201
9
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP1137L |
Pancreatic Polypeptide (human) acetate
|
Neuropeptide Y Receptor | GPCR/G Protein; Neuroscience |
Pancreatic Polypeptide (human) acetate 是一种 C 末端酰胺化的 36 个氨基酸肽,可作为神经肽 Y (NPY) Y4/Y5 受体激动剂。 | |||
TP1044L |
Pancreatic Polypeptide, rat acetate
|
Neuropeptide Y Receptor | GPCR/G Protein; Neuroscience |
Pancreatic Polypeptide, rat acetate 是 NPY 受体的激动剂,对 NPYR4 具有高亲和力。 | |||
TP1137 |
Pancreatic Polypeptide, human
Human pancreatic polypeptide |
||
Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract. | |||
TP1044 |
Pancreatic Polypeptide, rat
Rat pancreatic polypeptide |
||
Pancreatic Polypeptide, rat is an agonist of NPY receptor, with high affinity at NPYR4. Pancreatic polypeptide (PP) is a 36-amino acid, C-terminally amidated peptide, and is a member of the PP-fold peptide family. It is produced and secreted by the PP cel | |||
TP1731 |
Pancreatic Polypeptide, bovine
|
||
Agonist at Y4 neuropeptide Y receptors. | |||
TP1963 |
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
cpp1-7-npy19-23-ala31-aib32-gln34-hpancreatic-polypeptide,[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - hPancreatic Polypeptide |
||
Potent, selective peptide agonist for the neuropeptide Y Y5 receptor (IC50 values for inhibition of NPY binding to human Y5, Y1, Y2 and Y4 receptors are 0.24, 530, > 500, and 51 nM respectively, Ki at Y5 = 0.1 - 0.15 nM). Stimulates food intake in vivo. | |||
T76538 |
Pancreatic polypeptide
|
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Pancreatic polypeptide 是由胰腺内分泌的 PP 细胞所分泌的多肽,具有调节胰腺分泌功能、影响肝糖原储存及胃肠分泌的作用。 | |||
T83072 |
Antifreeze Polypeptide 6 (winter flounder)
|
||
Antifreeze Polypeptide 6 (winter flounder)为美洲拟鲽特有的抗冻多肽组成成分之一,主要作用是通过抑制冰核生长来降低血浆的凝固点。 | |||
T80209 |
Human membrane-bound PD-L1 polypeptide
|
PD-1/PD-L1 | Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation |
Human membrane-bound PD-L1 polypeptide 作为抗原,可诱导生成相应的PD-L1抗体。 | |||
T37589 |
GIP (3-42), human
Gastric Inhibitory Polypeptide (3-42) (human) |
IGF-1R | Tyrosine Kinase/Adaptors |
GIP (3-42), human (Gastric Inhibitory Polypeptide (3-42) (human)) 是一种多肽,可充当葡萄糖依赖性促胰岛素多肽 (GIP) 受体拮抗剂,在体内调节胰岛素分泌和 GIP 的代谢作用,可用于研究2型糖尿病。 | |||
T76308 |
Gastric Inhibitory Polypeptide (1-30), porcine
|
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Gastric Inhibitory Polypeptide (1-30), porcine 缺乏天然胃抑制多肽 (GIP) C 端 12 个氨基酸残基,能够增强胰岛素和生长抑素的释放而发挥生物活性。 | |||
T82332 |
Gastric Inhibitory Polypeptide (6-30) amide (human)
|
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Gastric Inhibitory Polypeptide (6-30) amide (human) 为一种肠促胰岛素激素,主要应用于糖尿病研究领域。 | |||
T83694 |
Gastric Inhibitory Peptide (1-42) (porcine) TFA
GIP (1-42),Glucose-dependent Insulinotropic Polypeptide (1-42) |
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胃抑制肽(GIP) (1-42)是一种内源性的42氨基酸肽类肠促素激素,能诱导胰岛素分泌。该激素在肠道神经内分泌K细胞和颌下腺中表达,并在餐后释放到循环中。GIP (1-42)抑制由组胺、五肽和胰岛素引起的胃酸和胃蛋白酶分泌,增加葡萄糖诱导的胰岛素释放,并在大鼠中刺激胃排空。 | |||
TP2315 |
glatiramer Acetate
|
Others | Others |
Glatiramer acetate 是髓鞘碱性蛋白的合成类似物和免疫调节剂,可用于多发性硬化症的研究。它能够诱导 T 辅助细胞 2 的特异性抑制细胞迁移到大脑并导致原位旁观者抑制。它能够于 MHC 分子强而杂乱的结合,因此与各种髓鞘抗原竞争,使其呈现给 T 细胞。 | |||
TP1054 |
PACAP (1-38), human, ovine, rat TFA
Pituitary Adenylate Cyclase Activating Polypeptide 38 (TFA) |
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PACAP (1-38), a novel neuropeptide isolated from the bovine hypothalamus is more active than vasoactive intestinal peptide (VIP) in stimulating adenylate cyclase (EC50=7 nM). PACAP 1-38 (10-9 M) increased substance P (SP), gastrin releasing peptide (GRP), | |||
T83696 |
Gastric Inhibitory Peptide 1 (3-42) (human) TFA
Glucose-dependent Insulinotropic Polypeptide 3-42,GIP-1 (3-42) |
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胃抑制肽1(GIP-1) (3-42)是肠促胰岛素激素GIP的一个肽段,同时也是GIP受体的拮抗剂。它通过血清二肽基肽酶4(DDP-4)从GIP中形成。GIP-1 (3-42) (100 nM)在减少BRIN-BD11胰腺细胞的胰岛素分泌方面起作用。在以25 nmol/kg剂量给药的ob/ob糖尿病小鼠模型中,它能增加血浆葡萄糖水平并降低血浆胰岛素水平。 | |||
T83905 |
Brain Natriuretic Peptide-32 (rat) acetate
BNP (14-45),B-type Natriuretic Peptide-32,Brain Natriuretic Polypeptide-32,BNP-32 |
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BNP-32(Brain natriuretic peptide-32)是心血管激素前体proBNP的肽段,能够结合大鼠血管平滑肌上的利钠肽受体(IC50 = 7.3 nM),并在同样的细胞中促进cGMP积累(EC50 = 170 nM)。BNP-32还能使经去甲肾上腺素预收缩的孤立大鼠主动脉条带松弛(EC50 = 6.7 nM),当以3 µg/kg的剂量给药时,能增加大鼠的尿量和尿液电解质排泄,并诱导低血压。 | |||
T75913 |
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic polypeptide TFA
|
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[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide 为高效且选择性的神经肽 YY5 受体激动剂,其与 hY5 受体的结合 IC50 值为 0.24 nM,已知可促进饮食摄入。 | |||
T40495 |
Elastase from porcine pancreas
弹性蛋白酶,EC 3.2.1.35 |
Others | Others |
Elastase from porcine pancreas 由 240 个氨基酸残基组成,是一种丝氨酸蛋白酶,可以水解蛋白质和多肽。它可诱发仓鼠气肿。 | |||
TP1878 |
PACAP (1-38), human, ovine, rat
Pituitary Adenylate Cyclase Activating Polypeptide 38,腺苷酸环化酶激活肽-38(抗原),PACAP 1-38 |
PACAP | GPCR/G Protein |
PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) 是含有 38 个氨基酸残基的神经肽。它能够结合 PACAP I 型受体(IC50:4 nM)、PACAP II 型受体 VIP1(IC50:2 nM)、PACAP II 型受体 VIP2(IC50:1 nM)。 | |||
T5443 |
JQ-1 (carboxylic acid)
JQ-1 carboxylic acid |
Epigenetic Reader Domain | Chromatin/Epigenetic |
JQ-1 (carboxylic acid) 是一种细胞渗透性 BRD4 抑制剂,对 BRD4(1) 和 BRD4(2) 的 IC50 分别为 77 和 33 nM。它是一种 (+)-JQ1 衍生物,可作为合成 PROTACs 的前体。 | |||
T37588 |
GIP (1-30) amide, porcine
|
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This GIP fragment has potent insulinotropic activity in the isolated, perfused rat pancreas but greatly reduced somatostatinotropic activity in the isolated perfused rat stomach. The site responsible for insulinotropic activity apparently lies between residues 19 and 30 of GIP. | |||
TP1389 |
Exendin-3/4 (64-86)
|
Others | Others |
Exendin-3/4 (64-86) 是一种多肽。 | |||
TP1711 |
5-Tamra-DRVYIHP
|
Others | Others |
5-Tamra-DRVYIHP 是一种含有用寡核苷酸标记的罗丹明衍生物的多肽。 | |||
TP2483L |
Cyclo(-RGDfC)acetate
Cyclo(-RGDfC)acetate(862772-11-0 free base) |
Others | Others |
Cyclo(-RGDfC)acetate 是一种整合素 avb3 亲和多肽,一种环状 RGDfc 序列。 | |||
TP2484L |
Cyclo(-RGDyC)acetate
|
Others | Others |
Cyclo(-RGDyC)acetate 是一种整合素 avb3 亲和多肽,一种环状 RGDyc 序列。 | |||
T38662 |
Fmoc-Gly-Thr(psi(Me,Me)pro)-OH
|
Others | Others |
Fmoc-Gly-Thr(psi(Me,Me)pro)-OH 是一个二肽。 | |||
TP1950L |
PEN(mouse) acetate
proSAAS(221-242) Acetate,PEN(mouse) acetate (1236955-25-1 Free base) |
Others | Others |
PEN(mouse) acetate (proSAAS(221-242) Acetate) (1236955-25-1 Free base)是一种多肽衍生物。 | |||
TP1071 |
Nociceptin
Orphanin FQ,孤菲肽 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Nociceptin (Orphanin FQ) 是一种 17 个氨基酸的多肽,是 nociceptin 受体的内源性配体,具有缓解疼痛的作用。 | |||
T40412L |
BAD (103-127) (human) acetate
BAD (103-127) (human) acetate (331762-68-6 Free base) |
Others | Others |
BAD (103-127) (human) acetate 是一种来自于 BAD 的 BH3结构域的25-mer Bad 多肽,可拮抗 Bcl-xl 的作用。 | |||
TP1843L |
Systemin acetate(137181-56-7 free base)
|
Others | Others |
Systemin acetate(137181-56-7 free base) 是一种 18 个氨基酸的多肽,序列为 AVQSKPPSKRDPPKMQTD,存在于茄科植物(如番茄和马铃薯)中。 | |||
TP1627L |
Prepro VIP (111-122), human acetate
Prepro VIP (111-122), human acetate(123025-94-5 free base) |
Others | Others |
Prepro VIP (111-122), human acetate(123025-94-5 free base) 是一种前血管活性肠多肽 (VIP) 衍生肽,对应于残基 111-122。 | |||
TP2320 |
Pramlintide acetate(151126-32-8 free base)
|
Others | Others |
Pramlintide acetate是人源淀粉样肽的多肽类似物。作为一种抗糖尿病药物,它在结直肠癌中展现出抗肿瘤活性。 | |||
T4579 |
Pentagastrin
五肽胃泌素,ICI-50123 |
Others; cholecystokinin | GPCR/G Protein; Others |
Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂,IC50=11 nM。它能够增强胃粘膜对酸的防御机制,并保护胃粘膜免受损伤。 | |||
TP1739L |
HEX3 acetate(688805-40-5 free base)
|
Others | Others |
HEX3 acetate(688805-40-5 free base) 是腺病毒六邻体的一个片段。 Hexon 是腺病毒的主要衣壳蛋白,由三个相同的多肽链组成。 | |||
TP1814L |
CEF4 acetate
CEF4 acetate(199727-68-9 free base) |
Others | Others |
CEF4 acetate (CEF4 acetate (199727-68-9 free base)) 是对应于甲型流感病毒核壳蛋白的氨基酸序列342-351的多肽。 | |||
T38617L |
Biotin-TAT (47-57) acetate
Biotin-TAT (47-57) acetate(1231898-25-1 free base) |
Others | Others |
Biotin-TAT (47-57) acetate 是一种生物素标记的 TAT 多肽和转录反式激活因子。 Biotin-TAT (47-57) acetate 是蛋白质转导结构域中使用广泛的肽之一。 | |||
TP1724L |
PUMA BH3 acetate
PUMA BH3 acetate(PUMA BH3 Free base) |
BCL | Apoptosis |
PUMA BH3 acetate (PUMA BH3 Free base) 是一种 p53 凋亡阳性调节因子 (PUMA) BH3 结构域多肽,可作为 Bak 的直接激活剂,Kd 为 26 nM。 | |||
TP1125 |
Insulin(cattle)
牛胰岛素,Insulin from bovine pancreas,胰岛素 |
IGF-1R | Tyrosine Kinase/Adaptors |
Insulin cattle (Insulin from bovine pancreas) 是一种在胰腺 β 细胞中产生的两链多肽激素,在很多哺乳动物细胞培养体系中用作生长因子。 | |||
TP1076L |
AUNP-12 acetate
AUNP-12 acetate (1353563-85-5 Free base) |
PD-1/PD-L1 | Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation |
AUNP-12 acetate 是一种 PD-1的多肽抑制剂,在抑制淋巴细胞增殖和效应功能上对 PD-1和 PD-2等效,具有免疫激活和良好的抗肿瘤活性。 | |||
T18723 |
Succinic anhydride
|
Others | Others |
Succinic anhydride 中的环状酸酐和不可裂解的 ADC 接头。它可以与化合物 4 反应,将前药连接到靶向多肽的胺或羟基 1 基团。 | |||
TP1410 |
Cecropin A
|
Antibacterial; Antibiotic | Microbiology/Virology |
Cecropin A 是37个氨基酸组成的线性多肽,表现出抗菌、抗炎和抗肿瘤的功效。 | |||
TP1155L |
Human growth hormone-releasing factor acetate
|
GHSR | GPCR/G Protein |
Human growth hormone-releasing factor acetate 是一种下丘脑多肽,通过与垂体前叶细胞上的 GHRH 受体 (GHRHR) 结合来刺激 GH 的产生和释放。 | |||
T31932 |
GJ071 oxalate
GJ 071,GJ-071,GJ071 |
Others | Others |
GJ071 oxalate 是一种无义抑制剂。无义抑制剂(NonSups)诱导“读出”,即在提前终止密码子处选择近同源tRNA,并将相应的氨基酸插入新生多肽中。 | |||
T37588L |
GIP (1-30) amide, porcine acetate
|
IGF-1R | Tyrosine Kinase/Adaptors |
GIP (1-30) amide, porcine acetate 是完全葡萄糖依赖性促胰岛素多肽 (GIP) 受体的激动剂。它可弱抑制胃酸分泌,强烈刺激胰岛素。 | |||
T76279 |
Retatrutide
LY3437943 |
Glucagon Receptor | GPCR/G Protein |
Retatrutide (LY3437943) 是胰高血糖素受体、葡萄糖依赖性促胰岛素多肽受体和胰高血糖素样肽-1 受体三重激动剂,对GCGR、GIPR 和 GLP-1R 具有抑制作用。Retatrutide 可用研究肥胖症。 | |||
TP1535L |
GPLGIAGQ acetate
GPLGIAGQ acetate(109053-09-0 Free base) |
MMP | Proteases/Proteasome |
GPLGIAGQ acetate 是一种 MMP2 可切割的多肽。GPLGIAGQ acetate 可用作脂质体和胶束纳米载体中的刺激敏感接头,以在光动力治疗中合成独特的 MMP2 靶向光敏剂。 | |||
T35373L |
Bulevirtide (Myrcludex B) acetate
|
HBV | Microbiology/Virology |
Bulevirtide (Myrcludex B) acetate 是一种病毒粒子进入抑制剂,可阻断病毒粒子的肝细胞进入途径,即肝钠/牛磺胆酸盐协同转运多肽 (NTCP) 受体。它可用于 HBV 和 HDV 感染研究。 | |||
TP1111 |
Tirzepatide
LY-3298176 |
Glucagon Receptor | GPCR/G Protein |
Tirzepatide (LY-3298176) 是葡萄糖依赖性多肽 (GIP) 和胰高血糖素样肽-1 (GLP-1) 受体双重激动剂,具有神经保护活性,可改善血压并降低低密度脂蛋白 (LDL) 胆固醇和甘油三酯,可以用于研究糖尿病和肥胖症。 | |||
T78105 |
PAC1R antagonist 1
|
PACAP | GPCR/G Protein |
PAC1R antagonist 1为一种具有口服活性的 PAC1 受体拮抗剂,可抑制由垂体腺苷酸环化酶激活多肽(PACAP)及神经损伤所诱导的异常性疼痛,可用于研究肿瘤和与免疫相关的疾病。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T21518 |
Colistin methanesulfonate sodium salt
粘杆菌素甲基磺酸钠,Colistin Methanesulfonate (sodium salt) |
Cell wall; Antibacterial | Immunology/Inflammation; Microbiology/Virology |
Colistin methanesulfonate sodium salt (Colistimethate Sodium) 是一种来自 Bacillus colistinus 的环状多肽抗生素,由多粘菌素 E1 和 E2 组成。 | |||
T1245 |
Colistin sulfate
Colistin sulfate (1066-17-7 free base),Polymixin E Sulfate,Polymyxin E Sulfate,硫酸粘杆菌素 |
Cell wall; Antibacterial; Antibiotic; Autophagy | Autophagy; Immunology/Inflammation; Microbiology/Virology |
Colistin sulfate (Colistin sulfate (1066-17-7 free base)) 是抑制革兰氏阴性细菌的一种多肽抗生素,与革兰氏阴性细菌的外细胞膜中的脂多糖和磷脂结合起作用。 | |||
T1130 |
Gramicidin
短杆菌肽,Gramicidinum,Gramicidine,Gramicidina |
MRP; Antibacterial; Antibiotic | Immunology/Inflammation; Microbiology/Virology |
Gramicidin (Gramicidine) 是一种抗菌肽。它通过组装成膜中的通道,增加其对阳离子的渗透性。 | |||
T0945 |
Cyclosporin A
环孢素,Cyclosporine A,Ciclosporin,Cyclosporine,环孢菌素 |
Phosphatase; Antibiotic; Complement System | Immunology/Inflammation; Metabolism; Microbiology/Virology |
Cyclosporin A 属于天然产物,是一种真菌的活性代谢产物,一种环状多肽。Cyclosporin A 是一种能与亲环素结合的免疫抑制剂,可以抑制 calcineurin (IC50=7 nM)。 | |||
T41042 |
Gramicidin C
|
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Gramicidin C, a naturally occurring polypeptide antibiotic, is isolated from B. brevis var. G.B. | |||
T38805 |
Euphol acetate
|
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Euphol acetate, a triterpene found in Euphorbia broteri, has demonstrated inhibitory effects on the hepatic transport proteins known as organic anion-transporting polypeptide 1/3 (OATP1B1/3). | |||
T25211 |
CC 1014
CC1014,CC-1014,NSC-356885,NSC356885,NSC 356885 |
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CC 1014 is a polypeptide antibiotic isolated from Penicillium lilacinum that inhibits phosphorylation of ADP, Mg ATPase. | |||
T17185 |
Tyrothricin
|
Others | Others |
Tyrothricin is a polypeptide antibiotic mixture isolated from Bacillus brevis and consists of tyrocidines and gramicidins. Tyrothricin displays activity against bacteria, fungi, and some viruses. | |||
T75974 |
Cecropin A TFA
|
||
Cecropin A TFA 是由 37 个氨基酸残基构成的线性抗菌肽,从 Hyalaphora cecropiapupae 得到,具有抗菌、抗炎和抗癌作用。 |