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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T80586 |
Anti-Mouse IL-1a Antibody (ALF-161)
|
Integrin | Cytoskeletal Signaling |
Anti-Mouse IL-1a Antibody 为针对小鼠IL-1a 的IgG1类免疫抑制单克隆抗体,源自Armenian Hamster。 | |||
T22232 |
Alfuzosin
SL 77499,UROXATRAL |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Alfuzosin (SL 77499) 是一种 α-1 肾上腺素能拮抗剂,用于治疗良性前列腺肥大和尿道功能障碍。 | |||
T0091 |
Alfuzosin hydrochloride
SL 77499-10,Alfuzosin HCl,盐酸阿夫唑嗪 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Alfuzosin hydrochloride (Alfuzosin HCl) 是一种 α1 肾上腺素受体拮抗剂,可用于良性前列腺增生(BPH)的研究。 | |||
T6374 |
Alfacalcidol
Bondiol,Etalpha,阿法骨化醇,1-hydroxy Vitamin D3,1.alpha.-Hydroxyvitamin D3,1-hydroxycholecalciferol |
Others | Others |
Alfacalcidol (Etalpha) 是一种维生素 D3 衍生物,是非选择性的维生素 D 受体活化剂,有用于骨质疏松研究的潜力。 | |||
T22254 |
Alflutinib
AST2818,ASK120067 |
EGFR; P450 | Angiogenesis; JAK/STAT signaling; Metabolism; Tyrosine Kinase/Adaptors |
Alflutinib (ASK120067) 是 EGFR 抑制剂。 它对 T790M 的性耐药突变以及 EGFR 活性突变具有抑制作用。它对于癌症疾病,特别是非小细胞肺癌(NSC-LC)方面具有研究潜力。 | |||
T1338 |
Sucralfate
硫糖铝,Sucrose octasulfate–aluminum complex |
FGFR; Others; Antibacterial; Prostaglandin Receptor | Angiogenesis; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Others; Tyrosine Kinase/Adaptors |
Sucralfate (Sucrose octasulfate–aluminum complex) 是一种口服活性胃保护剂。它抑制消化性活性,并与黏膜损伤时暴露的带负电荷的上皮下蛋白结合,形成一层粘性层,保护血管床和增殖区。它可用于预防和治疗胃肠道疾病。 | |||
T7349 |
Ralfinamide
(S)-2-[[4-[(2-氟苄基)氧基]苄基]氨基]丙酰胺,Priralfinamide,FCE-26742A |
Sodium Channel | Membrane transporter/Ion channel |
Ralfinamide (Priralfinamide) 是一种具有口服活性的,来源于 α-aminoamide 的钠离子通道阻滞剂, 在缓解疼痛方面有研究的价值。 | |||
TP1029 |
Thymalfasin
胸腺法新,Thymosin α1,醋酸胸腺α1 |
Others | Others |
Thymalfasin (Thymosin α1) 是一种免疫调节化合物,可增强 Thl 的免疫应答。 | |||
T7175 |
Alflutinib mesylate
甲磺酸伏美替尼,AST2818 mesylate |
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Alflutinib mesylate (AST2818 mesylate) 是一种不可逆的酪氨酸激酶抑制剂,可选择性抑制 EGFR 突变。 | |||
T7547 |
Ralfinamide mesylate
FCE-26742A (mesylate) |
Sodium Channel | Membrane transporter/Ion channel |
Ralfinamide mesylate (FCE-26742A (mesylate)) 是一种口服有效,来源于 α-aminoamide 的钠离子通道阻滞剂, 在缓解疼痛方面有研究价值。 | |||
T26592 |
Alfadolone acetate
GR 2,GR-2,R140,GR2R-140 |
||
Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist. | |||
T77087 | Mipeginterferon alfa-2b | ||
Mipeginterferon alfa-2b 是一种干扰素IFNA2b 类似物。包括一个 N 末端和 10 个赖氨酸 N6 在内的 11 个氨基,平均被取代掉 5 个。Mipeginterferon alfa-2b 的相对分子质量为 40 kDa。 | |||
T80565 |
Gulgafafusp alfa
|
||
Gulgafafusp alfa 为人源化IgG2κ类抗体,专一性靶向GLP1R(胰高血糖素样肽1受体)。 | |||
T25047 |
Alfetamine
alpha-allyl-phenethylamine |
||
Alfetamine is a chemical compound of the phenethylamine family. It is similar to imipramine and amitriptyline, two tricyclic antidepressants. | |||
T31392 |
Detralfate
|
||
Detralfate is a biochemical. | |||
T29860 |
Alfaprostol
|
||
Alfaprostol is a bioactive chemical. | |||
T81917 |
Lorukafusp alfa
hu14.18-IL2,EMD 273063,14.18 mAb |
||
Lorukafusp alfa(14.18 mAb; hu14.18-IL2)是一种由人源化14.18抗GD2抗体和IL210连接而成的免疫细胞因子。该化合物通过其hu14.18-IL2与肿瘤细胞表面的GD2结合,激活抗体依赖性细胞毒性(ADCC)和补体依赖性细胞毒性,以及与效应细胞上Fc受体结合并激活NK和T细胞的活性,从而显现出抗肿瘤效果。 | |||
T82449 |
Eramkafusp Alfa
|
||
Eramkafusp Alfa为针对小鼠B淋巴细胞上CD20 (MS4A1) 抗原的人源化IgG1单克隆抗体。 | |||
T81528 |
Peginterferon alfacon-2
|
||
Peginterferon alfacon-2为针对IFNAR1/2的人源化抗体。 | |||
T10279 |
Alfacalcidol-D6
|
Others | Others |
Alfacalcidol-D6 is a deuterated Alfacalcidol. Alfacalcidol is a non-selective VDR activator medication. | |||
T76236 | Rilunermin alfa | ||
Rilunermin alfa (SCB-313) 是一种活性化合物。Rilunermin alfa 可用于各种生化研究。 | |||
T77082 | Melredableukin alfa | ||
Melredableukin alfa (RO-7049665)是一种由人IgG1-κ通过多肽连接子与人突变白细胞介素2(IL2 mutin)融合形成的融合蛋白。它适用于乙型肝炎和溃疡性结肠炎的研究。 | |||
T76239 | Efrilacedase alfa | ||
Efrilacedase alfa 是一种活性化合物。Efrilacedase alfa 可用于各种生化研究。 | |||
T76853 | Ropeginterferon alfa-2b | ||
Ropeginterferon alfa-2b (Ropeginterferon alfa-2b-njft) 为单聚乙二醇化IFN-α类化合物,主要应用于骨髓增性肿瘤研究领域。 | |||
T76964 | Valanafusp alfa | ||
Valanafusp alfa (AGT-181) 是一种融合了抗人胰岛素受体 (HIR) 和人硬糖苷酶 (IDUA) 的嵌合单克隆抗体的脑穿透重组融合蛋白。该化合物主要应用于粘多糖病 I 型 (MPS I) 的研究领域。 | |||
T131401 |
Halfordamine
|
||
Halfordamine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131401。 | |||
T29859 |
Alfadolone
|
||
Alfadolone is an anesthetic derivative of pregnanedione. | |||
T125793 |
Malformin-B4
|
||
Malformin-B4 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125793,CAS号为 149596-55-4。 | |||
T80592 |
Ledelabricin alfa
|
Endogenous Metabolite | Metabolism |
Ledelabricin alfa为人蛋白多糖proteoglycan 4 (PRG4)亚型A的一种变体,主要功能为关节/边界润滑剂,常用于关节病变的研究。 | |||
T81622 |
Octocog alfa
|
||
Octocog alfa为第二代全长重组因子VIII,具有抗血友病A功能。 | |||
T82502 |
Efaprinermin alfa
OMP-336B11 |
||
Efaprinermin alfa (OMP-336B11),一种人源化单克隆抗体,靶向TNFRSF18。该化合物为GITR配体-Fc融合蛋白。 | |||
T25728 |
Limaprost alfadex
Opalmon,OP 1306 - alpha-cyclodextrin,Prorenal |
||
Limaprost alfadex is an oral medicine for the circulatory system (for confinement-related thromboangiitis ulcer, anaphrodisia, sharp pain and ischemia characteristics symptom, the improvement of subjective symptom and walking ability with postnatal lumbar | |||
T78241 |
Asfotase alfa
ENB-0040 |
||
Asfotase alfa (ENB-0040) 是一款针对骨骼的基因重组糖蛋白。该药物提升了Akp2−/−基因敲除小鼠的存活率、骨矿化及骨骼生长,并且缓解了脚部、胸部、下肢及颌骨矿化缺损。它主要用于对围产期、婴幼儿及青少年型低磷酸酶血症(HPP)进行研究。 | |||
T77169 |
Simlukafusp alfa
|
||
Simlukafusp alfa (FAP-IL2v) 是一种免疫细胞因子,包括一种抗成纤维细胞活化蛋白 α (FAPα) 的抗体和一种只结合 IL-2Rβγ的 IL-2变体。Simlukafusp alfa 是一种人IgG1抗体。 | |||
T77171 |
Efineptakin alfa
|
||
Efineptakin alfa (NT-17) 是一种长效重组人 IL-7。 Efineptakin alfa 支持人和小鼠体内 CD4+和 CD8+细胞的增殖和存活。 Efineptakin alfa 可用于胶质母细胞瘤的研究。 | |||
T81270 |
Ripafollitropin alfa (bovine)
|
||
Ripafollitropin alfa (bovine)为一种结合了重组促卵泡激素(FSH)与绒毛膜促性腺激素(HCG)的融合蛋白。 | |||
T82499 |
Efmoroctocog alfa
|
||
Efmoroctocog alfa,一种重组人凝血因子 VIII-Fc 融合蛋白(rFVIIIFc),主要应用于血友病 A 研究。 | |||
T82508 |
Eciskafusp alfa
|
PD-1/PD-L1 | Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation |
Eciskafusp alfa是一种针对程序性细胞死亡1(PDCD1,亦称PD-1)的顺式靶向IL2v免疫细胞因子。它优先选择抗原特异性干细胞样PD-1+ TCF-1+ CD8+ T细胞,并促使这些细胞分化成更高效的效应器细胞。Eciskafusp alfa主要用于癌症与慢性感染的研究领域。 | |||
T82498 |
Eftansomatropin alfa
|
||
Eftansomatropin alfa是一种融合蛋白,由GH1与IGHG4 Fc结合而成,旨在靶向生长激素受体(GSH)。 | |||
T22707 |
Dalfopristin (mesylate) (112362-50-2 free base)
Dalfopristin (mesylate) |
Others | Others |
Dalfopristin (mesylate) is a streptogramin antibiotic and a 50S ribosome inhibitor. Streptogramins are produced by a variety of Streptomyces sp as a mixture (ratio of 7:3) of two chemically unrelated compounds, type A and B. Dalfopristin, the type A Strep | |||
T76943 | Cepeginterferon alfa-2b | ||
Cepeginterferon alfa-2b是一种聚乙二醇化干扰素, 其聚乙二醇基由分子量为20 kDa的PEG构成。该化合物广泛应用于丙型肝炎病毒(HCV)、真性红细胞增多症(PV)和原发性血小板增多症(ET)等疾病的研究中。 | |||
T77038 | Interferon alfa | ||
Interferon alfa 是 I 型干扰素,可激活新基因,对靶细胞产生有效抗病毒和抗增殖活性。Interferon alfa 的信号传导需要 Stat1和 Stat2 的受体依赖性激活,形成异源二聚化 STAT。STAT 复合物与 DNA 结合蛋白 IRF-9 (p48) 结合并形成 ISGF-3 (IFN 刺激基因因子 3)。随后由 ISGF-3 进一步激活驱动基因,实现抗病毒功能。 | |||
T77112 | Onfekafusp alfa | ||
Onfekafusp alfa(L19TNF)是一款将工程化的L19抗体scFv与人TNF融合所得的同源三聚体。该化合物主要应用于恶性胶质瘤的研究。 | |||
T77131 | Clervonafusp alfa | ||
Clervonafusp alfa (VAL-1221) 作为一种融合蛋白,针对胞浆及溶酶体糖原进行靶向。该化合物结合了穿透细胞的抗体Fab部分与重组人酸性葡萄糖苷酶 (rhGAA),通过核苷转运体ENT-2进入细胞质,再利用甘露糖-6-磷酸受体(M6PRs)导向溶酶体。主要应用于晚发型庞贝病的研究领域。 | |||
TP2285 |
Quinupristin-Dalfopristin Complex (mesylate)
|
Others | Others |
Quinupristin-Dalfopristin Complex is a mixture of two streptogramin antibiotics. Quinupristin-dalfopristin complex is a mixture of two streptogramin antibiotics, dalfopristin, and quinupristin. Streptogramin antibiotics are divided into types A and B, whi | |||
T82616 |
Dalcinonacog alfa
CB-2679d,ISU-304,DalcA |
||
Dalcinonacog alfa为重组FIX因子,用于血友病B的科研之用。 | |||
T82887 |
Bifikafusp alfa
L19-IL2 |
||
Bifikafusp alfa (L19-IL2) 是一种由人类L19抗体与细胞因子白介素2 (IL2) 结合而成的免疫融合蛋白,特异性针对纤维连接蛋白的EDB区域,并表现出抗癌活性。 | |||
T82526 |
Drotrecogin alfa (activated)
|
||
Drotrecogin alfa activated (DrotAA)为重组人活化蛋白C(APC)。该化合物能够抑制由烟雾引起的大鼠肺微血管通透性上升及促炎细胞因子IL-1β水平增加,具有抗凝血与抗炎作用,并促进纤溶过程。Drotrecogin alfa activated主要用于重症脓毒症的实验研究。 | |||
T81573 |
Pabinafusp alfa
JR-141 |
||
Pabinafusp alfa (JR-141) 是由Iduronate 2-sulfatase和抗人转铁蛋白受体抗体结合而成的转铁蛋白受体靶向抗体。它具备穿透血脑屏障的能力,可防止粘多糖病II型(MPS II)小鼠中枢神经系统中硫酸肝素(HS)的积累。此外,Pabinafusp alfa能够促进小鼠的学习能力,并抑制中枢神经系统神经元的损伤。 | |||
T81256 |
Rozibafusp alfa
AMG-570 |
||
Rozibafusp alfa为靶向ICOSLG的IgG2-κ型抗体,结合TNFSF13B融合蛋白。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13592 |
Calf thymus DNA
DNA from calf thymus, Thymonucleic acid |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Calf thymus DNA (DNA from calf thymus, Thymonucleic acid) 是一种从牛胸腺中提取出来的高质量双链模板DNA,可广泛应用于DNA 结合抗癌剂和调节DNA 结构和功能的DNA 结合剂的研究。 | |||
TQ0152 |
Dalfopristin
RP54476,达福普汀 |
Antibacterial; Antibiotic | Microbiology/Virology |
Dalfopristin (RP54476) 是一种半合成的链霉素抗生素。 Quinupristin/Dalfopristin (Q/D) 用于治疗耐多药粪肠球菌感染。 | |||
T36489 |
Malformin A
|
||
Malformin A is a cyclopentapeptide fungal metabolite that has been found in A. niger and has diverse biological activities. It is a plant growth regulator that induces malformations in plant structure. Malformin A inhibits replication of tobacco mosaic virus (TMV) in local lesion and leaf-disc assays (IC50s = 19.7 and 45.4 μg/ml, respectively). It is cytotoxic to NCI-H460, MIA PaCa-2, MCF-7, SF-268, and WI-38 cancer cells (IC50s = 70, 50, 100, 70, and 100 nM, respectively), inhibits proliferati... | |||
T36961 |
Malformin C
|
||
Malformin C is a natural fungus-derived bicyclic pentapeptide that has antibacterial properties, particularly against species of Bacillus. Malformin C potently blocks the ability of bleomycin to induce G2 arrest in human T-cell leukemia-derived Jurkat cells (IC50 = 0.9 nM). It less potently abrogates colchicine-induced M phase arrest in Jurkat cells (IC50 = 24 nM). Malformin C inhibits cell growth dose-dependently in Colon 38 and HCT 115 cancer cells (IC50s = 0.27 and 0.18 μM, respectively) but ... |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-03962 |
AFM Protein, Human, Recombinant (His)
afamin,ALBA,ALB2,ALF |
Human | HEK293 Cells |
Afamin is an 87 kDa glycoprotein with five predicted N-glycosylation sites. Afamin's glycan abundance contributes to conformational and chemical inhomogeneity presenting great challenges for molecular structure determination. Afamin, a human plasma glycoprotein and putative transporter of hydrophobic molecules, has been shown to act as extracellular chaperone for poorly soluble, acylated Wnt proteins, forming a stable, soluble complex with functioning Wnt proteins. The 2.1-Å crystal structure of... | |||
TMPH-03424 |
Rotavirus A (strain Nebraska calf diarrhea virus) VP4 Protein (His & Myc)
|
RV-A | E. coli |
Rotavirus A (strain Nebraska calf diarrhea virus) VP4 Protein (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 33.2 kDa and the accession number is P17465. | |||
TMPH-03417 |
Rotavirus A (strain Nebraska calf diarrhea virus) VP6 Protein (His)
|
RV-A | E. coli |
Rotavirus A (strain Nebraska calf diarrhea virus) VP6 Protein (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 50.8 kDa and the accession number is A7J3A1. | |||
TMPY-04012 |
Influenza A H7N9 (A/Anhui/1-BALF_RG6/2013) Nucleoprotein/NP Protein (His)
NP Protein |
H7N9 | Baculovirus Insect Cells |
Influenza A H7N9 (A/Anhui/1-BALF_RG6/2013) Nucleoprotein/NP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.8 kDa and the accession number is A0A024E372. | |||
TMPH-03422 |
Rotavirus A (strain Nebraska calf diarrhea virus) VP7 Protein (His & Myc)
|
RV-A | E. coli |
Rotavirus A (strain Nebraska calf diarrhea virus) VP7 Protein (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 36.2 kDa and the accession number is P04511. |