首页工具

登录

搜索结果

Search Results for " anesthesia "

31

抑制剂 & 化合物

3

天然产物

如果没找到您满意的产品或者您对产品有其他要求，可以联系我们专业顾问为您提供针对性的合理建议。 QQ咨询网站留言咨询

Cat. No.	Product Name	Target	Signaling Pathways
T7045	Clonidine Nexiclon,Catapres,Kapvay,可乐定	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Clonidine (Kapvay) 是 alpha2 肾上腺素能激动剂。
T5326	Sugammadex sodium Org25969,Sugammadex (sodium),舒更葡糖钠	Others	Others
	Sugammadex sodium (Org25969) 是合成的 γ 环糊精衍生物，是一种新型的神经肌肉阻断逆转剂。
T0862	Diphenidol hydrochloride Diphenidol HCl,盐酸地芬尼多,Difenidol hydrochloride	Sodium Channel; AChR	Membrane transporter/Ion channel; Neuroscience
	Diphenidol hydrochloride (Difenidol hydrochloride) 是一种非选择性的毒蕈碱 M1-M4 受体拮抗剂，具有抗心律失常活性，用作抗眩晕药和止吐药。它也是神经细胞电压门控离子通道的有效非特异性阻滞剂。
T0364L	Dibucaine hydrochloride Cinchocaine HCl,Dibucaine HCl,盐酸地布卡因,Cinchocaine hydrochloride	Sodium Channel; AChR	Membrane transporter/Ion channel; Neuroscience
	Dibucaine hydrochloride (Cinchocaine hydrochloride) 是钠通道抑制剂和有效的 SChE 抑制剂。
T0364	Dibucaine 地布卡因,Cinchocaine	CaMK; Sodium Channel; AChR	Membrane transporter/Ion channel; Neuroscience
	Dibucaine (Cinchocaine) 是钠通道抑制剂和有效的SChE 抑制剂。
T33272	Mefenidil McN-2378,McN 2378	Others	Others
	Mefenidil (McN-2378) 是一种选择性脑血管扩张剂，在狗麻醉模型中显示出在不刺激 O2 摄取的情况下增加健康大脑中的 CBF。
T13142L	Theodrenaline hydrochloride Theodrenaline hydrochloride(13460-98-5 Free base)	SARS-CoV	Microbiology/Virology
	Theodrenaline hydrochloride 是一种靶向 SARS-CoV-2 的抑制剂，可用于研究由脊髓麻醉引起的低血压。
T19658	Enflurane NSC115944,Ethrane,NSC-115944,恩氟烷,Efrane,NSC 115944	Others	Others
	Enflurane (Efrane) 是一种挥发性麻醉剂，是 Chara australis 高电导 Ca2+ 激活的 K+ 通道的有效抑制剂。安氟醚是通过顶空气相色谱-质谱法监测卤化挥发性麻醉剂的内标。它可以快速调整麻醉深度，而脉搏或呼吸频率几乎没有变化。
T1198	Tetracaine hydrochloride 盐酸丁卡因,Amethocaine hydrochloride,Amethocalne HCl,Tetracaine HCl	Calcium Channel; Sodium Channel	Membrane transporter/Ion channel; Metabolism
	Tetracaine hydrochloride (Amethocalne HCl) 是一种钙通道蛋白抑制剂，可阻断肌浆网中 Ca2+的电压敏感释放。它主要用作眼科的止痒剂和局部用药，可用于表面和脊髓麻醉。
T2524	Dexmedetomidine	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Dexmedetomidine 是选择性、具有口服活性的 α2 肾上腺素能受体激动剂，Ki=1.08 nM。它对 α1 肾上腺素受体显示出 1620 倍的选择性。它具有抗焦虑活性，可用于研究促进睡眠和缓解疼痛。
T1787	Levobupivacaine	Sodium Channel	Membrane transporter/Ion channel
	Levobupivacaine 是一种氨基酰胺类局麻药，属于n-alkylsubstituted pipecoloxylidide 家族。它是bupivacaine 的 S-对映异构体。
T34753	Suxamethonium bromide L.T. 1,370 I.S.,Brevidil M
	Suxamethonium bromide can be used to cause short-term paralysis as part of general anesthesia.
T21099	Decamethonium iodide Decamethonium iodatum,Decamethonium diiodide,Dekamethoniumjodid
	Decamethonium is a neuromuscular blocking agent or depolarizing muscle relaxant, and is used in anesthesia to induce paralysis.
T29846	Alcuronium free base Alcuronium,Alcuronum,Diallylnortoxiferine,Alcuronium kation,Alloferine
	Alcuronium free base is a non-depolarizing skeletal muscle relaxant similar to Tubocurarine. It is used as an anesthesia adjuvant.
T28591	Ro 48-6791 Ro-486791,Ro 486791,Ro-48-6791,Ro486791,Ro48-6791
	Ro 48-6791, a GABA receptor agonist, is used potentially for anesthesia.
T3609	Dioxopromethazine Prothanon,Dioxoprothazine,盐酸二氧丙嗪	Others	Others
	Dioxopromethazine (Dioxoprothazine) 是一种口服具有活性的抗组胺药，能够抑制哮喘症状。
T25637	Laudexium methylsulfate Laudexium,Laudolissin methosulphate
	Laudexium methylsulfate is a neuromuscular blocking drug or skeletal muscle relaxant. It is used adjunctively in surgical anesthesia to facilitate endotracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilation.
T28259	Org-21465 Org21465,Org 21465
	Org-21465, a gamma-aminobutyric acid (GABA) receptor agonist, is used potentially for the use of anesthesia.
T31914	Gantacurium chloride GW 280430A,AV4430A,AV 4430A,GW280430,GW 280430,GW-0430
	Gantacurium chloride is a benzylisoquinoline alkaloid, which may be used as an adjuvant in anesthesia.
T0818L	Decamethonium
	Decamethonium (Syncurine) is a depolarizing muscle relaxant or neuromuscular blocking agent, and is used in anesthesia to induce paralysis.
T24690	Pyrromecaine HCl Bumecaine hydrochloride,Pyrromecaine
	Pyrromecaine is a local anesthetic used for surface anesthesia. Pyromecaine has a wide spectrum of antiarrhythmic action, exerts a favorable effect on the contractility of the left ventricle, and on the myocardial blood flow following the ligation of the
T31296	Decamethonium chloride Decamethylenebis(trimethylammonium chloride),Decamethonium dichloride
	Decamethonium is a depolarizing muscle relaxant or neuromuscular blocking agent,[1] and is used in anesthesia to induce paralysis.
T25636	Laudexium Laudexium ion,Laudexium cation
	Laudexium is a neuromuscular blocking drug or skeletal muscle relaxant in the category of non-depolarizing neuromuscular-blocking drugs. It is used adjunctively in surgical anesthesia to facilitate endotracheal intubation and to provide skeletal muscle re
T33638	Neostigmine Iodide SB 24,SB24,TL1321,TL 1321,TL-1321,SB-24
	Neostigmine Iodide is a parasympathic compound used as a reversible acetylcholinesterase inhibitor to improve muscle tone in patients with myasthenia gravis and in routine anesthesia to reverse the effects of non-depolarizing muscle relaxants such as rocu
T83124	Amylocaine
	Amylocaine为一种酯类局部麻醉药，能在给药部位附近产生可逆性麻木，主要应用于脊柱麻醉。
T82146	Hydroxydione
	Hydroxydione展现全身麻醉效应，作为一种神经活性类固醇，适用于麻醉研究。
T0029	Procaine Duracaine,Spinocaine,普鲁卡因,Novocaine,Vitamin H3,奴夫卡因	Histone Demethylase; DNA/RNA Synthesis; Sodium Channel	Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Membrane transporter/Ion channel
	Procaine (Vitamin H3) 是DNA 脱甲基剂，是一种酯类局部麻醉剂。它起效缓慢，作用持续时间短，主要用于浸润麻醉、周围神经阻滞和脊髓阻滞。
T37702	Pancuronium (bromide hydrate)
	Pancuronium is an aminosteroid antagonist of muscle-type nicotinic acetylcholine receptors (nAChRs) with an IC50value of 14.8 nM using patch clamp electrophysiology in BOSC23 cells expressing mouse nAChRs.1It acts as a non-depolarizing neuromuscular blocking agent.2Pancuronium enhances anesthesia induced by isoflurane , reducing immobilization with an ED50value of 1.62 μg/kg.3 1.Liu, M., and Dilger, J.P.Site selectivity of competitive antagonists for the mouse adult muscle nicotinic acetylcholin...
T33287	Mephentermine Sulfate sulfuric acid,MLS002153976,N,2-dimethyl-1-phenylpropan-2-amine,AC1NWAW7,Mephentermine sodium
	Mephentermine sulfate is a cardiac stimulant, before as a stimulant in psychiatry, has been used as a treatment for low blood pressure. Mephentermine sulfate is a sympathomimetic agent with specificity for alpha-1 adrenergic receptors. It is used to maint
T80638	Glycinexylidide GX	MEK	MAPK
	Glycinexylidide (GX) 是一种 Lidocaine 的活性代谢物。作为有效的局部麻醉药，Lidocaine 可以通过阻断复杂电压依赖性的钠通道来发挥作用。此外，它还能抑制胃癌细胞生长、迁移和侵袭。GX 显示出在麻醉、癌症治疗和心血管疾病研究中的应用潜力。
T69598	Isoproterenol-d7 HCl
	Isoproterenol-d7 is intended for use as an internal standard for the quantification of isoproterenol by GC- or LC-MS. Isoproterenol is an agonist of β1- and β2-adrenergic receptors (β1- and β2-ARs; Kis = 224 and 458 nM, respectively). It is selective for β1- and β2-ARs over β3-ARs (Ki = 1,570 nM). Isoproterenol inhibits contractions in isolated field-stimulated rat vas deferens (EC50 = 45.6 nM). In vivo, isoproterenol (0.33 mg/kg) decreases blood pressure and increases water intake in nephrectom...

化合物

Cat.No: T7045

Synonym: Nexiclon,Catapres,Kapvay,可乐定

Target: Adrenergic Receptor

Sugammadex sodium

Cat.No: T5326

Synonym: Org25969,Sugammadex (sodium),舒更葡糖钠

Target: Others

Diphenidol hydrochloride

Cat.No: T0862

Synonym: Diphenidol HCl,盐酸地芬尼多,Difenidol hydrochloride

Target: Sodium Channel, AChR

Dibucaine hydrochloride

Cat.No: T0364L

Synonym: Cinchocaine HCl,Dibucaine HCl,盐酸地布卡因,Cinchocaine hydrochloride

Target: Sodium Channel, AChR

Cat.No: T0364

Synonym: 地布卡因,Cinchocaine

Target: CaMK, Sodium Channel, AChR

Cat.No: T33272

Synonym: McN-2378,McN 2378

Target: Others

Theodrenaline hydrochloride

Cat.No: T13142L

Synonym: Theodrenaline hydrochloride(13460-98-5 Free base)

Target: SARS-CoV

Cat.No: T19658

Synonym: NSC115944,Ethrane,NSC-115944,恩氟烷,Efrane,NSC 115944

Target: Others

Tetracaine hydrochloride

Cat.No: T1198

Synonym: 盐酸丁卡因,Amethocaine hydrochloride,Amethocalne HCl,Tetracaine HCl

Target: Calcium Channel, Sodium Channel

Dexmedetomidine

Cat.No: T2524

Target: Adrenergic Receptor

Levobupivacaine

Cat.No: T1787

Target: Sodium Channel

Suxamethonium bromide

Cat.No: T34753

Synonym: L.T. 1,370 I.S.,Brevidil M

Decamethonium iodide

Cat.No: T21099

Synonym: Decamethonium iodatum,Decamethonium diiodide,Dekamethoniumjodid

Alcuronium free base

Cat.No: T29846

Synonym: Alcuronium,Alcuronum,Diallylnortoxiferine,Alcuronium kation,Alloferine

Cat.No: T28591

Synonym: Ro-486791,Ro 486791,Ro-48-6791,Ro486791,Ro48-6791

Dioxopromethazine

Cat.No: T3609

Synonym: Prothanon,Dioxoprothazine,盐酸二氧丙嗪

Target: Others

Laudexium methylsulfate

Cat.No: T25637

Synonym: Laudexium,Laudolissin methosulphate

Cat.No: T28259

Synonym: Org21465,Org 21465

Gantacurium chloride

Cat.No: T31914

Synonym: GW 280430A,AV4430A,AV 4430A,GW280430,GW 280430,GW-0430

Cat.No: T0818L

Pyrromecaine HCl

Cat.No: T24690

Synonym: Bumecaine hydrochloride,Pyrromecaine

Decamethonium chloride

Cat.No: T31296

Synonym: Decamethylenebis(trimethylammonium chloride),Decamethonium dichloride

Cat.No: T25636

Synonym: Laudexium ion,Laudexium cation

Neostigmine Iodide

Cat.No: T33638

Synonym: SB 24,SB24,TL1321,TL 1321,TL-1321,SB-24

Cat.No: T83124

Cat.No: T82146

Cat.No: T0029

Synonym: Duracaine,Spinocaine,普鲁卡因,Novocaine,Vitamin H3,奴夫卡因

Target: Histone Demethylase, DNA/RNA Synthesis, Sodium Channel

Pancuronium (bromide hydrate)

Cat.No: T37702

Mephentermine Sulfate

Cat.No: T33287

Synonym: sulfuric acid,MLS002153976,N,2-dimethyl-1-phenylpropan-2-amine,AC1NWAW7,Mephentermine sodium

Glycinexylidide

Cat.No: T80638

Synonym: GX

Target: MEK

Isoproterenol-d7 HCl

Cat.No: T69598

Cat. No.	Product Name	Target	Signaling Pathways
T0012	Cinchonine LA40221,(8R,9S)-Cinchonine,奎宁树,辛可宁	Apoptosis; P-gp; Parasite	Apoptosis; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
	Cinchonine (LA40221) 是金鸡纳树皮中的一种天然产物。它可激活内质网应激诱导的人肝癌细胞凋亡。它是一种酰胺类局部麻醉剂。
T5734	(+)-BORNEOL d-Borneol,(+)-冰片	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	(+)-BORNEOL (d-Borneol) 是一种天然的双环单萜，在中药中用于镇痛和麻醉；增强 GABA 受体活性，EC50 为 248 μM。
Fr16605	Lupinine 鲁冰花,羽扇豆碱	AChR; AChE	Neuroscience
	Lupinine 是一种能够抵消乙醇麻醉的生物碱。 Lupinine 是一种 AChE 和 BChE 抑制剂和潜在的 CD69 激活剂，存在于 Loranthus、Calia 和 Lupinus 物种中。它还可以抑制肝素。

天然产物

Cat.No: T0012

Synonym: LA40221,(8R,9S)-Cinchonine,奎宁树,辛可宁

Target: Apoptosis, P-gp, Parasite

Cat.No: T5734

Synonym: d-Borneol,(+)-冰片

Target: GABA Receptor

Cat.No: Fr16605

Synonym: 鲁冰花,羽扇豆碱

Target: AChR, AChE

我们的所有产品和服务仅用于科学研究，不能被用于人体，我们也不向个人提供产品和服务。

Copyright © 2015-2024 TargetMol Chemicals Inc. All rights reserved. 沪ICP备20019793号-4

沪公网安备 31010602006700号

沪公网安备 31010602006700号

TargetMol Loading

联系我们

电话：

400-820-0310

邮箱：

service@tsbiochem.com

QQ：

2881945090（终端用户）

2885109491（经销商）

经销：

终端：

地址：

上海市静安区江场三路238号8楼