Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2330 |
Rilpivirine
TMC278,R278474,利匹韦林,DB08864 |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Rilpivirine (R278474) 是一种二芳基嘧啶衍生物和非核苷逆转录酶抑制剂,具有抗 HIV-1 的抗病毒活性,用于治疗 HIV 感染。 | |||
T27154 |
Dexelvucitabine
D-D-4FC,DPC-817,RVT,beta-D-D-4FC,DFC |
Reverse Transcriptase | Microbiology/Virology |
Dexelvucitabine (RVT) 是一种胞苷类似物,一种口服有活性的核苷逆转录酶抑制剂。它是一种 2'-脱氧胞苷抗逆转录病毒剂。它是一种有效的抗 HIV-1病毒剂,这些病毒聚合酶中含有胸苷类似物和/或 M184V 突变。 | |||
T1404 |
Stavudine
d4T,Sanilvudine,BMY-27857,NSC 163661,司他夫定 |
Apoptosis; Nucleoside Antimetabolite/Analog; HIV Protease; NOD-like Receptor (NLR); Reverse Transcriptase; Autophagy | Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome |
Stavudine (BMY-27857) 是一种口服活性核苷逆转录酶抑制剂,还抑制线粒体 DNA 的复制,具有抗HIV-1和HIV-2的活性。它降低 NLRP3 炎症小体激活,调节淀粉样 β 自噬,诱导细胞凋亡。 | |||
T7700 |
Lersivirine
3-氰基-5-[[3,5-二乙基-1-(2-羟基乙基)-1H-吡唑-4-基]氧基]苯腈,Lersivirine(UK 453061),UK-453061 |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Lersivirine (UK-453061) 是非核苷逆转录的抑制剂 (NNRTI),有效抑制 NNRTI 耐药病毒。它对野生型人类免疫缺陷病毒和临床相关 NNRTI 耐药菌株显示出强大的抗逆转录病毒活性。 | |||
T1815 |
Dapivirine
R147681,达匹维林,TMC120 |
Apoptosis; HIV Protease; Reverse Transcriptase; Autophagy | Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome |
Dapivirine (R147681) 是一种二芳基嘧啶非核苷类逆转录酶抑制剂。 | |||
T1513 |
Telbivudine
NV 02B,L-Thymidine,Epavudine,替比夫定 |
Others; HBV; Reverse Transcriptase | Microbiology/Virology; Others |
Telbivudine (NV 02B) 是一种乙型肝炎病毒复制的抗病毒抑制剂,是一种具有口服活性的胸腺嘧啶核苷类似物。 | |||
T0110 |
Zalcitabine
Dideoxycytidine,ddC,扎西他滨,NSC 606170,Ro 24-2027/000,2',3'-Dideoxycytidine |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Zalcitabine (Dideoxycytidine) 是一种核苷类似物逆转录酶抑制剂,用于HIV 感染相关研究。 | |||
T3172 |
Trovirdine
曲韦定,LY300046 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Trovirdine (LY300046) 是一种硫脲类非核苷类逆转录酶抑制剂。 | |||
T2578 |
Didanosine
ddI,去羟肌苷,2',3'-Dideoxyinosine |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Didanosine (ddI) 是一种逆转录酶抑制剂,IC50为490nM。 | |||
T2393 |
Efavirenz
EFV,依非韦伦,DMP 266,依法韦仑,Sustiva,Stocrin,L-743726 |
HIV Protease; Reverse Transcriptase; Autophagy | Autophagy; Microbiology/Virology; Proteases/Proteasome |
Efavirenz (DMP 266) 是一种人类免疫缺陷病毒 1 非核苷类似物逆转录酶抑制剂。它也是一种野生型HIV-1 RT 抑制剂,Ki 为 2.93 nM,有效抑制 HIV-1 复制,IC95为 1.5 nM。 | |||
T31860 |
Fosdevirine
GSK-2248761A,IDX 899,GSK 2248761A,GSK 2248761,GSK-2248761,IDX-12899,GSK2248761,FDV,GSK2248761A |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Fosdevirine (GSK2248761) 是一种具有选择性和高效性的非核苷类逆转录酶 (NNRTI) 抑制剂 ,具有抗 HIV 活性,可用于研究迟发性癫痫等神经系统相关疾病。 | |||
T2551 |
Etravirine
TMC125,依曲韦林,R165335 |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Etravirine (R165335) 是一种非核苷逆转录酶抑制剂,具有抗 HIV 的作用。 | |||
T68103L |
Mk-6186 HCl
Mk-6186 HCl(1034474-19-5 Free base) |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
MK-6186 HCl,一种新型非核苷类逆转录酶抑制剂,具有抗病毒活性,可用于研究HIV。 | |||
T6214 |
Emtricitabine
恩曲他滨,FTC,Emtriva,BW1592 |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Emtricitabine (FTC) 是一种核苷逆转录酶抑制剂, 在 PBMC 细胞中的 EC50值为0.01 µM,可研究 HIV 感染。 | |||
T1267 |
Abacavir
Epzicom,Ziagen,阿巴卡韦,Abacavir sulfate |
Apoptosis; HIV Protease; Reverse Transcriptase | Apoptosis; Microbiology/Virology; Proteases/Proteasome |
Abacavir (Ziagen) 是一种核苷类似物逆转录酶抑制剂。 | |||
T68103 |
MK-6186
|
Reverse Transcriptase | Microbiology/Virology |
MK-6186 是一种新型非核苷类逆转录酶抑制剂,具有抗病毒活性,可用于研究病毒感染。 | |||
T60540 |
Netivudine
|
||
Netivudine 是一种有效的核苷类逆转录酶抑制剂(NRTIs),是一种核苷类似物,具有抗水痘带状疱疹病毒活性,可用于治疗人类免疫缺陷病毒(HIV)感染。Netivudine 通过抑制逆转录酶起作用,通过抑制作用减少体内的病毒载量,减缓疾病的进展。 | |||
T67804 |
KM-023
|
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
KM-023是一种新的第二代非核苷类逆转录酶抑制剂,可用于研究人类免疫缺陷病毒(HIV)1型感染。 | |||
T2279 |
Tizoxanide
替唑尼特,Desacetyl-nitazoxanide,TIZ |
Antiviral; HIV Protease; Antibacterial; Autophagy | Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome |
Tizoxanide (Desacetyl-nitazoxanide) 是 Nitazoxanide 活性代谢物,有抗HIV-1的活性。Nitazoxanide 可抗细菌和多种病毒复制。 | |||
T3632 |
Doravirine
多拉维林,多拉韦林,MK-1439 |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Doravirine (MK-1439) 是一种高度特异性的HIV-1非核苷逆转录酶抑制剂,对野生型以及K103N 和Y181C 逆转录酶突变体的IC50值分别为 4.5 nM,5.5 nM 和 6.1 nM。 | |||
T7212 |
Delavirdine mesylate
U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate) |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Delavirdine mesylate (BHAP-U 90152(mesylate)) 是一种口服活性非核苷逆转录酶抑制剂。它抑制 HIV-1 病毒复制,可以用于艾滋病的相关研究。它选择性地抑制 HIV-1 逆转录酶,其选择性超过 DNA 聚合酶 α 和 DNA 聚合酶 δ 。 | |||
T31860L |
(Iso)-Fosdevirine
(Iso)-Fosdevirine(Iso-1018450-26-4),(Iso)-GSK2248761 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
(Iso)-Fosdevirine ( (Iso)-GSK2248761) 是一种具有选择性和高效性的非核苷类逆转录酶 (NNRTI) 抑制剂 ,具有抗 HIV 活性,可用于研究迟发性癫痫等神经系统相关疾病。 | |||
T1595 |
Nevirapine
NSC 641530,奈韦拉平,BI-RG 587,奈伟拉平,NVP |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Nevirapine (NVP) 是一种 HIV-1逆转录酶非核苷抑制剂,Ki 值为 270 μM,可用于研究 HIV/AIDS。 | |||
T1675 |
Adefovir dipivoxil
Hepsera,GS 0840,阿德福韦酯,Preveon |
Others; HBV; Reverse Transcriptase | Microbiology/Virology; Others |
Adefovir dipivoxil (GS 0840) 是一种腺苷类似物,是核苷逆转录酶抑制剂 Adefovir 的口服前药,具有抗乙型肝炎病毒、疱疹病毒和人类免疫缺陷病毒的活性。 | |||
T2409L |
Tenofovir Disoproxil Fumarate
GS-1278 Disoproxil Fumarate,Tenofovir DF,富马酸替诺福韦酯 |
HBV; HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Tenofovir Disoproxil Fumarate (GS-1278 Disoproxil Fumarate) 是一种核苷酸逆转录酶抑制剂,有潜力研究艾滋病和慢性乙型肝炎。 | |||
T7447 |
Adefovir
|
HBV; Reverse Transcriptase; Telomerase | DNA Damage/DNA Repair; Microbiology/Virology |
Adefovir 是一种单磷酸腺苷类似物抗病毒剂,在细胞内转化为 Adefovir diphosphate 后可抑制HBVDNA 聚合酶。它在 HepG2.2.15 细胞系中对HBV 的IC50为 0.7 μM。它对多种病毒(包括HBV 和疱疹病毒)具有良好的抗病毒活性。 | |||
T16098 |
Islatravir
MK-8591 |
HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Islatravir (MK-8591) 是一种核苷逆转录酶抑制剂,是抗HIV-1药物,对 HIV-1 (WT),HIV-1 (M184V),HIV-1 (MDR) 的EC50值分别为 0.068 nM,3.1 nM 和 0.15 nM。 | |||
T29037 |
UC-781
NSC 675186,UC781,UC 781 |
Antiviral; HIV Protease | Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome |
UC-781 (NSC-675186) 是一种高效且具有选择性的人类免疫缺陷病毒 HIV-1 非核苷类逆转录酶(NNRTI)I抑制剂 ,C50 值为 5 nM。UC-781 具有抗病毒活性和耐药性。UC-781状态稳定,较低的 PH 或不同温度对其影响较小。 | |||
T14489 |
Azvudine
4-氨基-1-(4-C-叠氮基-2-脱氧-2-氟-BETA-D-呋喃阿拉伯糖基)-2(1H)-嘧啶酮,FNC,RO-0622 |
HCV Protease; HBV; HIV Protease; Reverse Transcriptase | Microbiology/Virology; Proteases/Proteasome |
Azvudine (FNC) 是一种有效的核苷逆转录酶抑制剂 (NRTI),对 HIV、HBV 和 HCV 具有抗病毒活性。它抑制耐 NRTI 的病毒株,高效抑制 HIV-1和 HIV-2。 | |||
T27625 |
IQP-0528
SJ-3991,SJ3991,IQP0528 |
Antiviral; HIV Protease; Reverse Transcriptase | Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome |
IQP-0528是一种高效的非核苷类逆转录酶抑制剂(NNRTI),通过阻断病毒进入,有可能用于治疗HIV 感染,并且作为杀微生物凝胶显示出抗病毒活性。IQP-0528对HIV-1和HIV-2都显示出抑制作用,对HIV-1的EC50为0.2 nM,对HIV-2的EC50为100 nM。 | |||
T28204 |
NSC-176377
NSC 176377 |
||
NSC-176377 is a non-nucleoside reverse transcriptase inhibitor. | |||
T2330L |
Rilpivirine HCl
Rilpivirine hydrochloride,TMC278,Rilpivirine,TMC-278,TMC 278. trade name Edurant |
||
Rilpivirine is a potent non-nucleoside reverse transcriptase inhibitor. | |||
T27542 |
HI-207
HI207,HI 207 |
||
HI-207 is an inhibitor of non-nucleoside reverse transcriptase. | |||
T24354 |
L 738372
L-738,372,L 738,372,L738372,L738,372,L-738372 |
||
L 738372 is a non-nucleoside inhibitor of HIV-1 reverse transcriptase. | |||
T24087 |
GCA-186
I-EBU-dM,IEBUdM,I EBU dM,GCA 186 |
||
GCA-186 is an effective non-nucleoside HIV-1 reverse transcriptase inhibitor. | |||
T70794 | Nevirapine dimer | ||
Nevirapine dimer is a non-nucleoside reverse transcriptase inhibitor (NNRTI). | |||
T33435 |
MK-4965
|
||
MK-4965 is a new type of non-nucleoside reverse transcriptase inhibitor with antiviral activity. | |||
T70851 |
U 88204
|
||
U 88204 is a non-nucleoside HIV-1 reverse transcriptase inhibitor. | |||
T68450 |
IDX-989
|
||
IDX-989 is an HIV-1 non-nucleoside reverse transcriptase inhibitor. | |||
T28833 |
SPD-756
SPD 756,BCH13520,BCH-13520,BCH 13520 |
||
SPD-756, a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection. | |||
T71566 |
MK-7445
|
||
MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase. | |||
T11814 |
Lamivudine 13C,15N2
|
Others | Others |
Lamivudine 13C,15N2, an impurity of Lamivudine (BCH-189), functions as an inhibitor of both HIV-1/2 reverse transcriptase and hepatitis B virus reverse transcriptase, classifying it as a nucleoside reverse transcriptase inhibitor (NRTIs). | |||
T27348 |
Fosalvudine tidoxil
HDP-990003,HDP990003,HDP 99.0003,HDP99.0003,HDP-99.0003,HDP 990003 |
||
Fosalvudine tidoxil, a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection. | |||
T28507 |
RDEA-427
RDEA 427 |
||
RDEA-427, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection. | |||
T26940 |
Calanolide A
NSC 675451,NSC675451,NSC-675451 |
||
Calanolide A, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection. | |||
T26946 |
Capravirine
S-1153,AG1549,S1153,AG-1549,AG 549 |
||
Capravirine, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection. | |||
T15776 |
Loviride
R 89439 |
Others | Others |
Loviride is a non-nucleoside reverse transcriptase inhibitor (IC50: 0.3 µM). Loviride inhibits HIV-1, HIV-2 and SIV replication in MT-4 cells. It is used for reverse transcriptase from HIV-1. | |||
T27512 |
GW-695634
GW5634,GW695634,GW-5634G,GW-5634 |
||
GW-695634, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection. | |||
T25501 |
HI-236
HI 236,D-PBT,D PBT,DPBT |
||
HI-236 is used as a non-nucleoside HIV-1 reverse-transcriptase inhibitor. | |||
T70156 |
K-5a2
|
||
K-5a2 is a novel human immunodeficiency virus type 1 (HIV-1) non-nucleoside reverse transcriptase inhibitor (NNRTI). |