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28

抑制剂 & 化合物

5

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T0517	Pancreatin Pancreatic enzymes,pancrelipase,胰酶	Others	Others
	Pancreatin (pancrelipase) 是一种含有胰腺消化酶的猪胰腺提取物。
T68056	Donetidine	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Donetidine 是一种组胺 H2 受体拮抗剂，可用于治疗消化系统疾病。
T34123	Pranazepide FR120480,FK 480,FR-120480	cholecystokinin	GPCR/G Protein
	Pranazepide (FK 480) 是一种小分子胆囊收缩素受体拮抗剂，可用于研究消化系统疾病和胰腺炎。
T1201	Sulpiride Aiglonyl,舒必利,Dogmatil,Sulpyrid,Dolmatil,Dobren	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Sulpiride (Aiglonyl) 是一种多巴胺 D2 受体拮抗剂，可用作抗抑郁药、抗精神病药和助消化剂发挥治疗作用。
T9420	prifinium bromide	Others	Others
	Prifinium bromide 是抗胆碱能试剂，能够改善痉挛，具有止吐效果。
T8385	Metoclopramide hydrochloride hydrate 盐酸甲氧氯普胺,甲氧氯普胺盐酸水合物,Metoclopramide monohydrochloride monohydrate	Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience
	Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) 是5-HT3和多巴胺D2受体拮抗剂，IC50值分别为 308 和 483 nM，可用于恶心呕吐、胃食管反流和胃轻瘫的研究。
T68035	Capeserod SL-650155,SL-65.0155	5-HT Receptor	GPCR/G Protein; Neuroscience
	Capeserod 是一种潜在的 5-HT4 receptor(5-羟色胺受体4)激动剂，可用于研究消化系统疾病和神经系统疾病。
T63806	CFTR corrector 8	CFTR	Membrane transporter/Ion channel
	CFTR corrector 8 is a highly effective modulator of the cystic fibrosis transmembrane conductance regulator (CFTR). This compound is specifically designed for utilization in research related to cystic fibrosis, a genetic disorder primarily affecting the lungs and digestive system [1].
T4994	Tocofersolan Vitamin E-TPGS,Tocophersolan,TPGS,D-α-Tocopherol polyethylene glycol 1000 succinate,托可索仑,维生素E聚乙二醇琥珀酸酯	Others	Others
	Tocofersolan (TPGS) 是合成的 α-生育酚的聚乙二醇衍生物。
T69984	Ticalopride	5-HT Receptor	GPCR/G Protein; Neuroscience
	Ticalopride是一种5-HT3 receptor激动剂，可用于治疗消化系统疾病、口颌疾病、耳鼻咽喉疾病，可用于研究神经性贪食症、胃食管反流和肠易激综合征。
T12404	CCK-A receptor inhibitor 1	cholecystokinin	GPCR/G Protein
	CCK-A receptor inhibitor 1 是一种有效的缩胆囊素 A (CCK-A) 受体抑制剂(IC50：340 nM）。CCK-A receptor inhibitor 1 可用于研究与消化系统相关的疾病。
T61699	Osunprotafib AC 484,Osunprotafib,AC484,ABBV-CLS-484	Phosphatase	Metabolism
	ABBV-CLS-484 (Osunprotafib) 是一种具有亚纳摩尔活性的有效的PTPN2抑制剂，具有抗肿瘤活性，可增强T细胞抗肿瘤免疫力。ABBV-CLS-484可用于治疗肿瘤、食管癌和消化系统疾病。
T0992	Carbenoxolone disodium Biogastrone,Duogastrone,甘珀酸钠,Bioral	Gap Junction Protein	Cytoskeletal Signaling
	Carbenoxolone disodium (Duogastrone) 是甘草酸的活性代谢物和人11β-HSD 和细菌3α, 20β-HSD 的抑制剂。它是一种缝隙连接的解耦剂，可抑制牛痘病毒生长，用于消化性、食道和口腔溃疡和炎症的相关研究。
T25206	Casokefamide beta Casomorphin 4027
	Casokefamide is a peripherally-specific, synthetic opioid pentapeptide. It was derived from the β-casomorphin sequence and designed with the intention of improving resistance to digestive enzymes so that it could be used as an antidiarrheal medicine.
T35788	Orlistat Degradation Product (sodium salt)
	Orlistat degradation product is a degradation product of the digestive lipase inhibitor orlistat . It is formed via hydrolytic and thermal degradation as well as digestion by human carboxyl ester lipase.
T78347	Serratia marcescens nuclease
	Serratia marcescens nuclease，为一种非特异性核酸酶，因具备强大消化DNA与RNA活性，应用范围广泛。
T80881	Valosin (porcine)
	Valosin (porcine)是一种含有25个氨基酸的生物活性肽，最近从猪肠中分离得到，主要用于消化系统研究。
T60813	Alizapride
	Alizapride 是多巴胺受体 (dopamine receptor) 的拮抗剂。Alizapride 可以用于人体消化系统疾病，是一种有效的止吐剂。
T82163	Human enteropeptidase-IN-3
	Human enteropeptidase-IN-3是一种肽类酶抑制剂，主要作用于肠肽酶，具有长效抑制功能。该化合物广泛应用于研究肠道消化相关疾病。
T72547	Plm IV inhibitor-2
	Plm IV inhibitor-2 是一种有效的Plm IV 抑制剂，对Plm IV、II 和 I 的IC50分别为24 nM、70 nM 和 0.3 μM。适用于研究Plasmodium 寄生虫引起的疟疾。
T0194L2	Chloroquine dihydrochloride Chloroquine HCl,NSC 14050,Aralen hydrochloride,NSC14050,Chloroquine hydrochloride,Aralen HCl,NSC-14050
	Chloroquine is a medication preventing and treating malaria in areas where malaria is known to be sensitive to its effects. It is also sometimes used for amebiasis that is occurring outside the intestines, rheumatoid arthritis, and lupus erythematosus. Ch
T37545	cis-9,10-Methyleneoctadecanoic Acid
	cis-9,10-Methyleneoctadecanoic acid is a cyclopropane fatty acid that has been found in bacteria and the digestive gland of P. globosa. It is a component of S. aureus cell membranes and levels decrease upon treatment with carvacrol. cis-9,10-Methyleneoctadecanoic acid is secreted by H. pylori and enhances histamine- and dibutyryl cAMP-stimulated acid secretion in isolated guinea pig parietal cells. It also activates protein kinase C (PKC) in a calcium-dependent manner.
T69215	Ambrein
	Ambrein is a triterpene alcohol that is the chief constituent of ambergris, a secretion from the digestive system of the sperm whale, and has been suggested as the possible active component producing the supposed aphrodisiac effects of ambergris. It serves as the biological precursor for a number of aromatic derivatives such as ambroxan and is thought to possess fixative properties for other odorants. It has been shown to act as an analgesic and it has been proven to increase sexual behavior in ...
T81182	Secretin (swine)
	Secretin (swine)为源自猪的神经内分泌激素，由十二指肠黏膜S细胞产生，具有27个氨基酸的多肽结构，并针对分泌素受体起作用。此激素在各类成熟肠内分泌细胞亚群中表达，受脂肪酸的促进。它主要激发胰腺释放水和碳酸氢盐，同时在消化系统、中枢神经系统和能量代谢方面具有广泛应用。
T77117	Toripalimab
	Toripalimab 是一个国产抗肿瘤 PD-1抗体。Toripalimab 是一种靶向 PD-1的选择性人源化单克隆抗体。Toripalimab 能够与 PD-1结合并阻断与其配体相互作用。Toripalimab 具有强效抗肿瘤作用，可用于黑色素瘤、肺癌、消化道肿瘤、肝胆和胰腺肿瘤、神经内分泌肿瘤、鼻咽癌和尿路上皮癌等肿瘤的研究。
T70882	Orlistat-d3
	Orlistat-d3 is intended for use as an internal standard for the quantification of orlistat by GC- or LC-MS. Orlistat is a digestive lipase inhibitor. It inhibits diacylglycerol lipase α (DAGLα), DAGLβ, α/β-hydrolase domain-containing protein 12 (ABHD12), ABHD16A, and platelet-activating factor acetylhydrolase (PAF-AH; IC50s = 0.06, 0.1, 0.08, 0.03, and 0.05 µM, respectively), as well as pancreatic lipase and hormone-sensitive lipase (IC50s = 0.65 and 2.1 µg/ml, respectively) but does not inhibit...
T31194	Dalapon Basfapon B,Dowpon M,Dawpon-Rae
	Dalapon is a selective herbicide used to control perennial grasses. The major use of dalapon is on food crops including sugarcane and sugar beets. Its use is no longer authorized in France. The National Institute for Occupational Safety and Health in the
T8761	[Leu15]-Gastrin I human Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2	Others	Others
	[Leu15]-Gastrin I human (Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2) 基因编码人体内的蛋白质 [Leu15]-胃泌素 I。在人类染色体中，GAST 基因定位于 17q21.2。胃窦中的 G 细胞产生 [Leu15]-胃泌素 I 的前体前胃泌素。前胃泌素经过裂解和加工产生胃泌素，它对整个胃肠道上皮细胞具有营养作用。胃泌素对消化系统的生长至关重要，并刺激壁细胞产生胃酸。胃泌素通过称为胆囊收缩素(CCK) 或 CCK-B 受体 (CCK-BR) 的 G 蛋白偶联受体发挥其功能。胃泌素的释放受到食物的刺激，尤其是蛋白质饮食，并受到非常低的 pH 值的抑制。萎缩性胃炎、幽门螺杆菌感染和长期服用质子泵抑制剂感染可能导致胃泌素过度表达。胃腺癌显示高水平的胃泌素。

化合物

Cat.No: T0517

Synonym: Pancreatic enzymes,pancrelipase,胰酶

Target: Others

Cat.No: T68056

Target: Histamine Receptor

Cat.No: T34123

Synonym: FR120480,FK 480,FR-120480

Target: cholecystokinin

Cat.No: T1201

Synonym: Aiglonyl,舒必利,Dogmatil,Sulpyrid,Dolmatil,Dobren

Target: Dopamine Receptor

prifinium bromide

Cat.No: T9420

Target: Others

Metoclopramide hydrochloride hydrate

Cat.No: T8385

Synonym: 盐酸甲氧氯普胺,甲氧氯普胺盐酸水合物,Metoclopramide monohydrochloride monohydrate

Target: Dopamine Receptor, 5-HT Receptor

Cat.No: T68035

Synonym: SL-650155,SL-65.0155

Target: 5-HT Receptor

CFTR corrector 8

Cat.No: T63806

Target: CFTR

Cat.No: T4994

Synonym: Vitamin E-TPGS,Tocophersolan,TPGS,D-α-Tocopherol polyethylene glycol 1000 succinate,托可索仑,维生素E聚乙二醇琥珀酸酯

Target: Others

Cat.No: T69984

Target: 5-HT Receptor

CCK-A receptor inhibitor 1

Cat.No: T12404

Target: cholecystokinin

Cat.No: T61699

Synonym: AC 484,Osunprotafib,AC484,ABBV-CLS-484

Target: Phosphatase

Carbenoxolone disodium

Cat.No: T0992

Synonym: Biogastrone,Duogastrone,甘珀酸钠,Bioral

Target: Gap Junction Protein

Cat.No: T25206

Synonym: beta Casomorphin 4027

Orlistat Degradation Product (sodium salt)

Cat.No: T35788

Serratia marcescens nuclease

Cat.No: T78347

Valosin (porcine)

Cat.No: T80881

Cat.No: T60813

Human enteropeptidase-IN-3

Cat.No: T82163

Plm IV inhibitor-2

Cat.No: T72547

Chloroquine dihydrochloride

Cat.No: T0194L2

Synonym: Chloroquine HCl,NSC 14050,Aralen hydrochloride,NSC14050,Chloroquine hydrochloride,Aralen HCl,NSC-14050

cis-9,10-Methyleneoctadecanoic Acid

Cat.No: T37545

Cat.No: T69215

Secretin (swine)

Cat.No: T81182

Cat.No: T77117

Cat.No: T70882

Cat.No: T31194

Synonym: Basfapon B,Dowpon M,Dawpon-Rae

[Leu15]-Gastrin I human

Cat.No: T8761

Synonym: Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
TN1148	Isopsoralenoside	Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Antibacterial	Endocrinology/Hormones; Microbiology/Virology
	Isopsoralenoside 是补骨脂多糖中的一种苯并呋喃苷。它在消化道内容物中可迅速代谢为补骨脂素。它具有雌激素样活性、促进成骨细胞增殖活性、抗肿瘤活性和抗菌活性。
TN1008	Psoralenoside	CaMK; Calcium Channel; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
	Psoralenoside 是源于补骨脂中的苯并呋喃苷，具有抗肿瘤、抗菌、促进成骨细胞增殖和雌激素样活性。它对组胺 H1、钙调素和电压门控 l 型钙通道具有较高的亲和力。
T2O2733	L-Cystine Cystine Acid,cystine,胱氨酸,L-胱氨酸	Antioxidant; Ferroptosis; Endogenous Metabolite	Apoptosis; Metabolism; oxidation-reduction
	L-Cystine (Cystine Acid) 是一种从半胱氨酸氨基酸硫醇侧链氧化获得的含硫衍生物。它起到抗氧化剂的作用，保护组织免受辐射和污染，减缓衰老过程。它还有助于蛋白质合成。
T2973	Astragaloside IV AST-IV,黄芪甲苷IV,AS-IV,黄芪皂苷 IV	MMP; ERK; Estrogen/progestogen Receptor; JNK	Endocrinology/Hormones; MAPK; Proteases/Proteasome
	Astragaloside IV (AS-IV) 是从黄芪中分离得到的一种皂苷，抑制ERK1/2和JNK 激活，在乳腺癌细胞 MDA-MB-231 中，下调(MMP)-2和(MMP)-9的信号通路。
T82725	Chrysanthellin A
	Chrysanthellin A, 主要皂苷化合物，源自Chrysanthellum americanum提取物，适用于研究消化功能障碍。

天然产物

Isopsoralenoside

Cat.No: TN1148

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Antibacterial

Cat.No: TN1008

Target: CaMK, Calcium Channel, Histamine Receptor

Cat.No: T2O2733

Synonym: Cystine Acid,cystine,胱氨酸,L-胱氨酸

Target: Antioxidant, Ferroptosis, Endogenous Metabolite

Astragaloside IV

Cat.No: T2973

Synonym: AST-IV,黄芪甲苷IV,AS-IV,黄芪皂苷 IV

Target: MMP, ERK, Estrogen/progestogen Receptor, JNK

Chrysanthellin A

Cat.No: T82725

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