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Targets Recommended: Apoptosis Endogenous Metabolite Prostaglandin Receptor Autophagy PROTAC Linker

28

抑制剂 & 化合物

13

天然产物

2

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T4546 Dinoprost tromethamine salt

Dinoprost Tromethamine,Zinoprost,Prostin F2 alpha,PGF2α THAM,Dinolytic,地诺前列素氨丁三醇,Prostaglandin F2α THAM

Apoptosis; Endogenous Metabolite; Prostaglandin Receptor; Autophagy; PROTAC Linker Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; Metabolism; PROTAC
Dinoprost tromethamine salt (PGF2α THAM) 是一种口服有效的前列腺素 F 受体激动剂。它是在子宫内膜腔上皮和黄体中局部产生的溶酶激素,在分娩过程中起关键作用。
T0002 Ethamsylate

Cyclonamine,Etamsylate,酚磺乙胺,Dicynene,Aglumin

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Ethamsylate (Dicynene) 通常用作止血药,增加毛细血管内皮阻力和血小板粘附,抑制前列腺素的生物合成和作用。
T4989 Fosfomycin Tromethamine

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin tromethamine 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T0048 Nikethamide

N,N-Diethylnicotinamide,Corvotone,Anacardone,烟酰乙胺,Corvin

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Nikethamide 是呼吸中枢激活剂,可用于研究呼吸衰竭。
T25986 Prinomide tromethamine

Others Others
Prinomide tromethamine 是一种抗风湿病的化合物。
T15772 Lodoxamide tromethamine

U-42585E

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Lodoxamide tromethamine 是一种的肥大细胞稳定剂,具有抗过敏特性,可用于治疗哮喘和过敏性结膜炎的研究。
T1212 Ketorolac tromethamine salt

酮咯酸氨丁三醇,Acular LS,Toradol,Ketorolac tris salt,Acular

COX Immunology/Inflammation; Neuroscience
Ketorolac tromethamine salt (Ketorolac tris salt) 是一种非甾体抗炎剂,是非选择性的 COX 抑制剂,对 COX-1 和 COX-2 的IC50值分别为 20 和 120 nM。
T0849 Pyrimethamine

Pirimecidan,RP 4753,Pirimetamin,乙胺嘧啶

DHFR; Antifolate; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Pyrimethamine (Pirimecidan) 是一种二氢叶酸还原酶的竞争性抑制剂,用作抗疟药。
T0023 Valethamate bromide

Ediposin,Epidozin,戊沙溴铵,Epidosin,Resitan

Others Others
Valethamate bromide (Resitan) 是快速作用的抗胆碱能解痉和肌萎缩剂,是一种酯,能够改善宫颈扩张加速分娩。
T7114 GALANTHAMINONE

(-)-Narwedine,氢溴酸加兰他敏,Narwedin

AChE Neuroscience
Galanthaminone ((-)-Narwedine) 是一种竞争性的、可逆的胆碱酯酶抑制剂,可作用于多种记忆障碍疾病的研究。
T25929 Pemetrexed tromethamine

Pemetrexed ditromethamine dihydrate

Pemetrexed tromethamine is a chemotherapy drug used for pleural mesothelioma and non-small cell lung cancer.
T71500 Palifosfamide tromethamine

IPM tromethamine,Isophosphoramide mustard tromethamine,ZIO-201 tromethamine,Isophosphoramide mustard tromethamine ; IPM tromethamine ; ZIO-201 tromethamine

Palifosfamide (tromethamine) 是一种具有潜在抗肿瘤活性的合成烷基化剂。作为异环磷酰胺 (ifosfamide) 稳定的活性代谢物,Palifosfamide (tromethamine) 通过GC 碱基对不可逆地烷基化和交联DNA,导致了DNA 复制的抑制,并导致细胞死亡。与异环磷酰胺相比,Palifosfamide (tromethamine)的毒性较小。
T25395 Ethamoxytriphetol

Ethamoxytriphetol is a non-steroidal estrogen antagonist.
T69724 Cilofexor tromethamine

Cilofexor, also known as GS-9674, is a farnesoid X receptor (FXR) agonist. The nonsteroidal FXR agonist cilofexor (GS-9674) improves markers of cholestasis and liver injury in patients with PSC. In clinical study, cilofexor was well tolerated and led to significant improvements in liver biochemistries and markers of cholestasis in patients with PSC.
TMIH-0223 Ethambutol.2HCl-d4

Ethambutol.2HCl-d4 是 Ethambutol.2HCl 的氘代化合物。
T75430 Succinic acid tromethamine

Succinic acid tromethamine 是一种口服活性抗焦虑剂,有效地参与三羧酸循环作为中间产物。它也广泛用作食品、化学和制药行业中多种重要工业化学品的前体。
T22570 Amthamine dihydrobromide

Others Others
H2 agonist
T31688 Ethambutol, (R,R)-

L-Ethambutol

Ethambutol, (R, R)- can be used to treat tuberculosis. It is usually used in combination with other tuberculosis medications. It may also be used to treat Mycobacterium avium complex, and Mycobacterium kansasii.
T67829 Compound AMTHAMINE DIHYDROBROMIDE

Compound AMTHAMINE DIHYDROBROMIDE 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67829,CAS号为 142437-67-0。
T11534L Haemanthamine hydrochloride (466-75-1 free base)

Haemanthamine hydrochloride

Others Others
Haemanthamine hydrochloride is an alkaloid isolated from the Amaryllidaceae plants with potent anticancer activity. It inhibits protein biosynthesis during the elongation stage of translation. It has antimalarial, pro-apoptotic, antiviral, antioxidant, an
T75326 ATP ditromethamine

ATP ditromethamine(Adenosine 5'-triphosphate ditromethamine)作为体内能量储存和代谢的核心物质,不仅为代谢过程提供必需能量,而且在细胞中担任辅酶角色。此外,它在免疫和炎症反应中,扮演着关键的内源性信号分子角色。
T69781 Methamilane maleate

Methamilane maleate is a Muscarinic agonist.
T125493 Athamantin

T69251 Methamilane methiodide

Methamilane methiodide is a Muscarinic agonist.
T7062 Ethambutol

Ethambutol 是一种抗分枝杆菌化合物,通过抑制阿拉伯糖基转移酶活性阻止细胞壁的形成。
T72146 Loxoprofenol-SRS tromethamine

HR1405–01

Loxoprofenol-SRS tromethamine (HR1405-01) 为Loxoprofen的活性代谢物,为一种可静脉注射的安全非甾体抗炎药(NSAID),展现出良好的抗炎及镇痛效果。
T31499 Dinitrosoethambutol

Ddeta

Dinitrosoethambutol is a biochemical.
T124710 Trachelanthamidine

Trachelanthamidine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124710。

化合物

Dinoprost tromethamine salt
Cat.No: T4546
Synonym: Dinoprost Tromethamine,Zinoprost,Prostin F2 alpha,PGF2α THAM,Dinolytic,地诺前列素氨丁三醇,Prostaglandin F2α THAM
Target: Apoptosis, Endogenous Metabolite, Prostaglandin Receptor, Autophagy, PROTAC Linker
Ethamsylate
Cat.No: T0002
Synonym: Cyclonamine,Etamsylate,酚磺乙胺,Dicynene,Aglumin
Target: Prostaglandin Receptor
Fosfomycin Tromethamine
Cat.No: T4989
Synonym:
Target: Antibacterial, Antibiotic
Nikethamide
Cat.No: T0048
Synonym: N,N-Diethylnicotinamide,Corvotone,Anacardone,烟酰乙胺,Corvin
Target: GABA Receptor
Prinomide tromethamine
Cat.No: T25986
Synonym:
Target: Others
Lodoxamide tromethamine
Cat.No: T15772
Synonym: U-42585E
Target: Histamine Receptor
Ketorolac tromethamine salt
Cat.No: T1212
Synonym: 酮咯酸氨丁三醇,Acular LS,Toradol,Ketorolac tris salt,Acular
Target: COX
Pyrimethamine
Cat.No: T0849
Synonym: Pirimecidan,RP 4753,Pirimetamin,乙胺嘧啶
Target: DHFR, Antifolate, Parasite
Valethamate bromide
Cat.No: T0023
Synonym: Ediposin,Epidozin,戊沙溴铵,Epidosin,Resitan
Target: Others
GALANTHAMINONE
Cat.No: T7114
Synonym: (-)-Narwedine,氢溴酸加兰他敏,Narwedin
Target: AChE
Pemetrexed tromethamine
Cat.No: T25929
Synonym: Pemetrexed ditromethamine dihydrate
Target:
Palifosfamide tromethamine
Cat.No: T71500
Synonym: IPM tromethamine,Isophosphoramide mustard tromethamine,ZIO-201 tromethamine,Isophosphoramide mustard tromethamine ; IPM tromethamine ; ZIO-201 tromethamine
Target:
Ethamoxytriphetol
Cat.No: T25395
Synonym:
Target:
Cilofexor tromethamine
Cat.No: T69724
Synonym:
Target:
Ethambutol.2HCl-d4
Cat.No: TMIH-0223
Synonym:
Target:
Succinic acid tromethamine
Cat.No: T75430
Synonym:
Target:
Amthamine dihydrobromide
Cat.No: T22570
Synonym:
Target: Others
Ethambutol, (R,R)-
Cat.No: T31688
Synonym: L-Ethambutol
Target:
Compound AMTHAMINE DIHYDROBROMIDE
Cat.No: T67829
Synonym:
Target:
Haemanthamine hydrochloride (466-75-1 free base)
Cat.No: T11534L
Synonym: Haemanthamine hydrochloride
Target: Others
ATP ditromethamine
Cat.No: T75326
Synonym:
Target:
Methamilane maleate
Cat.No: T69781
Synonym:
Target:
Athamantin
Cat.No: T125493
Synonym:
Target:
Methamilane methiodide
Cat.No: T69251
Synonym:
Target:
Ethambutol
Cat.No: T7062
Synonym:
Target:
Loxoprofenol-SRS tromethamine
Cat.No: T72146
Synonym: HR1405–01
Target:
Dinitrosoethambutol
Cat.No: T31499
Synonym: Ddeta
Target:
Trachelanthamidine
Cat.No: T124710
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T14865 Carboprost tromethamine

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Carboprost tromethamine 是合成的前列腺素 F2α的15-甲基类似物,能有效促进子宫的规律收缩,显着减少产中及产后出血量。
T0810 Ethambutol dihydrochloride

Ethambutol 2HCl,盐酸乙胺丁醇,Emb dihydrochloride,CL40881

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Ethambutol dihydrochloride (CL40881) 能抗分枝杆菌,可抑制阿拉伯糖基转移酶活性来阻止细胞壁形成。
TN6786 O-Desmethyl Galanthamine

Sanguinine,O-去甲基加兰他敏

AChE Neuroscience
O-Desmethyl Galanthamine (Sanguinine) 是一种加兰他敏型生物碱,是一种乙酰胆碱酯酶 (AChE) 抑制剂,其IC50=1.83 μM。
T0086 Galanthamine hydrobromide

Galantamine hydrobromide,Galanthamine HBr,氢溴酸加兰他敏

AChR; AChE Neuroscience
Galanthamine hydrobromide (Galantamine hydrobromide) 是一种长效的中枢活性 AChE 抑制剂,IC50为 410 nM。它是神经元烟碱型 ACh 受体的变构增强剂,IC50值为 0.35 µM,可用于阿尔茨海默症的研究。
T4S1725 Galanthamine

Galantamine,加兰他敏

Apoptosis; AChE Apoptosis; Neuroscience
Galanthamine (Galantamine) 是一种乙酰胆碱酯酶抑制剂,IC50为 500 nM。
TN6792 O-Acetylgalanthamine

Others Others
O-Acetylgalanthamine 是一种天然产物,已在 Narcissus pseudonarcissu 的鳞茎中发现。
T11351 Galanthamine N-Oxide

AChE Neuroscience
Galanthamine N-Oxide 是分离于Zephyranthes concolor 的球茎中的一种生物碱。它抑制电鳗乙酰胆碱酯酶,EC50=26.2 μM。它是TcAChE,hAChE 和 hBChE 酶活性位点中底物调节的显著抑制剂。
TN5158 Trachelanthamine

Others Others
Trachelanthamine is a natural product from Eupatorium fortunei.
TN7055 N-Desmethyl Galanthamine

N-Desmethyl Galanthamine 在生命科学相关研究中具有广泛的应用。
T83460 11-O-β-D-glucopyranosyl thamnosmonin

11-O-β-D-glucopyranosyl thamnosmonin是一种香豆素苷,能够从Angelica apaensis根部提取。该化合物对PAF、AA和ADP诱发的兔血小板聚集表现出轻度的抑制效果。
T73813 Haemanthamine hydrochloride

Haemanthamine hydrochloride 是从Amaryllidaceae 植物中分离出来的一种蛇毒碱样生物碱,具有强大的抗癌活性。Haemanthamine hydrochloride 靶向核糖体以在翻译的延长阶段抑制蛋白质的生物合成。Haemanthamine hydrochloride 具有促凋亡,抗氧化剂,抗病毒,抗疟疾和抗惊厥活性。
T11534 Haemanthamine

Others Others
Haemanthamine is an alkaloid isolated from the Amaryllidaceae plants with potent anticancer activity. It inhibits protein biosynthesis during the elongation stage of translation. It has antimalarial, pro-apoptotic, antiviral, antioxidant, and anticonvulsa
TN5886 Thamnosmonin

Thamnosmonin is a natural product from Citrus sinensis.

天然产物

Carboprost tromethamine
Cat.No: T14865
Synonym:
Target: Prostaglandin Receptor
Ethambutol dihydrochloride
Cat.No: T0810
Synonym: Ethambutol 2HCl,盐酸乙胺丁醇,Emb dihydrochloride,CL40881
Target: Antibacterial, Antibiotic, Antifungal
O-Desmethyl Galanthamine
Cat.No: TN6786
Synonym: Sanguinine,O-去甲基加兰他敏
Target: AChE
Galanthamine hydrobromide
Cat.No: T0086
Synonym: Galantamine hydrobromide,Galanthamine HBr,氢溴酸加兰他敏
Target: AChR, AChE
Galanthamine
Cat.No: T4S1725
Synonym: Galantamine,加兰他敏
Target: Apoptosis, AChE
O-Acetylgalanthamine
Cat.No: TN6792
Synonym:
Target: Others
Galanthamine N-Oxide
Cat.No: T11351
Synonym:
Target: AChE
Trachelanthamine
Cat.No: TN5158
Synonym:
Target: Others
N-Desmethyl Galanthamine
Cat.No: TN7055
Synonym:
Target:
11-O-β-D-glucopyranosyl thamnosmonin
Cat.No: T83460
Synonym:
Target:
Haemanthamine hydrochloride
Cat.No: T73813
Synonym:
Target:
Haemanthamine
Cat.No: T11534
Synonym:
Target: Others
Thamnosmonin
Cat.No: TN5886
Synonym:
Target:
Cat. No. Product Name Species Expression System
TMPY-00221 DPP4/CD26 Protein, Mouse, Recombinant (hFc)

dipeptidylpeptidase 4,Dpp-4,Cd26,THAM

Mouse HEK293 Cells
DPP4/CD26 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 112.9 kDa and the accession number is P28843.
TMPY-00074 DPP4/CD26 Protein, Mouse, Recombinant (His)

dipeptidylpeptidase 4,Dpp-4,Cd26,THAM

Mouse HEK293 Cells
DPP4/CD26 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 85.9 kDa and the accession number is P28843.

重组蛋白

DPP4/CD26 Protein, Mouse, Recombinant (hFc)
Cat.No: TMPY-00221
Species: Mouse
Expression System: HEK293 Cells
DPP4/CD26 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-00074
Species: Mouse
Expression System: HEK293 Cells
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