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Cat. No. Product Name Target Signaling Pathways
TN6783 Corysamine chloride

紫堇沙明碱,CORYSAMINE CHLORIDE(RG)

AChE Neuroscience
Corysamine chloride (CORYSAMINE CHLORIDE(RG)) 被确定可抑制 ACHE 的活性。
T5S2360 Corydaline

Corydalin,紫堇碱,延胡索甲素,(+)-Corydaline

P450; Virus Protease; Opioid Receptor; AChE Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Corydaline (Corydalin) 是从 Corydalis yanhusuo 提取的一种异喹啉生物碱,是一种新型促动力植物药的主要活性成分之一。它促进胃排空和小肠转运,促进胃的调节,具有抗乙酰胆碱酯酶、抗过敏和镇痛活性。
T5S2358 Dehydrocorydaline

Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline (13-Methylpalmatine) 是一种生物碱。它调节Bax,Bcl-2蛋白表达,激活caspase-7,caspase-8,并使PARP 失活。它能增强p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
T2S2362 Dehydrocorydaline nitrate

去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱

BCL; Others; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Others; Proteases/Proteasome
Dehydrocorydaline nitrate 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达,激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌、抗疟疾等功效。
T10990 Dehydrocorydaline chloride

盐酸脱氢紫堇碱,13-Methylpalmatine chloride

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline chloride (13-Methylpalmatine chloride) 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达;激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
T6S2356 Corynoline

紫蓳灵,堇醇灵碱,(+)-Corynoline

Nrf2; AChE Immunology/Inflammation; Neuroscience
Corynoline ((+)-Corynoline) 是可逆和非竞争性的乙酰胆碱酯酶抑制剂,IC50=30.6 μM。它可激活 Nrf2,具有抗炎作用。
TN2190 Scoulerine

Apoptosis; Beta-Secretase; BACE; Parasite Apoptosis; Microbiology/Virology; Neuroscience
Scoulerine 是抗有丝分裂化合物。它抑制细胞增殖,阻止细胞周期,并诱导癌细胞凋亡。它也是BACE1(淀粉样前体蛋白裂解酶 1) 的抑制剂。
TN1155 Corytuberine

Others Others
Corytuberine 具有促惊厥作用。 Corytuberine 的抗跳作用仅被纳洛酮抑制。
TN1526 Corydalmine

P450; Antifection Metabolism; Microbiology/Virology
Corydalmine exhibits antibacterial activities against Staphylococcus aureus and methicillin-resistant S. aureus strains.1-Corydalmine significantly inhibits spore germination of all the fungi at 100 to 1500 ppm. l-Corydalmine also exhibits potent analgesic activity in preclinical models, it is under development as an oral analgesic agent.
TN1484 Cheilanthifoline

NF-κB; Antifection Microbiology/Virology; NF-κB
Cheilanthifoline has anti-osteoclastogenic property, it gives significant inhibitions on receptor activator of nuclear factor-κB ligand-induced differentiation of mouse bone marrow-derived macrophages into multinucleated osteoclasts.
T5807 Stylopine hydrochloride

NOS; COX Immunology/Inflammation; Neuroscience
Stylopine hydrochloride 是一种生物碱类化合物,从紫堇属之植物块茎中分离得到,具有抗炎症和抗寄生虫作用。

天然产物

Corysamine chloride
Cat.No: TN6783
Synonym: 紫堇沙明碱,CORYSAMINE CHLORIDE(RG)
Target: AChE
Corydaline
Cat.No: T5S2360
Synonym: Corydalin,紫堇碱,延胡索甲素,(+)-Corydaline
Target: P450, Virus Protease, Opioid Receptor, AChE
Dehydrocorydaline
Cat.No: T5S2358
Synonym: Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Dehydrocorydaline nitrate
Cat.No: T2S2362
Synonym: 去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱
Target: BCL, Others, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Dehydrocorydaline chloride
Cat.No: T10990
Synonym: 盐酸脱氢紫堇碱,13-Methylpalmatine chloride
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Corynoline
Cat.No: T6S2356
Synonym: 紫蓳灵,堇醇灵碱,(+)-Corynoline
Target: Nrf2, AChE
Scoulerine
Cat.No: TN2190
Synonym:
Target: Apoptosis, Beta-Secretase, BACE, Parasite
Corytuberine
Cat.No: TN1155
Synonym:
Target: Others
Corydalmine
Cat.No: TN1526
Synonym:
Target: P450, Antifection
Cheilanthifoline
Cat.No: TN1484
Synonym:
Target: NF-κB, Antifection
Stylopine hydrochloride
Cat.No: T5807
Synonym:
Target: NOS, COX
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