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201

抑制剂 & 化合物

9

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1137L Pancreatic Polypeptide (human) acetate

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
Pancreatic Polypeptide (human) acetate 是一种 C 末端酰胺化的 36 个氨基酸肽,可作为神经肽 Y (NPY) Y4/Y5 受体激动剂。
TP1044L Pancreatic Polypeptide, rat acetate

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
Pancreatic Polypeptide, rat acetate 是 NPY 受体的激动剂,对 NPYR4 具有高亲和力。
TP1137 Pancreatic Polypeptide, human

Human pancreatic polypeptide

Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract.
TP1044 Pancreatic Polypeptide, rat

Rat pancreatic polypeptide

Pancreatic Polypeptide, rat is an agonist of NPY receptor, with high affinity at NPYR4. Pancreatic polypeptide (PP) is a 36-amino acid, C-terminally amidated peptide, and is a member of the PP-fold peptide family. It is produced and secreted by the PP cel
TP1731 Pancreatic Polypeptide, bovine

Agonist at Y4 neuropeptide Y receptors.
TP1963 [cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide

cpp1-7-npy19-23-ala31-aib32-gln34-hpancreatic-polypeptide,[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - hPancreatic Polypeptide

Potent, selective peptide agonist for the neuropeptide Y Y5 receptor (IC50 values for inhibition of NPY binding to human Y5, Y1, Y2 and Y4 receptors are 0.24, 530, > 500, and 51 nM respectively, Ki at Y5 = 0.1 - 0.15 nM). Stimulates food intake in vivo.
T76538 Pancreatic polypeptide

Pancreatic polypeptide 是由胰腺内分泌的 PP 细胞所分泌的多肽,具有调节胰腺分泌功能、影响肝糖原储存及胃肠分泌的作用。
T83072 Antifreeze Polypeptide 6 (winter flounder)

Antifreeze Polypeptide 6 (winter flounder)为美洲拟鲽特有的抗冻多肽组成成分之一,主要作用是通过抑制冰核生长来降低血浆的凝固点。
T80209 Human membrane-bound PD-L1 polypeptide

PD-1/PD-L1 Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation
Human membrane-bound PD-L1 polypeptide 作为抗原,可诱导生成相应的PD-L1抗体。
T37589 GIP (3-42), human

Gastric Inhibitory Polypeptide (3-42) (human)

IGF-1R Tyrosine Kinase/Adaptors
GIP (3-42), human (Gastric Inhibitory Polypeptide (3-42) (human)) 是一种多肽,可充当葡萄糖依赖性促胰岛素多肽 (GIP) 受体拮抗剂,在体内调节胰岛素分泌和 GIP 的代谢作用,可用于研究2型糖尿病。
T76308 Gastric Inhibitory Polypeptide (1-30), porcine

Gastric Inhibitory Polypeptide (1-30), porcine 缺乏天然胃抑制多肽 (GIP) C 端 12 个氨基酸残基,能够增强胰岛素和生长抑素的释放而发挥生物活性。
T82332 Gastric Inhibitory Polypeptide (6-30) amide (human)

Gastric Inhibitory Polypeptide (6-30) amide (human) 为一种肠促胰岛素激素,主要应用于糖尿病研究领域。
T83694 Gastric Inhibitory Peptide (1-42) (porcine) TFA

GIP (1-42),Glucose-dependent Insulinotropic Polypeptide (1-42)

胃抑制肽(GIP) (1-42)是一种内源性的42氨基酸肽类肠促素激素,能诱导胰岛素分泌。该激素在肠道神经内分泌K细胞和颌下腺中表达,并在餐后释放到循环中。GIP (1-42)抑制由组胺、五肽和胰岛素引起的胃酸和胃蛋白酶分泌,增加葡萄糖诱导的胰岛素释放,并在大鼠中刺激胃排空。
TP2315 glatiramer Acetate

Others Others
Glatiramer acetate 是髓鞘碱性蛋白的合成类似物和免疫调节剂,可用于多发性硬化症的研究。它能够诱导 T 辅助细胞 2 的特异性抑制细胞迁移到大脑并导致原位旁观者抑制。它能够于 MHC 分子强而杂乱的结合,因此与各种髓鞘抗原竞争,使其呈现给 T 细胞。
TP1054 PACAP (1-38), human, ovine, rat TFA

Pituitary Adenylate Cyclase Activating Polypeptide 38 (TFA)

PACAP (1-38), a novel neuropeptide isolated from the bovine hypothalamus is more active than vasoactive intestinal peptide (VIP) in stimulating adenylate cyclase (EC50=7 nM). PACAP 1-38 (10-9 M) increased substance P (SP), gastrin releasing peptide (GRP),
T83696 Gastric Inhibitory Peptide 1 (3-42) (human) TFA

Glucose-dependent Insulinotropic Polypeptide 3-42,GIP-1 (3-42)

胃抑制肽1(GIP-1) (3-42)是肠促胰岛素激素GIP的一个肽段,同时也是GIP受体的拮抗剂。它通过血清二肽基肽酶4(DDP-4)从GIP中形成。GIP-1 (3-42) (100 nM)在减少BRIN-BD11胰腺细胞的胰岛素分泌方面起作用。在以25 nmol/kg剂量给药的ob/ob糖尿病小鼠模型中,它能增加血浆葡萄糖水平并降低血浆胰岛素水平。
T83905 Brain Natriuretic Peptide-32 (rat) acetate

BNP (14-45),B-type Natriuretic Peptide-32,Brain Natriuretic Polypeptide-32,BNP-32

BNP-32(Brain natriuretic peptide-32)是心血管激素前体proBNP的肽段,能够结合大鼠血管平滑肌上的利钠肽受体(IC50 = 7.3 nM),并在同样的细胞中促进cGMP积累(EC50 = 170 nM)。BNP-32还能使经去甲肾上腺素预收缩的孤立大鼠主动脉条带松弛(EC50 = 6.7 nM),当以3 µg/kg的剂量给药时,能增加大鼠的尿量和尿液电解质排泄,并诱导低血压。
T75913 [cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic polypeptide TFA

[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide 为高效且选择性的神经肽 YY5 受体激动剂,其与 hY5 受体的结合 IC50 值为 0.24 nM,已知可促进饮食摄入。
T40495 Elastase from porcine pancreas

弹性蛋白酶,EC 3.2.1.35

Others Others
Elastase from porcine pancreas 由 240 个氨基酸残基组成,是一种丝氨酸蛋白酶,可以水解蛋白质和多肽。它可诱发仓鼠气肿。
TP1878 PACAP (1-38), human, ovine, rat

Pituitary Adenylate Cyclase Activating Polypeptide 38,腺苷酸环化酶激活肽-38(抗原),PACAP 1-38

PACAP GPCR/G Protein
PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) 是含有 38 个氨基酸残基的神经肽。它能够结合 PACAP I 型受体(IC50:4 nM)、PACAP II 型受体 VIP1(IC50:2 nM)、PACAP II 型受体 VIP2(IC50:1 nM)。
T5443 JQ-1 (carboxylic acid)

JQ-1 carboxylic acid

Epigenetic Reader Domain Chromatin/Epigenetic
JQ-1 (carboxylic acid) 是一种细胞渗透性 BRD4 抑制剂,对 BRD4(1) 和 BRD4(2) 的 IC50 分别为 77 和 33 nM。它是一种 (+)-JQ1 衍生物,可作为合成 PROTACs 的前体。
T37588 GIP (1-30) amide, porcine

This GIP fragment has potent insulinotropic activity in the isolated, perfused rat pancreas but greatly reduced somatostatinotropic activity in the isolated perfused rat stomach. The site responsible for insulinotropic activity apparently lies between residues 19 and 30 of GIP.
TP1389 Exendin-3/4 (64-86)

Others Others
Exendin-3/4 (64-86) 是一种多肽。
TP1711 5-Tamra-DRVYIHP

Others Others
5-Tamra-DRVYIHP 是一种含有用寡核苷酸标记的罗丹明衍生物的多肽。
TP2483L Cyclo(-RGDfC)acetate

Cyclo(-RGDfC)acetate(862772-11-0 free base)

Others Others
Cyclo(-RGDfC)acetate 是一种整合素 avb3 亲和多肽,一种环状 RGDfc 序列。
TP2484L Cyclo(-RGDyC)acetate

Others Others
Cyclo(-RGDyC)acetate 是一种整合素 avb3 亲和多肽,一种环状 RGDyc 序列。
T38662 Fmoc-Gly-Thr(psi(Me,Me)pro)-OH

Others Others
Fmoc-Gly-Thr(psi(Me,Me)pro)-OH 是一个二肽。
TP1950L PEN(mouse) acetate

proSAAS(221-242) Acetate,PEN(mouse) acetate (1236955-25-1 Free base)

Others Others
PEN(mouse) acetate (proSAAS(221-242) Acetate) (1236955-25-1 Free base)是一种多肽衍生物。
TP1071 Nociceptin

Orphanin FQ,孤菲肽

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Nociceptin (Orphanin FQ) 是一种 17 个氨基酸的多肽,是 nociceptin 受体的内源性配体,具有缓解疼痛的作用。
T40412L BAD (103-127) (human) acetate

BAD (103-127) (human) acetate (331762-68-6 Free base)

Others Others
BAD (103-127) (human) acetate 是一种来自于 BAD 的 BH3结构域的25-mer Bad 多肽,可拮抗 Bcl-xl 的作用。
TP1843L Systemin acetate(137181-56-7 free base)

Others Others
Systemin acetate(137181-56-7 free base) 是一种 18 个氨基酸的多肽,序列为 AVQSKPPSKRDPPKMQTD,存在于茄科植物(如番茄和马铃薯)中。
TP1627L Prepro VIP (111-122), human acetate

Prepro VIP (111-122), human acetate(123025-94-5 free base)

Others Others
Prepro VIP (111-122), human acetate(123025-94-5 free base) 是一种前血管活性肠多肽 (VIP) 衍生肽,对应于残基 111-122。
TP2320 Pramlintide acetate(151126-32-8 free base)

Others Others
Pramlintide acetate是人源淀粉样肽的多肽类似物。作为一种抗糖尿病药物,它在结直肠癌中展现出抗肿瘤活性。
T4579 Pentagastrin

五肽胃泌素,ICI-50123

Others; cholecystokinin GPCR/G Protein; Others
Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂,IC50=11 nM。它能够增强胃粘膜对酸的防御机制,并保护胃粘膜免受损伤。
TP1739L HEX3 acetate(688805-40-5 free base)

Others Others
HEX3 acetate(688805-40-5 free base) 是腺病毒六邻体的一个片段。 Hexon 是腺病毒的主要衣壳蛋白,由三个相同的多肽链组成。
TP1814L CEF4 acetate

CEF4 acetate(199727-68-9 free base)

Others Others
CEF4 acetate (CEF4 acetate (199727-68-9 free base)) 是对应于甲型流感病毒核壳蛋白的氨基酸序列342-351的多肽。
T38617L Biotin-TAT (47-57) acetate

Biotin-TAT (47-57) acetate(1231898-25-1 free base)

Others Others
Biotin-TAT (47-57) acetate 是一种生物素标记的 TAT 多肽和转录反式激活因子。 Biotin-TAT (47-57) acetate 是蛋白质转导结构域中使用广泛的肽之一。
TP1724L PUMA BH3 acetate

PUMA BH3 acetate(PUMA BH3 Free base)

BCL Apoptosis
PUMA BH3 acetate (PUMA BH3 Free base) 是一种 p53 凋亡阳性调节因子 (PUMA) BH3 结构域多肽,可作为 Bak 的直接激活剂,Kd 为 26 nM。
TP1125 Insulin(cattle)

牛胰岛素,Insulin from bovine pancreas,胰岛素

IGF-1R Tyrosine Kinase/Adaptors
Insulin cattle (Insulin from bovine pancreas) 是一种在胰腺 β 细胞中产生的两链多肽激素,在很多哺乳动物细胞培养体系中用作生长因子。
TP1076L AUNP-12 acetate

AUNP-12 acetate (1353563-85-5 Free base)

PD-1/PD-L1 Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation
AUNP-12 acetate 是一种 PD-1的多肽抑制剂,在抑制淋巴细胞增殖和效应功能上对 PD-1和 PD-2等效,具有免疫激活和良好的抗肿瘤活性。
T18723 Succinic anhydride

Others Others
Succinic anhydride 中的环状酸酐和不可裂解的 ADC 接头。它可以与化合物 4 反应,将前药连接到靶向多肽的胺或羟基 1 基团。
TP1410 Cecropin A

Antibacterial; Antibiotic Microbiology/Virology
Cecropin A 是37个氨基酸组成的线性多肽,表现出抗菌、抗炎和抗肿瘤的功效。
TP1155L Human growth hormone-releasing factor acetate

GHSR GPCR/G Protein
Human growth hormone-releasing factor acetate 是一种下丘脑多肽,通过与垂体前叶细胞上的 GHRH 受体 (GHRHR) 结合来刺激 GH 的产生和释放。
T31932 GJ071 oxalate

GJ 071,GJ-071,GJ071

Others Others
GJ071 oxalate 是一种无义抑制剂。无义抑制剂(NonSups)诱导“读出”,即在提前终止密码子处选择近同源tRNA,并将相应的氨基酸插入新生多肽中。
T37588L GIP (1-30) amide, porcine acetate

IGF-1R Tyrosine Kinase/Adaptors
GIP (1-30) amide, porcine acetate 是完全葡萄糖依赖性促胰岛素多肽 (GIP) 受体的激动剂。它可弱抑制胃酸分泌,强烈刺激胰岛素。
T76279 Retatrutide

LY3437943

Glucagon Receptor GPCR/G Protein
Retatrutide (LY3437943) 是胰高血糖素受体、葡萄糖依赖性促胰岛素多肽受体和胰高血糖素样肽-1 受体三重激动剂,对GCGR、GIPR 和 GLP-1R 具有抑制作用。Retatrutide 可用研究肥胖症。
TP1535L GPLGIAGQ acetate

GPLGIAGQ acetate(109053-09-0 Free base)

MMP Proteases/Proteasome
GPLGIAGQ acetate 是一种 MMP2 可切割的多肽。GPLGIAGQ acetate 可用作脂质体和胶束纳米载体中的刺激敏感接头,以在光动力治疗中合成独特的 MMP2 靶向光敏剂。
T35373L Bulevirtide (Myrcludex B) acetate

HBV Microbiology/Virology
Bulevirtide (Myrcludex B) acetate 是一种病毒粒子进入抑制剂,可阻断病毒粒子的肝细胞进入途径,即肝钠/牛磺胆酸盐协同转运多肽 (NTCP) 受体。它可用于 HBV 和 HDV 感染研究。
TP1111 Tirzepatide

LY-3298176

Glucagon Receptor GPCR/G Protein
Tirzepatide (LY-3298176) 是葡萄糖依赖性多肽 (GIP) 和胰高血糖素样肽-1 (GLP-1) 受体双重激动剂,具有神经保护活性,可改善血压并降低低密度脂蛋白 (LDL) 胆固醇和甘油三酯,可以用于研究糖尿病和肥胖症。
T78105 PAC1R antagonist 1

PACAP GPCR/G Protein
PAC1R antagonist 1为一种具有口服活性的 PAC1 受体拮抗剂,可抑制由垂体腺苷酸环化酶激活多肽(PACAP)及神经损伤所诱导的异常性疼痛,可用于研究肿瘤和与免疫相关的疾病。

化合物

Pancreatic Polypeptide (human) acetate
Cat.No: TP1137L
Synonym:
Target: Neuropeptide Y Receptor
Pancreatic Polypeptide, rat acetate
Cat.No: TP1044L
Synonym:
Target: Neuropeptide Y Receptor
Pancreatic Polypeptide, human
Cat.No: TP1137
Synonym: Human pancreatic polypeptide
Target:
Pancreatic Polypeptide, rat
Cat.No: TP1044
Synonym: Rat pancreatic polypeptide
Target:
Pancreatic Polypeptide, bovine
Cat.No: TP1731
Synonym:
Target:
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
Cat.No: TP1963
Synonym: cpp1-7-npy19-23-ala31-aib32-gln34-hpancreatic-polypeptide,[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - hPancreatic Polypeptide
Target:
Pancreatic polypeptide
Cat.No: T76538
Synonym:
Target:
Antifreeze Polypeptide 6 (winter flounder)
Cat.No: T83072
Synonym:
Target:
Human membrane-bound PD-L1 polypeptide
Cat.No: T80209
Synonym:
Target: PD-1/PD-L1
GIP (3-42), human
Cat.No: T37589
Synonym: Gastric Inhibitory Polypeptide (3-42) (human)
Target: IGF-1R
Gastric Inhibitory Polypeptide (1-30), porcine
Cat.No: T76308
Synonym:
Target:
Gastric Inhibitory Polypeptide (6-30) amide (human)
Cat.No: T82332
Synonym:
Target:
Gastric Inhibitory Peptide (1-42) (porcine) TFA
Cat.No: T83694
Synonym: GIP (1-42),Glucose-dependent Insulinotropic Polypeptide (1-42)
Target:
glatiramer Acetate
Cat.No: TP2315
Synonym:
Target: Others
PACAP (1-38), human, ovine, rat TFA
Cat.No: TP1054
Synonym: Pituitary Adenylate Cyclase Activating Polypeptide 38 (TFA)
Target:
Gastric Inhibitory Peptide 1 (3-42) (human) TFA
Cat.No: T83696
Synonym: Glucose-dependent Insulinotropic Polypeptide 3-42,GIP-1 (3-42)
Target:
Brain Natriuretic Peptide-32 (rat) acetate
Cat.No: T83905
Synonym: BNP (14-45),B-type Natriuretic Peptide-32,Brain Natriuretic Polypeptide-32,BNP-32
Target:
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic polypeptide TFA
Cat.No: T75913
Synonym:
Target:
Elastase from porcine pancreas
Cat.No: T40495
Synonym: 弹性蛋白酶,EC 3.2.1.35
Target: Others
PACAP (1-38), human, ovine, rat
Cat.No: TP1878
Synonym: Pituitary Adenylate Cyclase Activating Polypeptide 38,腺苷酸环化酶激活肽-38(抗原),PACAP 1-38
Target: PACAP
JQ-1 (carboxylic acid)
Cat.No: T5443
Synonym: JQ-1 carboxylic acid
Target: Epigenetic Reader Domain
GIP (1-30) amide, porcine
Cat.No: T37588
Synonym:
Target:
Exendin-3/4 (64-86)
Cat.No: TP1389
Synonym:
Target: Others
5-Tamra-DRVYIHP
Cat.No: TP1711
Synonym:
Target: Others
Cyclo(-RGDfC)acetate
Cat.No: TP2483L
Synonym: Cyclo(-RGDfC)acetate(862772-11-0 free base)
Target: Others
Cyclo(-RGDyC)acetate
Cat.No: TP2484L
Synonym:
Target: Others
Fmoc-Gly-Thr(psi(Me,Me)pro)-OH
Cat.No: T38662
Synonym:
Target: Others
PEN(mouse) acetate
Cat.No: TP1950L
Synonym: proSAAS(221-242) Acetate,PEN(mouse) acetate (1236955-25-1 Free base)
Target: Others
Nociceptin
Cat.No: TP1071
Synonym: Orphanin FQ,孤菲肽
Target: Opioid Receptor
BAD (103-127) (human) acetate
Cat.No: T40412L
Synonym: BAD (103-127) (human) acetate (331762-68-6 Free base)
Target: Others
Systemin acetate(137181-56-7 free base)
Cat.No: TP1843L
Synonym:
Target: Others
Prepro VIP (111-122), human acetate
Cat.No: TP1627L
Synonym: Prepro VIP (111-122), human acetate(123025-94-5 free base)
Target: Others
Pramlintide acetate(151126-32-8 free base)
Cat.No: TP2320
Synonym:
Target: Others
Pentagastrin
Cat.No: T4579
Synonym: 五肽胃泌素,ICI-50123
Target: Others, cholecystokinin
HEX3 acetate(688805-40-5 free base)
Cat.No: TP1739L
Synonym:
Target: Others
CEF4 acetate
Cat.No: TP1814L
Synonym: CEF4 acetate(199727-68-9 free base)
Target: Others
Biotin-TAT (47-57) acetate
Cat.No: T38617L
Synonym: Biotin-TAT (47-57) acetate(1231898-25-1 free base)
Target: Others
PUMA BH3 acetate
Cat.No: TP1724L
Synonym: PUMA BH3 acetate(PUMA BH3 Free base)
Target: BCL
Insulin(cattle)
Cat.No: TP1125
Synonym: 牛胰岛素,Insulin from bovine pancreas,胰岛素
Target: IGF-1R
AUNP-12 acetate
Cat.No: TP1076L
Synonym: AUNP-12 acetate (1353563-85-5 Free base)
Target: PD-1/PD-L1
Succinic anhydride
Cat.No: T18723
Synonym:
Target: Others
Cecropin A
Cat.No: TP1410
Synonym:
Target: Antibacterial, Antibiotic
Human growth hormone-releasing factor acetate
Cat.No: TP1155L
Synonym:
Target: GHSR
GJ071 oxalate
Cat.No: T31932
Synonym: GJ 071,GJ-071,GJ071
Target: Others
GIP (1-30) amide, porcine acetate
Cat.No: T37588L
Synonym:
Target: IGF-1R
Retatrutide
Cat.No: T76279
Synonym: LY3437943
Target: Glucagon Receptor
GPLGIAGQ acetate
Cat.No: TP1535L
Synonym: GPLGIAGQ acetate(109053-09-0 Free base)
Target: MMP
Bulevirtide (Myrcludex B) acetate
Cat.No: T35373L
Synonym:
Target: HBV
Tirzepatide
Cat.No: TP1111
Synonym: LY-3298176
Target: Glucagon Receptor
PAC1R antagonist 1
Cat.No: T78105
Synonym:
Target: PACAP
Cat. No. Product Name Target Signaling Pathways
T21518 Colistin methanesulfonate sodium salt

粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt)

Cell wall; Antibacterial Immunology/Inflammation; Microbiology/Virology
Colistin methanesulfonate sodium salt (Colistimethate Sodium) 是一种来自 Bacillus colistinus 的环状多肽抗生素,由多粘菌素 E1 和 E2 组成。
T1245 Colistin sulfate

Colistin sulfate (1066-17-7 free base),Polymixin E Sulfate,Polymyxin E Sulfate,硫酸粘杆菌素

Cell wall; Antibacterial; Antibiotic; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology
Colistin sulfate (Colistin sulfate (1066-17-7 free base)) 是抑制革兰氏阴性细菌的一种多肽抗生素,与革兰氏阴性细菌的外细胞膜中的脂多糖和磷脂结合起作用。
T1130 Gramicidin

短杆菌肽,Gramicidinum,Gramicidine,Gramicidina

MRP; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology
Gramicidin (Gramicidine) 是一种抗菌肽。它通过组装成膜中的通道,增加其对阳离子的渗透性。
T0945 Cyclosporin A

环孢素,Cyclosporine A,Ciclosporin,Cyclosporine,环孢菌素

Phosphatase; Antibiotic; Complement System Immunology/Inflammation; Metabolism; Microbiology/Virology
Cyclosporin A 属于天然产物,是一种真菌的活性代谢产物,一种环状多肽。Cyclosporin A 是一种能与亲环素结合的免疫抑制剂,可以抑制 calcineurin (IC50=7 nM)。
T41042 Gramicidin C

Gramicidin C, a naturally occurring polypeptide antibiotic, is isolated from B. brevis var. G.B.
T38805 Euphol acetate

Euphol acetate, a triterpene found in Euphorbia broteri, has demonstrated inhibitory effects on the hepatic transport proteins known as organic anion-transporting polypeptide 1/3 (OATP1B1/3).
T25211 CC 1014

CC1014,CC-1014,NSC-356885,NSC356885,NSC 356885

CC 1014 is a polypeptide antibiotic isolated from Penicillium lilacinum that inhibits phosphorylation of ADP, Mg ATPase.
T17185 Tyrothricin

Others Others
Tyrothricin is a polypeptide antibiotic mixture isolated from Bacillus brevis and consists of tyrocidines and gramicidins. Tyrothricin displays activity against bacteria, fungi, and some viruses.
T75974 Cecropin A TFA

Cecropin A TFA 是由 37 个氨基酸残基构成的线性抗菌肽,从 Hyalaphora cecropiapupae 得到,具有抗菌、抗炎和抗癌作用。

天然产物

Colistin methanesulfonate sodium salt
Cat.No: T21518
Synonym: 粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt)
Target: Cell wall, Antibacterial
Colistin sulfate
Cat.No: T1245
Synonym: Colistin sulfate (1066-17-7 free base),Polymixin E Sulfate,Polymyxin E Sulfate,硫酸粘杆菌素
Target: Cell wall, Antibacterial, Antibiotic, Autophagy
Gramicidin
Cat.No: T1130
Synonym: 短杆菌肽,Gramicidinum,Gramicidine,Gramicidina
Target: MRP, Antibacterial, Antibiotic
Cyclosporin A
Cat.No: T0945
Synonym: 环孢素,Cyclosporine A,Ciclosporin,Cyclosporine,环孢菌素
Target: Phosphatase, Antibiotic, Complement System
Gramicidin C
Cat.No: T41042
Synonym:
Target:
Euphol acetate
Cat.No: T38805
Synonym:
Target:
CC 1014
Cat.No: T25211
Synonym: CC1014,CC-1014,NSC-356885,NSC356885,NSC 356885
Target:
Tyrothricin
Cat.No: T17185
Synonym:
Target: Others
Cecropin A TFA
Cat.No: T75974
Synonym:
Target:
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