14
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7943 |
Fluphenazine decanoate
|
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Fluphenazine decanoate 是一种高度连续的多巴胺 D2受体阻滞剂,是一种长效吩噻嗪抗精神病药,用于精神分裂症的研究。 | |||
T2390 |
Cevimeline hydrochloride hemihydrate
|
AChR | Neuroscience |
Cevimeline hydrochloride hemihydrate 是乙酰胆碱的奎尼丁衍生物,也是选择性的和口服活性的毒蕈碱型M1和M3受体激动剂。它可穿过血脑屏障,刺激唾液腺分泌,用作口干症的催涎剂。 | |||
T0734 |
Antipyrine
安替比林,Phenazone,Phenazon |
COX | Immunology/Inflammation; Neuroscience |
Antipyrine (Phenazone) 是一种退烧剂和止痛剂。它可用作氧化药物代谢的探针药物,常用于评估人类的肝氧化能力。 | |||
T0979 |
Dequalinium chloride
Dequafungan,地喹氯铵,Danical,Decabis |
Potassium Channel; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel |
Dequalinium chloride (Decabis) 是一种apamin 敏感型的钾离子通道选择性阻断剂。 | |||
T0858 |
Flufenamic acid
Arlef,Nichisedan,氟灭酸,氟芬那酸,Achless |
Potassium Channel; Calcium Channel; Chloride channel; COX; AMPK; Parasite | Chromatin/Epigenetic; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling |
Flufenamic acid (Arlef) 是一种非甾体类抗炎剂,是一种邻氨基苯甲酸衍生物,具有镇痛、抗炎和解热的特性。 它用于肌肉骨骼和关节疾病。 | |||
T20570 |
Labetalol
Apo-Labetalol,Albetol,Trandate,Dilevalol,拉贝洛尔,Normodyne |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Labetalol (Apo-Labetalol) 是一种抗高血压药物,可用于心血管疾病的研究,如妊娠期高血压。它是一种口服具有活性的选择性 α1- 和非选择性 β-肾上腺素能受体 (adrenergic receptor) 竞争性拮抗剂。 | |||
T4553 |
Procaine penicillin G
普鲁卡因青霉素,Duphapen,Hydracillin,Hostacillin |
Antibiotic | Microbiology/Virology |
Procaine penicillin G (Duphapen) 是一种抗生素,可用于治疗多种细菌感染。具体来说,它用于梅毒、炭疽、口腔感染、肺炎、白喉、蜂窝组织炎和动物咬伤。 | |||
T34228 |
Quinethazone
Quinethazon,Hydromox,Aquamox,Quinethazonum,Chinethazonum |
||
Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels. | |||
T73979 | Tibezonium iodide | ||
Tibezonium iodide 是一种口咽部消毒剂,具有抗菌活性,可用于预防口腔感染。 | |||
T20188 |
Polynoxylin
Formaldehyde, urea polymer,Gabrite,Hygromull,HSDB 7203 |
||
Polynoxylin is an antiseptic. It is used for local treatment of the skin and the mouth. | |||
T69144 | Hexylcaine HCl | ||
Hexylcaine HCl also called cyclaine or osmocaine, is a short-acting local anesthetic. It acts by inhibiting sodium channel conduction. Overdose can lead to headache, tinnitus, numbness and tingling around the mouth and tongue, convulsions, inability to breathe, and decreased heart function. | |||
T21119 |
Cevimeline
AF-102B,西维美林,FKS 508,SNI 2011,HSDB 7286 |
||
Cevimeline, a parasympathomimetic and muscarinic agonist, affects M1 and M3 receptors. Cevimeline has been shown to treat dry mouth and Sj gren's syndrome. It is also used to reduce Xerostomia symptoms and increase salivary flow in head and neck cancer survivors after radiotherapy. | |||
T70855 | Favipiravir sodium | ||
Favipiravir sodium is a selective inhibitor of viral RNA-dependent RNA polymerase with activity against many RNA viruses, influenza viruses, West Nile virus, yellow fever virus, foot-and-mouth disease virus as well as other flaviviruses, arenaviruses, bunyaviruses and alphaviruses. | |||
T83704 |
A20FMDV2 TFA
|
||
A20FMDV2是一种由口蹄疫病毒(FMDV)血清型O的VP1衣壳蛋白上的α-螺旋RGD细胞相互作用域组成的肽,能够结合到αVβ6整合素上。该化合物在表达人αVβ6的H357舌鳞状细胞癌细胞中抑制αVβ6整合素依赖的细胞粘附(IC50 = 1.2 µM)。与111indium-DTPA耦合时,A20FMDV2(20 MBq)可结合于在乳腺癌小鼠异种移植模型中内源性表达的αVβ6整合素,用于放射成像分析。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1285 |
Anethole trithione
茴三硫,Anetholtrithion |
Others; AChR | Neuroscience; Others |
Anethole trithione (Anetholtrithion) 是硫杂环胆碱,是一种胆汁分泌刺激剂,可增强唾液分泌并增加 mAChR 受体,用于口干症的研究。 | |||
T1284 |
Megestrol acetate
SC10363,醋酸甲地孕酮,BDH1298 |
Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy | Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome |
Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。 |