82
20
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0510 |
Sulfaguanidine
Sulfaguine,Guanicil,磺胺脒 |
Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology |
Sulfaguanidine (Guanicil) 是一种具有口服活性的磺胺类抗菌剂和抗生素。它可用于肠道感染,例如细菌性痢疾的研究。 | |||
T1005 |
Amoxicillin
Amoxycillin,阿莫西林 |
Antibacterial; Antibiotic | Microbiology/Virology |
Amoxicillin (Amoxycillin) 是一种具有广谱抗菌活性和良好口服吸收的抗生素。 | |||
T7533 |
Taurolidine
|
Apoptosis; Others; Antibacterial; Antibiotic | Apoptosis; Microbiology/Virology; Others |
Taurolidine 是一种广谱抗菌剂,用于预防中心静脉导管相关感染。它具有抗真菌和抗肿瘤作用。 | |||
T6385 |
Amoxicillin Sodium
阿莫西林钠,Clavulanate |
Antibacterial; Antibiotic | Microbiology/Virology |
Amoxicillin Sodium (Clavulanate) 是一种有广谱抗菌活性,口服吸收好的抗生素。它能抑制细胞壁中多肽的生物合成,可抑制细胞生长。 | |||
T3117 |
Marbofloxacin
马波沙星,Marbofloxacine,Zeniquin,Marbocyl |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。 | |||
T0921 |
Sulfabenzamide
Sultrin,N-Sulfanilylbenzamide,苯甲酰磺胺 |
Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology |
Sulfabenzamide (N-Sulfanilylbenzamide) 是一种磺胺类抗菌剂,可单独使用或与磺胺噻唑和磺胺乙酰胺一起用作阴道内的局部抗菌制剂。 | |||
T1177 |
Sulfaquinoxaline
磺胺喹恶啉,Avicocid,磺胺喹噁啉,Sulphaquinoxaline,Sulfabenzpyrazine |
Others; Antibacterial; Antibiotic; Parasite | Microbiology/Virology; Others |
Sulfaquinoxaline (Sulfabenzpyrazine) 是一种兽用抗菌剂,对革兰氏阴性菌和革兰氏阳性菌均有活性。它能用于预防球虫病和细菌感染。 | |||
T1434 |
Clarithromycin
A-56268,克拉霉素 |
P450; ribosome; MRP; Antibacterial; Antibiotic; Autophagy | Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology |
Clarithromycin (A-56268) 具有广谱的抗菌活性。它抑制 CYP3A4催化的三唑仑 α-羟基化,IC50(Ki) 值为 56 (43) μM。它抑制 HERG 钾电流。它可削弱连接 hERG1 和 PI3K 的信号通路影响自噬流 。 | |||
TP1444 |
Magainin 2
蛙皮素 2 |
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Magainin 2是从非洲爪蟾皮肤中分离得到的一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌显示出抗生素活性,对原生动物也有活性。它通过优先与细菌膜中丰富的阴离子磷脂相互作用而发挥细胞毒性作用。 | |||
T19717 |
Cyclo-L-Trp-L-Trp
|
Antifungal | Microbiology/Virology |
Cyclo-L-Trp-L-Trp 是一种广谱抗真菌剂。它还诱导组蛋白的高度乙酰化。 | |||
T4989 |
Fosfomycin Tromethamine
|
Antibacterial; Antibiotic | Microbiology/Virology |
Fosfomycin tromethamine 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。 | |||
T0917 |
Sulfaquinoxaline sodium salt
SQ-Na,磺胺喹恶啉钠盐,Sulfaquinoxaline sodium,磺胺喹啉钠 |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Sulfaquinoxaline sodium salt (SQ-Na) 是一种兽用广谱抗菌剂,有抗革兰氏阴性菌和革兰氏阳性菌活性。Sulfaquinoxaline 能用于预防球虫病和细菌感染。 | |||
T1000L |
Chlorhexidine diacetate
醋酸氯己定,Hibitane diacetate,Chlorhexidine Acetate,Bactigras |
CAT; Antibacterial; Antibiotic; Antifection | Microbiology/Virology; oxidation-reduction |
Chlorhexidine diacetate (Bactigras) 是一种双胍类杀菌剂,能快速消灭革兰氏阳性菌和革兰氏阴性菌。它也用作漱口水以防止口腔菌斑。 | |||
T20702 |
Ormetoprim
Ro5-9754,奥美普林,Ro 5-9754,Ro-5-9754 |
Antibiotic | Microbiology/Virology |
Ormetoprim (Ro 5-9754) 是一种兽用抗菌剂,通常用于水产养殖和家禽行业,可以预防疾病在淡水水产养殖中的传播,促进家畜的生长。 | |||
T3125 |
Amikacin sulfate
Amikacin Sulfate Salt,阿米卡霉素硫酸,硫酸阿米卡星 |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Amikacin sulfate 是一种氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它抑制大多数革兰氏阴性细菌,还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。 | |||
T7865 |
Danofloxacin
达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine |
Others; DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。 | |||
T1233 |
Oxolinic acid
Emyrenil,Nidantin,NSC 110364,恶喹酸,Dioxacin,Urinox |
Dopamine Receptor; DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; GPCR/G Protein; Microbiology/Virology; Neuroscience |
Oxolinic acid (Nidantin) 是一种抗生素,对革兰氏阴性菌和革兰氏阳性菌均有效,可研究急性和慢性尿路感染。它是一种 DNA/RNA 合成抑制剂,也是一种多巴胺摄取抑制剂,能刺激小鼠的活跃过度。 | |||
T7419 |
Sutezolid
PNU-100480,U-100480,PF-02341272 |
Antibacterial; Antibiotic | Microbiology/Virology |
Sutezolid (U-100480) 是一种具有口服活性恶唑烷酮抗菌剂,通过抑制细菌蛋白质合成发挥作用。它有抗分枝杆菌活性,可研究耐药结核病。 | |||
T0195 |
Secnidazole
RP-14539,PM-185184,塞克硝唑 |
Antibiotic; Parasite | Microbiology/Virology |
Secnidazole (PM-185184) 是一种具有口服活性唑类抗生素,半衰期比甲硝唑更长。它有潜力研究细菌性阴道病。 | |||
T3131 |
Fosfomycin calcium
Phosphomycin calcium salt,Fosmicin,磷霉素钙 |
Antibacterial; Antibiotic | Microbiology/Virology |
Fosfomycin calcium (Phosphomycin calcium salt) 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。 | |||
T1005L |
Amoxicillin trihydrate
Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate |
Antibacterial; Antibiotic | Microbiology/Virology |
Amoxicillin trihydrate (Moxaline trihydrate) 是一种中谱β内酰胺抗菌素。 | |||
T0331 |
Moxifloxacin hydrochloride
盐酸莫西沙星,莫西沙星盐酸盐,BAY-128039,Moxifloxacin HCl,BAY12-8039 HCl |
Topoisomerase; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Moxifloxacin hydrochloride (BAY12-8039 HCl) 是一种口服有效的 8-甲氧基喹诺酮类抗菌药物,可研究感染性肺炎,急性细菌性鼻窦炎和慢性支气管炎的急性细菌性加重。 | |||
T6382 |
Amikacin disulfate
硫酸阿米卡星,Pierami,阿米卡星硫酸盐,BAY-416651 sulfate,BB-K8,Amikacin sulfate |
Antibacterial; Antibiotic | Microbiology/Virology |
Amikacin disulfate (BAY-416651 sulfate) 是氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它对大多数革兰氏阴性细菌都有效。它还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。 | |||
T6383 |
Amikacin hydrate
阿米卡星水合物,BAY416651 hydrate |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Amikacin hydrate (BAY416651 hydrate) 是氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。 | |||
T1733 |
Ciprofloxacin EP IMpurity A
Q-Acid,Fluoroquinolonic Acid,环丙羧酸,Ciprofloxacin Impurity A |
Antibiotic | Microbiology/Virology |
Ciprofloxacin EP IMpurity A (Fluoroquinolonic Acid) 是一种抗生素和抗菌剂。 | |||
T30785 |
Cefacetrile
Cefacetrilum,Cefacetrilo,Celospor,Cephacetrile,Cefacetril |
Antibiotic | Microbiology/Virology |
Cefacetrile (Cephacetrile) 是一种广谱的头孢类抗生素,具有抗菌活性,可用于研究革兰氏菌感染,作用与头孢噻吩作用。 | |||
T20022 |
Cephalexin monohydrate
Cephalexin hydrate,Cephacillin hydrate,Cefalexin hydrate |
Antibiotic | Microbiology/Virology |
Cephalexin monohydrate (Cephalexin hydrate) 是一种可口服的半合成头孢菌素类抗生素,具有显著的抗菌活性, 通过靶向青霉素结合蛋白 (PBPs)抑制细菌增殖。 | |||
T12512 |
PNU288034
|
Antifungal | Microbiology/Virology |
PNU288034 是一种有效的恶唑烷酮类抗生素,具有抗菌活性,可用于预防和治疗革兰氏菌感染。 | |||
TP1763L |
Magainin 1 acetate
|
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Magainin 1 acetate 是一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌表现出抗生素活性。 | |||
T14922 |
Cefodizime
|
Antibacterial; Antibiotic | Microbiology/Virology |
Cefodizime 是一种新型头孢菌素抗生素,具有广泛的生物活性。Cefodizime 对肾脏没有毒性且具有良好的耐受性和免疫调节活性,具有抗菌活性,可用于研究呼吸系统和泌尿系统的严重感染。 | |||
T25085 |
Amythiamicin B
|
||
Amythiamicin B is a novel antimicrobial antibiotic. | |||
T25037 | Aldecalmycin | ||
Aldecalmycin is a new antimicrobial antibiotic isolated from Streptomyces. | |||
T1070L |
Cefmetazole
Sodium, Cefmetazole,Cefmetazolum,Cefmetazolo |
||
Cefmetazole is a second-generation semi-synthetic β-lactam cephalosporin antibiotic with antimicrobial activity. | |||
T26479 |
A32390A
A-32390A,A 32390A |
||
A32390A, an antibiotic inhibitor, shows antimicrobial activity against gram-positive bacteria and fungi. | |||
T26455 |
A 83016F
A-83016F,A83016F |
||
A 83016F, an antibiotic from an actinomycete designated A83016, exhibits weak antimicrobial activity. | |||
T16382 |
Oleandomycin
|
Others | Others |
Oleandomycin is similar to Erythromycin has antimicrobial activity. Oleandomycin is a macrolide antibiotic structurally closely related to Erythromycin. | |||
T70429 |
TP-6076
|
||
TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A. baumannii. | |||
T31104 |
CS 461
CS461,CS-461 |
||
CS 461 is a cephalosporin antibiotic that has shown effective antimicrobial activity against a variety of bacteria in vitro and in vivo. | |||
T28046 |
Mirosamicin
A 11725 II,Antibiotic AR 5-2 |
||
Mirosamicin is a macrolide antibiotic, it has antimicrobial effect against gram-positive bacteria, some gram-negative bacteria and mycoplasma. | |||
T1466L |
Difloxacin HCl
|
||
Difloxacin 是第二代合成的氟喹诺酮抗菌抗生素。 | |||
T37350 |
TBI-223
|
||
TBI-223 is an orally bioavailable oxazolidinone antibiotic with antimicrobial properties. It exhibits potent activity against Mycobacterium tuberculosis (Mtb)[1][2]. | |||
T83042 | Antimicrobial agent-26 | ||
Antimicrobial agent-26?是一款降低抗生素耐药性的高效抗菌化合物。 | |||
T39683 |
Human β-defensin-3
Human β-defensin-3,HβD-3 |
||
Human β-defensin-3 (HβD-3) is an antibiotic antimicrobial peptide synthesized by epithelial cells. It exhibits potent antimicrobial properties and mitigates inflammatory cytokine responses. HβD-3 efficiently targets various microorganisms, displaying IC90 values ranging from 6 to 25 μg/ml. | |||
T80304 |
Aurein 5.2
|
Antibiotic | Microbiology/Virology |
Aurein 5.2是一种具有抗菌活性的抗生素肽类化合物。 | |||
T10330 |
Antibiotic-5d
|
Antibacterial | Microbiology/Virology |
Antibiotic-5d 是一种合成的抗菌化合物,对各种革兰氏阳性和革兰氏阴性细菌、真菌和酵母表现出中等的抗菌活性。 | |||
T78114 |
Phenethicillin sodium
α-Phenoxyethylpenicillin sodium,Pheneticillin sodium |
||
Phenethicillin (α-Phenoxyethylpenicillin) sodium为抗生素类青霉素类药物,表现出抗菌特性。 | |||
T80302 |
Aurein 3.2
|
Antibiotic | Microbiology/Virology |
Aurein 3.2为一种具备抗菌及抗肿瘤功能的生物活性肽。 | |||
T10306 |
Amoxicillin D4
Amoxycillin D4 |
Others | Others |
Amoxicillin D4 (Amoxycillin D4) is a deuterium-labeled Amoxicillin. Amoxicillin is an antibiotic with broad-spectrum antimicrobial activity. | |||
T80298 |
Aurein 2.4
|
Antibiotic | Microbiology/Virology |
Aurein 2.4为一种抗菌肽,对革兰氏阳性细菌显示出抗生素活性。 | |||
T80299 |
Aurein 2.5
|
Antibiotic | Microbiology/Virology |
Aurein 2.5,一种具备抗细菌及抗真菌活性的抗生素肽。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1313 |
Nitrofurantoin
Furadantine,呋喃妥因,Macrodantin,Furadonine |
Antibacterial; Antibiotic | Microbiology/Virology |
Nitrofurantoin (Furadantine) 是一种具有口服活性的广谱内酰胺酶抗菌剂。它是一种抗生素,可研究尿路感染。 | |||
T1032 |
Erythromycin
红霉素,E-Mycin |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Erythromycin (E-Mycin) 是由放线菌产生的大环内酯类抗生素。它结合细菌的 50S 核糖体亚基,通过阻断转肽和易位反应来抑制 RNA 依赖性蛋白的合成。 | |||
T6995 |
Ochromycinone
STA 21,STA21,STA-21 |
Antibacterial; STAT | JAK/STAT signaling; Microbiology/Virology; Stem Cells |
Ochromycinone (STA 21) 是一种天然抗生素,也是一种 STAT3抑制剂。它可抑制 STAT3DNA 结合活性,STAT3二聚化。它具有抗癌和抗菌活性。 | |||
T22308 |
Dimboa
2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one,丁布 |
Others; Antibacterial; Antibiotic; Antifungal | Microbiology/Virology; Others |
Dimboa (2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one) 是抗生素,是禾本科植物化学防御系统的一部分。 它对许多已研究的细菌和真菌菌株具有生长抑制特性。它表现出强大的自由基清除活性和较弱的铁 (III) 离子还原活性和有抗氧化活性。 | |||
T0146 |
Tioconazole
UK-20349,Vagistat,噻康唑 |
Antibiotic; Antifection; Antifungal | Microbiology/Virology |
Tioconazole (Vagistat) 是一种广谱性的抗真菌咪唑衍生物。它抑制几种皮肤真菌和几种酵母菌的 MIC50分别小于 3.12 mg/L 和 9 mg/L。 | |||
T8262 |
Fosfomycin sodium
Fosfomycin Disodium,磷霉素钠 |
Antibacterial; Antibiotic | Microbiology/Virology |
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。 | |||
T1153 |
Trimethoprim
NIH 204,BW 56-72,甲氧苄啶,NSC-106568 |
DHFR; DNA/RNA Synthesis; Antifolate; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology |
Trimethoprim (NSC-106568) 是抑菌抗生素,也是具有口服活性的二氢叶酸还原酶抑制剂。它对多种革兰氏阳性和革兰氏阴性需氧细菌具有活性,可用于尿路感染,肺孢子菌肺炎和志贺氏菌病的研究。 | |||
T15717 |
Lasalocid
Lasalocid-A,Antibiotic X-537A,Ionophore X-537A |
Antibacterial | Microbiology/Virology |
Lasalocid (Lasalocid-A) 是一种由链霉菌产生的离子载体抗生素,具有抗菌和寄生虫作用,常添加进饲料中。 | |||
T7148 |
JOSAMYCIN
EN-141,交沙霉素 |
Antibacterial; Antibiotic | Microbiology/Virology |
Josamycin (EN-141) 是一种大环内酯类抗生素,对多种病原体有抗菌活性。它对核糖体的解离常数Kd 为 5.5 nM。 | |||
T4136 |
Lapachol
Bethabarra wood,CI75490,黄钟花醌,Greenhartin,Tecomin |
Others; Influenza Virus; Antibacterial; Parasite; Antifungal | Microbiology/Virology; Others |
Lapachol (CI75490) 是从Tabebuia avellanedae 中分离得到的一种萘醌。它具有具有抗菌、抗炎、镇痛、抗肿瘤和抗生素特性。 | |||
T0950 |
Neomycin sulfate
Framycin sulfate,硫酸新霉素 |
Phospholipase; ribosome; Antibacterial; Antibiotic | Metabolism; Microbiology/Virology |
Neomycin sulfate (Framycin sulfate) 是一种广谱的氨基糖苷类抗生素。Neomycin sulfate 可以阻断细菌蛋白质的合成以发挥抗菌活性。Neomycin sulfate 常用于筛选具有 Neo 抗性基因的原核和真核细胞。 | |||
T8641 |
Vancomycin
|
Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology |
Vancomycin 是一种糖肽类抗生素,可以通过改变细胞膜的渗透性并选择性地抑制核糖核酸的合成以发挥抗菌活性。Vancomycin 可以用于治疗所有抗生素均无效的严重感染。 | |||
T20779 |
Kitasamycin tartrate
Leucomycin tartrate |
||
Kitasamycin tartrate, a macrolide antibiotic produced by Streptomyces kitasatoensis, has a wide spectrum of antimicrobial activity. | |||
T75443 | Tomaymycin | ||
Tomaymycin 是一种抗肿瘤抗生素。Tomaymycin 对革兰氏阳性菌具有抗菌活性。 | |||
T6402 |
Azomycin
2-Nitroimidazole,2-硝基咪唑,Ro 05-9129,Amicin |
Antibacterial; Antibiotic | Microbiology/Virology |
Azomycin (Ro 05-9129) 是一种可抑制有氧革兰氏阳性菌和革兰氏阴性菌的生长的抗生素。 | |||
T38241 |
2-Aminoimidazole
|
||
2-Aminoimidazole is a potent antibiofilm agent and adjuvant to antimicrobial treatments, which effectively disrupts bacterial self-protection mechanisms by inhibiting biofilm formation and genetically-encoded antibiotic resistance traits. Additionally, 2-Aminoimidazole acts as a weak noncompetitive inhibitor of human arginase I, with a Ki value of 3.6 mM[1][2][3]. | |||
T11233 | Erythromycin thiocyanate | Antibacterial | Microbiology/Virology |
Erythromycin thiocyanate acts by binding to bacterial 50S ribosomal subunits and inhibits RNA-dependent protein synthesis by blockage of transpeptidation and/or translocation reactions, without affecting synthesis of nucleic acid .Erythromycin thiocyanate | |||
T75753 |
Magainin 1 TFA
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Magainin 1 TFA (Magainin I TFA) 是从 Xenopus laevis 皮肤中分离出的一种抗菌和两亲性肽。Magainin 1 TFA 对多种革兰氏阴性和革兰氏阳性细菌均表现出抗生素活性。 | |||
T73673 |
Thiomarinol A
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Thiomarinol A (4-Hydroxythiomarinol C) 是一种有效的抗生素。Thiomarinol A 是二硫代吡咯酮和海藻酸的混合物。Thiomarinol A 显示出抗菌活性。Thiomarinol A 以剂量依赖性方式抑制 MRSA IleRS,Kiapp 值为 19 nM。 | |||
T35741 |
Gliovirin
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Gliovirin is a fungal metabolite that has been found inT. harzianumand has fungicidal, antimicrobial and anti-inflammatory activities.1It is active against the plant pathogenic fungusP. ultimum(MIC = 60 ng/ml) and the parasiteT. brucei brucei(IC50= 90 ng/ml), but has no effect on the plant pathogenic fungiR. solani,P. omnivorum,T. basicola,R. arrhizus, andV. dahliaeor the bacteriaB. thuringiensis,P. fluorescens, andX. malvacearumwhen used at concentrations up to 1,000 ng/ml.2,3Gliovirin decrease... |