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Cat. No. Product Name Target Signaling Pathways
T10380 AS19

5-HT Receptor GPCR/G Protein; Neuroscience
AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM). AS19 is selective for 5-HT7 over 5-HT1A, 5-HT1B, 5-HT1D, and 5-HT5A receptors (Kis: 89.7 nM, 490 nM, 6.6 nM and 98.5 nM, respectively).
T23819 Braco-19 trihydrochloride

BRAC-O19,BRACO19 hydrochloride,BRACO19 3HCl,BRACO 19,BRACO19 HCl

 Telomerase DNA Damage/DNA Repair
Braco-19 trihydrochloride (BRACO19 3HCl) 是一种端粒酶抑制剂，可阻止端粒酶的加帽和催化作用。 Braco-19 trihydrochloride 抑制 HAdV 病毒复制。
T15655 KFM19

Adenosine Receptor GPCR/G Protein; Neuroscience
KFM19 是一种具有强效性和选择性的腺苷受体 (A1-receptor) 拮抗剂(IC50 ： 50 nM)，可用于研究神经系统疾病。
T67950 S19-1035

NADPH Metabolism
S19-1035为AKR1C3(aldehyde ketone reductase 1C3)的高效特异性抑制剂，其IC50值为3.04 nM，主要应用于肿瘤研究。
T8931L ICCB-19 hydrochloride

ICCB-19 HCl（750621-52-4 free base）

 Apoptosis; Others; Autophagy; RIP kinase Apoptosis; Autophagy; NF-κB; Others
ICCB-19 hydrochloride (ICCB-19 HCl) 是RIPK1激酶活性的间接抑制剂。它是一种 TRADD 抑制剂，可与 TRADD 的 N 端结构域结合，破坏其与 TRADD-C 和 TRAF2 的结合，诱导自噬和长寿命蛋白质的降解。
T21083 TFIIH Modulator-19

TFIIH Modulator19,TFIIH Modulator 19

 Others Others
TFIIH Modulator-19 诱导毛发硫营养不良组 A 蛋白的二聚化以调节 TFIIH 转录活性。
T10123 VEGFR-2-IN-9

KDR-in-4

 VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR-2-IN-9 (KDR-in-4) 是一种高效的 KDR/VEGFR2 抑制剂（IC50：7 nM）,可用于研究乳腺癌。
T10341 Antitumor agent-19

Others Others
Antitumor agent-19 是一种肿瘤相关巨噬细胞的调节剂，在 RAW 264.7 细胞和 BMDM 细胞中的 EC50 分别为 17.18 μM 和 18.87 μM。
TP1563 Gap19

Gap Junction Protein Cytoskeletal Signaling
Gap19 是一种衍生自 Cx43 细胞质环九个氨基酸的肽，是选择性连接蛋白 43 半通道阻滞剂。它可以防止 C 末端与 CL 的分子内相互作用，具有保护心肌作用。
T9998 MIND4-19

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
MIND4-19 是一种具有抗肿瘤活性的 SIRT2 抑制剂。
T36711 FM19G11

FM19G11,HIF-1alpha/2alpha Inhibitor

 HIF Angiogenesis; Chromatin/Epigenetic
FM19G11 是一种低氧诱导因子 (HIF) α-亚基抑制剂（在低氧诱导的荧光素酶试验中 IC50 为 80 nM）。
T29017 TrxR1-IN-B19

TrxR1INB19,Go Y015,TrxR1 IN B19,Go-Y015

 Others Others
TrxR1-IN-B19 (TrxR1 IN B19) 是一种 TrxR1 抑制剂，通过靶向 TrxR1 和 ROS 介导的 ER 应激激活，通过小分子选择性杀死胃癌细胞。
T9936 ZX-J-19J

N-(2,3-Diphenyl-6-quinoxalinyl)octanamide

 Others Others
ZX-J-19J (N-(2,3-Diphenyl-6-quinoxalinyl)octanamide) 是 Cyclophilin J 的抑制剂，对肿瘤细胞生长有显着的抑制作用，与环孢素 A 相当，但比 5-氟尿嘧啶强得多。
TP2110L TAT-Gap19 acetate

Gap Junction Protein Cytoskeletal Signaling
TAT-Gap19 acetate 是 connexin43 hemichannel (Cx43 HC) 的特异性抑制剂。 它穿过血脑屏障并减轻小鼠的肝纤维化。它不抑制相应的 Cx43 GJC。
T40286 KRAS G12C inhibitor 19

Ras GPCR/G Protein; MAPK
KRAS G12C inhibitor 19 是一种有效的 KRAS G12C 抑制剂，在细胞实验中显示出抗肿瘤活性，科抑制肿瘤生长。
T72022 11β-HSD1 inibitor 19

11β-HSD1 inibitor 19 对 hHSD1 和 mHSD1 显示抑制活性，IC50 为 16 nM 和 10 nM。
TP1863L Glucagon (19-29), human acetate

Glucagon Receptor GPCR/G Protein
Glucagon (19-29), human acetate 是一种从胰高血糖素加工而来的 COOH 末端片段，是一种有效的胰岛素分泌抑制剂。
TP1053L Protein Kinase C 19-31 acetate

Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate

 PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Protein Kinase C 19-31 acetate(121545-65-1 free base) 是一种蛋白激酶 C (PKC) 的肽抑制剂，源自 PKCa 的假底物调节结构域（残基 19-31），在 25 位用丝氨酸取代野生型丙氨酸作为蛋白激酶 C 底物肽，用于测试蛋白激酶 C 活性。
T38360 NBC 19

Potent NLRP3 inflammasome inhibitor (IC50 = 60-80 nM). Inhibits nigericin- and ATP-induced IL-1β release. Baldwin et al (2017) Boron-Based Inhibitors of the NLRP3 Inflammasome. Cell Chem.Biol. 24 1321 PMID:28943355 |Redondo-Castro et al (2018) Development of a characterised tool kit for the interrogation of NLRP3 inflammasome-dependent responses. Sci.Rep. 8 5667 PMID:29618797
T37237 (±)19(20)-DiHDTE

(±)19(20)-DiHDTE is an oxylipin and an oxidative metabolite of docosapentaenoic acid . It is formed via cytochrome P450 (CYP) metabolism of DPA via a (±)19(20)-EpDTE intermediate.
T40185 BTK inhibitor 19

BTK inhibitor 19 is a highly selective, covalent BTK inhibitor ( IC 50 = 2.7 nM).
T41183 Helianorphin-19

Helianorphin-19 is a high affinity, potent and selective κ-opioid receptor (KOR) agonist (Ki = 25 nM; EC50= 45 nM). Helianorphin-19 exhibits approximately 200-fold selectivity for KOR over μ and δ-opioid receptors.In vivoHelianorphin-19 shows potent peripheral analgesic efficacy in a mouse model of visceral pain without affecting motor coordination/sedation.
T37239 (±)19(20)-EpDTE

(±)19(20)-EpDTE is an oxylipin and an oxidative metabolite of docosapentaenoic acid . It is formed via cytochrome P450 (CYP) metabolism of DPA and can be further metabolized to (±)19(20)-DiHDTE by epoxide hydrolase.
T40991 19-Heptatriacontanol

19-Heptatriacontanol,19-Hydroxyheptatriacontane
19-Heptatriacontanol is used to combine macromolecules and small molecules.
T36216 19(R)-HETE

19-HETE is one of the major cytochrome P450 (CYP450) metabolites of arachidonic acid that is released from the kidney in response to angiotensin II. When formed by the CYP2E1 isoform, 19-HETE is composed of 70% and 30% of the (S) and (R) stereoisomers, respectively. Both 19(S)- and 19(R)-HETE are potent vasodilators of renal preglomerular vessels. However, 19(R)-HETE at 1 μM completely blocks 20-HETE-induced vasoconstriction of renal arterioles, whereas 19(S)-HETE remains inactive.
T35850 19(S)-HETE

19-HETE is one of the major cytochrome P450 (CYP450) metabolites of arachidonic acid that is released from the kidney in response to angiotensin II. When formed by the CYP2E1 isoform, 19-HETE is composed of 70% and 30% of the (S) and (R) stereoisomers, respectively. Both 19(S)- and 19(R)-HETE are potent vasodilators of renal preglomerular vessels. 19(S)-HETE stimulates both renal sodium-potassium ATPase and volume absorption in the rabbit proximal straight tubule.
T37238 (±)19(20)-EpDPA

EDHF (endothelium-derived hyperpolarizing factor) is an unidentified mediator released from vascular endothelial cells in response to acetylcholine and bradykinin which is distinct from the NOS- (nitric oxide) and COX-derived (prostacyclin) vasodilators. Cytochrome P450 (CYP450) metabolism of polyunsaturated fatty acids produces epoxides such as (±)14(15)-EpETrE which are prime candidates for the actual active mediator. However, the CYP450 metabolites of eicosapentaenoic acid and docosahexaenoic...
T36217 19-hydroxy Cholesterol

19-hydroxy Cholesterol is formed during metabolic oxidation of cholesterol. It has been used as an internal standard for the quantitative determination of sterols by mass spectroscopic analysis.[1]
T35873 C19 Ceramide (d18:1/19:0)

C19 Ceramide (d18:1/19:0)
C19 Ceramide is a naturally occurring ceramide that has been found in J. juncea extracts as well as rat brain and mouse heart.[1],[2],[3] It is elevated in adult and decreased in juvenile whole rat brain extracts by 114 and 37%, respectively, following chronic ethanol exposure.[2] C19 Ceramide is also increased in mouse hearts following administration of angiotensin II.[3]
T35468 (±)19(20)-EDP Ethanolamide

(±)19(20)-EDP ethanolamide is an ω-3 endocannabinoid epoxide and cannabinoid (CB) receptor agonist (EC50s = 108 and 280 nM for CB1 and CB2, respectively). It is produced through direct epoxygenation of docosahexaenoyl ethanolamide by cytochrome P450 (CYP) epoxygenases. (±)19(20)-EDP ethanolamide (25 μM) reduces the viability of 143B metastatic osteosarcoma cells. It decreases the production of IL-6 and increases the production of IL-10 when used at concentrations ranging from 2.5 to 10 μM in BV-...
T39709 HPK1-IN-19

HPK1-IN-19
HPK1-IN-19 is an inhibitor of hematopoietic progenitor kinase 1 (HPK1).
T63125 Antiviral agent 19

Antiviral agent 19 (Compound 3) 是一种 Zika 病毒的选择性抑制剂 (EC50: 1.3 μM)，具有低细胞毒性。
T63652 DHODH-IN-19

DHODH-IN-19 是 DHODH 的有效抑制剂。其中 DHODH 是一种含铁的黄素依赖性酶，存在于人类线粒体的内膜中，对肿瘤生长具有抑制作用。DHODH-IN-19 对癌症和炎症疾病表现出研究潜力。
T63837 RET-IN-19

RET-IN-19 是 RET 的有效抑制剂，能够作用于 RET-wt (IC50: 6.8 nM) 和 RET V804M (IC50: 13.51 nM)，表现出抗癌效果。RET-IN-19 能够用于研究非小细胞肺癌 (NSCLC)。
T82126 ICMT-IN-19

ICMT-IN-19 (compound 53)为一种高效ICMT抑制剂，其半抑制浓度(IC50)为0.026 μM。
T63628 AChE-IN-19

AChE-IN-19 是 AChE 的高效抑制剂 (IC50: 0.56 μM)，对 Aβ 聚集也表现出抑制作用。AChE-IN-19 表现出神经保护作用，对 SH-SY5Y 细胞几乎没有毒性。AChE-IN-19 能够用于研究阿尔兹海默症。
T62891 α-Glucosidase-IN-19

α-Glucosidase-IN-19 (Compound 6B) 是一种口服具有活力的 α-glucosidase 抑制剂 (IC50: 3.63 μM)，具有抗糖尿病作用。
T80721 Zndm19

Zndm19为New Delhi Metallo-β-lactamase-1 (NDM-1)的抑制剂，适用于抗药性细菌感染研究。
T75067 Antimalarial agent 19

Parasite Microbiology/Virology
Antimalarial agent 19（compound 6e）是一种活性抗疟疾化合物，对K1型恶性疟原虫和伯氏疟原虫展现出较强的抑制效果，其EC50值分别为0.3 µM和15.3 µM。相较于γ-肝硫平，该化合物具有更好的水溶性、肠道渗透性以及微粒体稳定性。
T73319 BTK-IN-19

BTK-IN-19 是一种可逆的BTK 抑制剂，IC50<0.001 μM。
T72330 Antibacterial agent 19

Antibacterial agent 19 是一种有效的抗菌剂。Antibacterial agent 19 对K. pneumoniae，(M-R)S. aureus 和 (M-R,V-R)S. aureus 具有抗菌活性, 其 MIC 值为 0.022, 0.022 和 0.045 mg/mL。
T125260 19-Hydroxypseudovincadifformine

19-Hydroxypseudovincadifformine 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T125260。
T62579 HBV-IN-19

HBV-IN19 对乙型肝炎病毒 (HBV) 感染具有抑制作用。HBV-IN19 能够抑制 HBsAg 分泌和/或产生，可以用于 HBV 感染的研究 (如:慢性 HBV 感染)。
T62095 TRK-IN-19

TRK-IN-19 (Compound I-10 ) 是一种 TRK 的有效抑制剂，对 TRKA、TRKAG595R 的 IC50 值分别为 1.1 nM、5.3 nM。TRK-IN-19 对癌症疾病表现出潜在的研究价值。
T61257 Antifungal agent 19

Antifungal agent 19 显示出强大的抗真菌活性（EC50= 0.72 μM）。
T80909 Tyrosinase-IN-19

Tyrosinase Proteases/Proteasome
Tyrosinase-IN-19 是竞争性酪氨酸酶抑制剂，对ROS、ABTS+ 及DPPH 自由基展现显著的抗氧化活性。该化合物通过剂量依赖性方式有效抑制酪氨酸酶表达。
T80295 GLR-19

HSV Microbiology/Virology
GLR-19 为一种具有抗HIV功能的肽类化合物，亦展现出对HSV-2的抗病毒活性。
T79692 BChE-IN-19

BChE-IN-19 (Compound 7b) 是一种具有对 BChE 抑制活性（IC50=0.04 μM）的茚酮对位取代衍生物，可改善神经系统胆碱能调控，适用于抗阿尔茨海默病研究。
T61636 ATR-IN-19

ATR-IN-19 (Compound 15 R-configure) 是一种ATR 抑制剂。
T63904 ATX inhibitor 19

ATX inhibitor 19 是 ATX 的有效抑制剂 (IC50: 156 nM)。

化合物

AS19
Cat.No: T10380
Synonym:
Target: 5-HT Receptor
Braco-19 trihydrochloride
Cat.No: T23819
Synonym: BRAC-O19,BRACO19 hydrochloride,BRACO19 3HCl,BRACO 19,BRACO19 HCl
Target: Telomerase
KFM19
Cat.No: T15655
Synonym:
Target: Adenosine Receptor
S19-1035
Cat.No: T67950
Synonym:
Target: NADPH
ICCB-19 hydrochloride
Cat.No: T8931L
Synonym: ICCB-19 HCl（750621-52-4 free base）
Target: Apoptosis, Others, Autophagy, RIP kinase
TFIIH Modulator-19
Cat.No: T21083
Synonym: TFIIH Modulator19,TFIIH Modulator 19
Target: Others
VEGFR-2-IN-9
Cat.No: T10123
Synonym: KDR-in-4
Target: VEGFR
Antitumor agent-19
Cat.No: T10341
Synonym:
Target: Others
Gap19
Cat.No: TP1563
Synonym:
Target: Gap Junction Protein
MIND4-19
Cat.No: T9998
Synonym:
Target: Sirtuin
FM19G11
Cat.No: T36711
Synonym: FM19G11,HIF-1alpha/2alpha Inhibitor
Target: HIF
TrxR1-IN-B19
Cat.No: T29017
Synonym: TrxR1INB19,Go Y015,TrxR1 IN B19,Go-Y015
Target: Others
ZX-J-19J
Cat.No: T9936
Synonym: N-(2,3-Diphenyl-6-quinoxalinyl)octanamide
Target: Others
TAT-Gap19 acetate
Cat.No: TP2110L
Synonym:
Target: Gap Junction Protein
KRAS G12C inhibitor 19
Cat.No: T40286
Synonym:
Target: Ras
11β-HSD1 inibitor 19
Cat.No: T72022
Synonym:
Target:
Glucagon (19-29), human acetate
Cat.No: TP1863L
Synonym:
Target: Glucagon Receptor
Protein Kinase C 19-31 acetate
Cat.No: TP1053L
Synonym: Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate
Target: PKC
NBC 19
Cat.No: T38360
Synonym:
Target:
(±)19(20)-DiHDTE
Cat.No: T37237
Synonym:
Target:
BTK inhibitor 19
Cat.No: T40185
Synonym:
Target:
Helianorphin-19
Cat.No: T41183
Synonym:
Target:
(±)19(20)-EpDTE
Cat.No: T37239
Synonym:
Target:
19-Heptatriacontanol
Cat.No: T40991
Synonym: 19-Heptatriacontanol,19-Hydroxyheptatriacontane
Target:
19(R)-HETE
Cat.No: T36216
Synonym:
Target:
19(S)-HETE
Cat.No: T35850
Synonym:
Target:
(±)19(20)-EpDPA
Cat.No: T37238
Synonym:
Target:
19-hydroxy Cholesterol
Cat.No: T36217
Synonym:
Target:
C19 Ceramide (d18:1/19:0)
Cat.No: T35873
Synonym: C19 Ceramide (d18:1/19:0)
Target:
(±)19(20)-EDP Ethanolamide
Cat.No: T35468
Synonym:
Target:
HPK1-IN-19
Cat.No: T39709
Synonym: HPK1-IN-19
Target:
Antiviral agent 19
Cat.No: T63125
Synonym:
Target:
DHODH-IN-19
Cat.No: T63652
Synonym:
Target:
RET-IN-19
Cat.No: T63837
Synonym:
Target:
ICMT-IN-19
Cat.No: T82126
Synonym:
Target:
AChE-IN-19
Cat.No: T63628
Synonym:
Target:
α-Glucosidase-IN-19
Cat.No: T62891
Synonym:
Target:
Zndm19
Cat.No: T80721
Synonym:
Target:
Antimalarial agent 19
Cat.No: T75067
Synonym:
Target: Parasite
BTK-IN-19
Cat.No: T73319
Synonym:
Target:
Antibacterial agent 19
Cat.No: T72330
Synonym:
Target:
19-Hydroxypseudovincadifformine
Cat.No: T125260
Synonym:
Target:
HBV-IN-19
Cat.No: T62579
Synonym:
Target:
TRK-IN-19
Cat.No: T62095
Synonym:
Target:
Antifungal agent 19
Cat.No: T61257
Synonym:
Target:
Tyrosinase-IN-19
Cat.No: T80909
Synonym:
Target: Tyrosinase
GLR-19
Cat.No: T80295
Synonym:
Target: HSV
BChE-IN-19
Cat.No: T79692
Synonym:
Target:
ATR-IN-19
Cat.No: T61636
Synonym:
Target:
ATX inhibitor 19
Cat.No: T63904
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1118 Tormentic acid

2Α,19Α-二羟基熊果酸,委陵菜酸

 Immunology/Inflammation related Immunology/Inflammation
Tormentic acid 是一种分离自 Rosa rugosa 中的三萜，具有抗炎、降血脂和抗动脉粥样硬化活性。
TN1198 19-Hydroxybufalin

Others Others
19-Hydroxybufalin 是蟾二烯羟酸内酯，能够阻碍上皮间质转化，抑制 PC3 细胞的迁移和侵袭。
TN2237 Steviol-19-O-glucoside

Steviol-19-O-Glucoside,甜菊醇-19-葡萄糖苷

 Others Others
Steviol-19-O-glucoside 是甜叶菊 Stevia rebuadiana 中甜菊糖苷生物合成途径的天然产物。
T35609 19-O-Acetylchaetoglobosin A

19-O-Acetylchaetoglobosin A is a fungal metabolite originally isolated fromC. globosumthat has actin polymerization inhibitory and cytotoxic activities.1,2It inhibits actin polymerization in a cell-free assay when used at a concentration of 2 μM.219-O-Acetylchaetoglobosin A (3.2, 10, and 32 μg/ml) is cytotoxic to HeLa cervical cancer cells.1 1.Umeda, M., Ohtsubo, K., Saito, M., et al.Cytotoxicity of new cytochalasans from Chaetomium globosumExperientia31(4)435-438(1975) 2.Sekita, S., Yoshihira, ...
T35483 19,20-Epoxycytochalasin D

19,20-Epoxycytochalasin D is a fungal metabolite that has been found in the endophytic fungus Nemania sp. UM10M. It is active against the chloroquine-sensitive and -resistant strains of P. falciparum (MIC = 0.4 ng/ml for both) without inducing cytotoxicity in Vero cells. It is cytotoxic to BT-549, LLC-PK11, and P388 cells (IC50s = 7.84, 8.4, and 0.16 &#181M, respectively) but not SK-MEL, KB, or SKOV3 cells up to a concentration of 10 &#181M.
T83578 (19R,23E)-5b,19-Epoxy19-ethoxycucurbita-6,23-diene-3b,25-diol

(19R,23E)-5b,19-Epoxy19-ethoxycucurbita-6,23-diene-3b,25-diol 是一种葫芦烷型三萜。该化合物在 MTT 法检测中对癌细胞系 MCF-7、HepG2、Du145、Colon205 以及 HL-60 均未表现出抑制效果。
TN1199 19-Oxocinobufagin

Others Others
19-Oxocinobufagin is a natural product from Bufo bufo gargarizans Cantor.
T83435 19-Hydroxy-10-deacetylbaccatin III

19-Hydroxy-10-deacetylbaccatin III (compound 13) 是紫杉烷类化合物，显示出潜在的抗肿瘤作用。在 A498 和 NCI-H226 细胞系中，此化合物表现出轻微的细胞毒性效应。研究指出，当浓度为 30 μg/mL 时，19-Hydroxy-10-deacetylbaccatin III 对 A498 细胞和 NCI-H226 细胞的抑制率为 16.6% 和 32%。
TN1200 19-Oxocinobufotalin

Others Others
19-Oxocinobufotalin 3-adipoylarginine ester shows significant inhibition effect against human hepatocellular carcinoma cell line SMMC-7721 in vitro.
T83458 12E,14-Trien-19-oic acid

12E,14-Trien-19-oic acid 为一类二萜，源自不丹药用植物 shug chher。该化合物在血小板聚集研究中有应用。
TN3941 ent-17-Hydroxykaur-15-en-19-oic acid

Others Others
ent-17-Hydroxykaur-15-en-19-oic acid 是从香树叶中发现的天然化合物，对人前列腺细胞的IC50为17.63microg/mL。
TN1178 11,15-Dihydroxy-16-kauren-19-oic acid

Others Others
11,15-Dihydroxy-16-kauren-19-oic acid is a natural product
T83570 (23E)-5b,19-epoxycucurbita-6,23,25(26)-triene-3b-ol

(23E)-5b,19-epoxycucurbita-6,23,25(26)-triene-3b-ol，一种葫芦烷三萜，可从苦瓜籽中提取。
TN1401 Arjunetin

Others Others
Arjunetin, an insect feeding-deterrent and growth inhibitor, shows antioxidant and anti-inflammatory activities.
TN3651 Cichoriin

Others Others
Cichoriin 对SARS-CoV-2有明显活性，是治疗重症COVID-19的潜在候选物质。
T8070 Nonadecanoic acid

Others Others
Nonadecanoic acid 是19 C 长的饱和脂肪酸，是白蚁防御时分泌的主要物质。
T0194 Chloroquine phosphate

Chloroquine diphosphate,Aralen phosphate,磷酸氯喹,Chingamin phosphate

 SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine phosphate (Aralen phosphate) 是广泛用于疟疾和类风湿性关节炎的抗疟疾和抗炎剂。它是autophagy 和toll-like receptors 抑制剂，有效抑制SARS-CoV-2(COVID-19) 感染 (EC50=1.13 μM)。
T3921 Punicalagin

安石榴甙,安石榴苷

 SARS-CoV; HBV Microbiology/Virology
Punicalagin 是一种在石榴中发现的主要鞣花单宁，是可逆且非竞争性的3CLpro 抑制剂，有抗氧化、抗炎和抗癌作用。它有潜力研究 COVID-19 。
TN3948 ent-3Beta-Angeloyloxykaur-16-en-19-oic acid

Others Others
ent-3Beta-Angeloyloxykaur-16-en-19-oic acid是一种天然产物，属于菊科蟛蜞菊属，其产品编号为 TN3948，CAS号为 74635-61-3。ent-3Beta-Angeloyloxykaur-16-en-19-oic acid可用作对照参考。
TN3939 ent-16beta,17-dihydroxy-9(11)-kauren-19-oic acid

Others Others
ent-16beta,17-dihydroxy-9(11)-kauren-19-oic acid是一种天然产物，属于菊科苍耳属，其产品编号为 TN3939，CAS号为 55483-24-4。ent-16beta,17-dihydroxy-9(11)-kauren-19-oic acid可用作对照参考。
TN6493 19-O-beta-D-carboxyglucopyranosyl-12-O-beta-D-glucopyranosyl-11,16-dihydroxyabieta-8,11,13-triene

19-O-beta-D-carboxyglucopyranosyl-12-O-beta-D-glucopyranosyl-11,16-dihydroxyabieta-8,11,13-triene是一种天然产物，属于松科松属，其产品编号为 TN6493，CAS号为 1011714-20-7。19-O-beta-D-carboxyglucopyranosyl-12-O-beta-D-glucopyranosyl-11,16-dihydroxyabieta-8,11,13-triene可用作对照参考。
TN2757 2-Epitormentic acid

Others Others
2-Epitormentic acid是一种天然产物，属于蔷薇科委陵菜属，其产品编号为 TN2757，CAS号为 119725-19-8。2-Epitormentic acid可用作对照参考。
TN2700 2,3-dihydrosciadopitysin

Others Others
2,3-dihydrosciadopitysin是一种天然产物，属于罗汉松科罗汉松属，其产品编号为 TN2700，CAS号为 34421-19-7。2,3-dihydrosciadopitysin可用作对照参考。
TN2486 1-(3,4-Dimethoxyphenyl)propane-1,2-diol

Others Others
β-Aflatrem是一种天然产物，属于金粟兰科金粟兰属，其产品编号为 TN2486，CAS号为 20133-19-1。β-Aflatrem可用作对照参考。
TN3254 7alpha-Hydroxystigmasterol

Others Others
7alpha-Hydroxystigmasterol是一种天然产物，属于菊科苍耳属，其产品编号为 TN3254，CAS号为 64998-19-2。7alpha-Hydroxystigmasterol可用作对照参考。
T75670 Lacto-N-fucopentaose II

Lacto-N-fucopentaose II (LNFP II)作为人Lewis血型决定因子的半抗原，其单唾液神经节苷/糖脂以及唾液酰衍生物CA 19-9，都是胆胰恶性肿瘤中的分子肿瘤标记物(TM)。
TN3269 8,9-Didehydro-7-hydroxydolichodial

Others Others
8,9-Didehydro-7-hydroxydolichodial是一种天然产物，属于败酱科败酱属，其产品编号为 TN3269，CAS号为 97856-19-4。8,9-Didehydro-7-hydroxydolichodial可用作对照参考。
TN1194 16beta,17-Dihydroxy-ent-kaurane-19-oic acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
16beta,17-Dihydroxy-ent-kaurane-19-oic acid as an anti-HIV principle, it showed significant activity against HIV replication in H9 lymphocyte cells with an EC50 value of 0.8 microgram/mL. It also possesses the activities of decompression and blood viscosi
TN5637 5-(Z-Heptadec-8-enyl)resorcinol

5-(8-Heptadecenyl)-1,3-benzenediol
5-(Z-Heptadec-8-enyl)resorcinol是一种天然产物，属于紫金牛科紫金牛属，其产品编号为 TN5637，CAS号为 52483-19-9。5-(Z-Heptadec-8-enyl)resorcinol可用作对照参考。
T38262 Sphingosine (d14:1)

Sphingosine (d14:1) is a bioactive sphingolipid that has been found in B. mori (silkworm), P. clarkii (crayfish), and A. aurita (jellyfish) extracts. It increases the germination rate of N. rileyi, an entomopathogenic fungus, with an EC50 value of 10.2 nM. Sphingosine (d14:1) inhibits protein kinase C (PKC) in vitro (IC50 = 7.3 mol%) as well as superoxide generation induced by phorbol 12-myristate 13-acetate in neutrophils and reduces growth of CHO cells (IC50s = 19 and 8 μM, respectively).
T72581 SARS-CoV MPro-IN-2

SARS-CoVMPro-IN-2 是一种有效的SARS-CoV-2 Mpro 抑制剂，IC50sub>值为 72.07 nM。病毒的主要蛋白酶 Mpro 作为加工病毒多蛋白的主要酶，有助于 SARS-CoV-2 在宿主细胞中的复制和转录，并已被定性为药物发现的有吸引力的靶点。SARS-CoVMPro-IN-2 具有研究 COVID-19 的潜力。
T38069 Aquastatin A

Aquastatin A is a fungal metabolite originally isolated fromF. aquaeductuumthat has diverse biological activities.1It is active againstS. aureus(MIC = 32 μg/ml) and inhibits enoyl-acyl carrier protein reductase (Fabl; IC50= 3.2 μM) andS. aureusfatty acid synthesis (IC50= 3.5 μM).2Aquastatin A also inhibits the Na+/K+-ATPase and H+/K+-ATPase (IC50s = 7.1 and 6.2 μM, respectively), as well as protein tyrosine phosphatase 1B (PTP1B; IC50= 0.19 μM).1,3 1.Hamano, K., Kinoshita-Okami, M., Minagawa, K....

天然产物

Tormentic acid
Cat.No: TN1118
Synonym: 2Α,19Α-二羟基熊果酸,委陵菜酸
Target: Immunology/Inflammation related
19-Hydroxybufalin
Cat.No: TN1198
Synonym:
Target: Others
Steviol-19-O-glucoside
Cat.No: TN2237
Synonym: Steviol-19-O-Glucoside,甜菊醇-19-葡萄糖苷
Target: Others
19-O-Acetylchaetoglobosin A
Cat.No: T35609
Synonym:
Target:
19,20-Epoxycytochalasin D
Cat.No: T35483
Synonym:
Target:
(19R,23E)-5b,19-Epoxy19-ethoxycucurbita-6,23-diene-3b,25-diol
Cat.No: T83578
Synonym:
Target:
19-Oxocinobufagin
Cat.No: TN1199
Synonym:
Target: Others
19-Hydroxy-10-deacetylbaccatin III
Cat.No: T83435
Synonym:
Target:
19-Oxocinobufotalin
Cat.No: TN1200
Synonym:
Target: Others
12E,14-Trien-19-oic acid
Cat.No: T83458
Synonym:
Target:
ent-17-Hydroxykaur-15-en-19-oic acid
Cat.No: TN3941
Synonym:
Target: Others
11,15-Dihydroxy-16-kauren-19-oic acid
Cat.No: TN1178
Synonym:
Target: Others
(23E)-5b,19-epoxycucurbita-6,23,25(26)-triene-3b-ol
Cat.No: T83570
Synonym:
Target:
Arjunetin
Cat.No: TN1401
Synonym:
Target: Others
Cichoriin
Cat.No: TN3651
Synonym:
Target: Others
Nonadecanoic acid
Cat.No: T8070
Synonym:
Target: Others
Chloroquine phosphate
Cat.No: T0194
Synonym: Chloroquine diphosphate,Aralen phosphate,磷酸氯喹,Chingamin phosphate
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
Punicalagin
Cat.No: T3921
Synonym: 安石榴甙,安石榴苷
Target: SARS-CoV, HBV
ent-3Beta-Angeloyloxykaur-16-en-19-oic acid
Cat.No: TN3948
Synonym:
Target: Others
ent-16beta,17-dihydroxy-9(11)-kauren-19-oic acid
Cat.No: TN3939
Synonym:
Target: Others
19-O-beta-D-carboxyglucopyranosyl-12-O-beta-D-glucopyranosyl-11,16-dihydroxyabieta-8,11,13-triene
Cat.No: TN6493
Synonym:
Target:
2-Epitormentic acid
Cat.No: TN2757
Synonym:
Target: Others
2,3-dihydrosciadopitysin
Cat.No: TN2700
Synonym:
Target: Others
1-(3,4-Dimethoxyphenyl)propane-1,2-diol
Cat.No: TN2486
Synonym:
Target: Others
7alpha-Hydroxystigmasterol
Cat.No: TN3254
Synonym:
Target: Others
Lacto-N-fucopentaose II
Cat.No: T75670
Synonym:
Target:
8,9-Didehydro-7-hydroxydolichodial
Cat.No: TN3269
Synonym:
Target: Others
16beta,17-Dihydroxy-ent-kaurane-19-oic acid
Cat.No: TN1194
Synonym:
Target: HIV Protease
5-(Z-Heptadec-8-enyl)resorcinol
Cat.No: TN5637
Synonym: 5-(8-Heptadecenyl)-1,3-benzenediol
Target:
Sphingosine (d14:1)
Cat.No: T38262
Synonym:
Target:
SARS-CoV MPro-IN-2
Cat.No: T72581
Synonym:
Target:
Aquastatin A
Cat.No: T38069
Synonym:
Target:
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