Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T19714 |
Fenpyroximate
|
Others | Others |
Fenpyroximate 是一种有效的杀螨剂。 | |||
T2180 |
Hexythiazox
|
Parasite | Microbiology/Virology |
Hexythiazox 是一种螨类生长调节剂和噻唑烷类杀螨剂,对多种螨类具有长效杀虫作用,适用于植物从萌芽到结果的任何生长阶段。 | |||
T13536 |
Afoxolaner
|
Chloride channel; GABA Receptor; Parasite | Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience |
Afoxolaner 是一种异恶唑啉杀虫剂/杀螨剂,可对抗犬的肩胛硬蜱。 它作用于昆虫的 γ-氨基丁酸(GABA)受体谷氨酸受体,抑制 GABA 和谷氨酸调节的氯离子吸收,导致过度的神经元刺激和节肢动物死亡。 | |||
T27794 |
λ-Cyhalothrin
lambda-Cyhalothrin,Karate,λ-氯氟氰菊酯,Icon |
Sodium Channel; Parasite | Membrane transporter/Ion channel; Microbiology/Virology |
λ-Cyhalothrin (Icon) 是广谱的 II 型合成除虫菊酯杀虫剂,含有 α-氰基,用于防治多种害虫。它是一种钠通道神经毒素,靶向中枢神经系统中神经元膜。 | |||
T14571 |
Bifenazate
|
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
Bifenazate 是 GABA 受体的正向变构调节剂。 Bifenazate 是一种杀螨剂,可在 25 ppm 的浓度下控制 100% 的螨虫。 | |||
T4446 |
Tebufenpyrad
Pyranica,吡螨胺,MK239,Comanche |
Mitochondrial Metabolism | Metabolism |
Tebufenpyrad (Comanche) 是一种重要的农业化学杀螨剂,其作用类似于已知的线粒体毒物 rotenone。 | |||
T5839 |
Phosalone
|
Parasite | Microbiology/Virology |
Phosalone 是一种有机磷酸盐化学品,通常用作杀虫剂和杀螨剂。 | |||
T3493 |
Clofentezine
Bisclofentazin,Acaristop,Apollo,四螨嗪 |
Others | Others |
Clofentezine (Apollo) 是生长抑制剂,对螨虫具有显著的致死作用。 | |||
T7075 |
2-Chloronaphthoquinone
2-Chloro-1,4-naphthoquinone,2-氯-1,4-萘醌 |
Others | Others |
2-Chloronaphthoquinone (2-Chloro-1,4-naphthoquinone) 是一种取代的萘醌,用作杀虫剂和杀螨剂。 | |||
T1632 |
Amitraz
BTS-27419,NSC 324552,双甲脒 |
Adrenergic Receptor; Parasite; Monoamine Oxidase | GPCR/G Protein; Microbiology/Virology; Neuroscience |
Amitraz (NSC 324552) 是一种非系统性杀螨剂和杀虫剂,,可治疗犬蠕形螨。它具有α-肾上腺素能激动剂活性, 与中枢神经系统的章鱼胺受体相互作用, 抑制单胺氧化酶和前列腺素合成。 | |||
T2479 |
Tyrphostin A9
Malonoben,Tyrphostin 9,SF 6847,AG 17,RG-50872 |
EGFR; VEGFR; Influenza Virus; PDGFR | Angiogenesis; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Tyrphostin A9 (SF 6847) 是一种线粒体分裂诱导剂,是 PDGFR 抑制剂,具有抗流感病毒的活性。 | |||
T4055 |
Etoxazole
|
Others | Others |
Etoxazole 是一种杀螨剂/杀虫剂,通过抑制几丁质生物合成来控制螨虫。用作农药检测的标准。 | |||
T12987 |
Spirodiclofen
BAJ-2740,螺螨酯 |
Parasite | Microbiology/Virology |
Spirodiclofen (BAJ-2740) 是选择性非系统性的杀螨剂,来自新的化学类特酮酸衍生物, 与目前市面上的杀螨剂无交叉耐药, 具有额外的杀虫性能。 | |||
T5114 |
Pyridaben
|
Calcium Channel; Parasite | Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Pyridaben 是一种METI 杀螨剂,可抑制复合物 I 处的线粒体电子转运。它对多种螨虫具有活性,通过滤纸接触给药,在 25 mg/mL、100 mg/mL 和 200 mg/mL 的剂量下,分别诱导 100% 的C. malaccensis,D. farina 和T. putrescentia 死亡率。 | |||
T20539 |
Pirimiphos-methyl
R 33986,甲基嘧啶磷,AI3-27699,Caswell No. 334B,PP511,Actelic |
AChE; Parasite | Microbiology/Virology; Neuroscience |
Pirimiphos-methyl (AI3-27699) 是一种速效有机磷杀虫剂和杀螨剂,对目标生物的乙酰胆碱酯酶有抑制作用。甲基嘧啶磷常用于农粮贮藏过程中甲虫、鼻甲虫、飞蛾和蝽蛄的防治。 | |||
T28397 |
Phenaglycodol
Atadiol,Felixin,Puasital,Sedapsin,Acalmid |
||
Chlordimeform Hydrochloride is an acaricide. | |||
T20487 | Sulphenone | ||
Sulphenone is an agent of Acaricide. | |||
T31377 |
Demiditraz
PF 3814927,PF-3814927,PF3814927 |
||
Demiditraz(PF-3814927) is an acaricide (veterinary use). | |||
T21464 |
Methiocarb
Mercaptodimethur,Mesurol |
||
Methiocarb, a carbamate pesticide, is used as an insecticide, acaricide, bird repellent, and molluscicide. Methiocarb stimulates cholinergic by inhibiting reversibly acetylcholinesterase activity, making methiocarb a potent neurotoxin. | |||
T25241 | Chlorbenside | ||
Chlorbenside is a pesticide, also known as chlorparaside and chlorsulfacide, which is most commonly used as an acaricide being used to kill mites and ticks. | |||
T20559 |
Tetradifon
Roztoczol,Roztoczol extra,Roztozol,三氯杀螨砜 |
||
Tetradifon is a contact acaricide. | |||
T20729 |
Vamidothion
RP9895,Kilval,Trucidor,RP-9895,RP 10465,RP 9895 |
||
Vamidothion is a polar organophosphorus insecticide and acaricide | |||
T19847 |
Benzoximate
Citrazon |
||
Benzoximate is an insecticide and acaricide. | |||
T20139 |
Butocarboxim
CO 755,Drawin 755 |
||
Butocarboxime is used as an insecticide and acaricide. | |||
T25427 |
Fluenetil
TH 367-1,M2060,M 2060,M-2060,Caswell No. 462A |
||
Fluenetil, a biphenyl compound, is an acaricide introduced in 1965 by Montedison. | |||
T69570 |
Banamite
|
||
Banamite is an acaricide & monoamine oxidase inhibitor. | |||
T73723 |
Bifenazate-diazene
|
||
Bifenazate-diazene 是 Bifenazate 的主要降解产物。Bifenazate 是一种选择性杀螨剂和杀虫剂。 | |||
T25002 |
Acrinathrin
RU38702,Rufast,RU 38702,RU-38702 |
||
Acrinathrin is a pyrethroid used as an insecticide and an acaricide. Although resistance is developing, Acrinathrin is used to control the mite Varroa jacobsoni in beekeeping. | |||
T35419 |
τ-Fluvalinate
|
||
τ-Fluvalinate is a pyrethroid acaricide.1It induces tail currents in Western honeybee (A. mellifera) voltage-gated sodium channels (AmNav1) expressed inXenopusoocytes (EC50= 60 nM). It also induces tail currents in honeybee parasitic Varroa mite (V. destructor) Nav1 channels (VdNav1) expressed inXenopusoocytes (EC50= 160 nM) with a faster tail current decay than that of AmNav1 channels. Topical application of τ-fluvalinate (2 μl) in combination with coumaphos , atrazine , 2,4-DMPF, chlorpyrifos ... |