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Cat. No. Product Name Target Signaling Pathways
T0029 Procaine

Duracaine,Spinocaine,普鲁卡因,Novocaine,Vitamin H3,奴夫卡因

Histone Demethylase; DNA/RNA Synthesis; Sodium Channel Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Membrane transporter/Ion channel
Procaine (Vitamin H3) 是DNA 脱甲基剂,是一种酯类局部麻醉剂。它起效缓慢,作用持续时间短,主要用于浸润麻醉、周围神经阻滞和脊髓阻滞。
T0802 Procaine hydrochloride

Novocaine HCl,Procaine HCl,盐酸普鲁卡因

Histone Demethylase; 5-HT Receptor; DNA/RNA Synthesis; Sodium Channel; NMDAR; AChR Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Procaine hydrochloride (Novocaine HCl) 是DNA 脱甲基剂,是一种苯甲酸衍生物,具有局部麻醉和抗心律失常特性。
T4553 Procaine penicillin G

普鲁卡因青霉素,Duphapen,Hydracillin,Hostacillin

Antibiotic Microbiology/Virology
Procaine penicillin G (Duphapen) 是一种抗生素,可用于治疗多种细菌感染。具体来说,它用于梅毒、炭疽、口腔感染、肺炎、白喉、蜂窝组织炎和动物咬伤。
T69027 Procaine merethoxylline

Procaine merethoxylline is a noted sodium channel blocker with a variety of inhibitory effects.
T16466 Penicillin G Procaine

PGP

Others Others
Penicillin G Procaine is a β-lactam antibiotic and is a crystalline complex produced by chemically combining penicillin G with procaine.
T6443 Chloroprocaine hydrochloride

盐酸氯普鲁卡因,Chloroprocaine HCl

ATPase; Others Membrane transporter/Ion channel; Others
Chloroprocaine hydrochloride (Chloroprocaine HCl) 是一种 Na/K-ATPase 活性抑制剂,IC50为 13 mM,可阻断外周神经。
T0378 Oxybuprocaine hydrochloride

Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐

Sodium Channel Membrane transporter/Ion channel
Oxybuprocaine hydrochloride (Oxybuprocaine HCl) 是可逆的钠通道阻断剂,可防止角膜,结膜和巩膜中疼痛神经的冲动传播。Oxybuprocaine hydrochloride 专用于眼科与耳鼻喉科。
T60469 Chloroprocaine

Chloroprocaine (2-Chloroprocaine) 是一种有效的Na,K-ATPase 酶活性抑制剂(IC50 = 13 mM)。Chloroprocaine 是一种阻滞外周神经的局部麻醉剂。
T0378L Oxybuprocaine

Butoxyprocaine,BNX,Benoxinate,Novescine,Novesin

Oxybuprocaine is an ester-type local anesthetic that is used especially in ophthalmology and otolaryngology. Oxybuprocaine binds to sodium channels and reversibly stabilizes the neuronal membrane which decreases its permeability to sodium ions.
T0018 Procainamide hydrochloride

Procapan,Procainamide HCl,Pronestyl,Procanbid,盐酸普鲁卡因胺

DNA Methyltransferase; Sodium Channel; AChR; Autophagy Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Neuroscience
Procainamide hydrochloride (Procapan) 是一种用于研究心律失常的抗心律失常制剂。
T1144 Lidocaine hydrochloride

Lidocaine HCL,盐酸利多卡因,Lignocaine hydrochloride,Xyloneural,Lidothesin

Apoptosis; ERK; NF-κB; MEK; Sodium Channel Apoptosis; MAPK; Membrane transporter/Ion channel; NF-κB
Lidocaine hydrochloride (Lignocaine hydrochloride) 抑制涉及复杂电压和依赖性的钠通道。它通过调节 miR-145 表达和进一步抑制 MEK/ERK 和 NF-κB 信号通路来减少胃癌细胞的生长,迁移和侵袭。Lidocaine 是一种酰胺衍生物,是一种研究室性心律失常的药物和有效的肿瘤抑制剂。
T60513 NMDA-IN-2

NMDA-IN-2 (化合物 6b) 是普鲁卡因的衍生物。NMDA-IN-2是 NMDA 受体2B 亚型的抑制剂。

化合物

Procaine
Cat.No: T0029
Synonym: Duracaine,Spinocaine,普鲁卡因,Novocaine,Vitamin H3,奴夫卡因
Target: Histone Demethylase, DNA/RNA Synthesis, Sodium Channel
Procaine hydrochloride
Cat.No: T0802
Synonym: Novocaine HCl,Procaine HCl,盐酸普鲁卡因
Target: Histone Demethylase, 5-HT Receptor, DNA/RNA Synthesis, Sodium Channel, NMDAR, AChR
Procaine penicillin G
Cat.No: T4553
Synonym: 普鲁卡因青霉素,Duphapen,Hydracillin,Hostacillin
Target: Antibiotic
Procaine merethoxylline
Cat.No: T69027
Synonym:
Target:
Penicillin G Procaine
Cat.No: T16466
Synonym: PGP
Target: Others
Chloroprocaine hydrochloride
Cat.No: T6443
Synonym: 盐酸氯普鲁卡因,Chloroprocaine HCl
Target: ATPase, Others
Oxybuprocaine hydrochloride
Cat.No: T0378
Synonym: Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐
Target: Sodium Channel
Chloroprocaine
Cat.No: T60469
Synonym:
Target:
Oxybuprocaine
Cat.No: T0378L
Synonym: Butoxyprocaine,BNX,Benoxinate,Novescine,Novesin
Target:
Procainamide hydrochloride
Cat.No: T0018
Synonym: Procapan,Procainamide HCl,Pronestyl,Procanbid,盐酸普鲁卡因胺
Target: DNA Methyltransferase, Sodium Channel, AChR, Autophagy
Lidocaine hydrochloride
Cat.No: T1144
Synonym: Lidocaine HCL,盐酸利多卡因,Lignocaine hydrochloride,Xyloneural,Lidothesin
Target: Apoptosis, ERK, NF-κB, MEK, Sodium Channel
NMDA-IN-2
Cat.No: T60513
Synonym:
Target:
TargetMol Loading
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