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Search Results for " phenylephrine "

18

抑制剂 & 化合物

8

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T0453L	DL-Phenylephrine HCl Eyelo,DL-Phenylephrine hydrochloride
	DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.
T35576	Phenylephrine-3-O-Sulfate
	Phenylephrine-3-O-sulfate is metabolite of the α1A-adrenergic receptor agonist phenylephrine formed via sulfation.
T68997	L-Phenylephrine
	L-Phenylephrine is an alpha-adrenergic agonist used as a mydriatic, nasal decongestant, and cardiotonic agent.
T22033	ARC 239 dihydrochloride	Norepinephrine	Neuroscience
	ARC 239 dihydrochloride 是一种选择性 α2B 肾上腺素受体拮抗剂。
T12913	Siguazodan SKF 94836	PDE	Metabolism
	Siguazodan (SKF 94836) 是选择性的，口服有效的磷酸二酯酶 III 抑制剂，IC50为 117 nM。它可增加完整血小板中 cAMP 的积累，EC50为 18.88 μM。它也抑制苯肾上腺素诱导的 5-HT 释放，IC50为 4.2 μM。
T4563	Thonzylamine neohetramine,松齐拉敏	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Thonzylamine (neohetramine) 是可口服的H1组胺受体拮抗剂，具有抗组胺和抗过敏特性，可用于鼻充血、过敏性结膜炎和其他过敏性疾病的研究。
T23557	Talibegron hydrochloride ZD2079 hydrochloride,ZD 2079	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Talibegron hydrochloride (ZD2079 hydrochloride) 是一种β3肾上腺素能受体激动剂，对苯肾上腺素预收缩大鼠肠系膜动脉的 pD2为3.72。松弛大鼠肠系膜动脉和离体主动脉。在体内抑制瘦小鼠 ob 基因表达和循环瘦素水平。
T27164	DHP-218 PAK-9,PAK9,PAK 9,DHP218
	DHP-218 is a calcium channel antagonist. DHP-218 inhibits Calcium-induced contraction of the rat aorta in high K+ solution with the pA2 value of 9.11. The IC50 value for the inhibitory effects of DHP-218 in high K+-induced and phenylephrine-induced contra
T40563	Sandaracopimaric acid
	Sandaracopimaric acid is an anti-inflammatory diterpenoid compound that effectively reduces the contraction of phenylephrine-induced pulmonary arteries. With an EC50 of 43.93 μM, it exhibits noteworthy anti-inflammatory properties.
T30427	Berefrine
	Berefrine is an Oxazolidine prodrug of phenylephrine.
TP2086	AdTx1
	Selective, high affinity, non-competitive α1A adrenoceptor antagonist (Ki = 0.35 nM). Exhibits no significant activity against a range of other GPCRs, including α2A, β1 and β2 adrenoceptors. Antagonizes effects of phenylephrine on isolated rabbit prostate
T35987	CAY10563 CAY10563
	S-Nitrosothiols (RSNOs) are a class of molecules that function as exogenous and endogenous nitric oxide (NO) donors. RSNOs found in vivo include proteins such as S-nitrosohemoglobin and S-nitrosoalbumin, as well as low molecular weight species such as S-nitrosoglutathione (GSNO) and S-nitrosocysteine (CysNO). CAY10563 is a member of a new class of S-nitrosothiol species that act as an NO donors under acidic conditions. It decomposes with a half-life of one minute in 0.1 M phosphate buffer, pH 5....
T39281	AM404
	AM404 is a chemical compound that functions as an inhibitor of endocannabinoid reuptake. It effectively blocks the transport of anandamide, with IC50 values measured in the low micromolar range. Moreover, AM404 exhibits the ability to induce relaxation in rat isolated hepatic arteries contracted with Phenylephrine. This relaxation effect is quantified by a pEC50 value of 7.4 (corresponding to an EC50 of 0.04 μM). Additionally, AM404 possesses a neuroprotective effect.
T69127	Moxisylyte
	Moxisylyte, also known as thymoxamine, is a drug used in urology for the treatment of erectile dysfunction. It is an α1-adrenergic antagonist. Moxisylyte is also used for the short-term treatment of primary Reynaud's syndrome, a condition where the fingers and toes become discoloured in response to cold or emotional distress. Moxisylyte helps by improving blood circulation to the extremities. It is also used locally in the eye to reverse the mydriasis caused by phenylephrine and other sympathomi...
T73083	Nipradolol KT 210 ; K 351 ; Hypadil,Hypadil,KT 210,K 351
	Nipradolol (KT-210; K-351) 是一种有效的 α-1-肾上腺素能受体的阻滞剂。Nipradolol 还抑制白化兔模型中 Phenylephrine 诱导的眼压升高 (IOP)。Nipradolol 抑制去甲肾上腺素 (NA) 引起的肌肉收缩，对犬冠状动脉也有血管扩张剂活性。
T35989	CAY10565
	S-Nitrosothiols (RSNOs) are a class of molecules that function as exogenous and endogenous nitric oxide (NO) donors. RSNOs found in vivo include proteins such as S-nitrosohemoglobin and S-nitrosoalbumin, as well as low molecular weight species such as S-nitrosoglutathione (GSNO) and S-nitrosocysteine (CysNO). CAY10565 is a member of a new class of S-nitrosothiol species that act as NO donors under acidic conditions. It decomposes with a half-life of 130 minutes in 0.1 M phosphate buffer, pH 5.0,...
T35988	CAY10564
	S-Nitrosothiols (RSNOs) are a class of molecules that function as exogenous and endogenous nitric oxide (NO) donors. RSNOs found in vivo include proteins such as S-nitrosohemoglobin and S-nitrosoalbumin, as well as low molecular weight species such as S-nitrosoglutathione (GSNO) and S-nitrosocysteine (CysNO). CAY10564 is a member of a new class of S-nitrosothiol species that act as NO donors under acidic conditions. It decomposes with a half-life of one minute in 0.1 M phosphate buffer, pH 5.0, ...
T36070	(±)5(6)-EET
	5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes. In solution, 5(6)-EET degrades into 5,6-DiHET and 5(6)-δ-lactone, which can be converted to 5(6)-DiHET and quantified by GC-MS. In neuroendocrine cells, such as the anterior pituitary and pancreatic islets, 5(6)-EET has been implicated in the mobilization of calcium and hormone secretion. 5(6)-EET is an inhibitor of T-type voltage-gated calcium channels (Cav3) that inhib...

化合物

DL-Phenylephrine HCl

Cat.No: T0453L

Synonym: Eyelo,DL-Phenylephrine hydrochloride

Phenylephrine-3-O-Sulfate

Cat.No: T35576

L-Phenylephrine

Cat.No: T68997

ARC 239 dihydrochloride

Cat.No: T22033

Target: Norepinephrine

Cat.No: T12913

Synonym: SKF 94836

Target: PDE

Cat.No: T4563

Synonym: neohetramine,松齐拉敏

Target: Histamine Receptor

Talibegron hydrochloride

Cat.No: T23557

Synonym: ZD2079 hydrochloride,ZD 2079

Target: Adrenergic Receptor

Cat.No: T27164

Synonym: PAK-9,PAK9,PAK 9,DHP218

Sandaracopimaric acid

Cat.No: T40563

Cat.No: T30427

Cat.No: TP2086

Cat.No: T35987

Synonym: CAY10563

Cat.No: T39281

Cat.No: T69127

Cat.No: T73083

Synonym: KT 210 ; K 351 ; Hypadil,Hypadil,KT 210,K 351

Cat.No: T35989

Cat.No: T35988

Cat.No: T36070

Cat. No.	Product Name	Target	Signaling Pathways
T17310	Phenylephrine 去氧肾上腺素,L-Phenylephrine,去氧肾上腺素碱,(R)-(-)-Phenylephrine	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Phenylephrine ((R)-(-)-Phenylephrine) 是一种选择性的α1-肾上腺素受体激动剂，常用作减充血剂。
T0453	Phenylephrine hydrochloride NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride	Endogenous Metabolite; Adrenergic Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Phenylephrine hydrochloride (NCI-c55641) 是选择性的α1-肾上腺素能受体激动剂，对α1A，α1B 和α1D 受体的pKis 分为4.70，4.87和5.86。
T7634	3-Hydroxymandelic Acid	Endogenous Metabolite	Metabolism
	3-Hydroxymandelic Acid 是一种 Phenylephrine 的代谢物。其中 Phenylephrine 是 α 受体激动剂。
T5263	p-Hydroxymandelic acid 4-羟基扁桃酸,4-Hydroxymandelic acid	Others; Endogenous Metabolite	Metabolism; Others
	p-Hydroxymandelic acid (4-Hydroxymandelic acid) 是有价值的芳香类化学品，常用于生产药物和食品添加剂。
T2944	Danshensu sodium salt Sodium Danshensu,(±)-DanShenSu sodium salt,丹参素钠,(±)-DanShenSu sodium sal	P450; Autophagy	Autophagy; Metabolism
	Danshensu sodium salt (Sodium Danshensu) 是从中国草本丹参中提取的一种天然产物，可以抑制去氧肾上腺素和CaCl2 在无Ca2+ 培养基中引起的血管收缩。
TN1624	Ethyl cinnamate	Calcium Channel; ROS; NO Synthase	Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
	Ethyl cinnamate 是食品香料和化妆品添加剂，也是哺乳动物组织的优良清除剂。
TN1724	Harmalol hydrochloride Harmidol hydrochloride	P450; Antioxidant	Metabolism; oxidation-reduction
	Harmalol hydrochloride (Harmidol hydrochloride) 是一种可从Peganum harmala L.的种子中提取出来的β-咔啉生物碱。Harmalol hydrochloride 是Harmaline 的主要代谢产物，在转录和翻译后水平上显著抑制二恶英介导的 CYP1A1 诱导。Harmalol hydrochloride 在去氧肾上腺素或KCl 预先收缩的分离大鼠胸主动脉制剂中显示出血管松弛活性。 Harmalol hydrochloride 具有抗氧化活性.
TN5061	Stephanine	Adrenergic Receptor; Antifection	GPCR/G Protein; Microbiology/Virology; Neuroscience
	l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of 6.76. Stephanine shows significant antiplasmodial activities with IC(50) ranged from 1.2 uM to 52.3 uM. Stephanine and crebanine have high inhibitory activity against gram-positive animal pathogenic bacteria, with MIC values of 0.078-0.312g/l, but low inhibitory activity against gram-negative animal pathogenic bacteria, they also inhibit...

天然产物

Phenylephrine

Cat.No: T17310

Synonym: 去氧肾上腺素,L-Phenylephrine,去氧肾上腺素碱,(R)-(-)-Phenylephrine

Target: Adrenergic Receptor

Phenylephrine hydrochloride

Cat.No: T0453

Synonym: NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride

Target: Endogenous Metabolite, Adrenergic Receptor

3-Hydroxymandelic Acid

Cat.No: T7634

Target: Endogenous Metabolite

p-Hydroxymandelic acid

Cat.No: T5263

Synonym: 4-羟基扁桃酸,4-Hydroxymandelic acid

Target: Others, Endogenous Metabolite

Danshensu sodium salt

Cat.No: T2944

Synonym: Sodium Danshensu,(±)-DanShenSu sodium salt,丹参素钠,(±)-DanShenSu sodium sal

Target: P450, Autophagy

Ethyl cinnamate

Cat.No: TN1624

Target: Calcium Channel, ROS, NO Synthase

Harmalol hydrochloride

Cat.No: TN1724

Synonym: Harmidol hydrochloride

Target: P450, Antioxidant

Cat.No: TN5061

Target: Adrenergic Receptor, Antifection

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