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抑制剂 & 化合物

29

天然产物

6

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T126550 1-O-β-D-Glucopyranosylpaeonisuffrone

1-O-β-D-Glucopyranosylpaeonisuffrone 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126550。
T11153 EG00229

Others Others
EG00229 selectively inhibits VEGF-A binding to NRP1 b1 domain with an IC50 of 3 μM, but has no effect on VEGFA binding to VEGFR-1 and VEGFR-2. EG00229 is a neuropilin 1 (NRP1) receptor antagonist.

化合物

1-O-β-D-Glucopyranosylpaeonisuffrone
Cat.No: T126550
Synonym:
Target:
EG00229
Cat.No: T11153
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T6S1657 Paeonolide

Others Others
Paeonolide 是一种广泛存在于 Paeonia 属植物根中的植物糖苷,含有一个非还原性末端 α-1-阿拉伯吡喃糖苷。
T3773 Oxypaeoniflorin

氧化芍药苷,Oxypaeoniflora

Others Others
Oxypaeoniflorin (Oxypaeoniflora) 从 Paeoniae 中分离得到的单萜糖苷化合物,是一种抗氧化剂,是具有神经保护和抗炎作用。
TN1698 Glucotropaeolin potassium

金莲葡糖硫苷钾盐,Glucotropaeolin,Benzylglucosinolate potassium,Glucotropaeolin Potassium Salt

Others Others
Glucotropaeolin potassium (Benzylglucosinolate potassium) 存在于十字花科蔬菜中,并且 可适度减少动物的自发性DNA 损伤。
TN6926 Paeonoside

Others Others
Paeonoside 发现与P. suffruticosa 中,具有生物活性,可以促进成骨细胞分化过程中的伤口愈合和迁移。Paeonoside 具有一定的抗糖尿病活性,可防止脓毒症和败血症引起的死亡。Paeonoside 对 MC3T3-E1细胞的前成骨细胞没有细胞毒性作用,以剂量依赖性的方式显著恢复伤口区域并促进细胞迁移和促进碱性磷酸酶(ALP)染色及其活性。
T3S0870 Paederosidic acid methyl ester

鸡屎藤苷酸甲酯,紫草酸甲酯

ATPase; Potassium Channel; NO Synthase Immunology/Inflammation; Membrane transporter/Ion channel
Paederosidic acid methyl ester 是 ATP 敏感的 K+channel 通道激活剂,分离自 P. scandens。它通过激活脑中和脊髓水平中 ATP 敏感型 K+通道提高了痛觉阈值,表现出显著的中枢缓解疼痛活性。
T5739 Paederosidic acid

鸡屎藤苷酸,异戊二酸 紫草酸

Apoptosis; BCL Apoptosis
Paederosidic acid 是从鸡矢藤分离出的一种天然产物,通过诱导线粒体介导的凋亡抑制肺癌细胞,具有显着的抗肿瘤、抗惊厥和镇静作用。
TN1067 Galloylpaeoniflorin

6'-O-Galloyl paeoniflorin,没食子酰芍药苷

NF-κB; Androgen Receptor; ROS Endocrinology/Hormones; Immunology/Inflammation; NF-κB
Galloylpaeoniflorin (6'-O-Galloyl paeoniflorin) 是 NF-κB 抑制剂,同时也是 DNA 裂解抑制剂。
T6S1652 Benzoylpaeoniflorin

COX Immunology/Inflammation; Neuroscience
Benzoylpaeoniflorin 是一种从白芍中提取的天然化合物,可以降低细胞凋亡,对冠心病具有潜在的研究价值。
T4S1658 Benzoyloxypaeoniflorin

苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷

NF-κB; Tyrosinase NF-κB; Proteases/Proteasome
Benzoyloxypaeoniflorin (Benzoyloxypeoniflorin) 是一种酪氨酸酶抑制剂,分离于Paeonia suffruticosa 的根,对mushroom tyrosinase 的 IC50为 0.453 mM。它是一种NF-κB 抑制剂,它通过对血小板聚集和凝血的抑制作用,有助于改善血液循环。
T2230 Paeoniflorin

芍药苷,Peoniflorin

HSP; COX Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; Neuroscience
Paeoniflorin (Peoniflorin) 是从芍药根中提取的一种蒎烷单萜糖苷,具有抗癌作用、抗氧化应激、抗血小板聚集、血管扩张、降低血液粘度和抗炎活性等多种生物活性。它是一种热休克蛋白诱导剂,通过自噬途径保护 PC12 细胞免受 MPP+和酸性损伤。
T5S1645 Apiopaeonoside

丹皮酚新苷

Others Others
Apiopaeonoside 是一种天然产物,分离自Paeonia suffruticosa 根部。
T2900 Paeonol

丹皮酚,Peonol

MAO; Autophagy; Monoamine Oxidase Autophagy; Metabolism; Neuroscience
Paeonol (Peonol) 是一种从牡丹中提取的活性物质,可抑制 MAO-A 和 MAO-B,IC50 分别为 54.6 μM 和 42.5 μM。
T3S0872 Paederoside

Antiviral; HBV Immunology/Inflammation; Microbiology/Virology
Paederoside 是从Paederia pertomentosa 分离的一种单萜 S-甲基硫代碳酸酯。它抑制 Epstein-Barr 病毒的激活,有抗肿瘤促进作用。
T78469 α-Copaene

α-Copaene,一种倍半萜烃,具有水果挥发物性质,可作为橄榄实蝇(Bactrocera oleae)的产卵促进剂。
TN5855 2'-O-Benzoylpaeoniflorin

2'-O-Benzoylpaeoniflorin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5855,CAS号为 1456598-64-3。
TN2037 Paeonilactone C

(3S,3AR,6S,7AR)-3-[(苯甲酰基氧基)甲基]四氢-6-羟基-6-甲基-2,5(3H,4H)-苯并呋喃二酮,芍药内苷 C

Others Others
Paeonilactone C significantly protects primary cultures of rat cortical cells against H2O2-induced neurotoxicity.
TN5857 Debenzoylgalloylpaeoniflorin

Debenzoylgalloylpaeoniflorin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5857,CAS号为 262350-51-6。
TN2035 Paeonilactone A

(3R,3AR,6S,7AR)-四氢-6-羟基-3,6-二甲基-2,5(3H,4H)-苯并呋喃二酮,芍药内苷A

Others Others
Paeonilactone A是一种天然产物,属于芍药科芍药属,其产品编号为 TN2035,CAS号为 98751-79-2。Paeonilactone A可用作对照参考。
T83310 4-O-Methyldebenzoylpaeoniflorin

4-O-Methyldebenzoylpaeoniflorin为自Paeonia albiflora提取的自然化合物。
T75455 Paecilomide

Paecilomide,吡啶酮生物碱,是一种乙酰胆碱酯酶 (acetylcholinesterase) 抑制剂。
T38524 Paeoniflorin sulfite

During the sulfur-fumigation process of Paeoniae Radix Alba, Paeoniflorin, which serves as a principal constituent, can be converted into Paeoniflorin sulfite.
T82594 Debenzoylpaeoniflorgenin

Debenzoylpaeoniflorgenin是从Paeonia lactiflora中分离得到的天然化合物,该植物是Guizhitang的一个组成成份。
TN2416 8-Debenzoylpaeoniflorin

Others Others
8-Debenzoylpaeoniflorin is a natural product from plants
T37962 Paeoniflorgenin

Paeoniflorgenin is a deglucosylated metabolite of Paeoniflorin[1]. [1]. Hsiu SL, et, al. A deglucosylated metabolite of paeoniflorin of the root of Paeonia lactiflora and its pharmacokinetics in rats. Planta Med. 2003 Dec; 69(12): 1113-8.
TN2036 Paeonilactone B

(+)-Paeonilactone B

NADPH-oxidase Immunology/Inflammation
Paeonilactone B ((+)-Paeonilactone B) 是一种来自白芍的单萜类化合物,具有神经保护活性,抑制氧化应激,在大鼠皮质细胞在抑制 H2O2 诱导的神经毒性。
T81570 Paecilaminol

FKI-0550

Paecilaminol (FKI-0550) 为一种高效的 NADH 富马酸还原酶 (NADH-fumarate reductase) 抑制剂,其对蛔虫 (Ascaris suum) NADH 富马酸还原酶展现了 5.1 μM 的 IC50 值。
T82028 Isomaltopaeoniflorin

Isomaltopaeoniflorin为舒郁中草药配方的代谢产物,该配方用以抑制抑郁症样疾病。
TN2034 Paeoniflorigenone

Others; Caspase Apoptosis; Others; Proteases/Proteasome
Paeoniflorigenone is a depolarizing neuromuscular blocking agent, being similar to succinylcholine.
T5603 Phthalic acid

邻苯二甲酸,1,2-Benzenedioic acid

Others Others
Phthalic acid (1,2-Benzenedioic acid) 是一种邻苯二甲酸酯 (PAE) 的最终常见代谢形式。它可用于合成试剂,如间苯二甲酸 (IPA) 和对苯二甲酸 (TPA)。它广泛的用于邻苯二甲酸酯增塑剂的制备。

天然产物

Paeonolide
Cat.No: T6S1657
Synonym:
Target: Others
Oxypaeoniflorin
Cat.No: T3773
Synonym: 氧化芍药苷,Oxypaeoniflora
Target: Others
Glucotropaeolin potassium
Cat.No: TN1698
Synonym: 金莲葡糖硫苷钾盐,Glucotropaeolin,Benzylglucosinolate potassium,Glucotropaeolin Potassium Salt
Target: Others
Paeonoside
Cat.No: TN6926
Synonym:
Target: Others
Paederosidic acid methyl ester
Cat.No: T3S0870
Synonym: 鸡屎藤苷酸甲酯,紫草酸甲酯
Target: ATPase, Potassium Channel, NO Synthase
Paederosidic acid
Cat.No: T5739
Synonym: 鸡屎藤苷酸,异戊二酸 紫草酸
Target: Apoptosis, BCL
Galloylpaeoniflorin
Cat.No: TN1067
Synonym: 6'-O-Galloyl paeoniflorin,没食子酰芍药苷
Target: NF-κB, Androgen Receptor, ROS
Benzoylpaeoniflorin
Cat.No: T6S1652
Synonym:
Target: COX
Benzoyloxypaeoniflorin
Cat.No: T4S1658
Synonym: 苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷
Target: NF-κB, Tyrosinase
Paeoniflorin
Cat.No: T2230
Synonym: 芍药苷,Peoniflorin
Target: HSP, COX
Apiopaeonoside
Cat.No: T5S1645
Synonym: 丹皮酚新苷
Target: Others
Paeonol
Cat.No: T2900
Synonym: 丹皮酚,Peonol
Target: MAO, Autophagy, Monoamine Oxidase
Paederoside
Cat.No: T3S0872
Synonym:
Target: Antiviral, HBV
α-Copaene
Cat.No: T78469
Synonym:
Target:
2'-O-Benzoylpaeoniflorin
Cat.No: TN5855
Synonym:
Target:
Paeonilactone C
Cat.No: TN2037
Synonym: (3S,3AR,6S,7AR)-3-[(苯甲酰基氧基)甲基]四氢-6-羟基-6-甲基-2,5(3H,4H)-苯并呋喃二酮,芍药内苷 C
Target: Others
Debenzoylgalloylpaeoniflorin
Cat.No: TN5857
Synonym:
Target:
Paeonilactone A
Cat.No: TN2035
Synonym: (3R,3AR,6S,7AR)-四氢-6-羟基-3,6-二甲基-2,5(3H,4H)-苯并呋喃二酮,芍药内苷A
Target: Others
4-O-Methyldebenzoylpaeoniflorin
Cat.No: T83310
Synonym:
Target:
Paecilomide
Cat.No: T75455
Synonym:
Target:
Paeoniflorin sulfite
Cat.No: T38524
Synonym:
Target:
Debenzoylpaeoniflorgenin
Cat.No: T82594
Synonym:
Target:
8-Debenzoylpaeoniflorin
Cat.No: TN2416
Synonym:
Target: Others
Paeoniflorgenin
Cat.No: T37962
Synonym:
Target:
Paeonilactone B
Cat.No: TN2036
Synonym: (+)-Paeonilactone B
Target: NADPH-oxidase
Paecilaminol
Cat.No: T81570
Synonym: FKI-0550
Target:
Isomaltopaeoniflorin
Cat.No: T82028
Synonym:
Target:
Paeoniflorigenone
Cat.No: TN2034
Synonym:
Target: Others, Caspase
Phthalic acid
Cat.No: T5603
Synonym: 邻苯二甲酸,1,2-Benzenedioic acid
Target: Others
Cat. No. Product Name Species Expression System
TMPH-03166 Elastase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)

PAE,lasB,Pseudolysin,Neutral metalloproteinase,Elas...

Pseudomonas aeruginosa E. coli
Cleaves host elastin, collagen, IgG, and several complement components as well as endogenous pro-aminopeptidase. Autocatalyses processing of its pro-peptide. Processes the pro-peptide of pro-chitin-binding protein (cbpD). Involved in the pathogenesis of P.aeruginosa infections. Elastase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 49.1 kDa and the accession number is P14756.
TMPH-03080 Sialidase Protein, Paeniclostridium sordellii, Recombinant (hFc & Myc)

Paeniclostridium sordellii HEK293 Cells
Sialidases have been suggested to be pathogenic factors in microbial infections. Sialidase Protein, Paeniclostridium sordellii, Recombinant (hFc & Myc) is expressed in HEK293 mammalian cells with C-hFC-Myc tag. The predicted molecular weight is 70.7 kDa and the accession number is P15698.
TMPH-03067 Ole e 7 Protein, Olea europaea, Recombinant (GST)

Olea europaea E. coli
Ole e 7 Protein, Olea europaea, Recombinant (GST) is expressed in E. coli.
TMPH-03079 Sialidase Protein, Paeniclostridium sordellii, Recombinant (His & Myc)

Paeniclostridium sordellii E. coli
Sialidases have been suggested to be pathogenic factors in microbial infections. Sialidase Protein, Paeniclostridium sordellii, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 49.2 kDa and the accession number is P15698.
TMPH-03078 CGTases Protein, Paenibacillus macerans, Recombinant (His)

Cyclodextrin-glycosyltransferase,CGTase,Cyclomaltodextrin gl...

Bacillus macerans P. pastoris (Yeast)
CGTases Protein, Paenibacillus macerans, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 13.4 kDa and the accession number is P31835.
TMPH-03077 CGTases Protein, Paenibacillus macerans, Recombinant (E. coli, His)

CGTase,Cyclomaltodextrin glucanotransferase,Cyclodextrin-gly...

Paenibacillus macerans E. coli
N/A. CGTases Protein, Paenibacillus macerans, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 15.4 kDa and the accession number is P31835.

重组蛋白

Elastase Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
Cat.No: TMPH-03166
Species: Pseudomonas aeruginosa
Expression System: E. coli
Sialidase Protein, Paeniclostridium sordellii, Recombinant (hFc & Myc)
Cat.No: TMPH-03080
Species: Paeniclostridium sordellii
Expression System: HEK293 Cells
Ole e 7 Protein, Olea europaea, Recombinant (GST)
Cat.No: TMPH-03067
Species: Olea europaea
Expression System: E. coli
Sialidase Protein, Paeniclostridium sordellii, Recombinant (His & Myc)
Cat.No: TMPH-03079
Species: Paeniclostridium sordellii
Expression System: E. coli
CGTases Protein, Paenibacillus macerans, Recombinant (His)
Cat.No: TMPH-03078
Species: Bacillus macerans
Expression System: P. pastoris (Yeast)
CGTases Protein, Paenibacillus macerans, Recombinant (E. coli, His)
Cat.No: TMPH-03077
Species: Paenibacillus macerans
Expression System: E. coli
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