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Cat. No. Product Name Target Signaling Pathways
T2330 Rilpivirine

TMC278,R278474,利匹韦林,DB08864

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Rilpivirine (R278474) 是一种二芳基嘧啶衍生物和非核苷逆转录酶抑制剂,具有抗 HIV-1 的抗病毒活性,用于治疗 HIV 感染。
T27154 Dexelvucitabine

D-D-4FC,DPC-817,RVT,beta-D-D-4FC,DFC

Reverse Transcriptase Microbiology/Virology
Dexelvucitabine (RVT) 是一种胞苷类似物,一种口服有活性的核苷逆转录酶抑制剂。它是一种 2'-脱氧胞苷抗逆转录病毒剂。它是一种有效的抗 HIV-1病毒剂,这些病毒聚合酶中含有胸苷类似物和/或 M184V 突变。
T1404 Stavudine

d4T,Sanilvudine,BMY-27857,NSC 163661,司他夫定

Apoptosis; Nucleoside Antimetabolite/Analog; HIV Protease; NOD-like Receptor (NLR); Reverse Transcriptase; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Stavudine (BMY-27857) 是一种口服活性核苷逆转录酶抑制剂,还抑制线粒体 DNA 的复制,具有抗HIV-1和HIV-2的活性。它降低 NLRP3 炎症小体激活,调节淀粉样 β 自噬,诱导细胞凋亡。
T7700 Lersivirine

3-氰基-5-[[3,5-二乙基-1-(2-羟基乙基)-1H-吡唑-4-基]氧基]苯腈,Lersivirine(UK 453061),UK-453061

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Lersivirine (UK-453061) 是非核苷逆转录的抑制剂 (NNRTI),有效抑制 NNRTI 耐药病毒。它对野生型人类免疫缺陷病毒和临床相关 NNRTI 耐药菌株显示出强大的抗逆转录病毒活性。
T1815 Dapivirine

R147681,达匹维林,TMC120

Apoptosis; HIV Protease; Reverse Transcriptase; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Dapivirine (R147681) 是一种二芳基嘧啶非核苷类逆转录酶抑制剂。
T1513 Telbivudine

NV 02B,L-Thymidine,Epavudine,替比夫定

Others; HBV; Reverse Transcriptase Microbiology/Virology; Others
Telbivudine (NV 02B) 是一种乙型肝炎病毒复制的抗病毒抑制剂,是一种具有口服活性的胸腺嘧啶核苷类似物。
T0110 Zalcitabine

Dideoxycytidine,ddC,扎西他滨,NSC 606170,Ro 24-2027/000,2',3'-Dideoxycytidine

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Zalcitabine (Dideoxycytidine) 是一种核苷类似物逆转录酶抑制剂,用于HIV 感染相关研究。
T3172 Trovirdine

曲韦定,LY300046

HIV Protease Microbiology/Virology; Proteases/Proteasome
Trovirdine (LY300046) 是一种硫脲类非核苷类逆转录酶抑制剂。
T2578 Didanosine

ddI,去羟肌苷,2',3'-Dideoxyinosine

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Didanosine (ddI) 是一种逆转录酶抑制剂,IC50为490nM。
T2393 Efavirenz

EFV,依非韦伦,DMP 266,依法韦仑,Sustiva,Stocrin,L-743726

HIV Protease; Reverse Transcriptase; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Efavirenz (DMP 266) 是一种人类免疫缺陷病毒 1 非核苷类似物逆转录酶抑制剂。它也是一种野生型HIV-1 RT 抑制剂,Ki 为 2.93 nM,有效抑制 HIV-1 复制,IC95为 1.5 nM。
T31860 Fosdevirine

GSK-2248761A,IDX 899,GSK 2248761A,GSK 2248761,GSK-2248761,IDX-12899,GSK2248761,FDV,GSK2248761A

HIV Protease Microbiology/Virology; Proteases/Proteasome
Fosdevirine (GSK2248761) 是一种具有选择性和高效性的非核苷类逆转录酶 (NNRTI) 抑制剂 ,具有抗 HIV 活性,可用于研究迟发性癫痫等神经系统相关疾病。
T2551 Etravirine

TMC125,依曲韦林,R165335

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Etravirine (R165335) 是一种非核苷逆转录酶抑制剂,具有抗 HIV 的作用。
T68103L Mk-6186 HCl

Mk-6186 HCl(1034474-19-5 Free base)

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
MK-6186 HCl,一种新型非核苷类逆转录酶抑制剂,具有抗病毒活性,可用于研究HIV。
T6214 Emtricitabine

恩曲他滨,FTC,Emtriva,BW1592

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Emtricitabine (FTC) 是一种核苷逆转录酶抑制剂, 在 PBMC 细胞中的 EC50值为0.01 µM,可研究 HIV 感染。
T1267 Abacavir

Epzicom,Ziagen,阿巴卡韦,Abacavir sulfate

Apoptosis; HIV Protease; Reverse Transcriptase Apoptosis; Microbiology/Virology; Proteases/Proteasome
Abacavir (Ziagen) 是一种核苷类似物逆转录酶抑制剂。
T68103 MK-6186

Reverse Transcriptase Microbiology/Virology
MK-6186 是一种新型非核苷类逆转录酶抑制剂,具有抗病毒活性,可用于研究病毒感染。
T60540 Netivudine

Netivudine 是一种有效的核苷类逆转录酶抑制剂(NRTIs),是一种核苷类似物,具有抗水痘带状疱疹病毒活性,可用于治疗人类免疫缺陷病毒(HIV)感染。Netivudine 通过抑制逆转录酶起作用,通过抑制作用减少体内的病毒载量,减缓疾病的进展。
T67804 KM-023

HIV Protease Microbiology/Virology; Proteases/Proteasome
KM-023是一种新的第二代非核苷类逆转录酶抑制剂,可用于研究人类免疫缺陷病毒(HIV)1型感染。
T2279 Tizoxanide

替唑尼特,Desacetyl-nitazoxanide,TIZ

Antiviral; HIV Protease; Antibacterial; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Tizoxanide (Desacetyl-nitazoxanide) 是 Nitazoxanide 活性代谢物,有抗HIV-1的活性。Nitazoxanide 可抗细菌和多种病毒复制。
T3632 Doravirine

多拉维林,多拉韦林,MK-1439

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Doravirine (MK-1439) 是一种高度特异性的HIV-1非核苷逆转录酶抑制剂,对野生型以及K103N 和Y181C 逆转录酶突变体的IC50值分别为 4.5 nM,5.5 nM 和 6.1 nM。
T7212 Delavirdine mesylate

U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate)

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Delavirdine mesylate (BHAP-U 90152(mesylate)) 是一种口服活性非核苷逆转录酶抑制剂。它抑制 HIV-1 病毒复制,可以用于艾滋病的相关研究。它选择性地抑制 HIV-1 逆转录酶,其选择性超过 DNA 聚合酶 α 和 DNA 聚合酶 δ 。
T31860L (Iso)-Fosdevirine

(Iso)-Fosdevirine(Iso-1018450-26-4),(Iso)-GSK2248761

HIV Protease Microbiology/Virology; Proteases/Proteasome
(Iso)-Fosdevirine ( (Iso)-GSK2248761) 是一种具有选择性和高效性的非核苷类逆转录酶 (NNRTI) 抑制剂 ,具有抗 HIV 活性,可用于研究迟发性癫痫等神经系统相关疾病。
T1595 Nevirapine

NSC 641530,奈韦拉平,BI-RG 587,奈伟拉平,NVP

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Nevirapine (NVP) 是一种 HIV-1逆转录酶非核苷抑制剂,Ki 值为 270 μM,可用于研究 HIV/AIDS。
T1675 Adefovir dipivoxil

Hepsera,GS 0840,阿德福韦酯,Preveon

Others; HBV; Reverse Transcriptase Microbiology/Virology; Others
Adefovir dipivoxil (GS 0840) 是一种腺苷类似物,是核苷逆转录酶抑制剂 Adefovir 的口服前药,具有抗乙型肝炎病毒、疱疹病毒和人类免疫缺陷病毒的活性。
T2409L Tenofovir Disoproxil Fumarate

GS-1278 Disoproxil Fumarate,Tenofovir DF,富马酸替诺福韦酯

HBV; HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Tenofovir Disoproxil Fumarate (GS-1278 Disoproxil Fumarate) 是一种核苷酸逆转录酶抑制剂,有潜力研究艾滋病和慢性乙型肝炎。
T7447 Adefovir

HBV; Reverse Transcriptase; Telomerase DNA Damage/DNA Repair; Microbiology/Virology
Adefovir 是一种单磷酸腺苷类似物抗病毒剂,在细胞内转化为 Adefovir diphosphate 后可抑制HBVDNA 聚合酶。它在 HepG2.2.15 细胞系中对HBV 的IC50为 0.7 μM。它对多种病毒(包括HBV 和疱疹病毒)具有良好的抗病毒活性。
T16098 Islatravir

MK-8591

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Islatravir (MK-8591) 是一种核苷逆转录酶抑制剂,是抗HIV-1药物,对 HIV-1 (WT),HIV-1 (M184V),HIV-1 (MDR) 的EC50值分别为 0.068 nM,3.1 nM 和 0.15 nM。
T29037 UC-781

NSC 675186,UC781,UC 781

Antiviral; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
UC-781 (NSC-675186) 是一种高效且具有选择性的人类免疫缺陷病毒 HIV-1 非核苷类逆转录酶(NNRTI)I抑制剂 ,C50 值为 5 nM。UC-781 具有抗病毒活性和耐药性。UC-781状态稳定,较低的 PH 或不同温度对其影响较小。
T14489 Azvudine

4-氨基-1-(4-C-叠氮基-2-脱氧-2-氟-BETA-D-呋喃阿拉伯糖基)-2(1H)-嘧啶酮,FNC,RO-0622

HCV Protease; HBV; HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Azvudine (FNC) 是一种有效的核苷逆转录酶抑制剂 (NRTI),对 HIV、HBV 和 HCV 具有抗病毒活性。它抑制耐 NRTI 的病毒株,高效抑制 HIV-1和 HIV-2。
T27625 IQP-0528

SJ-3991,SJ3991,IQP0528

Antiviral; HIV Protease; Reverse Transcriptase Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
IQP-0528是一种高效的非核苷类逆转录酶抑制剂(NNRTI),通过阻断病毒进入,有可能用于治疗HIV 感染,并且作为杀微生物凝胶显示出抗病毒活性。IQP-0528对HIV-1和HIV-2都显示出抑制作用,对HIV-1的EC50为0.2 nM,对HIV-2的EC50为100 nM。
T28204 NSC-176377

NSC 176377

NSC-176377 is a non-nucleoside reverse transcriptase inhibitor.
T2330L Rilpivirine HCl

Rilpivirine hydrochloride,TMC278,Rilpivirine,TMC-278,TMC 278. trade name Edurant

Rilpivirine is a potent non-nucleoside reverse transcriptase inhibitor.
T27542 HI-207

HI207,HI 207

HI-207 is an inhibitor of non-nucleoside reverse transcriptase.
T24354 L 738372

L-738,372,L 738,372,L738372,L738,372,L-738372

L 738372 is a non-nucleoside inhibitor of HIV-1 reverse transcriptase.
T24087 GCA-186

I-EBU-dM,IEBUdM,I EBU dM,GCA 186

GCA-186 is an effective non-nucleoside HIV-1 reverse transcriptase inhibitor.
T70794 Nevirapine dimer

Nevirapine dimer is a non-nucleoside reverse transcriptase inhibitor (NNRTI).
T33435 MK-4965

MK-4965 is a new type of non-nucleoside reverse transcriptase inhibitor with antiviral activity.
T70851 U 88204

U 88204 is a non-nucleoside HIV-1 reverse transcriptase inhibitor.
T68450 IDX-989

IDX-989 is an HIV-1 non-nucleoside reverse transcriptase inhibitor.
T28833 SPD-756

SPD 756,BCH13520,BCH-13520,BCH 13520

SPD-756, a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.
T71566 MK-7445

MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.
T11814 Lamivudine 13C,15N2

Others Others
Lamivudine 13C,15N2, an impurity of Lamivudine (BCH-189), functions as an inhibitor of both HIV-1/2 reverse transcriptase and hepatitis B virus reverse transcriptase, classifying it as a nucleoside reverse transcriptase inhibitor (NRTIs).
T27348 Fosalvudine tidoxil

HDP-990003,HDP990003,HDP 99.0003,HDP99.0003,HDP-99.0003,HDP 990003

Fosalvudine tidoxil, a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.
T28507 RDEA-427

RDEA 427

RDEA-427, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.
T26940 Calanolide A

NSC 675451,NSC675451,NSC-675451

Calanolide A, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.
T26946 Capravirine

S-1153,AG1549,S1153,AG-1549,AG 549

Capravirine, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.
T15776 Loviride

R 89439

Others Others
Loviride is a non-nucleoside reverse transcriptase inhibitor (IC50: 0.3 µM). Loviride inhibits HIV-1, HIV-2 and SIV replication in MT-4 cells. It is used for reverse transcriptase from HIV-1.
T27512 GW-695634

GW5634,GW695634,GW-5634G,GW-5634

GW-695634, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.
T25501 HI-236

HI 236,D-PBT,D PBT,DPBT

HI-236 is used as a non-nucleoside HIV-1 reverse-transcriptase inhibitor.
T70156 K-5a2

K-5a2 is a novel human immunodeficiency virus type 1 (HIV-1) non-nucleoside reverse transcriptase inhibitor (NNRTI).

化合物

Rilpivirine
Cat.No: T2330
Synonym: TMC278,R278474,利匹韦林,DB08864
Target: HIV Protease, Reverse Transcriptase
Dexelvucitabine
Cat.No: T27154
Synonym: D-D-4FC,DPC-817,RVT,beta-D-D-4FC,DFC
Target: Reverse Transcriptase
Stavudine
Cat.No: T1404
Synonym: d4T,Sanilvudine,BMY-27857,NSC 163661,司他夫定
Target: Apoptosis, Nucleoside Antimetabolite/Analog, HIV Protease, NOD-like Receptor (NLR), Reverse Transcriptase, Autophagy
Lersivirine
Cat.No: T7700
Synonym: 3-氰基-5-[[3,5-二乙基-1-(2-羟基乙基)-1H-吡唑-4-基]氧基]苯腈,Lersivirine(UK 453061),UK-453061
Target: HIV Protease, Reverse Transcriptase
Dapivirine
Cat.No: T1815
Synonym: R147681,达匹维林,TMC120
Target: Apoptosis, HIV Protease, Reverse Transcriptase, Autophagy
Telbivudine
Cat.No: T1513
Synonym: NV 02B,L-Thymidine,Epavudine,替比夫定
Target: Others, HBV, Reverse Transcriptase
Zalcitabine
Cat.No: T0110
Synonym: Dideoxycytidine,ddC,扎西他滨,NSC 606170,Ro 24-2027/000,2',3'-Dideoxycytidine
Target: HIV Protease, Reverse Transcriptase
Trovirdine
Cat.No: T3172
Synonym: 曲韦定,LY300046
Target: HIV Protease
Didanosine
Cat.No: T2578
Synonym: ddI,去羟肌苷,2',3'-Dideoxyinosine
Target: HIV Protease, Reverse Transcriptase
Efavirenz
Cat.No: T2393
Synonym: EFV,依非韦伦,DMP 266,依法韦仑,Sustiva,Stocrin,L-743726
Target: HIV Protease, Reverse Transcriptase, Autophagy
Fosdevirine
Cat.No: T31860
Synonym: GSK-2248761A,IDX 899,GSK 2248761A,GSK 2248761,GSK-2248761,IDX-12899,GSK2248761,FDV,GSK2248761A
Target: HIV Protease
Etravirine
Cat.No: T2551
Synonym: TMC125,依曲韦林,R165335
Target: HIV Protease, Reverse Transcriptase
Mk-6186 HCl
Cat.No: T68103L
Synonym: Mk-6186 HCl(1034474-19-5 Free base)
Target: HIV Protease, Reverse Transcriptase
Emtricitabine
Cat.No: T6214
Synonym: 恩曲他滨,FTC,Emtriva,BW1592
Target: HIV Protease, Reverse Transcriptase
Abacavir
Cat.No: T1267
Synonym: Epzicom,Ziagen,阿巴卡韦,Abacavir sulfate
Target: Apoptosis, HIV Protease, Reverse Transcriptase
MK-6186
Cat.No: T68103
Synonym:
Target: Reverse Transcriptase
Netivudine
Cat.No: T60540
Synonym:
Target:
KM-023
Cat.No: T67804
Synonym:
Target: HIV Protease
Tizoxanide
Cat.No: T2279
Synonym: 替唑尼特,Desacetyl-nitazoxanide,TIZ
Target: Antiviral, HIV Protease, Antibacterial, Autophagy
Doravirine
Cat.No: T3632
Synonym: 多拉维林,多拉韦林,MK-1439
Target: HIV Protease, Reverse Transcriptase
Delavirdine mesylate
Cat.No: T7212
Synonym: U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate)
Target: HIV Protease, Reverse Transcriptase
(Iso)-Fosdevirine
Cat.No: T31860L
Synonym: (Iso)-Fosdevirine(Iso-1018450-26-4),(Iso)-GSK2248761
Target: HIV Protease
Nevirapine
Cat.No: T1595
Synonym: NSC 641530,奈韦拉平,BI-RG 587,奈伟拉平,NVP
Target: HIV Protease, Reverse Transcriptase
Adefovir dipivoxil
Cat.No: T1675
Synonym: Hepsera,GS 0840,阿德福韦酯,Preveon
Target: Others, HBV, Reverse Transcriptase
Tenofovir Disoproxil Fumarate
Cat.No: T2409L
Synonym: GS-1278 Disoproxil Fumarate,Tenofovir DF,富马酸替诺福韦酯
Target: HBV, HIV Protease, Reverse Transcriptase
Adefovir
Cat.No: T7447
Synonym:
Target: HBV, Reverse Transcriptase, Telomerase
Islatravir
Cat.No: T16098
Synonym: MK-8591
Target: HIV Protease, Reverse Transcriptase
UC-781
Cat.No: T29037
Synonym: NSC 675186,UC781,UC 781
Target: Antiviral, HIV Protease
Azvudine
Cat.No: T14489
Synonym: 4-氨基-1-(4-C-叠氮基-2-脱氧-2-氟-BETA-D-呋喃阿拉伯糖基)-2(1H)-嘧啶酮,FNC,RO-0622
Target: HCV Protease, HBV, HIV Protease, Reverse Transcriptase
IQP-0528
Cat.No: T27625
Synonym: SJ-3991,SJ3991,IQP0528
Target: Antiviral, HIV Protease, Reverse Transcriptase
NSC-176377
Cat.No: T28204
Synonym: NSC 176377
Target:
Rilpivirine HCl
Cat.No: T2330L
Synonym: Rilpivirine hydrochloride,TMC278,Rilpivirine,TMC-278,TMC 278. trade name Edurant
Target:
HI-207
Cat.No: T27542
Synonym: HI207,HI 207
Target:
L 738372
Cat.No: T24354
Synonym: L-738,372,L 738,372,L738372,L738,372,L-738372
Target:
GCA-186
Cat.No: T24087
Synonym: I-EBU-dM,IEBUdM,I EBU dM,GCA 186
Target:
Nevirapine dimer
Cat.No: T70794
Synonym:
Target:
MK-4965
Cat.No: T33435
Synonym:
Target:
U 88204
Cat.No: T70851
Synonym:
Target:
IDX-989
Cat.No: T68450
Synonym:
Target:
SPD-756
Cat.No: T28833
Synonym: SPD 756,BCH13520,BCH-13520,BCH 13520
Target:
MK-7445
Cat.No: T71566
Synonym:
Target:
Lamivudine 13C,15N2
Cat.No: T11814
Synonym:
Target: Others
Fosalvudine tidoxil
Cat.No: T27348
Synonym: HDP-990003,HDP990003,HDP 99.0003,HDP99.0003,HDP-99.0003,HDP 990003
Target:
RDEA-427
Cat.No: T28507
Synonym: RDEA 427
Target:
Calanolide A
Cat.No: T26940
Synonym: NSC 675451,NSC675451,NSC-675451
Target:
Capravirine
Cat.No: T26946
Synonym: S-1153,AG1549,S1153,AG-1549,AG 549
Target:
Loviride
Cat.No: T15776
Synonym: R 89439
Target: Others
GW-695634
Cat.No: T27512
Synonym: GW5634,GW695634,GW-5634G,GW-5634
Target:
HI-236
Cat.No: T25501
Synonym: HI 236,D-PBT,D PBT,DPBT
Target:
K-5a2
Cat.No: T70156
Synonym:
Target:
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