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Search Results for " neurodevelopmental "

6

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T12421 PF-04885614

Sodium Channel Membrane transporter/Ion channel
PF-04885614是一种有效的NaV1.8抑制剂。PF-04885614有用于神经系统疾病和神经发育疾病研究的潜力。
T77565 Fluparoxan hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Fluparoxan hydrochloride 是一种高度选择性和有效的α2-肾上腺素受体拮抗剂,可用于预防、改善或治疗神经发育障碍和神经退行性疾病。
T77566 (3aR,9aR)-Fluparoxan

Adrenergic Receptor GPCR/G Protein; Neuroscience
(3aR,9aR)-Fluparoxan 是一种高度选择性和有效的肾上腺素能受体α2B 拮抗剂,可用于预防、改善或治疗神经发育障碍和神经退行性疾病。
T39252 TAK-418

Histone Demethylase Chromatin/Epigenetic
TAK-418 是一种选择性、口服活性 LSD1/KDM1A 酶抑制剂,IC50 为 2.9 nM。TAK-418 能解锁异常表观遗传机制,改善神经发育障碍模型中的自闭症症状。
T39940 Plazinemdor

Plazinemdor is an NMDA receptor positive allosteric modulator with potential applications in psychiatric, neurological, neurodevelopmental disorders, and diseases of the nervous system.
T74649 Rugonersen

Rugonersen (RG6091; RO7248824) 是一种通过锁定核酸 (LNA) 技术修饰的反义寡核苷酸 (ASOs),目的在于降低泛素蛋白连接酶 E3A (UBE3A) 的沉默。它被用于研究由于神经元 E3 连接酶 UBE3A 缺失所导致的严重神经发育障碍——Angelman 综合征 (AS)。

化合物

PF-04885614
Cat.No: T12421
Synonym:
Target: Sodium Channel
Fluparoxan hydrochloride
Cat.No: T77565
Synonym:
Target: Adrenergic Receptor
(3aR,9aR)-Fluparoxan
Cat.No: T77566
Synonym:
Target: Adrenergic Receptor
TAK-418
Cat.No: T39252
Synonym:
Target: Histone Demethylase
Plazinemdor
Cat.No: T39940
Synonym:
Target:
Rugonersen
Cat.No: T74649
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2775 2-Methoxystypandrone

MMP; BCL; IκB/IKK; GSK-3; TNF; NOS; NF-κB; Wnt/beta-catenin; COX; JAK; STAT Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; JAK/STAT signaling; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
2-Methoxystypandrone displays an immunomodulatory effect in a cellular model, it blocks inflammatory responses by impairing NF-κB signaling to limit the inflammation and oxidative stress for preservation of BBB integrity. 2-Methoxystypandrone concomitant

天然产物

2-Methoxystypandrone
Cat.No: TN2775
Synonym:
Target: MMP, BCL, IκB/IKK, GSK-3, TNF, NOS, NF-κB, Wnt/beta-catenin, COX, JAK, STAT
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