝脏活性。
TN4833 Prostephanaberrine

Others Others
Prostephanaberrine is a natural product from Stephania japonica.
TN1435 Bayogenin 3-O-β-D-glucopyranoside

Bayogenin 3-O-beta-D-glucopyranoside,贝萼皂苷元-3- O-Β-D-吡喃葡萄糖苷

Others Others
Bayogenin 3-O-beta-D-glucopyranoside is a natural product from Polygala japonica Houtt.
TN5603 Spiratisanin B

Spiratisanin B is a natural product from Spiraea japonica.
T26029 Rabdosin A

Rabdosin A is a diterpenoid antitumor constituent from Rabdosia japonica.
TN5402 (-)-Pinoresinol 4-O-glucoside

(-)-松脂素 4-O-葡萄糖苷,金银花

(-)-Pinoresinol 4-O-glucoside is a natural product from Lonicera japonica THUNB.
T30156 Asebotoxin III

Asebotoxin III is a diterpenoid obtained from the leaves of Asebi, Pieris japonica.
T81429 Polygalasaponin LII

Polygalasaponin LII,一种三萜皂苷,由Polygala japonica Houtt的根中提取。
TN2218 Sophorabioside

Others Others
Sophorabioside is a natural product from Sophora japonica.
TN5048 Spiratisanin C

Others Others
Spiratisanin C is a natural product from Spiraea japonica.
T19093 2,3,4,5-Tetracaffeoyl-D-Glucaric acid

Others Others
2,3,4,5-Tetracaffeoyl-D-Glucaric acid, a derivative of caffeoyl-D-glucaric acid, has been isolated from Inula japonica Thunb.
TN5003 Sessilifoline A

Others Others
Sessilifoline A is a natural product from Stemona japonica.
TN3908 (E)-Aldosecologanin

金银花

Others Others
(E)-Aldosecologanin is a natural product from Lonicera japonica.
TN5047 Spiratisanin A

Others Others
Spiratisanin A is a natural product from Spiraea japonica.
TN4507 Matairesinoside

Others Others
Matairesinoside is a natural product from Styrax japonica.
TMA0537 4-Oxododecanedioic acid

Others Others
4-Oxododecanedioic acid is a natural product from Coniogramme japonica
TN1616 Epivogeloside

金银花,表断马钱子甙半缩醛内酯

Others Others
Epivogeloside is a product from Lonicera japonica.
TN5276 (Z)-Aldosecologanin (Centauroside)

金银花

Others Others
(Z)-Aldosecologanin is a natural product from Lonicera japonica.
TN4983 Secoxyloganin methyl ester

金银花

Others Others
Secoxyloganin methyl ester is a natural product from Lonicera japonica.
T80005 n-Butyl α-D-fructofuranoside

JNK MAPK
n-Butyl α-D-fructofuranoside,分离自Ulmus davidiana var. japonica的根皮,通过激活JNK促进Nrf2活性,并表现出抗炎效应。
T82312 Glaucocalyxin D

Glaucocalyxin D为ent-kauranoid类二萜化合物,源于香茶菜。其对多种人类肿瘤细胞系显示出细胞毒作用,应用于癌症研究。
TN3210 7,3'-Di-O-methylorobol

Others Others
7,3'-Di-O-methylorobol is a natural product from Sophora japonica L.
TN4038 Eupatolide

TNF; NOS; NF-κB; ROS; MAPK; Akt; COX; DNA/RNA Synthesis; Nrf2; PDGFR; NO Synthase; Prostaglandin Receptor; Autophagy Angiogenesis; Apoptosis; Autophagy; Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; MAPK; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Eupatolide 是从 Inula japonica 的花中分离出来的,具有抗炎活性。 Eupatolide 可用于研究乳腺癌细胞对 TRAIL 的耐药性。
TN4810 Platyphyllonol

Influenza Virus Microbiology/Virology
Platyphyllonol 来自赤杨树皮,对 KBNP-0028 (H9N2) 禽流感病毒表现出中等活性。
TN5484 Cinchonain Ib

Others Others
Cinchonain Ib 是从枇杷叶中分离出来的。 Cinchonain Ib 具有促胰岛素作用,可用于管理 2 型糖尿病的研究。
T83364 3-Acetyl-11-keto-ursolic acid

3-Acetyl-11-keto-ursolic acid (Compound 18)为Eriobotrya japonica叶中提取的三萜类化合物,其抑制11b-羟基类固醇脱氢酶1 (11b-HSD1) 的特性使其在抗糖尿病研究中具有应用潜力。
T0772 Troxerutin

曲克芦丁,Trihydroxyethylrutin,维脑路通

NOD-like Receptor (NLR) Immunology/Inflammation
Troxerutin (Trihydroxyethylrutin) 是一种天然生物类黄酮芦丁的三羟乙基化衍生物,也被称为维生素 P4,可抑制活性氧的产生并抑制 ER 应激介导的NOD 活化。
T75555 (6E,12E)-Tetradecadiene-8,10-diyne-1,3-diol

'(6E,12E)-Tetradecadiene-8,10-diyne-1,3-diol' 是从白术根中分离出的一种具有抗菌活性的化合物,对 MRSA 显示出 4 - 32 μg/mL 的最小抑菌浓度(MIC),表现出对抗性细菌感染研究的潜力。

天然产物

Maoyerabdosin
Cat.No: TN4495
Synonym:
Target: Others
Chelidonine
Cat.No: T5S0055
Synonym: Helidonine,Khelidonin,白屈菜碱,Stylophorin
Target: Apoptosis, Others, Influenza Virus
Secoxyloganin
Cat.No: T3S1534
Synonym: 断氧化马钱苷,幼枝含断氧化马钱子甙,金银花
Target: Anti-infection
Emodin 6-O-β-D-glucoside
Cat.No: TN6774
Synonym: 大黄素-6-O-β-D-葡萄糖苷,Glucoemodin
Target: Others
3'-​O-​Acetylhamaudol
Cat.No: T10117
Synonym:
Target: Others
Styraxlignolide F
Cat.No: TN2241
Synonym:
Target: Others
methyl chlorogenate
Cat.No: TN6726
Synonym:
Target: NF-κB
Protostemotinine
Cat.No: TN1129
Synonym:
Target: Others
(+)-Medicarpin
Cat.No: T13768
Synonym:
Target: Estrogen/progestogen Receptor
(-)-Pinoresinol
Cat.No: TN2079
Synonym:
Target: Others, TNF, NF-κB, COX
Butyl chlorogenate
Cat.No: TN7230
Synonym:
Target: Others
Comanthoside A
Cat.No: TN3689
Synonym: Comanthosid A
Target: Others
Glaucocalyxin B
Cat.No: TQ0309
Synonym: 蓝萼乙素 B,蓝萼乙素
Target: Autophagy
Polygalasaponin V
Cat.No: T4S0675
Synonym: 瓜子金皂苷V,瓜子金皂苷 V
Target: Others
(R)-Isomucronulatol
Cat.No: TN6967
Synonym: (-)-Isomucronulatol,2H-1-Benzopyran-7-ol
Target: Apoptosis
2'-Hydroxy-3,4-dimethoxychalcone
Cat.No: TN7225
Synonym:
Target: Antioxidant, Parasite
Sweroside
Cat.No: T6S2252
Synonym:
Target: Others
Prostephanaberrine
Cat.No: TN4833
Synonym:
Target: Others
Bayogenin 3-O-β-D-glucopyranoside
Cat.No: TN1435
Synonym: Bayogenin 3-O-beta-D-glucopyranoside,贝萼皂苷元-3- O-Β-D-吡喃葡萄糖苷
Target: Others
Spiratisanin B
Cat.No: TN5603
Synonym:
Target:
Rabdosin A
Cat.No: T26029
Synonym:
Target:
(-)-Pinoresinol 4-O-glucoside
Cat.No: TN5402
Synonym: (-)-松脂素 4-O-葡萄糖苷,金银花
Target:
Asebotoxin III
Cat.No: T30156
Synonym:
Target:
Polygalasaponin LII
Cat.No: T81429
Synonym:
Target:
Sophorabioside
Cat.No: TN2218
Synonym:
Target: Others
Spiratisanin C
Cat.No: TN5048
Synonym:
Target: Others
2,3,4,5-Tetracaffeoyl-D-Glucaric acid
Cat.No: T19093
Synonym:
Target: Others
Sessilifoline A
Cat.No: TN5003
Synonym:
Target: Others
(E)-Aldosecologanin
Cat.No: TN3908
Synonym: 金银花
Target: Others
Spiratisanin A
Cat.No: TN5047
Synonym:
Target: Others
Matairesinoside
Cat.No: TN4507
Synonym:
Target: Others
4-Oxododecanedioic acid
Cat.No: TMA0537
Synonym:
Target: Others
Epivogeloside
Cat.No: TN1616
Synonym: 金银花,表断马钱子甙半缩醛内酯
Target: Others
(Z)-Aldosecologanin (Centauroside)
Cat.No: TN5276
Synonym: 金银花
Target: Others
Secoxyloganin methyl ester
Cat.No: TN4983
Synonym: 金银花
Target: Others
n-Butyl α-D-fructofuranoside
Cat.No: T80005
Synonym:
Target: JNK
Glaucocalyxin D
Cat.No: T82312
Synonym:
Target:
7,3'-Di-O-methylorobol
Cat.No: TN3210
Synonym:
Target: Others
Eupatolide
Cat.No: TN4038
Synonym:
Target: TNF, NOS, NF-κB, ROS, MAPK, Akt, COX, DNA/RNA Synthesis, Nrf2, PDGFR, NO Synthase, Prostaglandin Receptor, Autophagy
Platyphyllonol
Cat.No: TN4810
Synonym:
Target: Influenza Virus
Cinchonain Ib
Cat.No: TN5484
Synonym:
Target: Others
3-Acetyl-11-keto-ursolic acid
Cat.No: T83364
Synonym:
Target:
Troxerutin
Cat.No: T0772
Synonym: 曲克芦丁,Trihydroxyethylrutin,维脑路通
Target: NOD-like Receptor (NLR)
(6E,12E)-Tetradecadiene-8,10-diyne-1,3-diol
Cat.No: T75555
Synonym:
Target:
TargetMol Loading
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