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91

抑制剂 & 化合物

14

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Cat. No. Product Name Target Signaling Pathways
TP1155L Human growth hormone-releasing factor acetate

GHSR GPCR/G Protein
Human growth hormone-releasing factor acetate 是一种下丘脑多肽,通过与垂体前叶细胞上的 GHRH 受体 (GHRHR) 结合来刺激 GH 的产生和释放。
TP1155 Human growth hormone-releasing factor

Growth Hormone Releasing Factor human

Human growth hormone-releasing factor stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on cells in the anterior pituitary.Growth hormone-releasing hormone is a hormone produced in the hypothalamus. The main role of growth hormo
T17103 TM-N1324

Others; GHSR GPCR/G Protein; Others
TM-N1324 是一种 GPR39 激动剂。 TM-N1324 在没有和存在 Zn2+ 的情况下分别以 280 nM 和 9 nM 的高效率和效力激活人 GPR39。 TM-N1324 对鼠 GPR39 表现出相似的效力,EC50 分别为 180 nM 和 5 nM。
T4384 Halofenozide

Others Others
Halofenozide 是一种新的昆虫生长调节剂 (IGR),具有苯甲酰肼结构,也是一种蜕皮激素 (ecdysteroid) 激动剂。可模拟天然昆虫蜕皮激素 20-羟基蜕皮激素的作用,
T16044 Methoprene

烯虫酯,ZR-515

Others Others
Methoprene (ZR-515) 是一种保幼激素模拟物和一种生物杀虫剂。Methoprene 作为昆虫生长调节剂,干扰昆虫的生命周期并阻止其成熟或繁殖。
T4648 TC-G-1008

GPR39-C3

GHSR GPCR/G Protein
TC-G-1008 (GPR39-C3) 是一种口服有活性的 GPR39激动剂,可作用于大鼠受体(EC50: 0.4 nM)和人类受体(EC50:0.8 nM)的。
T16508 PF-5190457

PF-05190457

GHSR GPCR/G Protein
PF-5190457 是具有选择性的、有效的生长素释放肽受体选择性的反向激动剂(pKi:8.36)。
TQ0022 Capromorelin Tartrate

卡普瑞林酒石酸盐,CP 424391-18

GHSR GPCR/G Protein
Capromorelin Tartrate (CP 424391-18) 是口服有活性的 growth hormone secretagogue receptor 有效激动剂,能够作用于 hGHS-R1a(Ki:7 nM)。
TP1035L Cyclic somatostatin Acetate(38916-34-6(free base))

Somatostatin (sheep), monoacetate (salt),Somatostatin-14,SRIF-14,monoacetate (salt)

Others Others
Cyclic somatostatin Acetate(38916-34-6(free base)) (Somatostatin-14) 是一种环状十四肽,可调节许多内分泌和神经系统功能。
T34684 Somatotropin (6-13)

Human growth hormone (6-13)

Somatotropin (6-13) is a growth hormone.
T75713 Human growth hormone-releasing factor TFA

Growth Hormone Releasing Factor human TFA 是下丘脑多肽,通过与GHRHR结合,刺激生长激素生成和释放。
T10319 Anamorelin

RC-1291,阿拉莫林,ONO-7643

GHSR GPCR/G Protein
Anamorelin (ONO-7643) 是新型ghrelin receptor 激动剂,根据FLIPR 检测,得到其EC50=0.74 nM。
T82322 GHRF, mouse

Mouse growth hormone-releasing factor

GHRF, mouse为含44个氨基酸的小鼠生长激素释放肽,能够促进生长激素的释放与合成。
T7112 Ibutamoren Mesylate

MK-0677,伊布莫仑甲磺酸盐,MK-677

GHSR GPCR/G Protein
Ibutamoren Mesylate (MK-0677) 是非肽段类生长激素促分泌素受体 (GHSR) 激动剂,也是一种口服有活性的生长激素 (GH) 促分泌素。
TP1035 Cyclic somatostatin

SRIF-14,合成生长抑素,环状生长激素抑制素,Somatostatin-14

Others Others
Cyclic somatostatin (SRIF-14) 是生长激素释放抑制因子,可用于研究胃十二指肠溃疡出血。
T7225 AnaMorelin hydrochloride

RC-1291 hydrochloride,阿拉莫林盐酸盐,ONO-7643 hydrochloride

GHSR GPCR/G Protein
AnaMorelin hydrochloride (RC-1291 hydrochloride) 是生长素受体激动剂,根据 FLIPR 检测,得到 EC50=0.74 nM。
TP2328L CJC-1295 acetate(863288-34-0 free base)

DAC:GRF acetate

GHSR GPCR/G Protein
CJC-1295 acetate(863288-34-0 free base) (DAC:GRF acetate) 是生长激素释放激素 (GHRH)(也称为生长激素释放因子 (GRF))和生长激素促分泌素 (GHS) 的合成类似物。
T34281 Relamorelin

BIM28131,RM 131,BIM-28131,BIM-28163,BIM 28163,BIM28163,BIM 28131

GHSR GPCR/G Protein
Relamorelin (RM-131)是一种具有选择性和有效性的生长素释放肽/生长激素促分泌素受体 (GHSR) 激动剂,是一种有效的生长素释放肽模拟物,对 GHS-1a 受体具有很高的亲和力。Relamorelin 是一种具有中枢渗透性的五肽,可增加生长激素水平,加速胃排空,具有研究恶病质的潜力。
TP2236L Cortistatin-8 acetate

Cortistatin-8 acetate(485803-62-1 Free base)

GHSR GPCR/G Protein
Cortistatin-8 acetate 是一种皮质抑素类似物,是一种GHS-R拮抗剂,对生长激素促分泌素受体有抑制作用。Cortistatin-8 acetate 是一种合成皮质抑素衍生的生长素释放肽受体配体,不会改变人类对酰化生长素释放肽或海沙瑞林的内分泌反应。
T2584 Octreotide

SMS 201-995,奥曲肽

Somatostatin GPCR/G Protein
Octreotide (SMS 201-995) 是一种有效的生长激素、胰高血糖素和胰岛素抑制剂。它主要与生长抑素 2、3 和 5 亚型受体结合,可增强 Gi 活性,降低胞内 cAMP 的产生。
T7809L Ipamorelin 2 Pivalic acid

NNC-26-0161

Others Others
Ipamorelin 2 Pivalic acid (NNC-26-0161) 是一种生长激素释放肽,可诱导大鼠纵向骨生长。
TP1426 His-[D-2-ME-Trp]-Ala

Others Others
His-[D-2-ME-Trp]-Ala 是生长激素海沙瑞林的一个片段。
T7815L AOD9604 acetate(221231-10-3 free base)

AOD-9604 acetate,AOD9604 acetate,AOD 9604 acetate

Others Others
AOD9604 acetate(221231-10-3 free base) 是一种基于人类生长激素的潜在抗肥胖肽。
T4119 Octreotide Acetate

醋酸奥曲肽,SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)

Somatostatin GPCR/G Protein
Octreotide Acetate (Sandostatin) 是一种长期有效的合成生长抑素八肽类似物,可抑制生长激素的分泌。
T3630 Relugolix

RVT-601,瑞卢戈利,TAK-385

GNRH Receptor GPCR/G Protein
Relugolix (RVT-601) 是口服有活性的非肽性促性腺激素释放激素的拮抗剂。同 TAK-013 相比,它对人和猴子的受体具有高亲和力和强拮抗活性,它们的 IC50值分别为0.33 nM 和0.32 nM。它可用于研究性激素依赖性疾病,如子宫肌瘤、子宫内膜异位症、前列腺癌等。
T11719 JMV 2959 hydrochloride (925238-89-7 free base)

JMV 2959 hydrochloride

GHSR GPCR/G Protein
JMV 2959 hydrochloride (925238-89-7 free base) 是一种生长激素促分泌素受体 1a 型 (GHS-R1a) 拮抗剂,在 LLC-PK1 细胞中的 IC50 为 32±3 nM。
TP1125 Insulin(cattle)

牛胰岛素,Insulin from bovine pancreas,胰岛素

IGF-1R Tyrosine Kinase/Adaptors
Insulin cattle (Insulin from bovine pancreas) 是一种在胰腺 β 细胞中产生的两链多肽激素,在很多哺乳动物细胞培养体系中用作生长因子。
T1669 Liothyronine sodium

3,3',5-Triiodo-L-thyronine sodium,Triostat,T3 Sodium salt,三碘代甲状腺素钠盐,Sodium L-3,3',5-triiodothyronine,Cytomel

Thyroid hormone receptor(THR) Endocrinology/Hormones
Liothyronine sodium (3,3',5-Triiodo-L-thyronine sodium) 是甲状腺激素,能够结合并激活 β1 甲状腺激素受体。
TP1570 Cortistatin-14

Somatostatin GPCR/G Protein
Cortistatin-14 是一种与生长抑素-14结构相似的神经肽,具有抗惊厥和神经保护作用,通过激活 sst(2)、生长素释放肽和 GABA(A/B) 受体损害小鼠的识别记忆巩固,可用于研究脓毒症引发的认知障碍。
T1167 Cyproterone acetate

Androcur,醋酸环丙氯地孕酮,Cyproterone 17-O-acetate,醋酸环丙孕酮

Androgen Receptor Endocrinology/Hormones
Cyproterone acetate (Cyproterone 17-O-acetate) 是能够抗雄激素(IC50=7.1 nM) 和孕激素合成的类固醇。它与 progesteron 和糖皮质激素受体有亲和力。
T11798 L-692429

MK-0751

GHSR; GPCR19 GPCR/G Protein
L-692429 (MK-0751) 是一种有效的非肽基生长激素促分泌素 (GHS) 激动剂,是一种苯并内酰胺的衍生物,可逆转糖皮质激素对 GH 分泌的抑制。L-692429 对 G 蛋白偶联受体 (G protein-coupled receptor)具有很高的亲和力,可用于研究肢端肥大症和肥胖。
T28812 SM-130686

SM 130686,SM130,686,SM 130,686

SM-130,686 is a potent, orally-active agonist of the ghrelin/growth hormone secretagogue receptor (GHSR) and growth hormone secretagogue. It has around half the potency of the endogenous agonist ghrelin as a stimulator of growth hormone release.
T32507 L-739943

L 739943,L739943

L-739943 is a growth hormone secretagogue.
T36377 Somatorelin (1-44) amide (human) (trifluoroacetate salt)

Somatorelin (1-44) amide is a synthetic peptide that corresponds to the full 44-amino acid sequence of growth hormone-releasing hormone (GHRH), a hormone that stimulates the production of growth hormone from the pituitary gland and is involved in the regulation of cell proliferation and differentiation.1,2Somatorelin induces growth hormone release similarly to GHRHin vitroandin vivo.1
T32435 L 163255

L-163255,L163255,L163,255,L-163,255,L 163,255

L 163255 is a type of growth hormone secretagogue (GHS).
T5025L2 Pralmorelin HCl

WAY-GPA 748,WAY-GPA-748 WAY-GPA748,Pralmorelin dihydrochloride

Pralmorelin HCl is regarded as a Growth Hormone Releasing Factor.
T26295 Trioxifene mesylate

LY 133314,LY-133314,LY133314

Trioxifene mesylate is an antiestrogen that suppresses growth hormone secretion.
T31734 BMS-604992

EX1314,EX-1314 HCl,EX-1314,BMS604992,EX-1314 hydrochloride, BMS-604992,EX 1314

EX-1314 (BMS-604992) is a growth hormone secretagogue receptor (GHSR) agonist.
T19567 Substituted piperidines-1

Others Others
Substituted piperidines-1 can promote the release of growth hormone in humans and animals.
T76318 GHRF, porcine

GHRF, porcine 是一种生长激素释放激素 (GHRH) 多肽 (porcine)。GHRF, porcine 与 GHRHR 受体结合并促进生长激素的释放。
T76317 [His1,Nle27] GHRF (1-32), amide, human

[His1,Nle27] GHRF (1-32), amide, human为一种生长激素释放激素(GHRH)类似物,对GHRHR受体具有较好的亲和力。
T32499 L-692429 HCl

L692,429,L-692429,L 692429,L-692,429,L692429,L 692,429

L-692,429 is a novel non-peptide growth hormone secretagin.
T11719L JMV 2959

Others Others
JMV 2959 is an antagonist of growth hormone secretagogue receptor type 1a (GHS-R1a) (IC50: 32 nM).
TP1302 Somatostatin

Somatostatin, also known as growth hormone-inhibiting hormone, is a naturally-occurring peptide hormone of 14 or 28 amino acid residues that regulates the endocrine system. It is secreted by the D cells of the islets to inhibit the release of insulin and
T70634 Psycholeine

Psycholeine is isolated from the tropical plant Psychotria oleoides; exhibits somatostatin antagonistic activity on growth hormone secretion.
T2584L1 Octreotide HCl

Octreotide hydrochloride, (-)-,Octreotide hydrochloride

Octreotide HCl is a potent, long-acting synthetic SOMATOSTATIN octapeptide analog that inhibits the secretion of growth hormone.
T35793 JMV3002

JMV3002

Ghrelin is an endogenous ligand for the growth hormone secretagogue receptor that stimulates food intake and transduces signals to hypothalamic regulatory nuclei that control energy homeostasis. JMV3002 is a potent ghrelin receptor antagonist with an IC50 value of 1.1 nM in vitro. At 80 μg/kg, JMV3002 inhibits hexarelin-stimulated food intake by as much as 98% in rats. JMV3002 alone does not elicit growth hormone release nor does it inhibit hexarelin-stimulated growth hormone secretion when test...
TNU0430 N6-(p-Methoxybenzyl)adenosine

Nucleoside Derivatives - 6-Modified purine nucleosides; Drugs and Inhibitors; plant growth regulator, plant hormone
T75157L Cimdelirsen sodium

Cimdelirsen (sodium) 为针对肝脏的反义寡核苷酸,通过减少生长激素受体(GHr)合成,抑制生长激素(GH)的过度分泌效应,进而降低肢端肥大症患者体内循环胰岛素样生长因子-1 (IGF-1)水平。
T78039 Acetyl-(D-Arg2)-GRF (1-29) amide (human)

Acetyl-(D-Arg2)-GRF (1-29) amide (human) 是一种针对人体的生长激素释放因子(GRF)拮抗剂,其主要作用是抑制生长激素(GH)的释放,广泛应用于内分泌学领域的研究。

化合物

Human growth hormone-releasing factor acetate
Cat.No: TP1155L
Synonym:
Target: GHSR
Human growth hormone-releasing factor
Cat.No: TP1155
Synonym: Growth Hormone Releasing Factor human
Target:
TM-N1324
Cat.No: T17103
Synonym:
Target: Others, GHSR
Halofenozide
Cat.No: T4384
Synonym:
Target: Others
Methoprene
Cat.No: T16044
Synonym: 烯虫酯,ZR-515
Target: Others
TC-G-1008
Cat.No: T4648
Synonym: GPR39-C3
Target: GHSR
PF-5190457
Cat.No: T16508
Synonym: PF-05190457
Target: GHSR
Capromorelin Tartrate
Cat.No: TQ0022
Synonym: 卡普瑞林酒石酸盐,CP 424391-18
Target: GHSR
Cyclic somatostatin Acetate(38916-34-6(free base))
Cat.No: TP1035L
Synonym: Somatostatin (sheep), monoacetate (salt),Somatostatin-14,SRIF-14,monoacetate (salt)
Target: Others
Somatotropin (6-13)
Cat.No: T34684
Synonym: Human growth hormone (6-13)
Target:
Human growth hormone-releasing factor TFA
Cat.No: T75713
Synonym:
Target:
Anamorelin
Cat.No: T10319
Synonym: RC-1291,阿拉莫林,ONO-7643
Target: GHSR
GHRF, mouse
Cat.No: T82322
Synonym: Mouse growth hormone-releasing factor
Target:
Ibutamoren Mesylate
Cat.No: T7112
Synonym: MK-0677,伊布莫仑甲磺酸盐,MK-677
Target: GHSR
Cyclic somatostatin
Cat.No: TP1035
Synonym: SRIF-14,合成生长抑素,环状生长激素抑制素,Somatostatin-14
Target: Others
AnaMorelin hydrochloride
Cat.No: T7225
Synonym: RC-1291 hydrochloride,阿拉莫林盐酸盐,ONO-7643 hydrochloride
Target: GHSR
CJC-1295 acetate(863288-34-0 free base)
Cat.No: TP2328L
Synonym: DAC:GRF acetate
Target: GHSR
Relamorelin
Cat.No: T34281
Synonym: BIM28131,RM 131,BIM-28131,BIM-28163,BIM 28163,BIM28163,BIM 28131
Target: GHSR
Cortistatin-8 acetate
Cat.No: TP2236L
Synonym: Cortistatin-8 acetate(485803-62-1 Free base)
Target: GHSR
Octreotide
Cat.No: T2584
Synonym: SMS 201-995,奥曲肽
Target: Somatostatin
Ipamorelin 2 Pivalic acid
Cat.No: T7809L
Synonym: NNC-26-0161
Target: Others
His-[D-2-ME-Trp]-Ala
Cat.No: TP1426
Synonym:
Target: Others
AOD9604 acetate(221231-10-3 free base)
Cat.No: T7815L
Synonym: AOD-9604 acetate,AOD9604 acetate,AOD 9604 acetate
Target: Others
Octreotide Acetate
Cat.No: T4119
Synonym: 醋酸奥曲肽,SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)
Target: Somatostatin
Relugolix
Cat.No: T3630
Synonym: RVT-601,瑞卢戈利,TAK-385
Target: GNRH Receptor
JMV 2959 hydrochloride (925238-89-7 free base)
Cat.No: T11719
Synonym: JMV 2959 hydrochloride
Target: GHSR
Insulin(cattle)
Cat.No: TP1125
Synonym: 牛胰岛素,Insulin from bovine pancreas,胰岛素
Target: IGF-1R
Liothyronine sodium
Cat.No: T1669
Synonym: 3,3',5-Triiodo-L-thyronine sodium,Triostat,T3 Sodium salt,三碘代甲状腺素钠盐,Sodium L-3,3',5-triiodothyronine,Cytomel
Target: Thyroid hormone receptor(THR)
Cortistatin-14
Cat.No: TP1570
Synonym:
Target: Somatostatin
Cyproterone acetate
Cat.No: T1167
Synonym: Androcur,醋酸环丙氯地孕酮,Cyproterone 17-O-acetate,醋酸环丙孕酮
Target: Androgen Receptor
L-692429
Cat.No: T11798
Synonym: MK-0751
Target: GHSR, GPCR19
SM-130686
Cat.No: T28812
Synonym: SM 130686,SM130,686,SM 130,686
Target:
L-739943
Cat.No: T32507
Synonym: L 739943,L739943
Target:
Somatorelin (1-44) amide (human) (trifluoroacetate salt)
Cat.No: T36377
Synonym:
Target:
L 163255
Cat.No: T32435
Synonym: L-163255,L163255,L163,255,L-163,255,L 163,255
Target:
Pralmorelin HCl
Cat.No: T5025L2
Synonym: WAY-GPA 748,WAY-GPA-748 WAY-GPA748,Pralmorelin dihydrochloride
Target:
Trioxifene mesylate
Cat.No: T26295
Synonym: LY 133314,LY-133314,LY133314
Target:
BMS-604992
Cat.No: T31734
Synonym: EX1314,EX-1314 HCl,EX-1314,BMS604992,EX-1314 hydrochloride, BMS-604992,EX 1314
Target:
Substituted piperidines-1
Cat.No: T19567
Synonym:
Target: Others
GHRF, porcine
Cat.No: T76318
Synonym:
Target:
[His1,Nle27] GHRF (1-32), amide, human
Cat.No: T76317
Synonym:
Target:
L-692429 HCl
Cat.No: T32499
Synonym: L692,429,L-692429,L 692429,L-692,429,L692429,L 692,429
Target:
JMV 2959
Cat.No: T11719L
Synonym:
Target: Others
Somatostatin
Cat.No: TP1302
Synonym:
Target:
Psycholeine
Cat.No: T70634
Synonym:
Target:
Octreotide HCl
Cat.No: T2584L1
Synonym: Octreotide hydrochloride, (-)-,Octreotide hydrochloride
Target:
JMV3002
Cat.No: T35793
Synonym: JMV3002
Target:
N6-(p-Methoxybenzyl)adenosine
Cat.No: TNU0430
Synonym:
Target:
Cimdelirsen sodium
Cat.No: T75157L
Synonym:
Target:
Acetyl-(D-Arg2)-GRF (1-29) amide (human)
Cat.No: T78039
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T20945 2,4-D

Hedonal,Macondray,2,4-D acid,Chloroxone,2,4-二氯苯氧乙酸

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
2,4-Dichlorophenoxyacetic acid (Hedonal) 是一种合成生长素,用作植物生长调节剂,也用作植物细胞培养基中的补充剂。它是除草剂中的一种活性成分,用于破坏肌动蛋白细胞骨架,以控制根系伸长和细胞生成。
T7931 16a,17a-Epoxy-4-Pregnen-3,20-Dione

Others Others
16a,17a-Epoxy-4-Pregnen-3,20-Dione 是一种合成孕激素,是黄体酮激素的代谢产物,它通过与黄体酮受体结合发挥作用,已被用于研究孕激素对生殖器官的影响,激素对细胞生长和发育的影响,以及激素对免疫系统的影响。
T2O2791 3-Indoleacetic acid

3-IAA,Indole-3-acetic acid,1H-Indole-3-acetic acid,3-吲哚乙酸,indolylacetic acid,IAA,indoleacetic acid

Others; Endogenous Metabolite Metabolism; Others
3-Indoleacetic acid (indolylacetic acid) 是常见的天然植物生长激素。它可以诱导植物细胞的伸长和分裂。
TMS2181 trans-Zeatin

(E)-Zeatin,玉米素

ERK; MEK; Endogenous Metabolite MAPK; Metabolism
trans-Zeatin ((E)-Zeatin) 是植物细胞分裂素,可抑制紫外线诱导的MEK/ERK 的活化,在细胞生长、分化和分裂中起着重要的作用。
T3S0507 Homovanillic acid

Homovaniuic acid,Vanilacetic acid,高香草酸,Vanillacetic acid

Others; Endogenous Metabolite Metabolism; Others
Homovanillic acid (Vanillacetic acid) 是一种多巴胺代谢物,它与乳糜泻、生长激素缺乏、芳香族氨基酸脱羧酶缺乏症以及脂联素还原酶缺乏症相关。
T7990 9-hydroxy-4-androstene-3,17-dione

Others Others
9-hydroxy-4-androstene-3,17-dione 是一种类固醇激素,具有抗肿瘤活性,可以抑制多种癌症细胞的生长,包括乳腺癌、前列腺癌和肺癌细胞。
T3O2749 L-Leucine

(S)-Leucine,Leu,L-亮氨酸,亮氨酸

mTOR PI3K/Akt/mTOR signaling
L-Leucine ((S)-Leucine) 是必需的支链氨基酸,能够激活 mTOR 信号通路。
T4939 Indole-3-pyruvic acid

3-(3-吲哚基)-2-氧代丙酸,3-(3-Indolyl)-2-oxopropanoic acid

Others Others
Indole-3-pyruvic acid (3-(3-Indolyl)-2-oxopropanoic acid) 是一种参与Indole-3-acetic acid 生物合成的化合物,Indole-3-acetic acid 是一种植物激素,在调节生长和对环境变化的反应中起重要作用。
T5088 3-Indoleacetic acid sodium

Indole-3-Acetic Acid sodium salt,Sodium 2-(1H-indol-3-yl)acetate,IAA sodium salt,吲哚乙酸钠,Heteroauxin sodium salt

Others; Endogenous Metabolite Metabolism; Others
3-Indoleacetic acid sodium (Heteroauxin sodium salt) 是一种天然存在的植物生长素类激素。能刺激细胞伸长和分裂,促进植物生长发育。然而,高浓度时,它表现出生长抑制作用,包括生长和阻止茎和根的生长。后一种效应形成了合成生长素被开发为农业除草剂和生物调节剂的基础。
T6368 Abscisic Acid

Abscisin II,Dormin,(+)-脱落酸,(+)-ABA,Abscisic Acid (Dormin)

Others; Proton pump; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
Abscisic Acid (Dormin) 是具有口服活性的植物激素,存在于蔬菜和水果中,也是内源性的哺乳动物激素。它是生长抑制剂,可以调节植物生长发育。他抑制质子泵,并导致 Ca2+依赖性的质膜去极化。它是 LANCL2 的天然配体,属于胰岛素敏感化合物,在糖尿病前期,2 型糖尿病和代谢综合征的研究中具有价值。
T3S0860 Gitogenin

UGT Metabolism
Gitogenin 是一种从Tribulus longipetalus 整株中分离出来的天然类固醇,是一种 UDP-葡萄糖醛酸转移酶 1A4 (UGT1A4) 和 α-葡萄糖苷酶的选择性抑制剂,其IC50分别为 0.69 µM (使用三氟拉嗪为底物) 和 37.2 μM,对人类主要细胞色素 P450 亚型的活性无抑制作用。
T80006 Emoghrelin

GHSR GPCR/G Protein
Emoghrelin是一种从Polygonum multiflorum(何首乌)提取的化合物,能够通过激活生长素释放肽受体来刺激生长激素的分泌。
T82277 GM1a Ganglioside oligosaccharide

GM1a Ganglioside oligosaccharide为ganglioside GM1的半合成形式,后者作为霍乱毒素的天然受体,在生长调节及激素诱导反应的耦合中具有关键功能。
T32326 Juvabione

Juvabione is the methyl ester of todomatuic acid, both of which are sesquiterpenes (C15) found in the wood of true firs of the genus Abies. They exist as part of a mixture of sesquiterpenes based on the bisabolane scaffold. Sesquiterpenes of this family,

天然产物

2,4-D
Cat.No: T20945
Synonym: Hedonal,Macondray,2,4-D acid,Chloroxone,2,4-二氯苯氧乙酸
Target: DNA/RNA Synthesis
16a,17a-Epoxy-4-Pregnen-3,20-Dione
Cat.No: T7931
Synonym:
Target: Others
3-Indoleacetic acid
Cat.No: T2O2791
Synonym: 3-IAA,Indole-3-acetic acid,1H-Indole-3-acetic acid,3-吲哚乙酸,indolylacetic acid,IAA,indoleacetic acid
Target: Others, Endogenous Metabolite
trans-Zeatin
Cat.No: TMS2181
Synonym: (E)-Zeatin,玉米素
Target: ERK, MEK, Endogenous Metabolite
Homovanillic acid
Cat.No: T3S0507
Synonym: Homovaniuic acid,Vanilacetic acid,高香草酸,Vanillacetic acid
Target: Others, Endogenous Metabolite
9-hydroxy-4-androstene-3,17-dione
Cat.No: T7990
Synonym:
Target: Others
L-Leucine
Cat.No: T3O2749
Synonym: (S)-Leucine,Leu,L-亮氨酸,亮氨酸
Target: mTOR
Indole-3-pyruvic acid
Cat.No: T4939
Synonym: 3-(3-吲哚基)-2-氧代丙酸,3-(3-Indolyl)-2-oxopropanoic acid
Target: Others
3-Indoleacetic acid sodium
Cat.No: T5088
Synonym: Indole-3-Acetic Acid sodium salt,Sodium 2-(1H-indol-3-yl)acetate,IAA sodium salt,吲哚乙酸钠,Heteroauxin sodium salt
Target: Others, Endogenous Metabolite
Abscisic Acid
Cat.No: T6368
Synonym: Abscisin II,Dormin,(+)-脱落酸,(+)-ABA,Abscisic Acid (Dormin)
Target: Others, Proton pump, Endogenous Metabolite
Gitogenin
Cat.No: T3S0860
Synonym:
Target: UGT
Emoghrelin
Cat.No: T80006
Synonym:
Target: GHSR
GM1a Ganglioside oligosaccharide
Cat.No: T82277
Synonym:
Target:
Juvabione
Cat.No: T32326
Synonym:
Target:
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