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Cat. No. | Product Name | Target | Signaling Pathways |
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T21468 |
CVT-2738
UNII-NYS3I6283H,CVT 2738,EC 610-916-8,CVT2738,RS-94287,N-(2,6-二甲基苯基)-1-哌嗪乙酰胺 |
Others | Others |
CVT-2738 (RS-94287) 是雷诺嗪的代谢物。 Ranolazine 是一种部分脂肪酸氧化 (pFOX) 抑制剂和抗心绞痛药物。 | |||
T78360 |
Glyceraldehyde phosphate dehydrogenase
GAPDH,G3PDH,GADPH |
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Glyceraldehyde phosphate dehydrogenase是一种酶,既是抗胸腺细胞剂也是抗凋亡剂的靶点,它负责催化过羟基自由基对还原型烟酰胺腺嘌呤二核苷酸(NADH)的链氧化反应。 | |||
T75537 | N-Acetyldopamine dimer-2 | ||
N-Acetyldopamine dimer-2(compound 2)是一种从蝉皮黄色粉末中分离出来的N-acetyldopamine二聚体,具有抗氧化和抗炎作用。它能抑制氧化低密度脂蛋白(LDL)的氧化、ROS的生成、NO的生成以及NF-κB的活性。 | |||
T35881 |
Resolvin E2
|
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Resolvin E2 (RvE2) is a member of the specialized pro-resolving mediator (SPM) family of bioactive lipids.1It is produced from eicosapentaenoic acidviaan 18-HEPE intermediate, which is formed by aspirin-acetylated COX-2-mediated oxidation of EPA, by 5-lipoxygenase (5-LO) in human polymorphonuclear (PMN) neutrophils.2,3RvE2 (20 ng/animal) inhibits increases in inflammatory exudate neutrophil infiltration in a mouse model of peritonitis induced by zymosan A .3Hepatic RvE2 levels are increased in m... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6S0139 |
Neobavaisoflavone
|
Apoptosis; DNA/RNA Synthesis | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Neobavaisoflavone 是一种从Psoralea corylifolia 的种子中分离出来的类黄酮。它具有抗炎,抗癌和抗氧化的作用。它在中至高浓度下可抑制 DNA 聚合酶,也可抑制血小板聚集。 | |||
TN6771 |
Malabaricone B
|
Others | Others |
Malabaricone B 是一种源自香料的酚类物质,它通过不依赖 p53 的途径诱导肺癌细胞中的线粒体损伤。 | |||
T2961 |
Notoginsenoside R1
Sanqi glucoside R1,Sanchinoside R1,三七皂苷R1 |
Apoptosis; ERK; Beta Amyloid | Apoptosis; MAPK; Neuroscience |
Notoginsenoside R1 (Sanchinoside R1) 是一种从三七中分离出来的皂苷,具有抗氧化、抗炎、抗血管生成和抗凋亡的活性。它有神经保护和抗缺血/再灌注损伤的心脏保护作用。 | |||
T5S2076 |
Senkyunolide I
|
Others; Caspase | Apoptosis; Others; Proteases/Proteasome |
Senkyunolide I 是从川芎中分离得到的一种天然产物,具有神经保护作用,与其抗氧化和抗凋亡特性有关。 | |||
T3376 |
Cynaroside
朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside |
Others; Influenza Virus; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Cynaroside (Luteolin 7-O-Glucoside) 是一个抗氧化类黄酮。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 32 nM。 | |||
T8160 |
EGCG Octaacetate
乙酰化表没食子儿茶素没食子酸酯,乙酰化EGCG |
Others; Antibacterial | Microbiology/Virology; Others |
EGCG Octaacetate 是表没食子儿茶素没食子酸酯的前药,对革兰氏阳性菌和革兰氏阴性菌有潜在抗菌可能。它可下调 PI3K/Akt/NFκB 磷酸化和 p65 乙酰化来降低促炎介质水平,减少小鼠结肠炎引起的结肠癌。 | |||
T6S1930 |
Schisanhenol
五味子酚,Schizanhenol,Gomisin-K3 |
Antioxidant | oxidation-reduction |
Schisanhenol (Schizanhenol) 是一种UGT2B7的抑制剂,是一种天然化合物。 | |||
T5S1172 |
Tiliroside
银椴甙,Tribuloside,银椴苷;椴树苷 |
Antioxidant | oxidation-reduction |
Tiliroside (Tribuloside) 是糖苷类黄酮,是 α-淀粉酶的非竞争性抑制剂(Ki:84.2 μM)。它抑制胃肠道中碳水化合物的消化和葡萄糖的吸收,具有抗糖尿病作用。 | |||
TL0009 |
coniferin
Coniferoside,松柏苷,Abietin |
Others; Antifungal | Microbiology/Virology; Others |
Coniferin (Abietin) 是一种松柏醇中的葡萄糖苷。它抑制真菌生长和黑化反应,具有 ATP 依赖性转运活性并具有抗氧化作用。 | |||
T3822 |
Bellidifolin
Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮 |
Others; HIV Protease | Microbiology/Virology; Others; Proteases/Proteasome |
Bellidifolin (Bellidifoline) 是从獐牙菜的茎中提取的一种呫吨酮,它能作为病毒蛋白 R 的抑制剂,具有保肝、降血糖、抗炎、抗氧化、抗肿瘤作用。 | |||
TN1962 |
Myricetin 3-O-galactoside
Myricetin 3-O-beta-D-galactopyranoside |
NOS; Xanthine Oxidase | Immunology/Inflammation; Metabolism |
Myricetin 3-O-galactoside (Myricetin 3-O-beta-D-galactopyranoside) 可抑制黄嘌呤氧化酶 (xanthine oxidase; XO) 活性,脂质过氧化并清除自由基。杨梅素3- o -半乳糖苷具有很多作用包括细胞毒性、抗氧化、抗基因毒性、抗感染性、抗炎作用和抗氧化活性,其主要作用是抑制诱导型一氧化氮合酶(iNOS)的合成。Myricetin 3-O-galactoside 抑制脂质过氧化的 IC50 为 160 μg/mL。 | |||
TN7229 |
Baihuaqianhuoside
Praeroside |
Others | Others |
Baihuaqianhuoside (Praeroside) 是一种香豆素苷。Baihuaqianhuoside 可以从西番莲和 Hindenia solanacea 的根部分离出来,是首次从 P. japonicum 身上分离出来的。Baihuaqianhuoside 在体外具有抗炎活性,可以用于炎症的研究。Baihuaqianhuoside 对1,1-二苯基-2-丙烯酰肼自由基的清除作用,以及对2,2'-偶氮双(2-脒基丙烷)二盐酸盐诱导的脂质体氧化的抑制作用。 | |||
TN5904 | 1,3,7-Trihydroxy-2-methoxyxanthone | ||
1,3,7-Trihydroxy-2-methoxyxanthone shows different anti-oxidation activities. | |||
TN1618 | Erigeroside | Others | Others |
Erigeroside has the protective effects on cerebral ischemia-reperfusion injury in rat, its ability of anti-oxidation and scavenging oxidation free radical may be one of its protective mechanisms. | |||
TN2367 |
Cyanidin 3-arabinoside
矢车菊素-3-阿拉伯糖苷,Cyanidin 3-monoarabinoside |
Others | Others |
Cyanidin 3-monoarabinoside has anti-oxidation and anti-tumor effects. | |||
TN3517 | Bisacurone | IL Receptor; IκB/IKK; TNF; NF-κB; ROS; Akt; PKC | Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; NF-κB; PI3K/Akt/mTOR signaling |
Bisacurone has anti-oxidant, anti-inflammatory, and anti-metastatic activities, it may have a protective effect against ethanol-induced liver injury by suppressing hepatic oxidation and inflammation. | |||
TN4589 |
Mulberrofuran K
|
Others | Others |
Mulberrofuran K shows potent anti-oxidation activities. | |||
TN4956 |
Scandoside
|
NF-κB; MAPK | MAPK; NF-κB |
Scandoside exerts anti-inflammatory effect via suppressing NF-κB and MAPK signaling pathways in LPS-induced RAW 264.7 macrophages.It also inhibits LDL-oxidation. | |||
TN6515 |
Selaginellin
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Selaginellin has a neuroprotective effect against L-glutamate-induced neurotoxicity through mechanisms related to anti-oxidation and anti-apoptosis via scavenging reactive oxygen species and up-regulating the expression of klotho gene. Selaginellin shows | |||
T4484 | 1,7-Dihydroxy-2,3-methylenedioxyxanthone | Prostaglandin Receptor; Antifection | GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology |
1,7-Dihydroxy-2,3-methylenedioxyxanthone has antiulcerogenic, anti-oxidation, and antihyperalgesic activities, it can inhibit the carrageenan-induced hyperalgesia. | |||
T2S1797 |
Santalol
檀香醇;白檀油萜醇;檀香脑,檀香醇 |
Antioxidant; Antifungal | Microbiology/Virology; oxidation-reduction |
Santalol 是一种檀香醇的 α 和 β-异构体混合物。 其中α-santalol 分离自檀香油中,是一种有前途的抗癌药,能够预防口腔癌、前列腺癌、乳腺癌和皮肤癌。 | |||
TN3725 |
Cucurbitadienol
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Cucurbitadienol has significant anti-inflammatory, anti-tumor effect, is also CucurbitacinBE compounds biosynthesis the key intermediate. Cucurbitadienol synthase, the first committed enzyme for cucurbitacin biosynthesis, is a distinct enzyme from cycloar | |||
T72508 | Palmatine hydroxide | ||
Palmatine hydroxide 是不可逆的口服活性IDO-1抑制剂,其对HEK 293-hIDO-1 和 rhIDO-1的IC50值分别为3 μM和157 μM。该化合物还能非竞争性抑制(WNV)NS2B-NS3蛋白酶,IC50值为96 μM。Palmatine hydroxide展现了抗癌、抗炎、神经保护、抗细菌和抗病毒的活性。 |