110
7
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T80024 |
Cationic Bovine Serum Albumin
cBSA, chemically modified cationic bovine serum albumin |
||
Cationic Bovine Serum Albumin(带正电荷的牛血清白蛋白)是由583个氨基酸组成的蛋白质,具有三个同源的全α结构域。该蛋白质与Tanshinone IIA联用,在缺血性脑卒中中展现出显著的神经保护作用。 | |||
T16939 |
Stains-All
|
Others | Others |
Stains-All 是一种能够研究钙调蛋白 (CaM) 和相关钙结合蛋白 (CaBP) 的各个钙结合位点的结构特征的便捷探针,是一种阳离子碳菁染料。 | |||
T19080 |
DOPE
1,2-二油酰-SN-甘油-3-磷酰乙醇胺 |
Others | Others |
DOPE (DOPE) 是一种阳离子脂质体的中性辅助脂质 (helper lipid),能够与阳离子磷脂结合,增强裸 siRNA 的转染效率。 | |||
T11086 |
DOTAP chloride
(2,3-二油氧基丙基)三甲基氯化铵,1,2-Dioleoyl-3-trimethylammonium-propane chloride |
Others | Others |
DOTAP chloride (1,2-Dioleoyl-3-trimethylammonium-propane chloride) 是高效的阳离子脂质,可以在不使用辅助脂质的情况下,作用于瞬时或者稳定转染 DNA (质粒、bacmids) 和修饰核酸 (反义寡核苷酸)。 | |||
T6439 |
Cetylpyridinium Chloride
西吡氯铵,Cetamium,Pristacin,Hexadecylpyridinium Chloride |
Others; HBV; Antibacterial | Microbiology/Virology; Others |
Cetylpyridinium Chloride (Hexadecylpyridinium Chloride) 是阳离子季铵,是一种广谱抗菌剂。它有效抑制 HBV 衣壳装配,IC50为 2.5 μM。它被用于杀虫剂和各种漱口水以及其他个人护理产品中。 | |||
T20639 |
Lauryl benzalkonium chloride
Lauralkonium chloride,NSC 85508,NSC85508,十二烷基二甲基苄基氯化铵,Benzododecinium chloride,NSC-85508 |
Others | Others |
Lauryl benzalkonium chloride (Benzododecinium chloride) 是阳离子表面活性剂的一种。 | |||
T31546 |
DLinDAP
D-Lin-DAP,D-LinDAP |
Others | Others |
DLinDAP (D-LinDAP) 是一种可离子化的阳离子脂质,可用于 SiRNA 的递送。 | |||
T17073 |
Thioflavin T
Basic Yellow 1,硫黄素 T,硫黄素T |
Others | Others |
Thioflavin T (Basic Yellow 1) 是阳离子 Benzothiazole 染料,在组织切片中能够淀粉样蛋白结合,增强荧光强度。 | |||
T5823 |
D-Lin-MC3-DMA
|
Others | Others |
D-Lin-MC3-DMA 是一种递送 siRNA 载体,是一种可离子化的氨基脂质类化合物。 | |||
T22981 |
Tetradecyltrimethylammonium bromide
MitMAB,Cetrimide,tetradecyl trimethyl ammonium bromide,十四烷基三甲基溴化铵 |
Dynamin | Cytoskeletal Signaling |
Tetradecyltrimethylammonium bromide (MitMAB) 是一种具有不对称结构的阳离子表面活性剂,是一种有机结构单元。 | |||
T5152 |
MKT-077
MKT 077,FJ-776,MKT077 |
HSP | Cytoskeletal Signaling; Metabolism |
MKT-077 (FJ-776) 是一种阳离子红花青染料,通过抑制 Hsp70 分子伴侣家族成员的能力,显示出对癌细胞系的抗增殖活性。 | |||
T15139 |
DLin-KC2-DMA
|
Others | Others |
DLin-KC2-DMA 是一种可用于siRNA 传递的阳离子,也是一种可电离的脂质。 | |||
T0336 |
Benzalkonium chloride
苯扎氯铵,Alkyldimethylbenzylammonium chloride |
Others; Antibacterial | Microbiology/Virology; Others |
Benzalkonium chloride (Alkyldimethylbenzylammonium chloride) 是一种含有季铵基团的阳离子表面活性剂,也是一种抗菌剂,在滴眼液中用作防腐剂。 | |||
T17109 |
TMRM Perchlorate
四甲基若丹明甲酯酸铵,T668 |
Others | Others |
TMRM Perchlorate (T668) 是细胞渗透性的阳离子亲脂性红色荧光染料 (λex=530 nm, λem=592 nm)。 | |||
T19067 |
Thionin acetate
硫堇(劳氏紫),Thionine acetate |
Others | Others |
Thionin acetate (Thionine acetate) 是一种异染阳离子组织学染料,普遍用于生物学染色。 | |||
T38604 |
C12-200
C12-200 |
Others | Others |
C12-200是一个基准的可离子化的阳离子类脂质与辅助类脂质一起,用于 mRNA 的传递。 | |||
TP1341L |
Polymyxin B nonapeptide acetate
Polymyxin B nonapeptide acetate(86408-36-8 free base) |
Antibacterial; Antibiotic | Microbiology/Virology |
Polymyxin B nonapeptide acetate(86408-36-8 free base) 是一种阳离子环肽。 Polyxin B 九肽是 polyxin B 经酶解产生的衍生物。与 polyxin B 相比,polyxin B 九肽毒性低,缺乏杀菌活性,仍具有破坏革兰氏阴性菌外膜的能力。 | |||
TP1300 |
GsMTx4 TFA (1209500-46-8 free base)
GsMTx4 TFA |
Piezo Channel | Membrane transporter/Ion channel |
GsMTx4 TFA (1209500-46-8 free base) (GsMTx4 TFA) 是一种蜘蛛毒肽,可选择性地抑制属于 Piezo 和 TRP 通道家族的阳离子可渗透机械敏感通道 (MSC)。 | |||
T2188 |
Thonzonium Bromide
嘧苯十六铵,通佐溴胺 |
Proton pump; Antibacterial; Autophagy | Autophagy; Membrane transporter/Ion channel; Microbiology/Virology |
Thonzonium bromide 是一种单阳离子表面活性剂,在结构上与 Farnesol 相似的抗菌剂。它以剂量依赖的方式抑制质子转运 (EC50=69 μM)。在体外可抑制 RANKL 诱导的破骨细胞形成和骨吸收,并在体内阻止 LPS 诱导的骨丢失。 | |||
T16698 |
Pyronin Y
C.I. 45005,派洛宁Y,派洛宁 Y,Pyronine G |
Others | Others |
Pyronin Y (Pyronine G) 是一种可插入 RNA 的阳离子染料,可以靶向包括 RNA,DNA 和细胞器的细胞结构。它能够与双链核酸(尤其是 RNA) 形成荧光复合物,半定量分析细胞 RNA。它可用于活细胞中核糖核蛋白复合物的特定 RNA 亚种的鉴定。 | |||
T7026L |
Kukoamine B mesylate
|
Antioxidant | oxidation-reduction |
Kukoamine B mesylate 是从地骨皮中提取得到的新型阳离子生物碱,具有抗氧化活性,抑制 Kupffer 和 RAW 264。7 细胞中的 LPS 内化,可用于研究急性炎症和糖尿病。 | |||
TF0112 |
DPPS
12-Dipalmitoyl-sn-glycero-3-PS sodium salt,DPPS-Na |
Others | Others |
DPPS (12-Dipalmitoyl-sn-glycero-3-PS sodium salt) 是一种阴离子二酰基磷脂,是磷脂酰丝氨酸(PS)的一种形式,是一种位于细胞膜内小叶的带负电荷的磷脂。DPPS 被用来制作阳离子囊泡和脂质体。 | |||
T12510 |
PNU-177864 hydrochloride
PNU-177864 (hydrochloride) |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
PNU-177864 hydrochloride 是选择性的,口服有效的多巴胺 D3 受体拮抗剂。PNU-177864 hydrochloride 具有与阳离子两亲药物一致的结构。PNU-177864 hydrochloride 可在体内诱导磷脂代谢,并显示出抗精神分裂症活性。 | |||
T8644 |
Elamipretide Triacetate
Elamipretide TriTFA |
Others | Others |
Elamipretide Triacetate (Elamipretide TriTFA) 是一种芳香族阳离子四肽,可轻松穿透细胞膜并短暂定位于线粒体内膜,在此与心磷脂结合。它已用于研究 Leber 遗传性视神经病变治疗的试验。 | |||
T18918 |
Azure B
Azure B chloride,天青 B |
MAO; Monoamine Oxidase | Metabolism; Neuroscience |
Azure B (Azure B chloride) 是一种 Methylene blue 的主要代谢物,是一种阳离子染料,用于 Azure 曙红染色剂以进行血液涂片染色。它是高选择性和可逆的抑制单胺氧化酶(MAO)-A 的抑制剂,对重组人的 MAO-A 和 MAO-B 的IC50分别为 11 和 968 nM。它具有显著的抗抑郁作用。 | |||
T12992 |
SPR741 acetate
SPR741 acetate,NAB741 acetate,SPR741 acetate (1179330-52-9 free base) |
Antibacterial | Microbiology/Virology |
SPR741 acetate 是衍生自多粘菌素 B 的阳离子肽,通过增加革兰氏阴性细菌外膜的通透性来抑制严重的革兰氏阴性细菌感从而展现出对革兰氏阴性菌的抗菌活性。SPR741 acetate 常与抗生素联合使用来治疗一些疾病。 | |||
T0900 |
Cetylpyridinium chloride monohydrate
Hexadecylpyridinium chloride monohydrate,十六烷基氯化吡啶 |
Antibacterial; Antibiotic | Microbiology/Virology |
Cetylpyridinium chloride monohydrate (Hexadecylpyridinium chloride monohydrate) 是阳离子季铵, 是一种能杀死细菌和其他微生物的防腐剂, 用于某些类型的漱口水, 牙膏, 咽喉和鼻腔喷雾剂中, 可有效预防牙斑和减少牙龈炎。 | |||
T8902 |
DOTMA
Trimethyl[2,3-(dioleyloxy)propyl]ammonium Chloride,N-(1-(2,3-dioleyloxy)propyl)-N,N,N-trimethylammonium |
Others | Others |
DOTMA (N-(1-(2,3-dioleyloxy)propyl)-N,N,N-trimethylammonium) 作为 tetra-methylated DOTA 类似物,是一种阳离子脂类,被用作基因治疗的非病毒载体。它已被用作脂质体的成分,可用于封装 siRNA、microRNA 和寡核苷酸,并用于体外基因转染。在体外和体内均表现出良好的基因转染效果。DOTMA 诱导脂质体上的正电荷,从而促进脂质体与细胞膜的有效相互作用。 | |||
TP1410 |
Cecropin A
|
Antibacterial; Antibiotic | Microbiology/Virology |
Cecropin A 是37个氨基酸组成的线性多肽,表现出抗菌、抗炎和抗肿瘤的功效。 | |||
T34825 |
Tetralysine
|
||
Tetralysine is a cationic moiety that may construct gene delivery vectors and DNA nanoparticles. | |||
T40550 |
Human β-defensin-1
Human β-defensin-1,HβD-1 |
||
Human β-defensin-1 (HβD-1) is a cysteine-rich cationic skin-antimicrobial peptide (SAP) produced by epithelial surfaces, circulatory cells, and cells of the reproductive tract. It exhibits antimicrobial activity against a wide range of sperm bacteria. | |||
T81644 |
NRC-16
|
||
NRC-16为具有生物活性的肽,属于(杀侧耳素样阳离子AMP)类化合物。 | |||
T74320 |
14:0 EPC chloride
|
||
14:0 EPC chloride 是一种酰基阳离子脂质,用于药物递送中的脂质体。 | |||
T39436 |
Omiganan
|
||
Omiganan is a cationic antimicrobial peptide with activity against both gram-positive and gram-negative bacteria, as well as Candida spp. isolates. This compound, serving as an analogue of indolicidin, is utilized for research purposes related to alcohol nose and acne. | |||
T25972 |
Polymyxin D2
|
||
Polymyxin D2 is a cationic lipopeptide antibiotic against many species of Gram-negative bacteria. | |||
T74292 |
Fluorescent DOTAP
|
||
Fluorescent DOTAP 是一种阳离子脂质,可用于研究核酸和蛋白质传递。 | |||
T20462 |
Lysyllysyllysine
Trilysine,Lys-lys-lys,L-Lysine, L-lysyl-L-lysyl- |
||
Lysyllysyllysine is a cationic moiety. It may be used in the construction of gene delivery vectors and DNA nanoparticles. | |||
TP1773 |
PGLa
|
||
PGLa is a cationic antimicrobial peptide (AMP) originally isolated from frog. It has been shown to have antibacterial,antifungal,and antiviral,activities. | |||
T74239 | DOSPA | ||
DOSPA 是一种阳离子脂质。DOSPA 制备 DNA 是一种很有前途的转染系统。 | |||
T74319 |
14:0 DAP
|
||
14:0 DAP (1,2-dimyristoyl-3-dimethylammonium-propane ) 是一种阳离子脂质,可用于药物递送。 | |||
T74313 | MVL5 | ||
MVL5 是一种不可降解的多价阳离子脂质。MVL5 是一种高效的 DNA 和 siRNA 载体。 | |||
T74246 |
Transfectam
|
||
Transfectam为一种阳离子脂质,能与DNA形成复合物,从而高效地将基因转入多种真核细胞。 | |||
TP1090 |
SPR741
NAB741 |
||
SPR741, formerly NAB741 (12), is a cationic peptide derived from polymyxin B and is one such potentiator molecule that is under development for the treatment of serious Gram-negative bacterial infections. | |||
TP1341 |
Polymyxin B nonapeptide
|
||
Polymyxin B nonapeptide, a cationic cyclic peptide derived by enzymatic processing from the naturally occurring peptide polymyxin B, is able to increase the permeability of the outer membrane of Gram-negative bacteria toward hydrophobic antibiotics probab | |||
TP1089 |
SPR741 TFA (1179330-52-9 free base)
NAB741 TFA,SPR741 TFA |
||
SPR741 TFA (NAB741 TFA) is a cationic peptide derived from polymyxin B and is a potentiator molecule. | |||
T37018 |
OH-Chol
|
||
OH-Chol is a cationic cholesterol derivative.1 OH-Chol, as a component of lipoplexes with DOPE , has been used for siRNA delivery and gene silencing in MCF-7 cells, as well as in mice via intravenous injection, resulting in lipoplex accumulation in the liver. It has also been used in cationic nanoparticles in combination with Tween 80 to transfect pDNA and siRNA into PC3 mouse xenografts via intratumoral injection and with Tween 80 and folate-PEG2000-DSPE in a KB mouse xenograft model for intrat... | |||
T38679 |
DODAP
|
||
DODAP, an ionizable cationic lipid, serves as a vital component in liposome formation. Its applications encompass the capability to encapsulate siRNA, immunostimulatory chemotherapeutic agents for in vitro and in vivo delivery, among others. | |||
T75331 |
Brilliant green
|
||
Brilliant green, a cationic dye, is utilized for coloring silk and wool. Additionally, it halts the propagation of mold, intestinal parasites, and fungus, proving effective against Gram-positive bacteria [1] [2]. | |||
T23810 |
BMX-001
MnTnBuOE-3-PyP 5+,manganese butoxyethyl pyridyl porphyrin,BMX001,manganese (III) ortho N-butoxyethylpyridylporphyrin |
||
BMX-001 is a third-generation, cationic, lipophilic, manganese (Mn), and porphyrin-based mimetic of the human mitochondrial manganese superoxide dismutase (MnSOD). It also has antioxidant and potential chemoprotective activities. | |||
T19044 |
Oxazine 1 perchlorate
|
Others | Others |
Oxazine 1 perchlorate is a symmetric cationic dye (λem=666 nm, λex=653 nm). |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15716 |
Lasalocid sodium
拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium |
Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology |
Lasalocid sodium (Lasalocid-A sodium) 是一种抗菌剂。 | |||
T1100 |
Polymyxin B Sulfate
Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX |
Antibacterial; Antibiotic | Microbiology/Virology |
Polymyxin B Sulfate (Poly-RX) 是一个阳离子型表面活性剂抗生素剂,能够提高细胞膜的渗透性。 | |||
T3092 |
Nigericin sodium salt
尼日利亚菌素,尼日利亚菌素钠盐 |
Potassium Channel; NOD-like Receptor (NLR); Antibacterial; Antibiotic; NOD | Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB |
Nigericin sodium salt 属于抗生素,是一种 NLRP3 激活剂,也是一种阳离子离子载体。Nigericin sodium 可以触发 NALP3 炎性体的激活,可抑制高尔基体功能并抑制革兰氏阳性菌的生长。 | |||
T83902 |
Polymyxin E1 sulfate
Colistin A sulfate |
||
Polymyxin E1,是一种肽类抗生素,也是原初从B. polymyxa分离得到的阳离子脂肽抗生素colistin的主要成分。对P. aeruginosa和E. coli具有活性(MICs分别为2和0.8 µg/ml)。 | |||
T83904 |
Polymyxin E2 sulfate
Colistin B sulfate |
||
Polymyxin E2 是一种肽类抗生素,也是最初从B. polymyxa分离出的阳离子脂肽抗生素colistin的主要成分。该化合物对植物致病菌X. oryzae具有活性(EC50 = 0.21 µg/ml),并且在温室研究中,当以200 µg/ml的浓度应用时,能够预防和逆转水稻细菌性叶枯病。 | |||
T83903 |
Polymyxin B2 sulfate
|
||
Polymyxin B2是一种抗生素,并且是从B. polymyxa分离出的阳离子脂肽抗生素polymyxin B的主要成分。该化合物对P. aeruginosa、A. baumannii、K. pneumoniae和E. cloacae菌株具有活性(MICs分别为1-2、0.5-1、0.25-0.5和0.25-1 µg/ml)。在体内实验中,以4 mg/kg剂量的Polymyxin B2能显著降低P. aeruginosa血液感染小鼠模型中的血液集落形成单位(CFUs)数量。 | |||
T83693 |
Magainin 2 TFA
MG2 |
||
Magainin 2是一种从非洲爪蟾(X. laevis)皮肤中分离出的阳离子肽,具有宿主防御和抗菌活性。该化合物对细菌E. coli、K. pneumoniae、S. epidermidis、S. aureus及真菌C. albicans表现出活性(MICs分别为5、10、10、50和80 µg/ml)。Magainin 2(20 µM)能降低猕猴桃花粉的萌发率和平均管长。在被单纯疱疹病毒1型(HSV-1)或2型(HSV-2)感染的Vero细胞中,它可减少病毒复制(EC50s分别为22.16和19.8 µM),同时不影响细胞活性,其50%细胞毒性浓度值(CC50)大于100 µM。 |