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21

抑制剂 & 化合物

3

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T10876	CPA inhibitor Carboxypeptidase inhibitor	Carboxypeptidase	Proteases/Proteasome
	CPA inhibitor (Carboxypeptidase inhibitor) 是一种有效的羧肽酶 A (CPA) 抑制剂，Ki 值为 0.32 μM。
T16263	N6-Cyclopentyladenosine UK-80882,CPA	Adenosine Receptor	GPCR/G Protein; Neuroscience
	N6-Cyclopentyladenosine (CPA) 是一个选择性的腺苷A1 受体 (Adenosine A1 receptor)的激动剂，可用于模拟腺苷A1受体的作用，对人A1、A2A 和 A3 受体的Ki 分别为 2.3 nM、790 nM 和 43 nM。N6-Cyclopentyladenosine (CPA) 可用于调节细胞信号传导、神经递质释放和其他生物学过程。
T27138	Declopramide OXI-104,IMO-B,3-Chloroprocainamide	Apoptosis	Apoptosis
	Declopramide (OXI-104) 是新型化学增敏剂，具有抗肿瘤活性，可诱导细胞凋亡，可用于研究结直肠癌和炎症性肠病。
TP1560	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm a highly efficient, selective and short-acting peptide V2 receptor agonist (V2R), with EC50s of hV2R and rV2R being 0.25 and 0.05 nM, respectively.
TP1473	Velmupressin c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively.
TP1205	Velmupressin acetate V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate
	c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively.
T21519	CCPA 2-chloro-N(6)cyclopentyladenosine,2-氯-N6-环戊基腺苷,2-CHLORO-N-CYCLOPENTYLADENOSINE	Adenosine Receptor	GPCR/G Protein; Neuroscience
	CCPA (2-chloro-N(6)cyclopentyladenosine) 是一种有效的选择性腺苷 A1 受体激动剂。
T22489	2'-MeCCPA 2-Chloro-N-cyclopentyl-2′-C-methyladenosine	HCV Protease; Adenosine Receptor	GPCR/G Protein; Microbiology/Virology; Neuroscience; Proteases/Proteasome
	2'-MeCCPA 是一种具有有效性和高选择性的 A1 腺苷受体 (A1AR) 激动剂，对 AR 的 K 值为 1.8 nM。2'-MeCCPA 抑制毛喉素刺激的腺苷酸环化酶活性，IC值为13.1 nM。2'-MeCCPA 具有镇痛活性，可用于研究 HCV 。
T20701	MCPA NSC-2351,Krezone,NSC2351,NSC 2351,U 46 M-Fluid,Raphone	Others	Others
	MCPA（Krezone）是一种高效的苯氧基除草剂。使用 MCPA 会对附近的水资源和土壤资源产生影响。
T77567	BCPA	Others	Others
	BCPA 是一种无细胞毒性的 Pin1 调节剂。BCPA 可调节破骨细胞活化，减弱 Pin1 蛋白的减少，从而抑制 RANKL 诱导的破骨细胞发生的受体激活物。BCPA 用于研究骨质疏松。
T1025	Tranylcypromine (2-PCPA) hydrochloride 反苯环丙胺盐酸盐,Tranylcypromine (2-PCPA) HCl,SKF-385 HCl	Histone Demethylase; MAO	Chromatin/Epigenetic; Metabolism; Neuroscience
	Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl) 是一种单胺氧化酶抑制剂，对治疗重度抑郁症、心境恶劣障碍和非典型抑郁症有效。
T60359	cis-4-Br-2,5-F2-PCPA
	cis-4-Br-2,5-F2-PCPA (S1024) 抑制 LSD1 和 LSD2，Ki 值分别为 94 nM 和 8.4 μM。癌症干细胞中 LSD1异常表达，cis-4-Br-2,5-F2-PCPA 能够通过增加 CCRF-CEM 细胞中二甲基化组蛋白 H3 的 K4 (H3K4) 水平，抑制 LSD1活性和癌细胞增殖。
T33228	MCPA-potassium
	MCPA-potassium is a bioactive chemical.
T41143	pCPA methyl ester hydrochloride 4-氯-DL-苯基丙氨酸甲酯盐酸盐,4-Chloro-DL-phenylalanine methyl ester hydrochloride	5-HT Receptor; Hydroxylase	GPCR/G Protein; Metabolism; Neuroscience
	pCPA methyl ester hydrochloride (4-Chloro-DL-phenylalanine methyl ester hydrochloride) 是色氨酸羟化酶抑制剂和5-HT 合成的抑制剂。 pCPA methyl ester hydrochloride 可穿过血脑屏障并降低 5-HT 中枢可用性。
T33227	MCPA-butyl Yamaclean M
	MCPA-butyl is a biochemical.
T82765	CcpA-IN-1	Antibiotic	Microbiology/Virology
	CcpA-IN-1为一种针对金黄色葡萄球菌的抗生素，具备高效的杀菌能力，其最小抑菌浓度（MICS）为460 nM。
T20948	MCPA-thioethyl HOK 7501,HOK7501,HOK-7501
	MCPA-thioethyl is a biochemical.
T74170	MOCPAC
	MOCPAC 是一种HDAC1特异性底物。
T81054	T-1-MCPAB	VEGFR	Angiogenesis; Tyrosine Kinase/Adaptors
	T-1-MCPAB为一种高效VEGFR-2抑制剂（IC50=0.135 µM），其显著抑制MCF7细胞迁移，适用于癌症相关研究。
T82684	Connexin mimetic peptide 40,37GAP26
	Connexin mimetic peptide 40,37GAP26是一种生物活性肽，对应Cx37和Cx40主要血管连接蛋白的胞外环GAP26结构域，命名基于Cx同源性为37,40Gap26。本化合物主要用于研究间隙连接对环吡嗪酸(CPA)通过啮齿动物髂动脉壁导致的内皮超极化扩散的影响。Cx37和Cx40形成的间隙连接斑块在内皮细胞中高度丰富，而Connexin mimetic peptide 40,37GAP26能抑制内膜下超极化。
T71327	Paraxanthine-d6
	Paraxanthine-d6 is intended for use as an internal standard for the quantification of paraxanthine by GC- or LC-MS. Paraxanthine is an active metabolite of caffeine. It is formed via N3-demethylation of caffeine by the cytochrome P450 (CYP) isoform CYP1A2. Paraxanthine is an adenosine A1 and A2 receptor antagonist. In vivo, paraxanthine increases striatal cGMP and extracellular striatal dopamine levels and locomotor activity, as well as inhibits motor depression induced by the adenosine A1 agoni...

化合物

CPA inhibitor

Cat.No: T10876

Synonym: Carboxypeptidase inhibitor

Target: Carboxypeptidase

N6-Cyclopentyladenosine

Cat.No: T16263

Synonym: UK-80882,CPA

Target: Adenosine Receptor

Cat.No: T27138

Synonym: OXI-104,IMO-B,3-Chloroprocainamide

Target: Apoptosis

c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm

Cat.No: TP1560

Cat.No: TP1473

Synonym: c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2

Velmupressin acetate

Cat.No: TP1205

Synonym: V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate

Cat.No: T21519

Synonym: 2-chloro-N(6)cyclopentyladenosine,2-氯-N6-环戊基腺苷,2-CHLORO-N-CYCLOPENTYLADENOSINE

Target: Adenosine Receptor

Cat.No: T22489

Synonym: 2-Chloro-N-cyclopentyl-2′-C-methyladenosine

Target: HCV Protease, Adenosine Receptor

Cat.No: T20701

Synonym: NSC-2351,Krezone,NSC2351,NSC 2351,U 46 M-Fluid,Raphone

Target: Others

Cat.No: T77567

Target: Others

Tranylcypromine (2-PCPA) hydrochloride

Cat.No: T1025

Synonym: 反苯环丙胺盐酸盐,Tranylcypromine (2-PCPA) HCl,SKF-385 HCl

Target: Histone Demethylase, MAO

cis-4-Br-2,5-F2-PCPA

Cat.No: T60359

Cat.No: T33228

pCPA methyl ester hydrochloride

Cat.No: T41143

Synonym: 4-氯-DL-苯基丙氨酸甲酯盐酸盐,4-Chloro-DL-phenylalanine methyl ester hydrochloride

Target: 5-HT Receptor, Hydroxylase

Cat.No: T33227

Synonym: Yamaclean M

Cat.No: T82765

Target: Antibiotic

Cat.No: T20948

Synonym: HOK 7501,HOK7501,HOK-7501

Cat.No: T74170

Cat.No: T81054

Target: VEGFR

Connexin mimetic peptide 40,37GAP26

Cat.No: T82684

Paraxanthine-d6

Cat.No: T71327

Cat. No.	Product Name	Target	Signaling Pathways
T2895	Lupeol Fagarasterol,羽扇豆醇,Monogynol B,Clerodol,(3β,13ξ)-Lup-20(29)-en-3-ol,Farganasterol	Apoptosis; Androgen Receptor; Akt	Apoptosis; Cytoskeletal Signaling; Endocrinology/Hormones; PI3K/Akt/mTOR signaling
	Lupeol (Monogynol B) 是一个活跃的五环三萜，具有抗氧化剂、抗肿瘤和抗炎活性。它是一种雄激素受体抑制剂，可研究癌症，特别是雄激素依赖表型和去势抵抗表型的前列腺癌。
T15027	Cyclopiazonic acid 环匹阿尼酸,环二氮酸	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Cyclopiazonic acid 是一种神经毒性次级代谢产物 (SM)，源于A. flavus，是一种纳摩尔内质网钙 ATP 酶抑制剂 (Ca2+ATPase; SERCA)，是植物细胞死亡的有效诱导剂。
T8093	2-Benzylsuccinic acid 2-苄基丁二酸,DL-Benzylsuccinic acid	Carboxypeptidase	Proteases/Proteasome
	2-Benzylsuccinic acid (DL-Benzylsuccinic acid) 是羧肽酶 A (CPA) 抑制剂。

天然产物

Cat.No: T2895

Synonym: Fagarasterol,羽扇豆醇,Monogynol B,Clerodol,(3β,13ξ)-Lup-20(29)-en-3-ol,Farganasterol

Target: Apoptosis, Androgen Receptor, Akt

Cyclopiazonic acid

Cat.No: T15027

Synonym: 环匹阿尼酸,环二氮酸

Target: Calcium Channel

2-Benzylsuccinic acid

Cat.No: T8093

Synonym: 2-苄基丁二酸,DL-Benzylsuccinic acid

Target: Carboxypeptidase

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