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Search Results for " uterus "

13

抑制剂 & 化合物

8

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T8984	FLTX1	Estrogen Receptor/ERR; Estrogen/progestogen Receptor	Endocrinology/Hormones
	FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under permeabilized and non-permeabilized conditions. Additionally, FLTX1 demonstrates strong antiestrogenic activity in breast cancer cells, resembling the potent antiestrogenic properties of Tamoxifen. Notably, FLTX1 does not exhibit any estrogenic agonistic effect on the uterus.
T35841	5-Benzyloxygramine	Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience
	5-Benzyloxygramine 是一种 N 蛋白、蛋白互作的原位稳定剂，具有抗病毒和稳定 N-NTD 蛋白的作用。它能够阻断多巴胺受体，可拮抗 5-HT 对大鼠子宫和兔耳的作用。
T1433	Ritodrine hydrochloride DU21220,盐酸利托君,Ritodrine HCl,NSC 291565	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Ritodrine hydrochloride (NSC 291565) 是一种 β-2肾上腺素受体激动剂。
T4996	Atosiban 阿托西班,RWJ22164,RW22164	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Atosiban (RW22164) 是一种脱氨基催产素类似物，是一种九肽，也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂，可用于自发早产的研究。
T5148	Atosiban acetate RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Atosiban acetate (RW22164) 是一种脱氨基催产素类似物，是一种九肽，也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂，可用于自发早产的研究。
T11794	L-368,899 hydrochloride	Others	Others
	L-368,899 hydrochloride, used as a tocolytic agent, is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptor, respectively.
T10273	AhR modulator-1	Others	Others
	AhR modulator-1 is a selective and orally active aryl hydrocarbon receptor (AhR) modulator. It inhibits metastasis, in part, by inhibiting prostatic VEGF production prior to tumor formation. It also possesses anti-estrogenic properties in rat uterus.
T36728	9-deoxy-9-methylene Prostaglandin E2 9-deoxy-9-methylene Prostaglandin E2
	9-deoxy-9-methylene Prostaglandin E2 (9-deoxy-9-methylene PGE2) is a stable, isosteric analog of PGE2 . 9-deoxy-9-methylene PGE2 retains the biological profile of PGE2 with fewer side effects. In the rat 9-deoxy-9-methylene PGE2 is equipotent to PGE2 in decreasing blood pressure. It also stimulates the gerbil colon and primate uterus at the same potency as PGE2.
T36925	Neuromedin C (porcine)
	Neuromedin C (porcine) 是一种铃蟾肽样神经肽，可从猪脊髓中获得。Neuromedin C (porcine) 对大鼠子宫具有收缩活性。Neuromedin C (porcine) 有研究神经系统相关疾病的潜力。
T76049	Demoxytocin
	Demoxytocin为一种异源性环肽，属于催产素类似物。其通过影响细胞膜通透性，提升平滑肌细胞内钙离子含量，进而加强平滑肌细胞收缩力，具备刺激子宫平滑肌收缩的能力，发挥催产素功能。此外，Demoxytocin在研究早产破裂引发的分娩刺激中有应用。
T37319	5β-Dihydroprogesterone
	5β-Dihydroprogesterone (5β-DHP) is a progesterone receptor agonist and metabolite of progesterone .1,2It is formed from progesterone by 5β-reductase.25β-DHP inhibits spontaneous contractions in isolated rat uterus when used at a concentration of 10 μg/ml, an effect that can be blocked by the progesterone receptor antagonist RU486 but not the GABAAreceptor antagonist picrotoxin .1It is a negative modulator of homooligomeric Ρ1 subunit-containing GABAAreceptors, inhibiting GABA-induced currents in...
T69696	TAS-108 citrate
	TAS-108, also known as SR16234, is a synthetic, antiestrogenic steroidal compound with potential antitumor activity. TAS-108 binds to and inhibits estrogenic receptor alpha (ERa), mainly expressed in the mammary gland and uterus and upregulated in estrogen-dependent tumors. Blockage of ERa by TAS-108 prevents the binding and effects of estrogen and may lead to an inhibition of estrogen-dependent cancer cell proliferation. TAS-108 also is a partial agonist of the estrogenic receptor beta (ERb), e...
T27970	Mabuterol free base Mabuterol,PB 868Cl	Others	Others
	Mabuterol is a selective agonist of β2 adrenoreceptor with no beta 1-stimulation. Mabuterol inhibited the positive inotropic effect of isoprenaline at 10(-7) g/ml and decreased the maximum driving frequency at 3 X 10(-6) g/ml. Mabuterol was 3 times more p

化合物

Cat.No: T8984

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor

5-Benzyloxygramine

Cat.No: T35841

Target: Dopamine Receptor, 5-HT Receptor

Ritodrine hydrochloride

Cat.No: T1433

Synonym: DU21220,盐酸利托君,Ritodrine HCl,NSC 291565

Target: Adrenergic Receptor

Cat.No: T4996

Synonym: 阿托西班,RWJ22164,RW22164

Target: Oxytocin Receptor, Vasopressin Receptor

Atosiban acetate

Cat.No: T5148

Synonym: RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班

Target: Oxytocin Receptor, Vasopressin Receptor

L-368,899 hydrochloride

Cat.No: T11794

Target: Others

AhR modulator-1

Cat.No: T10273

Target: Others

9-deoxy-9-methylene Prostaglandin E2

Cat.No: T36728

Synonym: 9-deoxy-9-methylene Prostaglandin E2

Neuromedin C (porcine)

Cat.No: T36925

Cat.No: T76049

5β-Dihydroprogesterone

Cat.No: T37319

TAS-108 citrate

Cat.No: T69696

Mabuterol free base

Cat.No: T27970

Synonym: Mabuterol,PB 868Cl

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T14865	Carboprost tromethamine	Prostaglandin Receptor	GPCR/G Protein; Immunology/Inflammation
	Carboprost tromethamine 是合成的前列腺素 F2α的15-甲基类似物，能有效促进子宫的规律收缩，显着减少产中及产后出血量。
T4S1518	Pseudoginsenoside RT1 拟人参皂苷 RT1,假人参皂苷RT1	Others	Others
	Pseudoginsenoside RT1 是分离自 Randia siamensis 中，具有鱼毒素作用。它可导致血压下降、心率加快和子宫自发收缩力增加。
T0478	Progesterone 孕酮,Pregn-4-ene-3,20-dione	Estrogen/progestogen Receptor; Progesterone Receptor; Opioid Receptor; Endogenous Metabolite	Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience; Others
	Progesterone (Pregn-4-ene-3,20-dione) 是类固醇激素，能够调节月经周期。
T15824	Lysergol	Antibacterial	Microbiology/Virology
	Lysergol 已被用作一种降血压、精神镇痛药以及刺激子宫和肠道的药物。 Lysergol 是从 Ipomoea muricata 的种子中分离出来的一种棒状生物碱，是药物和营养物质的生物增强剂，具有抗菌活性。
T6S0033	Crotonoside 巴豆苷；异鸟苷,巴豆苷,Isoguanosine,2-HYDROXYADENOSINE	Others; FLT; HDAC	Angiogenesis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Others; Tyrosine Kinase/Adaptors
	Crotonoside (Isoguanosine) 是从中草药巴豆中分离出来的一种天然产物。它抑制 FLT3 和 HDAC3/6，有治疗急性髓性白血病 (AML)的研究潜力。
T6S2140	β-Anhydroicaritin Anhydroicaritin,Beta-Anhydroicaritin,脱水淫羊藿素	MMP; Others; TNF; Interleukin	Apoptosis; Immunology/Inflammation; Others; Proteases/Proteasome
	β-Anhydroicaritin 是从乳香提取的一种天然产物，具有重要的生物学和药理学作用，如抗骨质疏松症，雌激素调节和抗肿瘤特性。它改善牙周组织的降解，抑制糖尿病大鼠 TNF-α 和 MMP-3 的合成和分泌。它抑制细胞内 Ca2+的升高，并显著降低 iNOS 蛋白的表达。
TN3605	Casegravol	Others	Others
	Casegravol shows antiproliferative activity against human gastric adenocarcinoma (MK-1), human uterus carcinoma (HeLa), and murine melanoma (B16F10) cells.
TN4839	Psidial A	Others	Others
	Psidial A shows activity to enzyme PTP1B; it also reduces tumor growth and stimulate uterus proliferation.

天然产物

Carboprost tromethamine

Cat.No: T14865

Target: Prostaglandin Receptor

Pseudoginsenoside RT1

Cat.No: T4S1518

Synonym: 拟人参皂苷 RT1,假人参皂苷RT1

Target: Others

Cat.No: T0478

Synonym: 孕酮,Pregn-4-ene-3,20-dione

Target: Estrogen/progestogen Receptor, Progesterone Receptor, Opioid Receptor, Endogenous Metabolite

Cat.No: T15824

Target: Antibacterial

Cat.No: T6S0033

Synonym: 巴豆苷；异鸟苷,巴豆苷,Isoguanosine,2-HYDROXYADENOSINE

Target: Others, FLT, HDAC

β-Anhydroicaritin

Cat.No: T6S2140

Synonym: Anhydroicaritin,Beta-Anhydroicaritin,脱水淫羊藿素

Target: MMP, Others, TNF, Interleukin

Cat.No: TN3605

Target: Others

Cat.No: TN4839

Target: Others

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